Gene Activity List


Gene Activity List

Gene Compound Assay Inh Ic50 Ki View
calcium channel, voltage-dependent, gamma subunit 3 THIORIDAZINE Calcium Channel Type L, Phenylalkylamine 97% .443uM .431uM View
calcium channel, voltage-dependent, gamma subunit 2 THIORIDAZINE Calcium Channel Type L, Phenylalkylamine 97% .443uM .431uM View
calcium channel, voltage-dependent, gamma subunit 1 THIORIDAZINE Calcium Channel Type L, Phenylalkylamine 97% .443uM .431uM View
calcium channel, voltage-dependent, beta 4 subunit THIORIDAZINE Calcium Channel Type L, Phenylalkylamine 97% .443uM .431uM View
calcium channel, voltage-dependent, beta 3 subunit THIORIDAZINE Calcium Channel Type L, Phenylalkylamine 97% .443uM .431uM View
protein kinase C, epsilon PACLITAXEL Phorbol Ester 19% NoneNone NoneNone View
calcium channel, voltage-dependent, beta 2 subunit THIORIDAZINE Calcium Channel Type L, Phenylalkylamine 97% .443uM .431uM View
calcium channel, voltage-dependent, L type, alpha 1S subunit THIORIDAZINE Calcium Channel Type L, Phenylalkylamine 97% .443uM .431uM View
calcium channel, voltage-dependent, alpha 1F subunit THIORIDAZINE Calcium Channel Type L, Phenylalkylamine 97% .443uM .431uM View
calcium channel, voltage-dependent, L type, alpha 1D subunit THIORIDAZINE Calcium Channel Type L, Phenylalkylamine 97% .443uM .431uM View
calcium channel, voltage-dependent, L type, alpha 1C subunit THIORIDAZINE Calcium Channel Type L, Phenylalkylamine 97% .443uM .431uM View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit THIORIDAZINE Calcium Channel Type L, Phenylalkylamine 97% .443uM .431uM View
calcium channel, voltage-dependent, beta 1 subunit THIORIDAZINE Calcium Channel Type L, Phenylalkylamine 97% .443uM .431uM View
calcium channel, voltage-dependent, L type, alpha 1E subunit THIORIDAZINE Calcium Channel Type L, Phenylalkylamine 97% .443uM .431uM View
calcium channel, voltage-dependent, N type, alpha 1B subunit THIORIDAZINE Calcium Channel Type L, Phenylalkylamine 97% .443uM .431uM View
calcium channel, voltage-dependent, alpha2/delta subunit 1 THIORIDAZINE Calcium Channel Type L, Phenylalkylamine 97% .443uM .431uM View
calcium channel, voltage-dependent, gamma subunit 8 DILTIAZEM Calcium Channel Type L, Benzothiazepine 97% .028uM .025uM View
calcium channel, voltage-dependent, gamma subunit 7 DILTIAZEM Calcium Channel Type L, Benzothiazepine 97% .028uM .025uM View
calcium channel, voltage-dependent, gamma subunit 6 DILTIAZEM Calcium Channel Type L, Benzothiazepine 97% .028uM .025uM View
calcium channel, voltage-dependent, gamma subunit 5 DILTIAZEM Calcium Channel Type L, Benzothiazepine 97% .028uM .025uM View
calcium channel, voltage-dependent, gamma subunit 4 DILTIAZEM Calcium Channel Type L, Benzothiazepine 97% .028uM .025uM View
calcium channel, voltage-dependent, gamma subunit 3 DILTIAZEM Calcium Channel Type L, Benzothiazepine 97% .028uM .025uM View
calcium channel, voltage-dependent, gamma subunit 2 DILTIAZEM Calcium Channel Type L, Benzothiazepine 97% .028uM .025uM View
calcium channel, voltage-dependent, gamma subunit 1 DILTIAZEM Calcium Channel Type L, Benzothiazepine 97% .028uM .025uM View
calcium channel, voltage-dependent, beta 4 subunit DILTIAZEM Calcium Channel Type L, Benzothiazepine 97% .028uM .025uM View
