Gene Activity List


Gene Activity List

Gene Compound Assay Inh Ic50 Ki View
calcium channel, voltage-dependent, gamma subunit 7 CHLORPROMAZINE Calcium Channel Type L, Benzothiazepine 91% 3.214uM 2.857uM View
calcium channel, voltage-dependent, gamma subunit 6 CHLORPROMAZINE Calcium Channel Type L, Benzothiazepine 91% 3.214uM 2.857uM View
calcium channel, voltage-dependent, gamma subunit 5 CHLORPROMAZINE Calcium Channel Type L, Benzothiazepine 91% 3.214uM 2.857uM View
calcium channel, voltage-dependent, gamma subunit 4 CHLORPROMAZINE Calcium Channel Type L, Benzothiazepine 91% 3.214uM 2.857uM View
calcium channel, voltage-dependent, gamma subunit 3 CHLORPROMAZINE Calcium Channel Type L, Benzothiazepine 91% 3.214uM 2.857uM View
calcium channel, voltage-dependent, gamma subunit 2 CHLORPROMAZINE Calcium Channel Type L, Benzothiazepine 91% 3.214uM 2.857uM View
calcium channel, voltage-dependent, gamma subunit 1 CHLORPROMAZINE Calcium Channel Type L, Benzothiazepine 91% 3.214uM 2.857uM View
calcium channel, voltage-dependent, L type, alpha 1S subunit CLOZAPINE Calcium Channel Type L, Phenylalkylamine 91% .612uM .595uM View
calcium channel, voltage-dependent, alpha 1F subunit CLOZAPINE Calcium Channel Type L, Phenylalkylamine 91% .612uM .595uM View
calcium channel, voltage-dependent, L type, alpha 1D subunit CLOZAPINE Calcium Channel Type L, Phenylalkylamine 91% .612uM .595uM View
calcium channel, voltage-dependent, L type, alpha 1C subunit CLOZAPINE Calcium Channel Type L, Phenylalkylamine 91% .612uM .595uM View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit CLOZAPINE Calcium Channel Type L, Phenylalkylamine 91% .612uM .595uM View
calcium channel, voltage-dependent, beta 1 subunit CLOZAPINE Calcium Channel Type L, Phenylalkylamine 91% .612uM .595uM View
calcium channel, voltage-dependent, L type, alpha 1E subunit CLOZAPINE Calcium Channel Type L, Phenylalkylamine 91% .612uM .595uM View
calcium channel, voltage-dependent, N type, alpha 1B subunit CLOZAPINE Calcium Channel Type L, Phenylalkylamine 91% .612uM .595uM View
calcium channel, voltage-dependent, alpha2/delta subunit 1 CLOZAPINE Calcium Channel Type L, Phenylalkylamine 91% .612uM .595uM View
5-hydroxytryptamine receptor 6 CARVEDILOL Serotonin 5-HT6 91% 1.519uM .705uM View
dopamine receptor 2 CLOZAPINE Dopamine D2L 91% .387uM .129uM View
opioid receptor, sigma 1 DEXFENFLURAMINE Sigma1 91% .516uM .217uM View
Cytochrome P450, subfamily IIC (mephenytoin 4-hydroxylase) BENZBROMARONE CYP450-2C9 Inhibition 91% .016uM NoneNone View
cytochrome P450, family 2, subfamily C, polypeptide 9 BENZBROMARONE CYP450-2C9 Inhibition 91% .016uM NoneNone View
opioid receptor, kappa 1 BENZOTHIAZYL DISULFIDE Opiate kappa 91% 1.243uM .497uM View
progesterone receptor DESOXIMETASONE Progesterone 91% .084uM .011uM View
progesterone receptor DESOXIMETASONE Progesterone 91% .084uM .011uM View
progesterone receptor FLUNISOLIDE Progesterone 91% .359uM .047uM View
progesterone receptor FLUNISOLIDE Progesterone 91% .359uM .047uM View
5-hydroxytryptamine (serotonin) receptor 1A FLUPHENAZINE Serotonin 5-HT1A 91% 1.644uM .939uM View
adrenergic receptor, alpha 2b BENZOTHIAZYL DISULFIDE Adrenergic alpha2C 91% 1.658uM .241uM View
