| calcium channel, voltage-dependent, gamma subunit 2 |
PERGOLIDE |
Calcium Channel Type L, Benzothiazepine |
78% |
3.301uM |
2.934uM |
View
|
| calcium channel, voltage-dependent, gamma subunit 1 |
PERGOLIDE |
Calcium Channel Type L, Benzothiazepine |
78% |
3.301uM |
2.934uM |
View
|
| calcium channel, voltage-dependent, beta 4 subunit |
PERGOLIDE |
Calcium Channel Type L, Benzothiazepine |
78% |
3.301uM |
2.934uM |
View
|
| calcium channel, voltage-dependent, beta 3 subunit |
PERGOLIDE |
Calcium Channel Type L, Benzothiazepine |
78% |
3.301uM |
2.934uM |
View
|
| calcium channel, voltage-dependent, beta 2 subunit |
PERGOLIDE |
Calcium Channel Type L, Benzothiazepine |
78% |
3.301uM |
2.934uM |
View
|
| calcium channel, voltage-dependent, L type, alpha 1S subunit |
PERGOLIDE |
Calcium Channel Type L, Benzothiazepine |
78% |
3.301uM |
2.934uM |
View
|
| calcium channel, voltage-dependent, alpha 1F subunit |
PERGOLIDE |
Calcium Channel Type L, Benzothiazepine |
78% |
3.301uM |
2.934uM |
View
|
| calcium channel, voltage-dependent, L type, alpha 1D subunit |
PERGOLIDE |
Calcium Channel Type L, Benzothiazepine |
78% |
3.301uM |
2.934uM |
View
|
| calcium channel, voltage-dependent, L type, alpha 1C subunit |
PERGOLIDE |
Calcium Channel Type L, Benzothiazepine |
78% |
3.301uM |
2.934uM |
View
|
| calcium channel, voltage-dependent, P/Q type, alpha 1A subunit |
PERGOLIDE |
Calcium Channel Type L, Benzothiazepine |
78% |
3.301uM |
2.934uM |
View
|
| calcium channel, voltage-dependent, beta 1 subunit |
PERGOLIDE |
Calcium Channel Type L, Benzothiazepine |
78% |
3.301uM |
2.934uM |
View
|
| Cytochrom P450-2C19 monooxygenase |
ROTENONE |
CYP450-2C19 Inhibition |
78% |
3.6486uM |
NoneNone |
View
|
| solute carrier family 6 (neurotransmitter transporter, noradrenalin), member 2 |
BW-723C86 |
Adrenergic, Norepinephrine Transporter |
78% |
3.6257uM |
3.5957uM |
View
|
| Cytochrom P450-2D6 monooxygenase |
CYCLIZINE |
CYP450-2D6 Inhibition |
78% |
6.2175uM |
NoneNone |
View
|
| epidermal growth factor receptor |
THIORIDAZINE |
Protein Tyrosine Kinase, EGF Receptor |
78% |
2.947uM |
NoneNone |
View
|
| mitogen activated protein kinase 14 |
ZAFIRLUKAST |
Protein Serine/Threonine Kinase, p38alpha |
78% |
.353uM |
NoneNone |
View
|
| mitogen-activated protein kinase 14 |
ZAFIRLUKAST |
Protein Serine/Threonine Kinase, p38alpha |
78% |
.353uM |
NoneNone |
View
|
| cholinergic receptor, muscarinic 3 |
MONTELUKAST |
Muscarinic M3 |
78% |
6.626uM |
1.404uM |
View
|
| cannabinoid receptor 1 (brain) |
FLUNARIZINE |
Cannabinoid CB1 |
78% |
3.028uM |
2.391uM |
View
|
| calcium channel, voltage-dependent, gamma subunit 8 |
DIMENHYDRINATE |
Calcium Channel Type L, Phenylalkylamine |
78% |
3.344uM |
3.251uM |
View
|
| calcium channel, voltage-dependent, gamma subunit 7 |
DIMENHYDRINATE |
Calcium Channel Type L, Phenylalkylamine |
78% |
3.344uM |
3.251uM |
View
|
| calcium channel, voltage-dependent, gamma subunit 6 |
DIMENHYDRINATE |
Calcium Channel Type L, Phenylalkylamine |
78% |
3.344uM |
3.251uM |
View
|
| calcium channel, voltage-dependent, gamma subunit 5 |
DIMENHYDRINATE |
Calcium Channel Type L, Phenylalkylamine |
78% |
3.344uM |
3.251uM |
View
|
| calcium channel, voltage-dependent, gamma subunit 4 |
DIMENHYDRINATE |
