Gene Activity List


Gene Activity List

Gene Compound Assay Inh Ic50 Ki View
Sigma-2 Receptor TAMOXIFEN Sigma2 78% .619uM .381uM View
calcium channel, voltage-dependent, gamma subunit 8 BENZTROPINE Calcium Channel Type L, Phenylalkylamine 78% 1.348uM 1.311uM View
calcium channel, voltage-dependent, gamma subunit 7 BENZTROPINE Calcium Channel Type L, Phenylalkylamine 78% 1.348uM 1.311uM View
calcium channel, voltage-dependent, gamma subunit 6 BENZTROPINE Calcium Channel Type L, Phenylalkylamine 78% 1.348uM 1.311uM View
calcium channel, voltage-dependent, gamma subunit 5 BENZTROPINE Calcium Channel Type L, Phenylalkylamine 78% 1.348uM 1.311uM View
calcium channel, voltage-dependent, gamma subunit 4 BENZTROPINE Calcium Channel Type L, Phenylalkylamine 78% 1.348uM 1.311uM View
calcium channel, voltage-dependent, gamma subunit 3 BENZTROPINE Calcium Channel Type L, Phenylalkylamine 78% 1.348uM 1.311uM View
calcium channel, voltage-dependent, gamma subunit 8 SPIRADOLINE Calcium Channel Type L, Phenylalkylamine 78% 5.24uM 5.095uM View
calcium channel, voltage-dependent, gamma subunit 7 SPIRADOLINE Calcium Channel Type L, Phenylalkylamine 78% 5.24uM 5.095uM View
calcium channel, voltage-dependent, gamma subunit 6 SPIRADOLINE Calcium Channel Type L, Phenylalkylamine 78% 5.24uM 5.095uM View
calcium channel, voltage-dependent, gamma subunit 5 SPIRADOLINE Calcium Channel Type L, Phenylalkylamine 78% 5.24uM 5.095uM View
calcium channel, voltage-dependent, gamma subunit 4 SPIRADOLINE Calcium Channel Type L, Phenylalkylamine 78% 5.24uM 5.095uM View
calcium channel, voltage-dependent, gamma subunit 3 SPIRADOLINE Calcium Channel Type L, Phenylalkylamine 78% 5.24uM 5.095uM View
calcium channel, voltage-dependent, gamma subunit 2 SPIRADOLINE Calcium Channel Type L, Phenylalkylamine 78% 5.24uM 5.095uM View
calcium channel, voltage-dependent, gamma subunit 1 SPIRADOLINE Calcium Channel Type L, Phenylalkylamine 78% 5.24uM 5.095uM View
calcium channel, voltage-dependent, beta 4 subunit SPIRADOLINE Calcium Channel Type L, Phenylalkylamine 78% 5.24uM 5.095uM View
calcium channel, voltage-dependent, beta 3 subunit SPIRADOLINE Calcium Channel Type L, Phenylalkylamine 78% 5.24uM 5.095uM View
calcium channel, voltage-dependent, beta 2 subunit SPIRADOLINE Calcium Channel Type L, Phenylalkylamine 78% 5.24uM 5.095uM View
calcium channel, voltage-dependent, L type, alpha 1S subunit SPIRADOLINE Calcium Channel Type L, Phenylalkylamine 78% 5.24uM 5.095uM View
calcium channel, voltage-dependent, alpha 1F subunit SPIRADOLINE Calcium Channel Type L, Phenylalkylamine 78% 5.24uM 5.095uM View
calcium channel, voltage-dependent, L type, alpha 1D subunit SPIRADOLINE Calcium Channel Type L, Phenylalkylamine 78% 5.24uM 5.095uM View
calcium channel, voltage-dependent, L type, alpha 1C subunit SPIRADOLINE Calcium Channel Type L, Phenylalkylamine 78% 5.24uM 5.095uM View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit SPIRADOLINE Calcium Channel Type L, Phenylalkylamine 78% 5.24uM 5.095uM View
calcium channel, voltage-dependent, beta 1 subunit SPIRADOLINE Calcium Channel Type L, Phenylalkylamine 78% 5.24uM 5.095uM View
calcium channel, voltage-dependent, gamma subunit 3 PROMAZINE Calcium Channel Type L, Benzothiazepine 77% 3.217uM 2.86uM View