adrenergic receptor, alpha 2c (Non-specific probe) BENZOTHIAZYL DISULFIDE Adrenergic alpha2C 91% 1.658uM .241uM View
dopamine receptor D3 DOXEPIN Dopamine D3 91% 1.393uM .473uM View
prostaglandin-endoperoxide synthase 1 MELOXICAM Cyclooxygenase COX-1 91% 1.319uM NoneNone View
prostaglandin-endoperoxide synthase 1 (prostaglandin G/H synthase and cyclooxygenase) MELOXICAM Cyclooxygenase COX-1 91% 1.319uM NoneNone View
adrenergic receptor, alpha 2a TRAZODONE Adrenergic alpha2A 91% .909uM .341uM View
adrenergic receptor, alpha 2b TOLPERISONE Adrenergic alpha2B 91% 1uM .456uM View
adrenergic receptor, alpha 2b HALOPERIDOL Adrenergic alpha2C 91% 1.845uM .268uM View
adrenergic receptor, alpha 2c (Non-specific probe) HALOPERIDOL Adrenergic alpha2C 91% 1.845uM .268uM View
epidermal growth factor receptor GENTIAN VIOLET Protein Tyrosine Kinase, EGF Receptor 91% .473uM NoneNone View
sodium channel, voltage-gated, type IV, beta VERAPAMIL Sodium Channel, Site 2 91% 2.005uM 1.83uM View
sodium channel associated protein 1 VERAPAMIL Sodium Channel, Site 2 91% 2.005uM 1.83uM View
sodium channel associated protein 2 VERAPAMIL Sodium Channel, Site 2 91% 2.005uM 1.83uM View
sodium channel, voltage-gated, type III, beta VERAPAMIL Sodium Channel, Site 2 91% 2.005uM 1.83uM View
sodium channel, voltage-gated, type I, alpha VERAPAMIL Sodium Channel, Site 2 91% 2.005uM 1.83uM View
sodium channel, voltage-gated, type IX, alpha VERAPAMIL Sodium Channel, Site 2 91% 2.005uM 1.83uM View
sodium channel, voltage-gated, type VII, alpha VERAPAMIL Sodium Channel, Site 2 91% 2.005uM 1.83uM View
amiloride-sensitive cation channel 5, intestinal VERAPAMIL Sodium Channel, Site 2 91% 2.005uM 1.83uM View
sodium channel, voltage-gated, type III, beta VERAPAMIL Sodium Channel, Site 2 91% 2.005uM 1.83uM View
sodium channel, voltage-gated, type VIII, alpha polypeptide VERAPAMIL Sodium Channel, Site 2 91% 2.005uM 1.83uM View
sodium channel, voltage-gated, type XI, alpha VERAPAMIL Sodium Channel, Site 2 91% 2.005uM 1.83uM View
sodium channel, voltage-gated, type I, beta VERAPAMIL Sodium Channel, Site 2 91% 2.005uM 1.83uM View
sodium channel, voltage-gated, type 10, alpha polypeptide VERAPAMIL Sodium Channel, Site 2 91% 2.005uM 1.83uM View
sodium channel, voltage-gated, type IV, alpha polypeptide VERAPAMIL Sodium Channel, Site 2 91% 2.005uM 1.83uM View
sodium channel, voltage-gated, type V, alpha polypeptide VERAPAMIL Sodium Channel, Site 2 91% 2.005uM 1.83uM View
sodium channel, voltage-gated, type II, beta VERAPAMIL Sodium Channel, Site 2 91% 2.005uM 1.83uM View
sodium channel, nonvoltage-gated 1 alpha VERAPAMIL Sodium Channel, Site 2 91% 2.005uM 1.83uM View
sodium channel, nonvoltage-gated 1 gamma VERAPAMIL Sodium Channel, Site 2 91% 2.005uM 1.83uM View
sodium channel, nonvoltage-gated 1 beta VERAPAMIL Sodium Channel, Site 2 91% 2.005uM 1.83uM View
sodium channel, voltage-gated, type 2, alpha 1 polypeptide VERAPAMIL Sodium Channel, Site 2 91% 2.005uM 1.83uM View
sodium channel, voltage-gated, type XI, alpha VERAPAMIL Sodium Channel, Site 2 91% 2.005uM 1.83uM View
sodium channel, nonvoltage-gated 1, gamma VERAPAMIL Sodium Channel, Site 2 91% 2.005uM 1.83uM View
sodium channel, nonvoltage-gated 1, delta VERAPAMIL Sodium Channel, Site 2 91% 2.005uM 1.83uM View