calcium channel, voltage-dependent, beta 3 subunit DILTIAZEM Calcium Channel Type L, Benzothiazepine 97% .028uM .025uM View
calcium channel, voltage-dependent, beta 2 subunit DILTIAZEM Calcium Channel Type L, Benzothiazepine 97% .028uM .025uM View
calcium channel, voltage-dependent, L type, alpha 1S subunit DILTIAZEM Calcium Channel Type L, Benzothiazepine 97% .028uM .025uM View
calcium channel, voltage-dependent, alpha 1F subunit DILTIAZEM Calcium Channel Type L, Benzothiazepine 97% .028uM .025uM View
calcium channel, voltage-dependent, L type, alpha 1D subunit DILTIAZEM Calcium Channel Type L, Benzothiazepine 97% .028uM .025uM View
calcium channel, voltage-dependent, L type, alpha 1C subunit DILTIAZEM Calcium Channel Type L, Benzothiazepine 97% .028uM .025uM View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit DILTIAZEM Calcium Channel Type L, Benzothiazepine 97% .028uM .025uM View
calcium channel, voltage-dependent, beta 1 subunit DILTIAZEM Calcium Channel Type L, Benzothiazepine 97% .028uM .025uM View
calcium channel, voltage-dependent, L type, alpha 1E subunit DILTIAZEM Calcium Channel Type L, Benzothiazepine 97% .028uM .025uM View
calcium channel, voltage-dependent, N type, alpha 1B subunit DILTIAZEM Calcium Channel Type L, Benzothiazepine 97% .028uM .025uM View
calcium channel, voltage-dependent, alpha2/delta subunit 1 DILTIAZEM Calcium Channel Type L, Benzothiazepine 97% .028uM .025uM View
calcium channel, voltage-dependent, alpha2/delta subunit 1 CLOMIPHENE Calcium Channel Type L, Benzothiazepine 96% .789uM .701uM View
v-erb-b2 erythroblastic leukemia viral oncogene homolog 2, neuro/glioblastoma derived oncogene homolog (avian) CADMIUM ACETATE Protein Tyrosine Kinase, HER2 Receptor 96% 1.186uM NoneNone View
v-erb-b2 erythroblastic leukemia viral oncogene homolog 2, neuro/glioblastoma derived oncogene homolog (avian) CADMIUM ACETATE Protein Tyrosine Kinase, HER2 Receptor 96% 1.186uM NoneNone View
solute carrier family 6 (neurotransmitter transporter, dopamine), member 3 HALOPROGIN Dopamine Transporter 96% 1.969uM 1.565uM View
adrenergic receptor, alpha 2a HALOPROGIN Adrenergic alpha2A 96% 1.222uM .458uM View
5-hydroxytryptamine (serotonin) receptor 2B TROGLITAZONE Serotonin 5-HT2B 96% 1.312uM .835uM View
cholinergic receptor, muscarinic 1 GENTIAN VIOLET Muscarinic M1 96% 1.095uM .264uM View
5-hydroxytryptamine (serotonin) receptor 2B VERAPAMIL Serotonin 5-HT2B 96% .165uM .105uM View
histamine receptor H 1 MIANSERIN Histamine H1, Central 96% .001506uM .000175uM View
adrenergic receptor, alpha 2b MEPAZINE Adrenergic alpha2B 96% .397uM .181uM View
dopamine receptor D3 METHYSERGIDE Dopamine D3 96% .172uM .059uM View
Cytochrom P450-2C19 monooxygenase 1-(2-FLUOROBENZOYL)-4-(PHENYLMETHYL)-PIPERIDINE CYP450-2C19 Inhibition 96% .5uM NoneNone View
histamine receptor H 1 MEPAZINE Histamine H1, Central 96% .027uM .003126uM View
adrenergic receptor, alpha 2a RISPERIDONE Imidazoline I2, Central 96% .02uM .013uM View
adrenergic receptor, alpha 2c (Non-specific probe) RISPERIDONE Imidazoline I2, Central 96% .02uM .013uM View
epidermal growth factor receptor LEVODOPA Protein Tyrosine Kinase, EGF Receptor 96% 2.88uM NoneNone View
prostaglandin-endoperoxide synthase 2 DEXKETOPROFEN Cyclooxygenase COX-2 96% .23uM NoneNone View