calcium channel, voltage-dependent, gamma subunit 2 PROMAZINE Calcium Channel Type L, Benzothiazepine 77% 3.217uM 2.86uM View
calcium channel, voltage-dependent, gamma subunit 1 PROMAZINE Calcium Channel Type L, Benzothiazepine 77% 3.217uM 2.86uM View
calcium channel, voltage-dependent, beta 4 subunit PROMAZINE Calcium Channel Type L, Benzothiazepine 77% 3.217uM 2.86uM View
calcium channel, voltage-dependent, beta 3 subunit PROMAZINE Calcium Channel Type L, Benzothiazepine 77% 3.217uM 2.86uM View
calcium channel, voltage-dependent, beta 2 subunit PROMAZINE Calcium Channel Type L, Benzothiazepine 77% 3.217uM 2.86uM View
calcium channel, voltage-dependent, L type, alpha 1S subunit PROMAZINE Calcium Channel Type L, Benzothiazepine 77% 3.217uM 2.86uM View
calcium channel, voltage-dependent, alpha 1F subunit PROMAZINE Calcium Channel Type L, Benzothiazepine 77% 3.217uM 2.86uM View
calcium channel, voltage-dependent, L type, alpha 1D subunit PROMAZINE Calcium Channel Type L, Benzothiazepine 77% 3.217uM 2.86uM View
calcium channel, voltage-dependent, L type, alpha 1C subunit PROMAZINE Calcium Channel Type L, Benzothiazepine 77% 3.217uM 2.86uM View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit PROMAZINE Calcium Channel Type L, Benzothiazepine 77% 3.217uM 2.86uM View
calcium channel, voltage-dependent, beta 1 subunit PROMAZINE Calcium Channel Type L, Benzothiazepine 77% 3.217uM 2.86uM View
calcium channel, voltage-dependent, L type, alpha 1E subunit PROMAZINE Calcium Channel Type L, Benzothiazepine 77% 3.217uM 2.86uM View
calcium channel, voltage-dependent, N type, alpha 1B subunit PROMAZINE Calcium Channel Type L, Benzothiazepine 77% 3.217uM 2.86uM View
calcium channel, voltage-dependent, alpha2/delta subunit 1 PROMAZINE Calcium Channel Type L, Benzothiazepine 77% 3.217uM 2.86uM View
sodium channel, voltage-gated, type XI, alpha PROMAZINE Sodium Channel, Site 2 77% 2.573uM 2.347uM View
sodium channel, voltage-gated, type I, beta PROMAZINE Sodium Channel, Site 2 77% 2.573uM 2.347uM View
sodium channel, voltage-gated, type 10, alpha polypeptide PROMAZINE Sodium Channel, Site 2 77% 2.573uM 2.347uM View
sodium channel, voltage-gated, type IV, alpha polypeptide PROMAZINE Sodium Channel, Site 2 77% 2.573uM 2.347uM View
sodium channel, voltage-gated, type V, alpha polypeptide PROMAZINE Sodium Channel, Site 2 77% 2.573uM 2.347uM View
sodium channel, voltage-gated, type II, beta PROMAZINE Sodium Channel, Site 2 77% 2.573uM 2.347uM View
sodium channel, nonvoltage-gated 1 alpha PROMAZINE Sodium Channel, Site 2 77% 2.573uM 2.347uM View
sodium channel, nonvoltage-gated 1 gamma PROMAZINE Sodium Channel, Site 2 77% 2.573uM 2.347uM View
sodium channel, nonvoltage-gated 1 beta PROMAZINE Sodium Channel, Site 2 77% 2.573uM 2.347uM View
sodium channel, voltage-gated, type 2, alpha 1 polypeptide PROMAZINE Sodium Channel, Site 2 77% 2.573uM 2.347uM View
sodium channel, voltage-gated, type XI, alpha PROMAZINE Sodium Channel, Site 2 77% 2.573uM 2.347uM View
sodium channel, nonvoltage-gated 1, gamma PROMAZINE Sodium Channel, Site 2 77% 2.573uM 2.347uM View
sodium channel, nonvoltage-gated 1, delta PROMAZINE Sodium Channel, Site 2 77% 2.573uM 2.347uM View