sodium channel, nonvoltage-gated 1, beta (Liddle syndrome) VERAPAMIL Sodium Channel, Site 2 91% 2.005uM 1.83uM View
calcium channel, voltage-dependent, beta 4 subunit TAMOXIFEN Calcium Channel Type L, Phenylalkylamine 92% 2.042uM 1.985uM View
calcium channel, voltage-dependent, beta 3 subunit TAMOXIFEN Calcium Channel Type L, Phenylalkylamine 92% 2.042uM 1.985uM View
calcium channel, voltage-dependent, beta 2 subunit TAMOXIFEN Calcium Channel Type L, Phenylalkylamine 92% 2.042uM 1.985uM View
calcium channel, voltage-dependent, L type, alpha 1S subunit TAMOXIFEN Calcium Channel Type L, Phenylalkylamine 92% 2.042uM 1.985uM View
calcium channel, voltage-dependent, alpha 1F subunit TAMOXIFEN Calcium Channel Type L, Phenylalkylamine 92% 2.042uM 1.985uM View
calcium channel, voltage-dependent, L type, alpha 1D subunit TAMOXIFEN Calcium Channel Type L, Phenylalkylamine 92% 2.042uM 1.985uM View
calcium channel, voltage-dependent, L type, alpha 1C subunit TAMOXIFEN Calcium Channel Type L, Phenylalkylamine 92% 2.042uM 1.985uM View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit TAMOXIFEN Calcium Channel Type L, Phenylalkylamine 92% 2.042uM 1.985uM View
calcium channel, voltage-dependent, beta 1 subunit TAMOXIFEN Calcium Channel Type L, Phenylalkylamine 92% 2.042uM 1.985uM View
calcium channel, voltage-dependent, L type, alpha 1E subunit TAMOXIFEN Calcium Channel Type L, Phenylalkylamine 92% 2.042uM 1.985uM View
calcium channel, voltage-dependent, N type, alpha 1B subunit TAMOXIFEN Calcium Channel Type L, Phenylalkylamine 92% 2.042uM 1.985uM View
calcium channel, voltage-dependent, alpha2/delta subunit 1 TAMOXIFEN Calcium Channel Type L, Phenylalkylamine 92% 2.042uM 1.985uM View
adrenergic receptor, beta 3 TAMOXIFEN Adrenergic beta3 92% 7.703uM 5.778uM View
calcium channel, voltage-dependent, gamma subunit 8 CISAPRIDE Calcium Channel Type L, Phenylalkylamine 92% .53uM .515uM View
calcium channel, voltage-dependent, gamma subunit 7 CISAPRIDE Calcium Channel Type L, Phenylalkylamine 92% .53uM .515uM View
calcium channel, voltage-dependent, gamma subunit 6 CISAPRIDE Calcium Channel Type L, Phenylalkylamine 92% .53uM .515uM View
calcium channel, voltage-dependent, gamma subunit 5 CISAPRIDE Calcium Channel Type L, Phenylalkylamine 92% .53uM .515uM View
calcium channel, voltage-dependent, gamma subunit 4 CISAPRIDE Calcium Channel Type L, Phenylalkylamine 92% .53uM .515uM View
calcium channel, voltage-dependent, gamma subunit 3 CISAPRIDE Calcium Channel Type L, Phenylalkylamine 92% .53uM .515uM View
calcium channel, voltage-dependent, gamma subunit 2 CISAPRIDE Calcium Channel Type L, Phenylalkylamine 92% .53uM .515uM View
calcium channel, voltage-dependent, gamma subunit 1 CISAPRIDE Calcium Channel Type L, Phenylalkylamine 92% .53uM .515uM View
calcium channel, voltage-dependent, beta 4 subunit CISAPRIDE Calcium Channel Type L, Phenylalkylamine 92% .53uM .515uM View
calcium channel, voltage-dependent, beta 3 subunit CISAPRIDE Calcium Channel Type L, Phenylalkylamine 92% .53uM .515uM View
calcium channel, voltage-dependent, beta 2 subunit CISAPRIDE Calcium Channel Type L, Phenylalkylamine 92% .53uM .515uM View
calcium channel, voltage-dependent, L type, alpha 1S subunit CISAPRIDE Calcium Channel Type L, Phenylalkylamine 92% .53uM .515uM View
