Gene Activity List


Gene Activity List

Gene Compound Assay Inh Ic50 Ki View
sodium channel, voltage-gated, type IX, alpha DICYCLOMINE Sodium Channel, Site 2 94% 1.353uM 1.234uM View
sodium channel, voltage gated, type VIII, alpha DICYCLOMINE Sodium Channel, Site 2 94% 1.353uM 1.234uM View
sodium channel, voltage-gated, type VII, alpha DICYCLOMINE Sodium Channel, Site 2 94% 1.353uM 1.234uM View
sodium channel, voltage-gated, type V, alpha (long QT syndrome 3) DICYCLOMINE Sodium Channel, Site 2 94% 1.353uM 1.234uM View
sodium channel, voltage-gated, type IV, beta DICYCLOMINE Sodium Channel, Site 2 94% 1.353uM 1.234uM View
sodium channel, voltage-gated, type IV, alpha DICYCLOMINE Sodium Channel, Site 2 94% 1.353uM 1.234uM View
sodium channel, voltage-gated, type III, alpha DICYCLOMINE Sodium Channel, Site 2 94% 1.353uM 1.234uM View
sodium channel, voltage-gated, type II, beta DICYCLOMINE Sodium Channel, Site 2 94% 1.353uM 1.234uM View
sodium channel, voltage-gated, type II, alpha 2 DICYCLOMINE Sodium Channel, Site 2 94% 1.353uM 1.234uM View
sodium channel, voltage-gated, type I, beta DICYCLOMINE Sodium Channel, Site 2 94% 1.353uM 1.234uM View
sodium channel, voltage-gated, type I, alpha DICYCLOMINE Sodium Channel, Site 2 94% 1.353uM 1.234uM View
progesterone receptor TRIAMCINOLONE ACETONIDE Progesterone 94% .179uM .023uM View
progesterone receptor TRIAMCINOLONE ACETONIDE Progesterone 94% .179uM .023uM View
cholinergic receptor, muscarinic 2 CLOZAPINE Muscarinic M2 94% .476uM .169uM View
adrenergic receptor, alpha 2a THIMEROSAL Adrenergic alpha2A 94% .532uM .2uM View
adrenergic receptor, beta 1 TIMOLOL Adrenergic beta1 94% .002603uM .001503uM View
adrenergic, beta-1-, receptor TIMOLOL Adrenergic beta1 94% .002603uM .001503uM View
calcium channel, voltage-dependent, beta 3 subunit FLUOXETINE Calcium Channel Type L, Phenylalkylamine 94% 1.126uM 1.095uM View
calcium channel, voltage-dependent, beta 2 subunit FLUOXETINE Calcium Channel Type L, Phenylalkylamine 94% 1.126uM 1.095uM View
calcium channel, voltage-dependent, L type, alpha 1S subunit FLUOXETINE Calcium Channel Type L, Phenylalkylamine 94% 1.126uM 1.095uM View
calcium channel, voltage-dependent, alpha 1F subunit FLUOXETINE Calcium Channel Type L, Phenylalkylamine 94% 1.126uM 1.095uM View
calcium channel, voltage-dependent, L type, alpha 1D subunit FLUOXETINE Calcium Channel Type L, Phenylalkylamine 94% 1.126uM 1.095uM View
calcium channel, voltage-dependent, L type, alpha 1C subunit FLUOXETINE Calcium Channel Type L, Phenylalkylamine 94% 1.126uM 1.095uM View
protein kinase D1 LAMOTRIGINE Phorbol Ester 2% NoneNone NoneNone View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit FLUOXETINE Calcium Channel Type L, Phenylalkylamine 94% 1.126uM 1.095uM View
calcium channel, voltage-dependent, beta 1 subunit FLUOXETINE Calcium Channel Type L, Phenylalkylamine 94% 1.126uM 1.095uM View
calcium channel, voltage-dependent, L type, alpha 1E subunit FLUOXETINE Calcium Channel Type L, Phenylalkylamine 94% 1.126uM 1.095uM View
calcium channel, voltage-dependent, N type, alpha 1B subunit FLUOXETINE Calcium Channel Type L, Phenylalkylamine 94% 1.126uM 1.095uM View