sodium channel, nonvoltage-gated 1, beta (Liddle syndrome) PROMAZINE Sodium Channel, Site 2 77% 2.573uM 2.347uM View
sodium channel, nonvoltage-gated 1 alpha PROMAZINE Sodium Channel, Site 2 77% 2.573uM 2.347uM View
sodium channel, voltage-gated, type X, alpha PROMAZINE Sodium Channel, Site 2 77% 2.573uM 2.347uM View
sodium channel, voltage-gated, type IX, alpha PROMAZINE Sodium Channel, Site 2 77% 2.573uM 2.347uM View
sodium channel, voltage gated, type VIII, alpha PROMAZINE Sodium Channel, Site 2 77% 2.573uM 2.347uM View
sodium channel, voltage-gated, type VII, alpha PROMAZINE Sodium Channel, Site 2 77% 2.573uM 2.347uM View
sodium channel, voltage-gated, type V, alpha (long QT syndrome 3) PROMAZINE Sodium Channel, Site 2 77% 2.573uM 2.347uM View
sodium channel, voltage-gated, type IV, beta PROMAZINE Sodium Channel, Site 2 77% 2.573uM 2.347uM View
sodium channel, voltage-gated, type IV, alpha PROMAZINE Sodium Channel, Site 2 77% 2.573uM 2.347uM View
sodium channel, voltage-gated, type III, alpha PROMAZINE Sodium Channel, Site 2 77% 2.573uM 2.347uM View
sodium channel, voltage-gated, type II, beta PROMAZINE Sodium Channel, Site 2 77% 2.573uM 2.347uM View
sodium channel, voltage-gated, type II, alpha 2 PROMAZINE Sodium Channel, Site 2 77% 2.573uM 2.347uM View
sodium channel, voltage-gated, type I, beta PROMAZINE Sodium Channel, Site 2 77% 2.573uM 2.347uM View
sodium channel, voltage-gated, type I, alpha PROMAZINE Sodium Channel, Site 2 77% 2.573uM 2.347uM View
sodium channel, voltage-gated, type IV, beta PROMAZINE Sodium Channel, Site 2 77% 2.573uM 2.347uM View
sodium channel associated protein 1 PROMAZINE Sodium Channel, Site 2 77% 2.573uM 2.347uM View
sodium channel associated protein 2 PROMAZINE Sodium Channel, Site 2 77% 2.573uM 2.347uM View
sodium channel, voltage-gated, type III, beta PROMAZINE Sodium Channel, Site 2 77% 2.573uM 2.347uM View
sodium channel, voltage-gated, type I, alpha PROMAZINE Sodium Channel, Site 2 77% 2.573uM 2.347uM View
sodium channel, voltage-gated, type IX, alpha PROMAZINE Sodium Channel, Site 2 77% 2.573uM 2.347uM View
sodium channel, voltage-gated, type VII, alpha PROMAZINE Sodium Channel, Site 2 77% 2.573uM 2.347uM View
amiloride-sensitive cation channel 5, intestinal PROMAZINE Sodium Channel, Site 2 77% 2.573uM 2.347uM View
calcium channel, voltage-dependent, L type, alpha 1E subunit PAROXETINE Calcium Channel Type L, Phenylalkylamine 76% .747uM .726uM View
calcium channel, voltage-dependent, N type, alpha 1B subunit PAROXETINE Calcium Channel Type L, Phenylalkylamine 76% .747uM .726uM View
calcium channel, voltage-dependent, alpha2/delta subunit 1 PAROXETINE Calcium Channel Type L, Phenylalkylamine 76% .747uM .726uM View
carbonic anhydrase 5a, mitochondrial ROSIGLITAZONE Carbonic Anhydrase 76% 4.069uM NoneNone View
carbonic anhydrase 3 ROSIGLITAZONE Carbonic Anhydrase 76% 4.069uM NoneNone View
carbonic anhydrase 2 ROSIGLITAZONE Carbonic Anhydrase 76% 4.069uM NoneNone View
carbonic anhydrase 4 ROSIGLITAZONE Carbonic Anhydrase 76% 4.069uM NoneNone View
carbonic anhydrase XI ROSIGLITAZONE Carbonic Anhydrase 76% 4.069uM NoneNone View
carbonic anhydrase IX ROSIGLITAZONE Carbonic Anhydrase 76% 4.069uM NoneNone View
carbonic anhydrase VIII ROSIGLITAZONE Carbonic Anhydrase 76% 4.069uM NoneNone View