calcium channel, voltage-dependent, alpha 1F subunit CISAPRIDE Calcium Channel Type L, Phenylalkylamine 92% .53uM .515uM View
calcium channel, voltage-dependent, L type, alpha 1D subunit CISAPRIDE Calcium Channel Type L, Phenylalkylamine 92% .53uM .515uM View
calcium channel, voltage-dependent, L type, alpha 1C subunit CISAPRIDE Calcium Channel Type L, Phenylalkylamine 92% .53uM .515uM View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit CISAPRIDE Calcium Channel Type L, Phenylalkylamine 92% .53uM .515uM View
calcium channel, voltage-dependent, beta 1 subunit CISAPRIDE Calcium Channel Type L, Phenylalkylamine 92% .53uM .515uM View
calcium channel, voltage-dependent, L type, alpha 1E subunit CISAPRIDE Calcium Channel Type L, Phenylalkylamine 92% .53uM .515uM View
calcium channel, voltage-dependent, N type, alpha 1B subunit CISAPRIDE Calcium Channel Type L, Phenylalkylamine 92% .53uM .515uM View
calcium channel, voltage-dependent, alpha2/delta subunit 1 CISAPRIDE Calcium Channel Type L, Phenylalkylamine 92% .53uM .515uM View
calcium channel, voltage-dependent, gamma subunit 3 DICYCLOMINE Calcium Channel Type L, Phenylalkylamine 92% .11uM .107uM View
calcium channel, voltage-dependent, gamma subunit 2 DICYCLOMINE Calcium Channel Type L, Phenylalkylamine 92% .11uM .107uM View
glycine receptor, alpha 1 subunit IVERMECTIN Glycine, Strychnine-Sensitive 92% .3747uM .2118uM View
glycine receptor, beta subunit IVERMECTIN Glycine, Strychnine-Sensitive 92% .3747uM .2118uM View
glycine receptor, alpha 2 subunit IVERMECTIN Glycine, Strychnine-Sensitive 92% .3747uM .2118uM View
cholinergic receptor, muscarinic 5 IVERMECTIN Muscarinic M5 92% 3.608uM 2.5922uM View
Cytochrom P450-2D6 monooxygenase LISURIDE CYP450-2D6 Inhibition 92% .016uM NoneNone View
cytochrome P450, family 3, subfamily a, polypeptide 13 ERGOTAMINE CYP450-3A4 Inhibition 92% 1uM NoneNone View
calcium channel, voltage-dependent, gamma subunit 8 PROMAZINE Calcium Channel Type L, Phenylalkylamine 92% 1.193uM 1.16uM View
calcium channel, voltage-dependent, gamma subunit 7 PROMAZINE Calcium Channel Type L, Phenylalkylamine 92% 1.193uM 1.16uM View
calcium channel, voltage-dependent, gamma subunit 6 PROMAZINE Calcium Channel Type L, Phenylalkylamine 92% 1.193uM 1.16uM View
calcium channel, voltage-dependent, gamma subunit 5 PROMAZINE Calcium Channel Type L, Phenylalkylamine 92% 1.193uM 1.16uM View
calcium channel, voltage-dependent, gamma subunit 4 PROMAZINE Calcium Channel Type L, Phenylalkylamine 92% 1.193uM 1.16uM View
calcium channel, voltage-dependent, gamma subunit 3 PROMAZINE Calcium Channel Type L, Phenylalkylamine 92% 1.193uM 1.16uM View
calcium channel, voltage-dependent, gamma subunit 2 PROMAZINE Calcium Channel Type L, Phenylalkylamine 92% 1.193uM 1.16uM View
calcium channel, voltage-dependent, gamma subunit 1 PROMAZINE Calcium Channel Type L, Phenylalkylamine 92% 1.193uM 1.16uM View
calcium channel, voltage-dependent, beta 4 subunit PROMAZINE Calcium Channel Type L, Phenylalkylamine 92% 1.193uM 1.16uM View
calcium channel, voltage-dependent, beta 3 subunit PROMAZINE Calcium Channel Type L, Phenylalkylamine 92% 1.193uM 1.16uM View