prostaglandin-endoperoxide synthase 2 (prostaglandin G/H synthase and cyclooxygenase) DEXKETOPROFEN Cyclooxygenase COX-2 96% .23uM NoneNone View
adrenergic receptor, alpha 2a SERTRALINE Adrenergic alpha2A 96% .2888uM .1083uM View
cholinergic receptor, muscarinic 5 SERTRALINE Muscarinic M5 96% .5073uM .3645uM View
ATPase, Na+/K+ transporting, beta 2 polypeptide DIGOXIN ATPase, Na+/K+ 96% 1.647uM NoneNone View
ATPase, (Na+)/K+ transporting, beta 4 polypeptide DIGOXIN ATPase, Na+/K+ 96% 1.647uM NoneNone View
ATPase, Na+/K+ transporting, alpha 4 polypeptide DIGOXIN ATPase, Na+/K+ 96% 1.647uM NoneNone View
ATPase, Na+/K+ transporting, alpha 3 polypeptide DIGOXIN ATPase, Na+/K+ 96% 1.647uM NoneNone View
ATPase, Na+/K+ transporting, alpha 2 polypeptide DIGOXIN ATPase, Na+/K+ 96% 1.647uM NoneNone View
ATPase, Na+/K+ transporting, alpha 1 polypeptide DIGOXIN ATPase, Na+/K+ 96% 1.647uM NoneNone View
ATPase, Na+/K+ transporting, beta 1 polypeptide DIGOXIN ATPase, Na+/K+ 96% 1.647uM NoneNone View
ATPase, Na+/K+ transporting, beta 3 polypeptide DIGOXIN ATPase, Na+/K+ 96% 1.647uM NoneNone View
cholinergic receptor, muscarinic 5 KETOTIFEN Muscarinic M5 96% .374uM .269uM View
adrenergic receptor, alpha 2b NORTRIPTYLINE Adrenergic alpha2C 96% .203uM .03uM View
adrenergic receptor, alpha 2c (Non-specific probe) NORTRIPTYLINE Adrenergic alpha2C 96% .203uM .03uM View
estrogen receptor 1 NORETHINDRONE Estrogen ERalpha 96% .808uM .231uM View
estrogen receptor 1 NORETHINDRONE Estrogen ERalpha 96% .808uM .231uM View
nuclear receptor subfamily 3, group C, member 1 NORETHINDRONE Glucocorticoid 96% .433uM .197uM View
adrenergic receptor, alpha 2a OXICONAZOLE Adrenergic alpha2A 96% 4.0827uM 1.531uM View
cholinergic receptor, muscarinic 3 EBASTINE Muscarinic M3 96% .6475uM .1372uM View
cholinergic receptor, muscarinic 4 EBASTINE Muscarinic M4 96% .8279uM .1155uM View
dopamine receptor D3 RABEPRAZOLE Dopamine D3 96% 2.326uM .79uM View
adrenergic receptor, alpha 2b CETYLPYRIDINIUM BROMIDE Adrenergic alpha2C 96% 1.497uM .217uM View
adrenergic receptor, alpha 2c (Non-specific probe) CETYLPYRIDINIUM BROMIDE Adrenergic alpha2C 96% 1.497uM .217uM View
A3 adenosine receptor CETYLPYRIDINIUM BROMIDE Adenosine A3 96% 4.758uM 2.689uM View
prostaglandin-endoperoxide synthase 2 VALDECOXIB Cyclooxygenase COX-2 96% .208uM NoneNone View
prostaglandin-endoperoxide synthase 2 (prostaglandin G/H synthase and cyclooxygenase) VALDECOXIB Cyclooxygenase COX-2 96% .208uM NoneNone View
adrenergic receptor, beta 2 SOTALOL Adrenergic beta2 96% .4339uM .2983uM View
adrenergic receptor, alpha 2b PHENTOLAMINE Adrenergic alpha2C 96% .11uM .016uM View
adrenergic receptor, alpha 2c (Non-specific probe) PHENTOLAMINE Adrenergic alpha2C 96% .11uM .016uM View
5-hydroxytryptamine (serotonin) receptor 2A ASTEMIZOLE Serotonin 5-HT2A 96% .02uM .005575uM View
5-hydroxytryptamine (serotonin) receptor 2C ASTEMIZOLE Serotonin 5-HT2C 96% .179uM .094uM View
mu-opioid receptor MOR ASTEMIZOLE Opiate mu 96% 1.492uM .606uM View
adrenergic receptor, alpha 2b ASTEMIZOLE Adrenergic alpha2C 96% 1.959uM .285uM View
5-hydroxytryptamine (serotonin) receptor 2B MOSAPRIDE Serotonin 5-HT2B 95% .2959uM .1883uM View
5-hydroxytryptamine (serotonin) receptor 2A VERAPAMIL Serotonin 5-HT2A 95% .442uM .126uM View