Calcium Channel Type L, Phenylalkylamine |
78% |
3.344uM |
3.251uM |
View
|
| calcium channel, voltage-dependent, gamma subunit 3 |
DIMENHYDRINATE |
Calcium Channel Type L, Phenylalkylamine |
78% |
3.344uM |
3.251uM |
View
|
| calcium channel, voltage-dependent, gamma subunit 2 |
DIMENHYDRINATE |
Calcium Channel Type L, Phenylalkylamine |
78% |
3.344uM |
3.251uM |
View
|
| calcium channel, voltage-dependent, gamma subunit 1 |
DIMENHYDRINATE |
Calcium Channel Type L, Phenylalkylamine |
78% |
3.344uM |
3.251uM |
View
|
| sodium channel, voltage-gated, type III, beta |
PROMAZINE |
Sodium Channel, Site 2 |
77% |
2.573uM |
2.347uM |
View
|
| sodium channel, voltage-gated, type VIII, alpha polypeptide |
PROMAZINE |
Sodium Channel, Site 2 |
77% |
2.573uM |
2.347uM |
View
|
| 5-hydroxytryptamine (serotonin) receptor 2C |
TERCONAZOLE |
Serotonin 5-HT2C |
77% |
6.961uM |
3.646uM |
View
|
| adrenergic receptor, alpha 1d (Non-specific probe) |
TERCONAZOLE |
Adrenergic alpha1D |
77% |
14.385uM |
7.07uM |
View
|
| cholinergic receptor, muscarinic 2 |
PROCHLORPERAZINE |
Muscarinic M2 |
77% |
3.112uM |
1.107uM |
View
|
| A3 adenosine receptor |
TROGLITAZONE |
Adenosine A3 |
77% |
5.208uM |
2.943uM |
View
|
| adrenergic receptor, alpha 1d (Non-specific probe) |
ECONAZOLE |
Adrenergic alpha1D |
77% |
8.897uM |
4.373uM |
View
|
| calcium channel, voltage-dependent, gamma subunit 8 |
SULCONAZOLE |
Calcium Channel Type L, Dihydropyridine |
77% |
2.427uM |
1.56uM |
View
|
| calcium channel, voltage-dependent, gamma subunit 7 |
SULCONAZOLE |
Calcium Channel Type L, Dihydropyridine |
77% |
2.427uM |
1.56uM |
View
|
| calcium channel, voltage-dependent, gamma subunit 6 |
SULCONAZOLE |
Calcium Channel Type L, Dihydropyridine |
77% |
2.427uM |
1.56uM |
View
|
| calcium channel, voltage-dependent, gamma subunit 5 |
SULCONAZOLE |
Calcium Channel Type L, Dihydropyridine |
77% |
2.427uM |
1.56uM |
View
|
| calcium channel, voltage-dependent, gamma subunit 4 |
SULCONAZOLE |
Calcium Channel Type L, Dihydropyridine |
77% |
2.427uM |
1.56uM |
View
|
| Protein-tyrosine kinase, Fyn |
BETA-NAPHTHOFLAVONE |
Protein Tyrosine Kinase, Fyn |
77% |
2.5149uM |
NoneNone |
View
|
| epidermal growth factor receptor |
PERHEXILINE |
Protein Tyrosine Kinase, EGF Receptor |
77% |
1.4852uM |
NoneNone |
View
|
| Cytochrom P450-2C19 monooxygenase |
BUPROPION |
CYP450-2C19 Inhibition |
77% |
1.9983uM |
NoneNone |
View
|
| 5-hydroxytryptamine receptor 6 |
PROPAFENONE |
Serotonin 5-HT6 |
77% |
1.863uM |
.865uM |
View
|
| solute carrier family 6 (neurotransmitter transporter, serotonin), member 4 |
AMBROXOL |
Serotonin Transporter |
77% |
3.391uM |
1.802uM |
View
|
| Protein-tyrosine kinase, Fyn |
TERFENADINE |
Protein Tyrosine Kinase, Fyn |
77% |
6.123uM |
NoneNone |
View
|
| mu-opioid receptor MOR |
DOMPERIDONE |
Opiate mu |
77% |
4.218uM |
1.712uM |
View
|
| histamine receptor H 2 |
IMATINIB |
Histamine H2 |
77% |
1.963uM |
1.93uM |
View
|
| dopamine receptor D3 |
CYCLIZINE |
Dopamine D3 |
77% |
2.992uM |
1.016uM |
View
|
| Cytochrom P450-2D6 monooxygenase |
LOPERAMIDE |
CYP450-2D6 Inhibition |
77% |
2uM |
NoneNone |
View
|
| Cytochrom P450-2C19 monooxygenase |
ETHYLESTRENOL |
CYP450-2C19 Inhibition |
77% |
1.2907uM |
NoneNone |
View
|