calcium channel, voltage-dependent, beta 2 subunit PROMAZINE Calcium Channel Type L, Phenylalkylamine 92% 1.193uM 1.16uM View
calcium channel, voltage-dependent, L type, alpha 1S subunit PROMAZINE Calcium Channel Type L, Phenylalkylamine 92% 1.193uM 1.16uM View
calcium channel, voltage-dependent, alpha 1F subunit PROMAZINE Calcium Channel Type L, Phenylalkylamine 92% 1.193uM 1.16uM View
calcium channel, voltage-dependent, L type, alpha 1D subunit PROMAZINE Calcium Channel Type L, Phenylalkylamine 92% 1.193uM 1.16uM View
calcium channel, voltage-dependent, L type, alpha 1C subunit PROMAZINE Calcium Channel Type L, Phenylalkylamine 92% 1.193uM 1.16uM View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit PROMAZINE Calcium Channel Type L, Phenylalkylamine 92% 1.193uM 1.16uM View
calcium channel, voltage-dependent, beta 1 subunit PROMAZINE Calcium Channel Type L, Phenylalkylamine 92% 1.193uM 1.16uM View
calcium channel, voltage-dependent, L type, alpha 1E subunit PROMAZINE Calcium Channel Type L, Phenylalkylamine 92% 1.193uM 1.16uM View
calcium channel, voltage-dependent, N type, alpha 1B subunit PROMAZINE Calcium Channel Type L, Phenylalkylamine 92% 1.193uM 1.16uM View
calcium channel, voltage-dependent, alpha2/delta subunit 1 PROMAZINE Calcium Channel Type L, Phenylalkylamine 92% 1.193uM 1.16uM View
dopamine receptor D3 QUETIAPINE Dopamine D3 92% 1.1632uM .3951uM View
adrenergic receptor, alpha 1a EPINEPHRINE Adrenergic alpha1A 92% .628uM .254uM View
opioid receptor, sigma 1 TERCONAZOLE Sigma1 92% .508uM .214uM View
5-hydroxytryptamine (serotonin) receptor 1A SUMATRIPTAN Serotonin 5-HT1A 92% .804uM .459uM View
cholinergic receptor, muscarinic 2 PAROXETINE Muscarinic M2 92% .532uM .189uM View
adrenergic receptor, alpha 2b CYPROHEPTADINE Adrenergic alpha2C 92% 1.275uM .185uM View
adrenergic receptor, alpha 2c (Non-specific probe) CYPROHEPTADINE Adrenergic alpha2C 92% 1.275uM .185uM View
solute carrier family 6 (neurotransmitter transporter, serotonin), member 4 PIPAMAZINE Serotonin Transporter 92% .651uM .346uM View
adrenergic receptor, alpha 2a ECONAZOLE Adrenergic alpha2A 92% 4.325uM 1.622uM View
cytochrome P450, family 3, subfamily a, polypeptide 13 ECONAZOLE CYP450-3A4 Inhibition 92% .05uM NoneNone View
calcium channel, voltage-dependent, alpha 1F subunit MICONAZOLE Calcium Channel Type L, Dihydropyridine 92% 6.266uM 4.028uM View
calcium channel, voltage-dependent, L type, alpha 1D subunit MICONAZOLE Calcium Channel Type L, Dihydropyridine 92% 6.266uM 4.028uM View
calcium channel, voltage-dependent, L type, alpha 1C subunit MICONAZOLE Calcium Channel Type L, Dihydropyridine 92% 6.266uM 4.028uM View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit MICONAZOLE Calcium Channel Type L, Dihydropyridine 92% 6.266uM 4.028uM View
calcium channel, voltage-dependent, beta 1 subunit MICONAZOLE Calcium Channel Type L, Dihydropyridine 92% 6.266uM 4.028uM View
calcium channel, voltage-dependent, L type, alpha 1E subunit MICONAZOLE Calcium Channel Type L, Dihydropyridine 92% 6.266uM 4.028uM View
calcium channel, voltage-dependent, N type, alpha 1B subunit MICONAZOLE Calcium Channel Type L, Dihydropyridine 92% 6.266uM 4.028uM View
calcium channel, voltage-dependent, alpha2/delta subunit 1 MICONAZOLE Calcium Channel Type L, Dihydropyridine 92% 6.266uM 4.028uM View