calcium channel, voltage-dependent, alpha2/delta subunit 1 FLUOXETINE Calcium Channel Type L, Phenylalkylamine 94% 1.126uM 1.095uM View
calcium channel, voltage-dependent, gamma subunit 8 FLUOXETINE Calcium Channel Type L, Phenylalkylamine 94% 1.126uM 1.095uM View
calcium channel, voltage-dependent, gamma subunit 7 FLUOXETINE Calcium Channel Type L, Phenylalkylamine 94% 1.126uM 1.095uM View
calcium channel, voltage-dependent, gamma subunit 6 FLUOXETINE Calcium Channel Type L, Phenylalkylamine 94% 1.126uM 1.095uM View
calcium channel, voltage-dependent, gamma subunit 5 FLUOXETINE Calcium Channel Type L, Phenylalkylamine 94% 1.126uM 1.095uM View
calcium channel, voltage-dependent, gamma subunit 4 FLUOXETINE Calcium Channel Type L, Phenylalkylamine 94% 1.126uM 1.095uM View
calcium channel, voltage-dependent, gamma subunit 3 FLUOXETINE Calcium Channel Type L, Phenylalkylamine 94% 1.126uM 1.095uM View
calcium channel, voltage-dependent, gamma subunit 2 FLUOXETINE Calcium Channel Type L, Phenylalkylamine 94% 1.126uM 1.095uM View
calcium channel, voltage-dependent, gamma subunit 1 FLUOXETINE Calcium Channel Type L, Phenylalkylamine 94% 1.126uM 1.095uM View
calcium channel, voltage-dependent, beta 4 subunit FLUOXETINE Calcium Channel Type L, Phenylalkylamine 94% 1.126uM 1.095uM View
cholinergic receptor, muscarinic 4 FLUPHENAZINE Muscarinic M4 94% 3.468uM .484uM View
progesterone receptor FLUOCINONIDE Progesterone 94% .022uM .002904uM View
progesterone receptor FLUOCINONIDE Progesterone 94% .022uM .002904uM View
5-hydroxytryptamine receptor 6 DOXEPIN Serotonin 5-HT6 94% .32uM .149uM View
prostaglandin-endoperoxide synthase 1 TOLMETIN Cyclooxygenase COX-1 94% .041uM NoneNone View
prostaglandin-endoperoxide synthase 1 (prostaglandin G/H synthase and cyclooxygenase) TOLMETIN Cyclooxygenase COX-1 94% .041uM NoneNone View
prostaglandin-endoperoxide synthase 1 MECLOFENAMIC ACID Cyclooxygenase COX-1 94% .203uM NoneNone View
prostaglandin-endoperoxide synthase 1 (prostaglandin G/H synthase and cyclooxygenase) MECLOFENAMIC ACID Cyclooxygenase COX-1 94% .203uM NoneNone View
gamma-aminobutyric acid (GABA-A) receptor, subunit alpha 4 ZALEPLON GABAA, Benzodiazepine, Central 94% .412uM .336uM View
sodium channel associated protein 2 DIETHYLSTILBESTROL Sodium Channel, Site 2 94% 4.735uM 4.246uM View
sodium channel, voltage-gated, type III, beta DIETHYLSTILBESTROL Sodium Channel, Site 2 94% 4.735uM 4.246uM View
sodium channel, voltage-gated, type I, alpha DIETHYLSTILBESTROL Sodium Channel, Site 2 94% 4.735uM 4.246uM View
sodium channel, voltage-gated, type IX, alpha DIETHYLSTILBESTROL Sodium Channel, Site 2 94% 4.735uM 4.246uM View
calcium channel, voltage-dependent, alpha2/delta subunit 1 U-78517F Calcium Channel Type L, Benzothiazepine 93% 1.65uM 1.466uM View
solute carrier family 6 (neurotransmitter transporter, noradrenalin), member 2 CLOTRIMAZOLE Adrenergic, Norepinephrine Transporter 93% 7.936uM 7.87uM View
5-hydroxytryptamine (serotonin) receptor 2B CHLORPROMAZINE Serotonin 5-HT2B 93% .126uM .08uM View
adrenergic receptor, alpha 2b CHLORPROMAZINE Adrenergic alpha2C 93% .374uM .054uM View
adrenergic receptor, alpha 2c (Non-specific probe) CHLORPROMAZINE Adrenergic alpha2C 93% .374uM .054uM View