| Cytochrom P450-2C19 monooxygenase |
RAPAMYCIN |
CYP450-2C19 Inhibition |
77% |
4uM |
NoneNone |
View
|
| Cytochrom P450-2C19 monooxygenase |
RESVERATROL |
CYP450-2C19 Inhibition |
77% |
3uM |
NoneNone |
View
|
| A3 adenosine receptor |
HYDROXYPROGESTERONE |
Adenosine A3 |
77% |
4.73uM |
2.674uM |
View
|
| 5-hydroxytryptamine (serotonin) receptor 2A |
DIPHENIDOL |
Serotonin 5-HT2A |
77% |
2.586uM |
.739uM |
View
|
| estrogen receptor 1 |
ETHYLESTRENOL |
Estrogen ERalpha |
77% |
1.121uM |
.32uM |
View
|
| estrogen receptor 1 |
ETHYLESTRENOL |
Estrogen ERalpha |
77% |
1.121uM |
.32uM |
View
|
| adrenergic receptor, alpha 2a |
MOXONIDINE |
Imidazoline I2, Central |
77% |
1.4764uM |
.9843uM |
View
|
| adrenergic receptor, alpha 2c (Non-specific probe) |
MOXONIDINE |
Imidazoline I2, Central |
77% |
1.4764uM |
.9843uM |
View
|
| Protein-tyrosine kinase, Fyn |
METHYLDOPA |
Protein Tyrosine Kinase, Fyn |
77% |
5.176uM |
NoneNone |
View
|
| calcium channel, voltage-dependent, gamma subunit 8 |
LISURIDE |
Calcium Channel Type L, Benzothiazepine |
77% |
3.522uM |
3.131uM |
View
|
| calcium channel, voltage-dependent, gamma subunit 7 |
LISURIDE |
Calcium Channel Type L, Benzothiazepine |
77% |
3.522uM |
3.131uM |
View
|
| calcium channel, voltage-dependent, gamma subunit 6 |
LISURIDE |
Calcium Channel Type L, Benzothiazepine |
77% |
3.522uM |
3.131uM |
View
|
| calcium channel, voltage-dependent, gamma subunit 5 |
LISURIDE |
Calcium Channel Type L, Benzothiazepine |
77% |
3.522uM |
3.131uM |
View
|
| calcium channel, voltage-dependent, gamma subunit 4 |
LISURIDE |
Calcium Channel Type L, Benzothiazepine |
77% |
3.522uM |
3.131uM |
View
|
| calcium channel, voltage-dependent, gamma subunit 3 |
LISURIDE |
Calcium Channel Type L, Benzothiazepine |
77% |
3.522uM |
3.131uM |
View
|
| calcium channel, voltage-dependent, gamma subunit 2 |
LISURIDE |
Calcium Channel Type L, Benzothiazepine |
77% |
3.522uM |
3.131uM |
View
|
| calcium channel, voltage-dependent, gamma subunit 1 |
LISURIDE |
Calcium Channel Type L, Benzothiazepine |
77% |
3.522uM |
3.131uM |
View
|
| calcium channel, voltage-dependent, beta 4 subunit |
LISURIDE |
Calcium Channel Type L, Benzothiazepine |
77% |
3.522uM |
3.131uM |
View
|
| calcium channel, voltage-dependent, beta 3 subunit |
LISURIDE |
Calcium Channel Type L, Benzothiazepine |
77% |
3.522uM |
3.131uM |
View
|
| calcium channel, voltage-dependent, beta 2 subunit |
LISURIDE |
Calcium Channel Type L, Benzothiazepine |
77% |
3.522uM |
3.131uM |
View
|
| calcium channel, voltage-dependent, L type, alpha 1S subunit |
LISURIDE |
Calcium Channel Type L, Benzothiazepine |
77% |
3.522uM |
3.131uM |
View
|
| calcium channel, voltage-dependent, alpha 1F subunit |
LISURIDE |
Calcium Channel Type L, Benzothiazepine |
77% |
3.522uM |
3.131uM |
View
|
| calcium channel, voltage-dependent, L type, alpha 1D subunit |
LISURIDE |
Calcium Channel Type L, Benzothiazepine |
77% |
3.522uM |
3.131uM |
View
|
| calcium channel, voltage-dependent, L type, alpha 1C subunit |
LISURIDE |
Calcium Channel Type L, Benzothiazepine |
77% |
3.522uM |
3.131uM |
View
|
| calcium channel, voltage-dependent, P/Q type, alpha 1A subunit |
LISURIDE |
Calcium Channel Type L, Benzothiazepine |
77% |
3.522uM |
3.131uM |
View
|