carbonic anhydrase VII ROSIGLITAZONE Carbonic Anhydrase 76% 4.069uM NoneNone View
carbonic anhydrase VA, mitochondrial ROSIGLITAZONE Carbonic Anhydrase 76% 4.069uM NoneNone View
carbonic anhydrase IV ROSIGLITAZONE Carbonic Anhydrase 76% 4.069uM NoneNone View
carbonic anhydrase III, muscle specific ROSIGLITAZONE Carbonic Anhydrase 76% 4.069uM NoneNone View
carbonic anhydrase I ROSIGLITAZONE Carbonic Anhydrase 76% 4.069uM NoneNone View
carbonic anhydrase XIV ROSIGLITAZONE Carbonic Anhydrase 76% 4.069uM NoneNone View
carbonic anhydrase VB, mitochondrial ROSIGLITAZONE Carbonic Anhydrase 76% 4.069uM NoneNone View
carbonic anhydrase XII ROSIGLITAZONE Carbonic Anhydrase 76% 4.069uM NoneNone View
carbonic anhydrase VI ROSIGLITAZONE Carbonic Anhydrase 76% 4.069uM NoneNone View
carbonic anhydrase II ROSIGLITAZONE Carbonic Anhydrase 76% 4.069uM NoneNone View
adrenergic receptor, alpha 1b PROPAFENONE Adrenergic alpha1B 76% 2.558uM 1.416uM View
calcium channel, voltage-dependent, gamma subunit 8 PENTAMIDINE Calcium Channel Type L, Phenylalkylamine 76% 1.391uM 1.352uM View
calcium channel, voltage-dependent, gamma subunit 7 PENTAMIDINE Calcium Channel Type L, Phenylalkylamine 76% 1.391uM 1.352uM View
calcium channel, voltage-dependent, gamma subunit 6 PENTAMIDINE Calcium Channel Type L, Phenylalkylamine 76% 1.391uM 1.352uM View
calcium channel, voltage-dependent, gamma subunit 5 PENTAMIDINE Calcium Channel Type L, Phenylalkylamine 76% 1.391uM 1.352uM View
calcium channel, voltage-dependent, gamma subunit 4 PENTAMIDINE Calcium Channel Type L, Phenylalkylamine 76% 1.391uM 1.352uM View
calcium channel, voltage-dependent, gamma subunit 3 PENTAMIDINE Calcium Channel Type L, Phenylalkylamine 76% 1.391uM 1.352uM View
calcium channel, voltage-dependent, gamma subunit 2 PENTAMIDINE Calcium Channel Type L, Phenylalkylamine 76% 1.391uM 1.352uM View
calcium channel, voltage-dependent, gamma subunit 1 PENTAMIDINE Calcium Channel Type L, Phenylalkylamine 76% 1.391uM 1.352uM View
calcium channel, voltage-dependent, beta 4 subunit PENTAMIDINE Calcium Channel Type L, Phenylalkylamine 76% 1.391uM 1.352uM View
calcium channel, voltage-dependent, beta 3 subunit PENTAMIDINE Calcium Channel Type L, Phenylalkylamine 76% 1.391uM 1.352uM View
calcium channel, voltage-dependent, beta 2 subunit PENTAMIDINE Calcium Channel Type L, Phenylalkylamine 76% 1.391uM 1.352uM View
calcium channel, voltage-dependent, L type, alpha 1S subunit PENTAMIDINE Calcium Channel Type L, Phenylalkylamine 76% 1.391uM 1.352uM View
calcium channel, voltage-dependent, alpha 1F subunit PENTAMIDINE Calcium Channel Type L, Phenylalkylamine 76% 1.391uM 1.352uM View
calcium channel, voltage-dependent, L type, alpha 1D subunit PENTAMIDINE Calcium Channel Type L, Phenylalkylamine 76% 1.391uM 1.352uM View
calcium channel, voltage-dependent, L type, alpha 1C subunit PENTAMIDINE Calcium Channel Type L, Phenylalkylamine 76% 1.391uM 1.352uM View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit PENTAMIDINE Calcium Channel Type L, Phenylalkylamine 76% 1.391uM 1.352uM View
calcium channel, voltage-dependent, beta 1 subunit PENTAMIDINE Calcium Channel Type L, Phenylalkylamine 76% 1.391uM 1.352uM View