adrenergic receptor, alpha 2a GUANFACINE Imidazoline I2, Central 95% .045uM .03uM View
adrenergic receptor, alpha 2c (Non-specific probe) GUANFACINE Imidazoline I2, Central 95% .045uM .03uM View
5-hydroxytryptamine (serotonin) receptor 1A MIANSERIN Serotonin 5-HT1A 95% .872uM .498uM View
cholinergic receptor, muscarinic 5 MIANSERIN Muscarinic M5 95% .32uM .23uM View
Cytochrom P450-2C19 monooxygenase 1-(2-METHOXYBENZOYL)-4-(PHENYLMETHYL)-PIPERIDINE CYP450-2C19 Inhibition 95% .8uM NoneNone View
solute carrier family 6 (neurotransmitter transporter, serotonin), member 4 PROPRANOLOL Serotonin Transporter 95% .38uM .202uM View
cholinergic receptor, muscarinic 3 QUINACRINE Muscarinic M3 95% 1.255uM .266uM View
solute carrier family 6 (neurotransmitter transporter, noradrenalin), member 2 SERTRALINE Adrenergic, Norepinephrine Transporter 95% .9848uM .9766uM View
adrenergic receptor, alpha 1b SERTRALINE Adrenergic alpha1B 95% .605uM .3349uM View
androgen receptor CYPROTERONE ACETATE Testosterone 95% .047uM .031uM View
adrenergic receptor, beta 3 LEVOBUNOLOL Adrenergic beta3 95% .34uM .255uM View
5-hydroxytryptamine (serotonin) receptor 2A ORPHENADRINE Serotonin 5-HT2A 95% .436uM .125uM View
adrenergic receptor, alpha 2b EBASTINE Adrenergic alpha2C 95% .2757uM .0401uM View
adrenergic receptor, alpha 2c (Non-specific probe) EBASTINE Adrenergic alpha2C 95% .2757uM .0401uM View
lymphocyte protein tyrosine kinase (mapped) CETYLPYRIDINIUM BROMIDE Protein Tyrosine Kinase, Lck 95% 3.182uM NoneNone View
5-hydroxytryptamine (serotonin) receptor 2C PHENTOLAMINE Serotonin 5-HT2C 95% .396uM .207uM View
5-hydroxytryptamine (serotonin) receptor 2A PHENTOLAMINE Serotonin 5-HT2A 95% .359uM .103uM View
5-hydroxytryptamine (serotonin) receptor 2A BENZETHONIUM CHLORIDE Serotonin 5-HT2A 95% .129uM .037uM View
solute carrier family 6 (neurotransmitter transporter, serotonin), member 4 BENZETHONIUM CHLORIDE Serotonin Transporter 95% 2.438uM 1.295uM View
calcium channel, voltage-dependent, alpha2/delta subunit 1 BENZETHONIUM CHLORIDE Calcium Channel Type L, Phenylalkylamine 95% .452uM .439uM View
calcium channel, voltage-dependent, gamma subunit 8 BENZETHONIUM CHLORIDE Calcium Channel Type L, Phenylalkylamine 95% .452uM .439uM View
calcium channel, voltage-dependent, gamma subunit 7 BENZETHONIUM CHLORIDE Calcium Channel Type L, Phenylalkylamine 95% .452uM .439uM View
calcium channel, voltage-dependent, gamma subunit 6 BENZETHONIUM CHLORIDE Calcium Channel Type L, Phenylalkylamine 95% .452uM .439uM View
calcium channel, voltage-dependent, gamma subunit 5 BENZETHONIUM CHLORIDE Calcium Channel Type L, Phenylalkylamine 95% .452uM .439uM View
calcium channel, voltage-dependent, gamma subunit 4 BENZETHONIUM CHLORIDE Calcium Channel Type L, Phenylalkylamine 95% .452uM .439uM View
calcium channel, voltage-dependent, gamma subunit 3 BENZETHONIUM CHLORIDE Calcium Channel Type L, Phenylalkylamine 95% .452uM .439uM View
calcium channel, voltage-dependent, gamma subunit 2 BENZETHONIUM CHLORIDE Calcium Channel Type L, Phenylalkylamine 95% .452uM .439uM View
calcium channel, voltage-dependent, gamma subunit 1 BENZETHONIUM CHLORIDE Calcium Channel Type L, Phenylalkylamine 95% .452uM .439uM View