| calcium channel, voltage-dependent, beta 1 subunit |
LISURIDE |
Calcium Channel Type L, Benzothiazepine |
77% |
3.522uM |
3.131uM |
View
|
| calcium channel, voltage-dependent, L type, alpha 1E subunit |
LISURIDE |
Calcium Channel Type L, Benzothiazepine |
77% |
3.522uM |
3.131uM |
View
|
| calcium channel, voltage-dependent, N type, alpha 1B subunit |
LISURIDE |
Calcium Channel Type L, Benzothiazepine |
77% |
3.522uM |
3.131uM |
View
|
| calcium channel, voltage-dependent, alpha2/delta subunit 1 |
LISURIDE |
Calcium Channel Type L, Benzothiazepine |
77% |
3.522uM |
3.131uM |
View
|
| epidermal growth factor receptor |
TERFENADINE |
Protein Tyrosine Kinase, EGF Receptor |
76% |
3.566uM |
NoneNone |
View
|
| epidermal growth factor receptor |
ZAFIRLUKAST |
Protein Tyrosine Kinase, EGF Receptor |
76% |
5.751uM |
NoneNone |
View
|
| angiotensin 1 converting enzyme 1 |
IODOQUINOL |
Protease, Angiotensin Converting Enzyme |
76% |
.906uM |
NoneNone |
View
|
| angiotensin I converting enzyme (peptidyl-dipeptidase A) 1 |
IODOQUINOL |
Protease, Angiotensin Converting Enzyme |
76% |
.906uM |
NoneNone |
View
|
| nitric oxide synthase 3 (endothelial cell) |
CHLORZOXAZONE |
Nitric Oxide Synthase, Constitutive (cNOS) |
76% |
2.794uM |
NoneNone |
View
|
| nitric oxide synthase 3, endothelial cell |
CHLORZOXAZONE |
Nitric Oxide Synthase, Constitutive (cNOS) |
76% |
2.794uM |
NoneNone |
View
|
| cholinergic receptor, muscarinic 4 |
CINNARIZINE |
Muscarinic M4 |
76% |
3.66uM |
.51uM |
View
|
| Cytochrome P450, subfamily IIC (mephenytoin 4-hydroxylase) |
ALPHA-ERGOCRYPTINE |
CYP450-2C9 Inhibition |
76% |
6uM |
NoneNone |
View
|
| cytochrome P450, family 2, subfamily C, polypeptide 9 |
ALPHA-ERGOCRYPTINE |
CYP450-2C9 Inhibition |
76% |
6uM |
NoneNone |
View
|
| Cytochrome P450, subfamily IIC (mephenytoin 4-hydroxylase) |
RWJ-68354 |
CYP450-2C9 Inhibition |
76% |
1uM |
NoneNone |
View
|
| cytochrome P450, family 2, subfamily C, polypeptide 9 |
RWJ-68354 |
CYP450-2C9 Inhibition |
76% |
1uM |
NoneNone |
View
|
| Cytochrome P450, subfamily IIC (mephenytoin 4-hydroxylase) |
PHENYLHYDRAZINE |
CYP450-2C9 Inhibition |
76% |
6uM |
NoneNone |
View
|
| cytochrome P450, family 2, subfamily C, polypeptide 9 |
PHENYLHYDRAZINE |
CYP450-2C9 Inhibition |
76% |
6uM |
NoneNone |
View
|
| Cytochrom P450-2C19 monooxygenase |
NOSCAPINE |
CYP450-2C19 Inhibition |
76% |
.4003uM |
NoneNone |
View
|
| adrenergic receptor, alpha 2b |
BERBERINE CHLORIDE |
Adrenergic alpha2C |
76% |
2.837uM |
.412uM |
View
|
| adrenergic receptor, alpha 2c (Non-specific probe) |
BERBERINE CHLORIDE |
Adrenergic alpha2C |
76% |
2.837uM |
.412uM |
View
|
| phosphodiesterase 3B |
MILRINONE |
Phosphodiesterase PDE3 |
76% |
.9585uM |
NoneNone |
View
|
| phosphodiesterase 3A |
MILRINONE |
Phosphodiesterase PDE3 |
76% |
.9585uM |
NoneNone |
View
|
| melanocortin 5 receptor |
DIGITONIN |
Melanocortin MC5 |
76% |
3.88uM |
3.639uM |
View
|
| sodium channel, voltage-gated, type IV, beta |
MAPROTILINE |
Sodium Channel, Site 2 |
76% |
2.572uM |
2.346uM |
View
|
| sodium channel associated protein 1 |
MAPROTILINE |
Sodium Channel, Site 2 |
76% |
2.572uM |
2.346uM |
View
|
| sodium channel associated protein 2 |
MAPROTILINE |
Sodium Channel, Site 2 |
76% |
2.572uM |
2.346uM |