thromboxane A synthase 1 1-BENZYLIMIDAZOLE Thromboxane Synthetase 93% .602uM NoneNone View
thromboxane A synthase 1 (platelet, cytochrome P450, family 5, subfamily A) 1-BENZYLIMIDAZOLE Thromboxane Synthetase 93% .602uM NoneNone View
adrenergic receptor, alpha 2a TAMOXIFEN Adrenergic alpha2A 93% 1.935uM .726uM View
chemokine (C-C motif) receptor 2 NIFEDIPINE Chemokine CCR2B 93% 2.191uM .847uM View
solute carrier family 6 (neurotransmitter transporter, serotonin), member 4 CISAPRIDE Serotonin Transporter 93% .384uM .204uM View
dopamine receptor D1A CLOMIPRAMINE Dopamine D1 93% 1.113uM .557uM View
dopamine receptor 2 CLOMIPRAMINE Dopamine D2L 93% .413uM .138uM View
5-hydroxytryptamine receptor 6 BENZOTHIAZYL DISULFIDE Serotonin 5-HT6 93% 5.276uM 2.45uM View
A3 adenosine receptor BENZOTHIAZYL DISULFIDE Adenosine A3 93% .347uM .196uM View
solute carrier family 6 (neurotransmitter transporter, dopamine), member 3 BENZOTHIAZYL DISULFIDE Dopamine Transporter 93% .245uM .194uM View
5-hydroxytryptamine (serotonin) receptor 2A FLUOXETINE Serotonin 5-HT2A 93% .194uM .055uM View
cholinergic receptor, muscarinic 1 FLUPHENAZINE Muscarinic M1 93% 2.683uM .646uM View
adrenergic receptor, alpha 1d (Non-specific probe) FLUPHENAZINE Adrenergic alpha1D 93% .033uM .016uM View
5-hydroxytryptamine (serotonin) receptor 2C FLUPHENAZINE Serotonin 5-HT2C 93% .067uM .035uM View
v-erb-b2 erythroblastic leukemia viral oncogene homolog 2, neuro/glioblastoma derived oncogene homolog (avian) CAFFEIC ACID PHENETHYL ESTER Protein Tyrosine Kinase, HER2 Receptor 93% 1.329uM NoneNone View
v-erb-b2 erythroblastic leukemia viral oncogene homolog 2, neuro/glioblastoma derived oncogene homolog (avian) CAFFEIC ACID PHENETHYL ESTER Protein Tyrosine Kinase, HER2 Receptor 93% 1.329uM NoneNone View
adrenergic receptor, beta 2 R-(+)-PROPRANOLOL Adrenergic beta2 93% .076uM .052uM View
mitogen activated protein kinase 1 ISOTRETINOIN Protein Serine/Threonine Kinase, ERK2 93% .462uM NoneNone View
mitogen-activated protein kinase 1 ISOTRETINOIN Protein Serine/Threonine Kinase, ERK2 93% .462uM NoneNone View
5-hydroxytryptamine (serotonin) receptor 2C MOSAPRIDE Serotonin 5-HT2C 93% .3966uM .2077uM View
adrenergic receptor, alpha 2a BROMOCRIPTINE Imidazoline I2, Central 93% .053uM .035uM View
adrenergic receptor, alpha 2c (Non-specific probe) BROMOCRIPTINE Imidazoline I2, Central 93% .053uM .035uM View
adrenergic receptor, alpha 2a VERAPAMIL Adrenergic alpha2A 93% .579uM .217uM View
adrenergic receptor, alpha 2a LYSERGOL Adrenergic alpha2A 93% .18uM .067uM View
cholinergic receptor, muscarinic 2 MEPAZINE Muscarinic M2 93% .565uM .201uM View
5-hydroxytryptamine (serotonin) receptor 2B MEXILETINE Serotonin 5-HT2B 93% 1.138uM .724uM View
Cytochrom P450-2C19 monooxygenase 1-(2-CHLOROBENZOYL)-4-(PHENYLMETHYL)-PIPERIDINE CYP450-2C19 Inhibition 93% .2uM NoneNone View
solute carrier family 6 (neurotransmitter transporter, serotonin), member 4 MITOTANE Serotonin Transporter 93% 3.015uM 1.601uM View
prostaglandin-endoperoxide synthase 2 N,N'-DIPHENYL-P-PHENYLENEDIAMINE Cyclooxygenase COX-2 93% .58uM NoneNone View