calcium channel, voltage-dependent, beta 4 subunit BENZETHONIUM CHLORIDE Calcium Channel Type L, Phenylalkylamine 95% .452uM .439uM View
calcium channel, voltage-dependent, beta 3 subunit BENZETHONIUM CHLORIDE Calcium Channel Type L, Phenylalkylamine 95% .452uM .439uM View
calcium channel, voltage-dependent, beta 2 subunit BENZETHONIUM CHLORIDE Calcium Channel Type L, Phenylalkylamine 95% .452uM .439uM View
calcium channel, voltage-dependent, L type, alpha 1S subunit BENZETHONIUM CHLORIDE Calcium Channel Type L, Phenylalkylamine 95% .452uM .439uM View
calcium channel, voltage-dependent, alpha 1F subunit BENZETHONIUM CHLORIDE Calcium Channel Type L, Phenylalkylamine 95% .452uM .439uM View
calcium channel, voltage-dependent, L type, alpha 1D subunit BENZETHONIUM CHLORIDE Calcium Channel Type L, Phenylalkylamine 95% .452uM .439uM View
calcium channel, voltage-dependent, L type, alpha 1C subunit BENZETHONIUM CHLORIDE Calcium Channel Type L, Phenylalkylamine 95% .452uM .439uM View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit BENZETHONIUM CHLORIDE Calcium Channel Type L, Phenylalkylamine 95% .452uM .439uM View
calcium channel, voltage-dependent, beta 1 subunit BENZETHONIUM CHLORIDE Calcium Channel Type L, Phenylalkylamine 95% .452uM .439uM View
calcium channel, voltage-dependent, L type, alpha 1E subunit BENZETHONIUM CHLORIDE Calcium Channel Type L, Phenylalkylamine 95% .452uM .439uM View
calcium channel, voltage-dependent, N type, alpha 1B subunit BENZETHONIUM CHLORIDE Calcium Channel Type L, Phenylalkylamine 95% .452uM .439uM View
adrenergic receptor, alpha 2a PHENTOLAMINE Adrenergic alpha2A 95% .006uM .00225uM View
calcium channel, voltage-dependent, gamma subunit 8 NISOLDIPINE Calcium Channel Type L, Dihydropyridine 95% .000741uM .000476uM View
calcium channel, voltage-dependent, gamma subunit 7 NISOLDIPINE Calcium Channel Type L, Dihydropyridine 95% .000741uM .000476uM View
calcium channel, voltage-dependent, gamma subunit 6 NISOLDIPINE Calcium Channel Type L, Dihydropyridine 95% .000741uM .000476uM View
calcium channel, voltage-dependent, gamma subunit 5 NISOLDIPINE Calcium Channel Type L, Dihydropyridine 95% .000741uM .000476uM View
5-hydroxytryptamine (serotonin) receptor 2B GUANFACINE Serotonin 5-HT2B 74% 2.098uM 1.335uM View
calcium channel, voltage-dependent, gamma subunit 4 NISOLDIPINE Calcium Channel Type L, Dihydropyridine 95% .000741uM .000476uM View
calcium channel, voltage-dependent, gamma subunit 3 NISOLDIPINE Calcium Channel Type L, Dihydropyridine 95% .000741uM .000476uM View
calcium channel, voltage-dependent, gamma subunit 2 NISOLDIPINE Calcium Channel Type L, Dihydropyridine 95% .000741uM .000476uM View
calcium channel, voltage-dependent, gamma subunit 1 NISOLDIPINE Calcium Channel Type L, Dihydropyridine 95% .000741uM .000476uM View
calcium channel, voltage-dependent, N type, alpha 1B subunit TAMOXIFEN Calcium Channel Type L, Benzothiazepine 95% 1.44uM 1.28uM View
calcium channel, voltage-dependent, alpha2/delta subunit 1 TAMOXIFEN Calcium Channel Type L, Benzothiazepine 95% 1.44uM 1.28uM View
calcium channel, voltage-dependent, gamma subunit 8 TAMOXIFEN Calcium Channel Type L, Benzothiazepine 95% 1.44uM 1.28uM View
calcium channel, voltage-dependent, gamma subunit 7 TAMOXIFEN Calcium Channel Type L, Benzothiazepine 95% 1.44uM 1.28uM View