View
|
| sodium channel, voltage-gated, type III, beta |
MAPROTILINE |
Sodium Channel, Site 2 |
76% |
2.572uM |
2.346uM |
View
|
| sodium channel, voltage-gated, type I, alpha |
MAPROTILINE |
Sodium Channel, Site 2 |
76% |
2.572uM |
2.346uM |
View
|
| sodium channel, voltage-gated, type IX, alpha |
MAPROTILINE |
Sodium Channel, Site 2 |
76% |
2.572uM |
2.346uM |
View
|
| sodium channel, voltage-gated, type VII, alpha |
MAPROTILINE |
Sodium Channel, Site 2 |
76% |
2.572uM |
2.346uM |
View
|
| amiloride-sensitive cation channel 5, intestinal |
MAPROTILINE |
Sodium Channel, Site 2 |
76% |
2.572uM |
2.346uM |
View
|
| sodium channel, voltage-gated, type III, beta |
MAPROTILINE |
Sodium Channel, Site 2 |
76% |
2.572uM |
2.346uM |
View
|
| sodium channel, voltage-gated, type VIII, alpha polypeptide |
MAPROTILINE |
Sodium Channel, Site 2 |
76% |
2.572uM |
2.346uM |
View
|
| sodium channel, voltage-gated, type XI, alpha |
MAPROTILINE |
Sodium Channel, Site 2 |
76% |
2.572uM |
2.346uM |
View
|
| sodium channel, voltage-gated, type I, beta |
MAPROTILINE |
Sodium Channel, Site 2 |
76% |
2.572uM |
2.346uM |
View
|
| sodium channel, voltage-gated, type 10, alpha polypeptide |
MAPROTILINE |
Sodium Channel, Site 2 |
76% |
2.572uM |
2.346uM |
View
|
| sodium channel, voltage-gated, type IV, alpha polypeptide |
MAPROTILINE |
Sodium Channel, Site 2 |
76% |
2.572uM |
2.346uM |
View
|
| sodium channel, voltage-gated, type V, alpha polypeptide |
MAPROTILINE |
Sodium Channel, Site 2 |
76% |
2.572uM |
2.346uM |
View
|
| sodium channel, voltage-gated, type II, beta |
MAPROTILINE |
Sodium Channel, Site 2 |
76% |
2.572uM |
2.346uM |
View
|
| sodium channel, nonvoltage-gated 1 alpha |
MAPROTILINE |
Sodium Channel, Site 2 |
76% |
2.572uM |
2.346uM |
View
|
| sodium channel, nonvoltage-gated 1 gamma |
MAPROTILINE |
Sodium Channel, Site 2 |
76% |
2.572uM |
2.346uM |
View
|
| sodium channel, nonvoltage-gated 1 beta |
MAPROTILINE |
Sodium Channel, Site 2 |
76% |
2.572uM |
2.346uM |
View
|
| sodium channel, voltage-gated, type 2, alpha 1 polypeptide |
MAPROTILINE |
Sodium Channel, Site 2 |
76% |
2.572uM |
2.346uM |
View
|
| sodium channel, voltage-gated, type XI, alpha |
MAPROTILINE |
Sodium Channel, Site 2 |
76% |
2.572uM |
2.346uM |
View
|
| sodium channel, nonvoltage-gated 1, gamma |
MAPROTILINE |
Sodium Channel, Site 2 |
76% |
2.572uM |
2.346uM |
View
|
| sodium channel, nonvoltage-gated 1, delta |
MAPROTILINE |
Sodium Channel, Site 2 |
76% |
2.572uM |
2.346uM |
View
|
| sodium channel, nonvoltage-gated 1, beta (Liddle syndrome) |
MAPROTILINE |
Sodium Channel, Site 2 |
76% |
2.572uM |
2.346uM |
View
|
| sodium channel, nonvoltage-gated 1 alpha |
MAPROTILINE |
Sodium Channel, Site 2 |
76% |
2.572uM |
2.346uM |
View
|
| sodium channel, voltage-gated, type X, alpha |
MAPROTILINE |
Sodium Channel, Site 2 |
76% |
2.572uM |
2.346uM |
View
|
| sodium channel, voltage-gated, type IX, alpha |
MAPROTILINE |
Sodium Channel, Site 2 |
76% |
2.572uM |
2.346uM |
View
|
| sodium channel, voltage gated, type VIII, alpha |
MAPROTILINE |
Sodium Channel, Site 2 |
76% |
2.572uM |
2.346uM |
View
|
| sodium channel, voltage-gated, type VII, alpha |
MAPROTILINE |
Sodium Channel, Site 2 |
76% |
2.572uM |
2.346uM |
View
|