calcium channel, voltage-dependent, L type, alpha 1E subunit PENTAMIDINE Calcium Channel Type L, Phenylalkylamine 76% 1.391uM 1.352uM View
calcium channel, voltage-dependent, N type, alpha 1B subunit PENTAMIDINE Calcium Channel Type L, Phenylalkylamine 76% 1.391uM 1.352uM View
calcium channel, voltage-dependent, alpha2/delta subunit 1 PENTAMIDINE Calcium Channel Type L, Phenylalkylamine 76% 1.391uM 1.352uM View
calcium channel, voltage-dependent, gamma subunit 8 PERGOLIDE Calcium Channel Type L, Phenylalkylamine 76% .913uM .887uM View
calcium channel, voltage-dependent, gamma subunit 7 PERGOLIDE Calcium Channel Type L, Phenylalkylamine 76% .913uM .887uM View
calcium channel, voltage-dependent, gamma subunit 6 PERGOLIDE Calcium Channel Type L, Phenylalkylamine 76% .913uM .887uM View
calcium channel, voltage-dependent, gamma subunit 5 PERGOLIDE Calcium Channel Type L, Phenylalkylamine 76% .913uM .887uM View
calcium channel, voltage-dependent, gamma subunit 4 PERGOLIDE Calcium Channel Type L, Phenylalkylamine 76% .913uM .887uM View
calcium channel, voltage-dependent, gamma subunit 3 PERGOLIDE Calcium Channel Type L, Phenylalkylamine 76% .913uM .887uM View
calcium channel, voltage-dependent, gamma subunit 2 PERGOLIDE Calcium Channel Type L, Phenylalkylamine 76% .913uM .887uM View
solute carrier family 6 (neurotransmitter transporter, dopamine), member 3 BW-723C86 Dopamine Transporter 76% 2.6846uM 2.133uM View
dopamine receptor D3 TRANS-PLATINUM(II)DIAMMINE DICHLORIDE Dopamine D3 76% 3.3237uM 1.1288uM View
cholinergic receptor, muscarinic 3 PERHEXILINE Muscarinic M3 76% 3.1186uM .661uM View
sodium channel, nonvoltage-gated 1, beta (Liddle syndrome) DOXORUBICIN Sodium Channel, Site 2 75% 15.245uM 13.668uM View
sodium channel, nonvoltage-gated 1 alpha DOXORUBICIN Sodium Channel, Site 2 75% 15.245uM 13.668uM View
sodium channel, voltage-gated, type X, alpha DOXORUBICIN Sodium Channel, Site 2 75% 15.245uM 13.668uM View
sodium channel, voltage-gated, type IX, alpha DOXORUBICIN Sodium Channel, Site 2 75% 15.245uM 13.668uM View
sodium channel, voltage gated, type VIII, alpha DOXORUBICIN Sodium Channel, Site 2 75% 15.245uM 13.668uM View
5-hydroxytryptamine receptor 6 AMLODIPINE Serotonin 5-HT6 75% 2.898uM 1.346uM View
solute carrier family 6 (neurotransmitter transporter, noradrenalin), member 2 LOVASTATIN Adrenergic, Norepinephrine Transporter 75% 8.753uM 8.68uM View
opioid receptor, delta 1 AMIODARONE Opiate delta 75% 8.014uM 2.825uM View
5-hydroxytryptamine (serotonin) receptor 3a CHLORPROMAZINE Serotonin 5-HT3 75% 7.365uM 1.655uM View
5-hydroxytryptamine (serotonin) receptor 3b CHLORPROMAZINE Serotonin 5-HT3 75% 7.365uM 1.655uM View
aldo-keto reductase family 1, member B4 (aldose reductase) ZOMEPIRAC Aldose Reductase 75% 1.29uM NoneNone View
aldo-keto reductase family 1, member B1 (aldose reductase) ZOMEPIRAC Aldose Reductase 75% 1.29uM NoneNone View
aldo-keto reductase family 7, member A2 (aflatoxin aldehyde reductase) ZOMEPIRAC Aldose Reductase 75% 1.29uM NoneNone View
aldo-keto reductase family 7, member A3 (aflatoxin aldehyde reductase) ZOMEPIRAC Aldose Reductase 75% 1.29uM NoneNone View
melanocortin 5 receptor TAMOXIFEN Melanocortin MC5 75% 26.529uM 24.886uM View