calcium channel, voltage-dependent, gamma subunit 6 TAMOXIFEN Calcium Channel Type L, Benzothiazepine 95% 1.44uM 1.28uM View
calcium channel, voltage-dependent, gamma subunit 5 TAMOXIFEN Calcium Channel Type L, Benzothiazepine 95% 1.44uM 1.28uM View
calcium channel, voltage-dependent, gamma subunit 4 TAMOXIFEN Calcium Channel Type L, Benzothiazepine 95% 1.44uM 1.28uM View
calcium channel, voltage-dependent, gamma subunit 3 TAMOXIFEN Calcium Channel Type L, Benzothiazepine 95% 1.44uM 1.28uM View
calcium channel, voltage-dependent, gamma subunit 2 TAMOXIFEN Calcium Channel Type L, Benzothiazepine 95% 1.44uM 1.28uM View
calcium channel, voltage-dependent, gamma subunit 1 TAMOXIFEN Calcium Channel Type L, Benzothiazepine 95% 1.44uM 1.28uM View
calcium channel, voltage-dependent, beta 4 subunit TAMOXIFEN Calcium Channel Type L, Benzothiazepine 95% 1.44uM 1.28uM View
calcium channel, voltage-dependent, beta 3 subunit TAMOXIFEN Calcium Channel Type L, Benzothiazepine 95% 1.44uM 1.28uM View
calcium channel, voltage-dependent, beta 2 subunit TAMOXIFEN Calcium Channel Type L, Benzothiazepine 95% 1.44uM 1.28uM View
calcium channel, voltage-dependent, L type, alpha 1S subunit TAMOXIFEN Calcium Channel Type L, Benzothiazepine 95% 1.44uM 1.28uM View
calcium channel, voltage-dependent, alpha 1F subunit TAMOXIFEN Calcium Channel Type L, Benzothiazepine 95% 1.44uM 1.28uM View
calcium channel, voltage-dependent, L type, alpha 1D subunit TAMOXIFEN Calcium Channel Type L, Benzothiazepine 95% 1.44uM 1.28uM View
calcium channel, voltage-dependent, L type, alpha 1C subunit TAMOXIFEN Calcium Channel Type L, Benzothiazepine 95% 1.44uM 1.28uM View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit TAMOXIFEN Calcium Channel Type L, Benzothiazepine 95% 1.44uM 1.28uM View
calcium channel, voltage-dependent, beta 1 subunit TAMOXIFEN Calcium Channel Type L, Benzothiazepine 95% 1.44uM 1.28uM View
calcium channel, voltage-dependent, L type, alpha 1E subunit TAMOXIFEN Calcium Channel Type L, Benzothiazepine 95% 1.44uM 1.28uM View
opioid receptor, kappa 1 TAMOXIFEN Opiate kappa 95% 15.629uM 6.252uM View
5-hydroxytryptamine (serotonin) receptor 1A ERGONOVINE Serotonin 5-HT1A 95% .008126uM .004643uM View
opioid receptor, sigma 1 DICYCLOMINE Sigma1 95% .00489uM .002055uM View
opioid receptor, sigma 1 CLEMASTINE Sigma1 95% .034uM .014uM View
adrenergic receptor, alpha 2b CLEMASTINE Adrenergic alpha2B 95% .311uM .142uM View
adrenergic receptor, alpha 2b CLOMIPRAMINE Adrenergic alpha2C 95% 1.413uM .205uM View
adrenergic receptor, alpha 2c (Non-specific probe) CLOMIPRAMINE Adrenergic alpha2C 95% 1.413uM .205uM View
adrenergic receptor, beta 2 CARVEDILOL Adrenergic beta2 95% .000241uM .000166uM View
calcium channel, voltage-dependent, gamma subunit 8 CARVEDILOL Calcium Channel Type L, Phenylalkylamine 95% .389uM .378uM View
calcium channel, voltage-dependent, gamma subunit 7 CARVEDILOL Calcium Channel Type L, Phenylalkylamine 95% .389uM .378uM View
calcium channel, voltage-dependent, gamma subunit 6 CARVEDILOL Calcium Channel Type L, Phenylalkylamine 95% .389uM .378uM View
calcium channel, voltage-dependent, gamma subunit 5 CARVEDILOL Calcium Channel Type L, Phenylalkylamine 95% .389uM .378uM View