| sodium channel, voltage-gated, type V, alpha (long QT syndrome 3) |
MAPROTILINE |
Sodium Channel, Site 2 |
76% |
2.572uM |
2.346uM |
View
|
| sodium channel, voltage-gated, type IV, beta |
MAPROTILINE |
Sodium Channel, Site 2 |
76% |
2.572uM |
2.346uM |
View
|
| sodium channel, voltage-gated, type IV, alpha |
MAPROTILINE |
Sodium Channel, Site 2 |
76% |
2.572uM |
2.346uM |
View
|
| sodium channel, voltage-gated, type III, alpha |
MAPROTILINE |
Sodium Channel, Site 2 |
76% |
2.572uM |
2.346uM |
View
|
| sodium channel, voltage-gated, type II, beta |
MAPROTILINE |
Sodium Channel, Site 2 |
76% |
2.572uM |
2.346uM |
View
|
| solute carrier family 6 (neurotransmitter transporter, dopamine), member 3 |
CLEMASTINE |
Dopamine Transporter |
89% |
.678uM |
.538uM |
View
|
| adrenergic receptor, alpha 1d (Non-specific probe) |
CLEMASTINE |
Adrenergic alpha1D |
89% |
.032uM |
.015uM |
View
|
| 5-hydroxytryptamine (serotonin) receptor 1B |
CLEMASTINE |
Serotonin 5-HT1B |
89% |
.359uM |
.22uM |
View
|
| calcium channel, voltage-dependent, gamma subunit 4 |
CLEMASTINE |
Calcium Channel Type L, Phenylalkylamine |
89% |
.508uM |
.493uM |
View
|
| calcium channel, voltage-dependent, gamma subunit 3 |
CLEMASTINE |
Calcium Channel Type L, Phenylalkylamine |
89% |
.508uM |
.493uM |
View
|
| calcium channel, voltage-dependent, gamma subunit 2 |
CLEMASTINE |
Calcium Channel Type L, Phenylalkylamine |
89% |
.508uM |
.493uM |
View
|
| calcium channel, voltage-dependent, gamma subunit 1 |
CLEMASTINE |
Calcium Channel Type L, Phenylalkylamine |
89% |
.508uM |
.493uM |
View
|
| calcium channel, voltage-dependent, beta 4 subunit |
CLEMASTINE |
Calcium Channel Type L, Phenylalkylamine |
89% |
.508uM |
.493uM |
View
|
| calcium channel, voltage-dependent, beta 3 subunit |
CLEMASTINE |
Calcium Channel Type L, Phenylalkylamine |
89% |
.508uM |
.493uM |
View
|
| calcium channel, voltage-dependent, beta 2 subunit |
CLEMASTINE |
Calcium Channel Type L, Phenylalkylamine |
89% |
.508uM |
.493uM |
View
|
| calcium channel, voltage-dependent, L type, alpha 1S subunit |
CLEMASTINE |
Calcium Channel Type L, Phenylalkylamine |
89% |
.508uM |
.493uM |
View
|
| calcium channel, voltage-dependent, alpha 1F subunit |
CLEMASTINE |
Calcium Channel Type L, Phenylalkylamine |
89% |
.508uM |
.493uM |
View
|
| calcium channel, voltage-dependent, L type, alpha 1D subunit |
CLEMASTINE |
Calcium Channel Type L, Phenylalkylamine |
89% |
.508uM |
.493uM |
View
|
| calcium channel, voltage-dependent, L type, alpha 1C subunit |
CLEMASTINE |
Calcium Channel Type L, Phenylalkylamine |
89% |
.508uM |
.493uM |
View
|
| calcium channel, voltage-dependent, P/Q type, alpha 1A subunit |
CLEMASTINE |
Calcium Channel Type L, Phenylalkylamine |
89% |
.508uM |
.493uM |
View
|
| calcium channel, voltage-dependent, beta 1 subunit |
CLEMASTINE |
Calcium Channel Type L, Phenylalkylamine |
89% |
.508uM |
.493uM |
View
|
| calcium channel, voltage-dependent, L type, alpha 1E subunit |
CLEMASTINE |
Calcium Channel Type L, Phenylalkylamine |
89% |
.508uM |
.493uM |
View
|
| adrenergic receptor, alpha 2b |
DOMPERIDONE |
Adrenergic alpha2C |
89% |
1.011uM |
.147uM |
View
|
| adrenergic receptor, alpha 2c (Non-specific probe) |
DOMPERIDONE |
Adrenergic alpha2C |
89% |
1.011uM |
.147uM |
View
|