prostaglandin-endoperoxide synthase 2 (prostaglandin G/H synthase and cyclooxygenase) N,N'-DIPHENYL-P-PHENYLENEDIAMINE Cyclooxygenase COX-2 93% .58uM NoneNone View
cholinergic receptor, muscarinic 4 IRINOTECAN Muscarinic M4 93% 1.556uM .217uM View
Protein-tyrosine kinase, Fyn ITRACONAZOLE Protein Tyrosine Kinase, Fyn 93% 3.89uM NoneNone View
adrenergic receptor, beta 3 PROPRANOLOL Adrenergic beta3 93% .132uM .099uM View
nuclear receptor subfamily 3, group C, member 1 NORETHINDRONE ACETATE Glucocorticoid 93% .646uM .293uM View
adrenergic receptor, alpha 2b OLANZAPINE Adrenergic alpha2C 93% .531uM .077uM View
adrenergic receptor, alpha 2c (Non-specific probe) OLANZAPINE Adrenergic alpha2C 93% .531uM .077uM View
histamine receptor H 1 OLANZAPINE Histamine H1, Central 93% .013uM .001473uM View
5-hydroxytryptamine (serotonin) receptor 2B ONDANSETRON Serotonin 5-HT2B 93% .717uM .456uM View
tachykinin receptor 2 EBASTINE Tachykinin NK2 93% 1.9329uM .6443uM View
Cytochrome P450, subfamily IIC (mephenytoin 4-hydroxylase) SULFAPHENAZOLE CYP450-2C9 Inhibition 93% .2uM NoneNone View
cytochrome P450, family 2, subfamily C, polypeptide 9 SULFAPHENAZOLE CYP450-2C9 Inhibition 93% .2uM NoneNone View
prostaglandin-endoperoxide synthase 1 RESVERATROL Cyclooxygenase COX-1 93% .625uM NoneNone View
prostaglandin-endoperoxide synthase 1 (prostaglandin G/H synthase and cyclooxygenase) RESVERATROL Cyclooxygenase COX-1 93% .625uM NoneNone View
v-erb-b2 erythroblastic leukemia viral oncogene homolog 2, neuro/glioblastoma derived oncogene homolog (avian) CETYLPYRIDINIUM BROMIDE Protein Tyrosine Kinase, HER2 Receptor 93% 1.878uM NoneNone View
v-erb-b2 erythroblastic leukemia viral oncogene homolog 2, neuro/glioblastoma derived oncogene homolog (avian) CETYLPYRIDINIUM BROMIDE Protein Tyrosine Kinase, HER2 Receptor 93% 1.878uM NoneNone View
phosphodiesterase 4A, cAMP specific CANDESARTAN Phosphodiesterase PDE4 93% .2761uM NoneNone View
phosphodiesterase 4C, cAMP-specific CANDESARTAN Phosphodiesterase PDE4 93% .2761uM NoneNone View
phosphodiesterase 4D CANDESARTAN Phosphodiesterase PDE4 93% .2761uM NoneNone View
phosphodiesterase 4B, cAMP specific CANDESARTAN Phosphodiesterase PDE4 93% .2761uM NoneNone View
mitogen activated protein kinase 14 NOVARTIS P-38 INHIBITOR Protein Serine/Threonine Kinase, p38alpha 93% .1868uM NoneNone View
mitogen-activated protein kinase 14 NOVARTIS P-38 INHIBITOR Protein Serine/Threonine Kinase, p38alpha 93% .1868uM NoneNone View
5-hydroxytryptamine (serotonin) receptor 2B METOCLOPRAMIDE Serotonin 5-HT2B 93% .63uM .401uM View
solute carrier family 6 (neurotransmitter transporter, noradrenalin), member 2 ECONAZOLE Adrenergic, Norepinephrine Transporter 93% 2.435uM 2.415uM View
acetylcholinesterase (YT blood group) ECONAZOLE Acetylcholinesterase 93% 13.677uM NoneNone View
adrenergic receptor, alpha 1b CITALOPRAM Adrenergic alpha1B 74% 3.288uM 1.82uM View
collagen-like tail subunit (single strand of homotrimer) of asymmetric acetylcholinesterase ECONAZOLE Acetylcholinesterase 93% 13.677uM NoneNone View
acetylcholinesterase ECONAZOLE Acetylcholinesterase 93% 13.677uM NoneNone View
Cytochrome P450, subfamily IIC (mephenytoin 4-hydroxylase) MICONAZOLE CYP450-2C9 Inhibition 93% .2uM NoneNone View