calcium channel, voltage-dependent, gamma subunit 4 CARVEDILOL Calcium Channel Type L, Phenylalkylamine 95% .389uM .378uM View
calcium channel, voltage-dependent, gamma subunit 3 CARVEDILOL Calcium Channel Type L, Phenylalkylamine 95% .389uM .378uM View
calcium channel, voltage-dependent, gamma subunit 2 CARVEDILOL Calcium Channel Type L, Phenylalkylamine 95% .389uM .378uM View
calcium channel, voltage-dependent, gamma subunit 1 CARVEDILOL Calcium Channel Type L, Phenylalkylamine 95% .389uM .378uM View
calcium channel, voltage-dependent, beta 4 subunit CARVEDILOL Calcium Channel Type L, Phenylalkylamine 95% .389uM .378uM View
calcium channel, voltage-dependent, beta 3 subunit CARVEDILOL Calcium Channel Type L, Phenylalkylamine 95% .389uM .378uM View
calcium channel, voltage-dependent, beta 2 subunit CARVEDILOL Calcium Channel Type L, Phenylalkylamine 95% .389uM .378uM View
calcium channel, voltage-dependent, L type, alpha 1S subunit CARVEDILOL Calcium Channel Type L, Phenylalkylamine 95% .389uM .378uM View
calcium channel, voltage-dependent, alpha 1F subunit CARVEDILOL Calcium Channel Type L, Phenylalkylamine 95% .389uM .378uM View
calcium channel, voltage-dependent, L type, alpha 1D subunit CARVEDILOL Calcium Channel Type L, Phenylalkylamine 95% .389uM .378uM View
calcium channel, voltage-dependent, L type, alpha 1C subunit CARVEDILOL Calcium Channel Type L, Phenylalkylamine 95% .389uM .378uM View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit CARVEDILOL Calcium Channel Type L, Phenylalkylamine 95% .389uM .378uM View
adrenergic receptor, alpha 2a FLUNARIZINE Adrenergic alpha2A 95% .581uM .218uM View
adrenergic receptor, alpha 1a GUANABENZ Adrenergic alpha1A 95% .391uM .158uM View
5-hydroxytryptamine (serotonin) receptor 2B PIPAMAZINE Serotonin 5-HT2B 95% .049uM .031uM View
Cytochrom P450-2C19 monooxygenase 1-(2-METHYLBENZOYL)-4-(PHENYLMETHYL)-PIPERIDINE CYP450-2C19 Inhibition 95% .6uM NoneNone View
adrenergic receptor, alpha 2a MONTELUKAST Adrenergic alpha2A 95% 3.919uM 1.47uM View
opioid receptor, sigma 1 TRIHEXYPHENIDYL Sigma1 95% .108uM .045uM View
5-hydroxytryptamine (serotonin) receptor 1A CYPROHEPTADINE Serotonin 5-HT1A 95% .122uM .07uM View
nuclear receptor subfamily 3, group C, member 1 PREDNISONE Glucocorticoid 95% 1.146uM .521uM View
Cytochrom P450-1A2 monooxygenase BENZO[A]PYRENE CYP450-1A2 Inhibition 95% .04uM NoneNone View
adrenergic receptor, alpha 2b AURANOFIN Adrenergic alpha2B 95% .796uM .363uM View
solute carrier family 6 (neurotransmitter transporter, noradrenalin), member 2 SULCONAZOLE Adrenergic, Norepinephrine Transporter 95% 2.027uM 2.01uM View
estrogen receptor 1 BETA-ESTRADIOL 3-BENZOATE Estrogen ERalpha 95% .065uM .018uM View
estrogen receptor 1 BETA-ESTRADIOL 3-BENZOATE Estrogen ERalpha 95% .065uM .018uM View
adrenergic receptor, alpha 2b CELECOXIB Adrenergic alpha2B 95% 1.516uM .692uM View
dopamine receptor D1A AMITRIPTYLINE Dopamine D1 95% .355uM .178uM View
cholinergic receptor, muscarinic 5 AMOXAPINE Muscarinic M5 95% .856uM .615uM View
arachidonate 15-lipoxygenase, second type U-78517F Lipoxygenase 15-LO 95% 5.67uM NoneNone View
arachidonate 15-lipoxygenase U-78517F Lipoxygenase 15-LO 95% 5.67uM NoneNone View
arachidonate 15-lipoxygenase U-78517F Lipoxygenase 15-LO 95% 5.67uM NoneNone View