| cholinergic receptor, muscarinic 2 |
PENTAMIDINE |
Muscarinic M2 |
89% |
1.425uM |
.507uM |
View
|
| adrenergic receptor, alpha 2b |
EPINEPHRINE |
Adrenergic alpha2B |
89% |
.869uM |
.397uM |
View
|
| adrenergic receptor, alpha 2a |
METOCLOPRAMIDE |
Imidazoline I2, Central |
89% |
.708uM |
.472uM |
View
|
| adrenergic receptor, alpha 2c (Non-specific probe) |
METOCLOPRAMIDE |
Imidazoline I2, Central |
89% |
.708uM |
.472uM |
View
|
| calcium channel, voltage-dependent, gamma subunit 8 |
MICONAZOLE |
Calcium Channel Type L, Phenylalkylamine |
89% |
3.788uM |
3.683uM |
View
|
| calcium channel, voltage-dependent, gamma subunit 7 |
MICONAZOLE |
Calcium Channel Type L, Phenylalkylamine |
89% |
3.788uM |
3.683uM |
View
|
| calcium channel, voltage-dependent, gamma subunit 6 |
MICONAZOLE |
Calcium Channel Type L, Phenylalkylamine |
89% |
3.788uM |
3.683uM |
View
|
| calcium channel, voltage-dependent, gamma subunit 5 |
MICONAZOLE |
Calcium Channel Type L, Phenylalkylamine |
89% |
3.788uM |
3.683uM |
View
|
| calcium channel, voltage-dependent, gamma subunit 4 |
MICONAZOLE |
Calcium Channel Type L, Phenylalkylamine |
89% |
3.788uM |
3.683uM |
View
|
| calcium channel, voltage-dependent, gamma subunit 3 |
MICONAZOLE |
Calcium Channel Type L, Phenylalkylamine |
89% |
3.788uM |
3.683uM |
View
|
| calcium channel, voltage-dependent, gamma subunit 2 |
MICONAZOLE |
Calcium Channel Type L, Phenylalkylamine |
89% |
3.788uM |
3.683uM |
View
|
| calcium channel, voltage-dependent, gamma subunit 1 |
MICONAZOLE |
Calcium Channel Type L, Phenylalkylamine |
89% |
3.788uM |
3.683uM |
View
|
| calcium channel, voltage-dependent, beta 4 subunit |
MICONAZOLE |
Calcium Channel Type L, Phenylalkylamine |
89% |
3.788uM |
3.683uM |
View
|
| calcium channel, voltage-dependent, beta 3 subunit |
MICONAZOLE |
Calcium Channel Type L, Phenylalkylamine |
89% |
3.788uM |
3.683uM |
View
|
| calcium channel, voltage-dependent, beta 2 subunit |
MICONAZOLE |
Calcium Channel Type L, Phenylalkylamine |
89% |
3.788uM |
3.683uM |
View
|
| calcium channel, voltage-dependent, L type, alpha 1S subunit |
MICONAZOLE |
Calcium Channel Type L, Phenylalkylamine |
89% |
3.788uM |
3.683uM |
View
|
| calcium channel, voltage-dependent, alpha 1F subunit |
MICONAZOLE |
Calcium Channel Type L, Phenylalkylamine |
89% |
3.788uM |
3.683uM |
View
|
| calcium channel, voltage-dependent, L type, alpha 1D subunit |
MICONAZOLE |
Calcium Channel Type L, Phenylalkylamine |
89% |
3.788uM |
3.683uM |
View
|
| calcium channel, voltage-dependent, L type, alpha 1C subunit |
MICONAZOLE |
Calcium Channel Type L, Phenylalkylamine |
89% |
3.788uM |
3.683uM |
View
|
| calcium channel, voltage-dependent, P/Q type, alpha 1A subunit |
MICONAZOLE |
Calcium Channel Type L, Phenylalkylamine |
89% |
3.788uM |
3.683uM |
View
|
| calcium channel, voltage-dependent, beta 1 subunit |
MICONAZOLE |
Calcium Channel Type L, Phenylalkylamine |
89% |
3.788uM |
3.683uM |
View
|
| calcium channel, voltage-dependent, L type, alpha 1E subunit |
MICONAZOLE |
Calcium Channel Type L, Phenylalkylamine |
89% |
3.788uM |
3.683uM |
View
|
| calcium channel, voltage-dependent, N type, alpha 1B subunit |
MICONAZOLE |
Calcium Channel Type L, Phenylalkylamine |
89% |
3.788uM |
3.683uM |
View
|