calcium channel, voltage-dependent, gamma subunit 8 MICONAZOLE Calcium Channel Type L, Dihydropyridine 92% 6.266uM 4.028uM View
calcium channel, voltage-dependent, gamma subunit 7 MICONAZOLE Calcium Channel Type L, Dihydropyridine 92% 6.266uM 4.028uM View
calcium channel, voltage-dependent, gamma subunit 6 MICONAZOLE Calcium Channel Type L, Dihydropyridine 92% 6.266uM 4.028uM View
calcium channel, voltage-dependent, gamma subunit 5 MICONAZOLE Calcium Channel Type L, Dihydropyridine 92% 6.266uM 4.028uM View
calcium channel, voltage-dependent, gamma subunit 4 MICONAZOLE Calcium Channel Type L, Dihydropyridine 92% 6.266uM 4.028uM View
calcium channel, voltage-dependent, gamma subunit 3 MICONAZOLE Calcium Channel Type L, Dihydropyridine 92% 6.266uM 4.028uM View
calcium channel, voltage-dependent, gamma subunit 2 MICONAZOLE Calcium Channel Type L, Dihydropyridine 92% 6.266uM 4.028uM View
calcium channel, voltage-dependent, gamma subunit 1 MICONAZOLE Calcium Channel Type L, Dihydropyridine 92% 6.266uM 4.028uM View
calcium channel, voltage-dependent, beta 4 subunit MICONAZOLE Calcium Channel Type L, Dihydropyridine 92% 6.266uM 4.028uM View
calcium channel, voltage-dependent, beta 3 subunit MICONAZOLE Calcium Channel Type L, Dihydropyridine 92% 6.266uM 4.028uM View
calcium channel, voltage-dependent, beta 2 subunit MICONAZOLE Calcium Channel Type L, Dihydropyridine 92% 6.266uM 4.028uM View
calcium channel, voltage-dependent, L type, alpha 1S subunit MICONAZOLE Calcium Channel Type L, Dihydropyridine 92% 6.266uM 4.028uM View
ATPase, Na+/K+ transporting, alpha 4 polypeptide OUABAIN ATPase, Na+/K+ 92% .678uM NoneNone View
ATPase, Na+/K+ transporting, alpha 3 polypeptide OUABAIN ATPase, Na+/K+ 92% .678uM NoneNone View
ATPase, Na+/K+ transporting, alpha 2 polypeptide OUABAIN ATPase, Na+/K+ 92% .678uM NoneNone View
calcium channel, voltage-dependent, gamma subunit 5 THIORIDAZINE Calcium Channel Type L, Benzothiazepine 91% .469uM .417uM View
calcium channel, voltage-dependent, gamma subunit 4 THIORIDAZINE Calcium Channel Type L, Benzothiazepine 91% .469uM .417uM View
calcium channel, voltage-dependent, gamma subunit 3 THIORIDAZINE Calcium Channel Type L, Benzothiazepine 91% .469uM .417uM View
calcium channel, voltage-dependent, gamma subunit 2 THIORIDAZINE Calcium Channel Type L, Benzothiazepine 91% .469uM .417uM View
calcium channel, voltage-dependent, gamma subunit 1 THIORIDAZINE Calcium Channel Type L, Benzothiazepine 91% .469uM .417uM View
calcium channel, voltage-dependent, beta 4 subunit THIORIDAZINE Calcium Channel Type L, Benzothiazepine 91% .469uM .417uM View
Cytochrome P450, subfamily IIC (mephenytoin 4-hydroxylase) TANNIC ACID CYP450-2C9 Inhibition 91% 4.6074uM NoneNone View
cytochrome P450, family 2, subfamily C, polypeptide 9 TANNIC ACID CYP450-2C9 Inhibition 91% 4.6074uM NoneNone View
A3 adenosine receptor ZAFIRLUKAST Adenosine A3 91% 1.363uM .77uM View
lymphocyte protein tyrosine kinase (mapped) BITHIONOL Protein Tyrosine Kinase, Lck 91% 2.255uM NoneNone View
adrenergic receptor, alpha 1d (Non-specific probe) BENZTROPINE Adrenergic alpha1D 91% .052uM .026uM View
adrenergic receptor, alpha 1a CINNARIZINE Adrenergic alpha1A 91% 1.919uM .777uM View