cytochrome P450, family 2, subfamily C, polypeptide 9 MICONAZOLE CYP450-2C9 Inhibition 93% .2uM NoneNone View
dopamine receptor D3 DIETHYLSTILBESTROL Dopamine D3 93% 8.796uM 2.987uM View
solute carrier family 6 (neurotransmitter transporter, noradrenalin), member 2 ETHINYLESTRADIOL Adrenergic, Norepinephrine Transporter 93% .959uM .951uM View
mitogen activated protein kinase 1 LIPOPOLYSACCHARIDE E. COLI O55:B5 Protein Serine/Threonine Kinase, ERK2 93% .3208uM NoneNone View
mitogen-activated protein kinase 1 LIPOPOLYSACCHARIDE E. COLI O55:B5 Protein Serine/Threonine Kinase, ERK2 93% .3208uM NoneNone View
sodium channel, voltage-gated, type I, alpha MESTRANOL Sodium Channel, Site 2 93% 5.601uM 5.021uM View
sodium channel, voltage-gated, type IV, beta MESTRANOL Sodium Channel, Site 2 93% 5.601uM 5.021uM View
sodium channel associated protein 1 MESTRANOL Sodium Channel, Site 2 93% 5.601uM 5.021uM View
sodium channel associated protein 2 MESTRANOL Sodium Channel, Site 2 93% 5.601uM 5.021uM View
sodium channel, voltage-gated, type III, beta MESTRANOL Sodium Channel, Site 2 93% 5.601uM 5.021uM View
sodium channel, voltage-gated, type I, alpha MESTRANOL Sodium Channel, Site 2 93% 5.601uM 5.021uM View
sodium channel, voltage-gated, type IX, alpha MESTRANOL Sodium Channel, Site 2 93% 5.601uM 5.021uM View
sodium channel, voltage-gated, type VII, alpha MESTRANOL Sodium Channel, Site 2 93% 5.601uM 5.021uM View
amiloride-sensitive cation channel 5, intestinal MESTRANOL Sodium Channel, Site 2 93% 5.601uM 5.021uM View
sodium channel, voltage-gated, type III, beta MESTRANOL Sodium Channel, Site 2 93% 5.601uM 5.021uM View
sodium channel, voltage-gated, type VIII, alpha polypeptide MESTRANOL Sodium Channel, Site 2 93% 5.601uM 5.021uM View
sodium channel, voltage-gated, type XI, alpha MESTRANOL Sodium Channel, Site 2 93% 5.601uM 5.021uM View
sodium channel, voltage-gated, type I, beta MESTRANOL Sodium Channel, Site 2 93% 5.601uM 5.021uM View
sodium channel, voltage-gated, type 10, alpha polypeptide MESTRANOL Sodium Channel, Site 2 93% 5.601uM 5.021uM View
sodium channel, voltage-gated, type IV, alpha polypeptide MESTRANOL Sodium Channel, Site 2 93% 5.601uM 5.021uM View
sodium channel, voltage-gated, type V, alpha polypeptide MESTRANOL Sodium Channel, Site 2 93% 5.601uM 5.021uM View
sodium channel, voltage-gated, type II, beta MESTRANOL Sodium Channel, Site 2 93% 5.601uM 5.021uM View
sodium channel, nonvoltage-gated 1 alpha MESTRANOL Sodium Channel, Site 2 93% 5.601uM 5.021uM View
sodium channel, nonvoltage-gated 1 gamma MESTRANOL Sodium Channel, Site 2 93% 5.601uM 5.021uM View
sodium channel, nonvoltage-gated 1 beta MESTRANOL Sodium Channel, Site 2 93% 5.601uM 5.021uM View
sodium channel, voltage-gated, type 2, alpha 1 polypeptide MESTRANOL Sodium Channel, Site 2 93% 5.601uM 5.021uM View
sodium channel, voltage-gated, type XI, alpha MESTRANOL Sodium Channel, Site 2 93% 5.601uM 5.021uM View
sodium channel, nonvoltage-gated 1, gamma MESTRANOL Sodium Channel, Site 2 93% 5.601uM 5.021uM View
sodium channel, nonvoltage-gated 1, delta MESTRANOL Sodium Channel, Site 2 93% 5.601uM 5.021uM View