bradykinin receptor, beta 2 TAMOXIFEN Bradykinin B2 75% 20.356uM 12.048uM View
bradykinin receptor B2 TAMOXIFEN Bradykinin B2 75% 20.356uM 12.048uM View
progesterone receptor TAMOXIFEN Progesterone 75% 19.846uM 2.589uM View
progesterone receptor TAMOXIFEN Progesterone 75% 19.846uM 2.589uM View
solute carrier family 6 (neurotransmitter transporter, serotonin), member 4 THIMEROSAL Serotonin Transporter 75% 2.015uM 1.07uM View
phosphodiesterase 5A, cGMP-specific DIPYRIDAMOLE Phosphodiesterase PDE5 75% 2.831uM NoneNone View
phosphodiesterase 5A, cGMP-specific DIPYRIDAMOLE Phosphodiesterase PDE5 75% 2.831uM NoneNone View
prostaglandin-endoperoxide synthase 1 IPRIFLAVONE Cyclooxygenase COX-1 75% 2.9443uM NoneNone View
prostaglandin-endoperoxide synthase 1 (prostaglandin G/H synthase and cyclooxygenase) IPRIFLAVONE Cyclooxygenase COX-1 75% 2.9443uM NoneNone View
aldo-keto reductase family 1, member B4 (aldose reductase) DICUMAROL Aldose Reductase 75% 4.093uM NoneNone View
aldo-keto reductase family 1, member B1 (aldose reductase) DICUMAROL Aldose Reductase 75% 4.093uM NoneNone View
aldo-keto reductase family 7, member A2 (aflatoxin aldehyde reductase) DICUMAROL Aldose Reductase 75% 4.093uM NoneNone View
aldo-keto reductase family 7, member A3 (aflatoxin aldehyde reductase) DICUMAROL Aldose Reductase 75% 4.093uM NoneNone View
5-hydroxytryptamine (serotonin) receptor 2B TOLNAFTATE Serotonin 5-HT2B 75% 2.007uM 1.277uM View
adrenergic receptor, alpha 2b MOSAPRIDE Adrenergic alpha2B 75% 1.908uM .871uM View
mitogen activated protein kinase 14 ISOTRETINOIN Protein Serine/Threonine Kinase, p38alpha 75% 2.529uM NoneNone View
mitogen-activated protein kinase 14 ISOTRETINOIN Protein Serine/Threonine Kinase, p38alpha 75% 2.529uM NoneNone View
5-hydroxytryptamine (serotonin) receptor 2A GUANFACINE Serotonin 5-HT2A 75% 3.014uM .861uM View
potassium voltage-gated channel, subfamily H (eag-related), member 1 FLUPHENAZINE Potassium Channel HERG 75% 5.7058uM 4.6746uM View
potassium voltage-gated channel, subfamily H (eag-related), member 1 FLUPHENAZINE Potassium Channel HERG 75% 5.7058uM 4.6746uM View
potassium voltage-gated channel, subfamily H, member 8 FLUPHENAZINE Potassium Channel HERG 75% 5.7058uM 4.6746uM View
potassium voltage-gated channel, subfamily H (eag-related), member 6 FLUPHENAZINE Potassium Channel HERG 75% 5.7058uM 4.6746uM View
potassium voltage-gated channel, subfamily H (eag-related), member 7 FLUPHENAZINE Potassium Channel HERG 75% 5.7058uM 4.6746uM View
potassium voltage-gated channel, subfamily H (eag-related), member 2 FLUPHENAZINE Potassium Channel HERG 75% 5.7058uM 4.6746uM View
potassium voltage-gated channel, subfamily H (eag-related), member 5 FLUPHENAZINE Potassium Channel HERG 75% 5.7058uM 4.6746uM View
potassium voltage-gated channel, subfamily H (eag-related), member 3 FLUPHENAZINE Potassium Channel HERG 75% 5.7058uM 4.6746uM View
potassium voltage-gated channel, subfamily H (eag-related), member 4 FLUPHENAZINE Potassium Channel HERG 75% 5.7058uM 4.6746uM View
cholinergic receptor, muscarinic 5 TRANS-PLATINUM(II)DIAMMINE DICHLORIDE Muscarinic M5 75% 5.9254uM 4.2571uM View
Cytochrom P450-2D6 monooxygenase METHAPYRILENE CYP450-2D6 Inhibition 75% 2.7564uM NoneNone View