| calcium channel, voltage-dependent, alpha2/delta subunit 1 |
MICONAZOLE |
Calcium Channel Type L, Phenylalkylamine |
89% |
3.788uM |
3.683uM |
View
|
| prostaglandin-endoperoxide synthase 1 |
KETOPROFEN |
Cyclooxygenase COX-1 |
89% |
.014uM |
NoneNone |
View
|
| prostaglandin-endoperoxide synthase 1 (prostaglandin G/H synthase and cyclooxygenase) |
KETOPROFEN |
Cyclooxygenase COX-1 |
89% |
.014uM |
NoneNone |
View
|
| calcium channel, voltage-dependent, gamma subunit 8 |
ECONAZOLE |
Calcium Channel Type L, Phenylalkylamine |
89% |
3.014uM |
2.93uM |
View
|
| calcium channel, voltage-dependent, gamma subunit 7 |
ECONAZOLE |
Calcium Channel Type L, Phenylalkylamine |
89% |
3.014uM |
2.93uM |
View
|
| amiloride-sensitive cation channel 5, intestinal |
PERGOLIDE |
Sodium Channel, Site 2 |
88% |
1.728uM |
1.577uM |
View
|
| sodium channel, voltage-gated, type III, beta |
PERGOLIDE |
Sodium Channel, Site 2 |
88% |
1.728uM |
1.577uM |
View
|
| sodium channel, voltage-gated, type VIII, alpha polypeptide |
PERGOLIDE |
Sodium Channel, Site 2 |
88% |
1.728uM |
1.577uM |
View
|
| sodium channel, voltage-gated, type XI, alpha |
PERGOLIDE |
Sodium Channel, Site 2 |
88% |
1.728uM |
1.577uM |
View
|
| sodium channel, voltage-gated, type I, beta |
PERGOLIDE |
Sodium Channel, Site 2 |
88% |
1.728uM |
1.577uM |
View
|
| sodium channel, voltage-gated, type 10, alpha polypeptide |
PERGOLIDE |
Sodium Channel, Site 2 |
88% |
1.728uM |
1.577uM |
View
|
| sodium channel, voltage-gated, type IV, alpha polypeptide |
PERGOLIDE |
Sodium Channel, Site 2 |
88% |
1.728uM |
1.577uM |
View
|
| sodium channel, voltage-gated, type V, alpha polypeptide |
PERGOLIDE |
Sodium Channel, Site 2 |
88% |
1.728uM |
1.577uM |
View
|
| sodium channel, voltage-gated, type II, beta |
PERGOLIDE |
Sodium Channel, Site 2 |
88% |
1.728uM |
1.577uM |
View
|
| sodium channel, nonvoltage-gated 1 alpha |
PERGOLIDE |
Sodium Channel, Site 2 |
88% |
1.728uM |
1.577uM |
View
|
| sodium channel, nonvoltage-gated 1 gamma |
PERGOLIDE |
Sodium Channel, Site 2 |
88% |
1.728uM |
1.577uM |
View
|
| sodium channel, nonvoltage-gated 1 beta |
PERGOLIDE |
Sodium Channel, Site 2 |
88% |
1.728uM |
1.577uM |
View
|
| sodium channel, voltage-gated, type 2, alpha 1 polypeptide |
PERGOLIDE |
Sodium Channel, Site 2 |
88% |
1.728uM |
1.577uM |
View
|
| sodium channel, voltage-gated, type XI, alpha |
PERGOLIDE |
Sodium Channel, Site 2 |
88% |
1.728uM |
1.577uM |
View
|
| sodium channel, nonvoltage-gated 1, gamma |
PERGOLIDE |
Sodium Channel, Site 2 |
88% |
1.728uM |
1.577uM |
View
|
| sodium channel, nonvoltage-gated 1, delta |
PERGOLIDE |
Sodium Channel, Site 2 |
88% |
1.728uM |
1.577uM |
View
|
| sodium channel, nonvoltage-gated 1, beta (Liddle syndrome) |
PERGOLIDE |
Sodium Channel, Site 2 |
88% |
1.728uM |
1.577uM |
View
|
| sodium channel, nonvoltage-gated 1 alpha |
PERGOLIDE |
Sodium Channel, Site 2 |
88% |
1.728uM |
1.577uM |
View
|
| sodium channel, voltage-gated, type X, alpha |
PERGOLIDE |
Sodium Channel, Site 2 |
88% |
1.728uM |
1.577uM |
View
|
| sodium channel, voltage-gated, type IX, alpha |
PERGOLIDE |
Sodium Channel, Site 2 |
88% |
1.728uM |
1.577uM |
View
|
| phosphodiesterase 4A, cAMP specific |
GW-1929 |
Phosphodiesterase PDE4 |
88% |
7.45uM |
NoneNone |
View
|