sodium channel, nonvoltage-gated 1, beta (Liddle syndrome) MESTRANOL Sodium Channel, Site 2 93% 5.601uM 5.021uM View
sodium channel, nonvoltage-gated 1 alpha MESTRANOL Sodium Channel, Site 2 93% 5.601uM 5.021uM View
sodium channel, voltage-gated, type X, alpha MESTRANOL Sodium Channel, Site 2 93% 5.601uM 5.021uM View
sodium channel, voltage-gated, type IX, alpha MESTRANOL Sodium Channel, Site 2 93% 5.601uM 5.021uM View
sodium channel, voltage gated, type VIII, alpha MESTRANOL Sodium Channel, Site 2 93% 5.601uM 5.021uM View
sodium channel, voltage-gated, type VII, alpha MESTRANOL Sodium Channel, Site 2 93% 5.601uM 5.021uM View
sodium channel, voltage-gated, type V, alpha (long QT syndrome 3) MESTRANOL Sodium Channel, Site 2 93% 5.601uM 5.021uM View
sodium channel, voltage-gated, type IV, beta MESTRANOL Sodium Channel, Site 2 93% 5.601uM 5.021uM View
sodium channel, voltage-gated, type IV, alpha MESTRANOL Sodium Channel, Site 2 93% 5.601uM 5.021uM View
sodium channel, voltage-gated, type III, alpha MESTRANOL Sodium Channel, Site 2 93% 5.601uM 5.021uM View
sodium channel, voltage-gated, type II, beta MESTRANOL Sodium Channel, Site 2 93% 5.601uM 5.021uM View
sodium channel, voltage-gated, type II, alpha 2 MESTRANOL Sodium Channel, Site 2 93% 5.601uM 5.021uM View
sodium channel, voltage-gated, type I, beta MESTRANOL Sodium Channel, Site 2 93% 5.601uM 5.021uM View
adrenergic receptor, alpha 2c (Non-specific probe) ERGOTAMINE Imidazoline I2, Central 93% .003645uM .00243uM View
calcium channel, voltage-dependent, beta 2 subunit TERCONAZOLE Calcium Channel Type L, Benzothiazepine 93% 3.008uM 2.674uM View
calcium channel, voltage-dependent, L type, alpha 1S subunit TERCONAZOLE Calcium Channel Type L, Benzothiazepine 93% 3.008uM 2.674uM View
calcium channel, voltage-dependent, alpha 1F subunit TERCONAZOLE Calcium Channel Type L, Benzothiazepine 93% 3.008uM 2.674uM View
calcium channel, voltage-dependent, L type, alpha 1D subunit TERCONAZOLE Calcium Channel Type L, Benzothiazepine 93% 3.008uM 2.674uM View
calcium channel, voltage-dependent, L type, alpha 1C subunit TERCONAZOLE Calcium Channel Type L, Benzothiazepine 93% 3.008uM 2.674uM View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit TERCONAZOLE Calcium Channel Type L, Benzothiazepine 93% 3.008uM 2.674uM View
calcium channel, voltage-dependent, beta 1 subunit TERCONAZOLE Calcium Channel Type L, Benzothiazepine 93% 3.008uM 2.674uM View
calcium channel, voltage-dependent, L type, alpha 1E subunit TERCONAZOLE Calcium Channel Type L, Benzothiazepine 93% 3.008uM 2.674uM View
calcium channel, voltage-dependent, N type, alpha 1B subunit TERCONAZOLE Calcium Channel Type L, Benzothiazepine 93% 3.008uM 2.674uM View
calcium channel, voltage-dependent, alpha2/delta subunit 1 TERCONAZOLE Calcium Channel Type L, Benzothiazepine 93% 3.008uM 2.674uM View
calcium channel, voltage-dependent, gamma subunit 8 TERCONAZOLE Calcium Channel Type L, Benzothiazepine 93% 3.008uM 2.674uM View
calcium channel, voltage-dependent, gamma subunit 7 TERCONAZOLE Calcium Channel Type L, Benzothiazepine 93% 3.008uM 2.674uM View
calcium channel, voltage-dependent, gamma subunit 6 TERCONAZOLE Calcium Channel Type L, Benzothiazepine 93% 3.008uM 2.674uM View