Cytochrom P450-1A2 monooxygenase PROPAFENONE CYP450-1A2 Inhibition 75% 3.292uM NoneNone View
adrenergic receptor, beta 3 SULOCTIDIL Adrenergic beta3 75% 4.9963uM 3.7472uM View
solute carrier family 6 (neurotransmitter transporter, serotonin), member 4 LEVOBUNOLOL Serotonin Transporter 75% 4.898uM 2.602uM View
5-hydroxytryptamine (serotonin) receptor 2B DIMENHYDRINATE Serotonin 5-HT2B 75% 1.724uM 1.097uM View
mitogen activated protein kinase 14 MONTELUKAST Protein Serine/Threonine Kinase, p38alpha 75% .856uM NoneNone View
mitogen-activated protein kinase 14 MONTELUKAST Protein Serine/Threonine Kinase, p38alpha 75% .856uM NoneNone View
platelet-activating factor receptor CILOSTAMIDE Platelet Activating Factor (PAF) 75% 3.687uM 1.917uM View
cholinergic receptor, muscarinic 4 FLUNARIZINE Muscarinic M4 75% 5.656uM .789uM View
dopamine receptor D4 THIORIDAZINE Dopamine D4.2 75% 1.468uM .515uM View
calcium channel, voltage-dependent, L type, alpha 1E subunit SPIRADOLINE Calcium Channel Type L, Phenylalkylamine 78% 5.24uM 5.095uM View
calcium channel, voltage-dependent, N type, alpha 1B subunit SPIRADOLINE Calcium Channel Type L, Phenylalkylamine 78% 5.24uM 5.095uM View
calcium channel, voltage-dependent, alpha2/delta subunit 1 SPIRADOLINE Calcium Channel Type L, Phenylalkylamine 78% 5.24uM 5.095uM View
acetylcholinesterase (YT blood group) BUTENAFINE Acetylcholinesterase 78% 6.9071uM NoneNone View
collagen-like tail subunit (single strand of homotrimer) of asymmetric acetylcholinesterase BUTENAFINE Acetylcholinesterase 78% 6.9071uM NoneNone View
acetylcholinesterase BUTENAFINE Acetylcholinesterase 78% 6.9071uM NoneNone View
cholinergic receptor, muscarinic 1 QUETIAPINE Muscarinic M1 78% 2.615uM .6298uM View
A3 adenosine receptor VX-745 Adenosine A3 78% 8.547uM 4.831uM View
dopamine receptor D3 TERCONAZOLE Dopamine D3 78% 4.712uM 1.6uM View
adrenergic receptor, alpha 2a SEMUSTINE Adrenergic alpha2A 78% 4.809uM 1.803uM View
histamine receptor H 1 METERGOLINE Histamine H1, Central 78% 4.133uM .48uM View
cholinergic receptor, muscarinic 5 PENTAMIDINE Muscarinic M5 78% 2.885uM 2.073uM View
5-hydroxytryptamine (serotonin) receptor 2C PENTAMIDINE Serotonin 5-HT2C 78% 3.278uM 1.717uM View
adrenergic receptor, alpha 2a PRAZOSIN Imidazoline I2, Central 78% .949uM .633uM View
adrenergic receptor, alpha 2c (Non-specific probe) PRAZOSIN Imidazoline I2, Central 78% .949uM .633uM View
Protein-tyrosine kinase, Fyn PROCHLORPERAZINE Protein Tyrosine Kinase, Fyn 78% 5.684uM NoneNone View
calcium channel, voltage-dependent, gamma subunit 8 PERGOLIDE Calcium Channel Type L, Benzothiazepine 78% 3.301uM 2.934uM View
calcium channel, voltage-dependent, gamma subunit 7 PERGOLIDE Calcium Channel Type L, Benzothiazepine 78% 3.301uM 2.934uM View
calcium channel, voltage-dependent, gamma subunit 6 PERGOLIDE Calcium Channel Type L, Benzothiazepine 78% 3.301uM 2.934uM View
calcium channel, voltage-dependent, gamma subunit 5 PERGOLIDE Calcium Channel Type L, Benzothiazepine 78% 3.301uM 2.934uM View
calcium channel, voltage-dependent, gamma subunit 4 PERGOLIDE Calcium Channel Type L, Benzothiazepine 78% 3.301uM 2.934uM View
calcium channel, voltage-dependent, gamma subunit 3 PERGOLIDE Calcium Channel Type L, Benzothiazepine 78% 3.301uM 2.934uM View