solute carrier family 6 (neurotransmitter transporter, dopamine), member 3 PEMOLINE Dopamine Transporter 91% .5213uM .4142uM View
adrenergic receptor, alpha 1b FLUNARIZINE Adrenergic alpha1B 91% 1.096uM .606uM View
angiotensin 1 converting enzyme 1 QUINAPRIL Protease, Angiotensin Converting Enzyme 91% 4.008uM NoneNone View
angiotensin I converting enzyme (peptidyl-dipeptidase A) 1 QUINAPRIL Protease, Angiotensin Converting Enzyme 91% 4.008uM NoneNone View
adrenergic receptor, alpha 1d (Non-specific probe) QUETIAPINE Adrenergic alpha1D 91% .0966uM .0475uM View
opioid receptor, sigma 1 TERBINAFINE Sigma1 91% .5602uM .2354uM View
cholinergic receptor, muscarinic 1 TERCONAZOLE Muscarinic M1 91% 5.709uM 1.375uM View
arachidonate 15-lipoxygenase, second type TERCONAZOLE Lipoxygenase 15-LO 91% 2.446uM NoneNone View
arachidonate 15-lipoxygenase TERCONAZOLE Lipoxygenase 15-LO 91% 2.446uM NoneNone View
arachidonate 15-lipoxygenase TERCONAZOLE Lipoxygenase 15-LO 91% 2.446uM NoneNone View
adrenergic receptor, alpha 2a SEMUSTINE Imidazoline I2, Central 91% 1.615uM 1.077uM View
adrenergic receptor, alpha 2c (Non-specific probe) SEMUSTINE Imidazoline I2, Central 91% 1.615uM 1.077uM View
adrenergic receptor, alpha 1a PENTAMIDINE Adrenergic alpha1A 91% 1.212uM .491uM View
adrenergic receptor, alpha 1d (Non-specific probe) METERGOLINE Adrenergic alpha1D 91% .136uM .067uM View
cholinergic receptor, muscarinic 4 PROCHLORPERAZINE Muscarinic M4 91% 1.363uM .19uM View
Cytochrome P450, subfamily IIC (mephenytoin 4-hydroxylase) FLUVASTATIN CYP450-2C9 Inhibition 91% .4uM NoneNone View
cytochrome P450, family 2, subfamily C, polypeptide 9 FLUVASTATIN CYP450-2C9 Inhibition 91% .4uM NoneNone View
solute carrier family 6 (neurotransmitter transporter, noradrenalin), member 2 CYPROHEPTADINE Adrenergic, Norepinephrine Transporter 91% .564uM .559uM View
opioid receptor, sigma 1 NOVARTIS P-38 INHIBITOR Sigma1 91% .7951uM .3342uM View
adenosine A2a receptor ECONAZOLE Adenosine A2A 91% 14.616uM 8.206uM View
Cytochrom P450-1A2 monooxygenase ECONAZOLE CYP450-1A2 Inhibition 91% .3uM NoneNone View
dopamine receptor D4 MICONAZOLE Dopamine D4.2 91% 15.27uM 5.354uM View
melanocortin 4 receptor MICONAZOLE Melanocortin MC4 91% 12.448uM 11.97uM View
prostaglandin-endoperoxide synthase 2 INDOMETHACIN Cyclooxygenase COX-2 91% .84uM NoneNone View
prostaglandin-endoperoxide synthase 2 (prostaglandin G/H synthase and cyclooxygenase) INDOMETHACIN Cyclooxygenase COX-2 91% .84uM NoneNone View
cholinergic receptor, muscarinic 4 DEXCHLORPHENIRAMINE Muscarinic M4 91% 1.976uM .276uM View
adrenergic receptor, alpha 2b DEXCHLORPHENIRAMINE Adrenergic alpha2B 91% 4.607uM 2.103uM View
5-hydroxytryptamine (serotonin) receptor 2B SULCONAZOLE Serotonin 5-HT2B 91% 3.02uM 1.922uM View
adrenergic receptor, alpha 2a SULCONAZOLE Adrenergic alpha2A 91% 4.043uM 1.516uM View
5-hydroxytryptamine (serotonin) receptor 2A LY-294002 Serotonin 5-HT2A 91% 2.796uM .799uM View
progesterone receptor MEDROXYPROGESTERONE Progesterone 91% .711uM .093uM View
thromboxane A synthase 1 HEXACHLOROPHENE Thromboxane Synthetase 91% 3.087uM NoneNone View
thromboxane A synthase 1 (platelet, cytochrome P450, family 5, subfamily A) HEXACHLOROPHENE Thromboxane Synthetase 91% 3.087uM NoneNone View