calcium channel, voltage-dependent, gamma subunit 5 TERCONAZOLE Calcium Channel Type L, Benzothiazepine 93% 3.008uM 2.674uM View
calcium channel, voltage-dependent, gamma subunit 4 TERCONAZOLE Calcium Channel Type L, Benzothiazepine 93% 3.008uM 2.674uM View
calcium channel, voltage-dependent, gamma subunit 3 TERCONAZOLE Calcium Channel Type L, Benzothiazepine 93% 3.008uM 2.674uM View
calcium channel, voltage-dependent, gamma subunit 2 TERCONAZOLE Calcium Channel Type L, Benzothiazepine 93% 3.008uM 2.674uM View
calcium channel, voltage-dependent, gamma subunit 1 TERCONAZOLE Calcium Channel Type L, Benzothiazepine 93% 3.008uM 2.674uM View
calcium channel, voltage-dependent, beta 4 subunit TERCONAZOLE Calcium Channel Type L, Benzothiazepine 93% 3.008uM 2.674uM View
calcium channel, voltage-dependent, beta 3 subunit TERCONAZOLE Calcium Channel Type L, Benzothiazepine 93% 3.008uM 2.674uM View
cholinergic receptor, muscarinic 1 PROCHLORPERAZINE Muscarinic M1 93% 1.013uM .244uM View
dopamine receptor D3 METOCLOPRAMIDE Dopamine D3 93% .2uM .068uM View
opioid receptor, sigma 1 PIPAMAZINE Sigma1 93% .114uM .048uM View
dopamine receptor 2 CYPROHEPTADINE Dopamine D2L 93% .164uM .055uM View
A3 adenosine receptor DISULFIRAM Adenosine A3 93% .356uM .201uM View
calcium channel, voltage-dependent, L type, alpha 1E subunit EBASTINE Calcium Channel Type L, Dihydropyridine 92% .1436uM .0923uM View
calcium channel, voltage-dependent, N type, alpha 1B subunit EBASTINE Calcium Channel Type L, Dihydropyridine 92% .1436uM .0923uM View
calcium channel, voltage-dependent, alpha2/delta subunit 1 EBASTINE Calcium Channel Type L, Dihydropyridine 92% .1436uM .0923uM View
adrenergic receptor, alpha 1a PROMETHAZINE Adrenergic alpha1A 92% .079uM .032uM View
5-hydroxytryptamine (serotonin) receptor 2A CETYLPYRIDINIUM BROMIDE Serotonin 5-HT2A 92% 3.173uM .907uM View
adrenergic receptor, alpha 2a RALOXIFENE Adrenergic alpha2A 92% 1.664uM .624uM View
dopamine receptor 2 RALOXIFENE Dopamine D2L 92% 1.174uM .391uM View
solute carrier family 6 (neurotransmitter transporter, noradrenalin), member 2 4-NONYLPHENOL Adrenergic, Norepinephrine Transporter 92% 1.254uM 1.244uM View
opioid receptor, kappa 1 ASTEMIZOLE Opiate kappa 92% 6.616uM 2.646uM View
5-hydroxytryptamine (serotonin) receptor 2A CLOMIPHENE Serotonin 5-HT2A 92% 3.308uM .945uM View
5-hydroxytryptamine (serotonin) receptor 2C CLOMIPHENE Serotonin 5-HT2C 92% 1.272uM .666uM View
adrenergic receptor, beta 3 PROPAFENONE Adrenergic beta3 92% .424uM .318uM View
androgen receptor TIBOLONE Testosterone 92% .113uM .0754uM View
5-hydroxytryptamine (serotonin) receptor 2B S-(-)-PROPRANOLOL Serotonin 5-HT2B 92% .411uM .262uM View
sodium channel, voltage-gated, type V, alpha (long QT syndrome 3) ITRACONAZOLE Sodium Channel, Site 2 92% 2.577uM 2.351uM View
sodium channel, voltage-gated, type IV, beta ITRACONAZOLE Sodium Channel, Site 2 92% 2.577uM 2.351uM View
sodium channel, voltage-gated, type IV, alpha ITRACONAZOLE Sodium Channel, Site 2 92% 2.577uM 2.351uM View
sodium channel, voltage-gated, type III, alpha ITRACONAZOLE Sodium Channel, Site 2 92% 2.577uM 2.351uM View