Gene Activity List


Gene Activity List

Gene Compound Assay Inh Ic50 Ki View
calcium channel, voltage-dependent, beta 4 subunit NITRENDIPINE Calcium Channel Type L, Dihydropyridine 100% .000383uM .000246uM View
calcium channel, voltage-dependent, beta 3 subunit NITRENDIPINE Calcium Channel Type L, Dihydropyridine 100% .000383uM .000246uM View
calcium channel, voltage-dependent, beta 2 subunit NITRENDIPINE Calcium Channel Type L, Dihydropyridine 100% .000383uM .000246uM View
calcium channel, voltage-dependent, L type, alpha 1S subunit NITRENDIPINE Calcium Channel Type L, Dihydropyridine 100% .000383uM .000246uM View
calcium channel, voltage-dependent, alpha 1F subunit NITRENDIPINE Calcium Channel Type L, Dihydropyridine 100% .000383uM .000246uM View
calcium channel, voltage-dependent, L type, alpha 1D subunit NITRENDIPINE Calcium Channel Type L, Dihydropyridine 100% .000383uM .000246uM View
calcium channel, voltage-dependent, L type, alpha 1C subunit NITRENDIPINE Calcium Channel Type L, Dihydropyridine 100% .000383uM .000246uM View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit NITRENDIPINE Calcium Channel Type L, Dihydropyridine 100% .000383uM .000246uM View
calcium channel, voltage-dependent, beta 1 subunit NITRENDIPINE Calcium Channel Type L, Dihydropyridine 100% .000383uM .000246uM View
calcium channel, voltage-dependent, L type, alpha 1E subunit NITRENDIPINE Calcium Channel Type L, Dihydropyridine 100% .000383uM .000246uM View
calcium channel, voltage-dependent, N type, alpha 1B subunit NITRENDIPINE Calcium Channel Type L, Dihydropyridine 100% .000383uM .000246uM View
calcium channel, voltage-dependent, alpha2/delta subunit 1 NITRENDIPINE Calcium Channel Type L, Dihydropyridine 100% .000383uM .000246uM View
adrenergic receptor, alpha 1b QUETIAPINE Adrenergic alpha1B 100% .0245uM .0136uM View
adrenergic receptor, alpha 1d (Non-specific probe) PROMAZINE Adrenergic alpha1D 100% .013uM .00618uM View
adrenergic receptor, alpha 2b PROMAZINE Adrenergic alpha2B 100% .018uM .008418uM View
adrenergic receptor, alpha 2b METERGOLINE Adrenergic alpha2B 100% .016uM .007516uM View
calcium channel, voltage-dependent, gamma subunit 8 METERGOLINE Calcium Channel Type L, Phenylalkylamine 100% .278uM .27uM View
calcium channel, voltage-dependent, gamma subunit 7 METERGOLINE Calcium Channel Type L, Phenylalkylamine 100% .278uM .27uM View
calcium channel, voltage-dependent, gamma subunit 6 METERGOLINE Calcium Channel Type L, Phenylalkylamine 100% .278uM .27uM View
calcium channel, voltage-dependent, gamma subunit 5 METERGOLINE Calcium Channel Type L, Phenylalkylamine 100% .278uM .27uM View
calcium channel, voltage-dependent, gamma subunit 4 METERGOLINE Calcium Channel Type L, Phenylalkylamine 100% .278uM .27uM View
calcium channel, voltage-dependent, gamma subunit 3 METERGOLINE Calcium Channel Type L, Phenylalkylamine 100% .278uM .27uM View
calcium channel, voltage-dependent, gamma subunit 2 METERGOLINE Calcium Channel Type L, Phenylalkylamine 100% .278uM .27uM View
calcium channel, voltage-dependent, gamma subunit 1 METERGOLINE Calcium Channel Type L, Phenylalkylamine 100% .278uM .27uM View
aldo-keto reductase family 7, member A3 (aflatoxin aldehyde reductase) SULINDAC SULFONE Aldose Reductase 100% .269uM NoneNone View
solute carrier family 6 (neurotransmitter transporter, noradrenalin), member 2 PAROXETINE Adrenergic, Norepinephrine Transporter 100% .086uM .086uM View
cholinergic receptor, muscarinic 5 PAROXETINE Muscarinic M5 100% .123uM .089uM View
solute carrier family 6 (neurotransmitter transporter, serotonin), member 4 PAROXETINE Serotonin Transporter 100% .00008uM .000043uM View
5-hydroxytryptamine (serotonin) receptor 1B SUMATRIPTAN Serotonin 5-HT1B 100% .018uM .008191uM View
opioid receptor, delta 1 NALTREXONE Opiate delta 100% .251uM .088uM View
opioid receptor, kappa 1 NALTREXONE Opiate kappa 100% .018uM .007175uM View
sodium channel, voltage-gated, type X, alpha PROCHLORPERAZINE Sodium Channel, Site 2 100% 1.265uM 1.154uM View
sodium channel, voltage-gated, type IX, alpha PROCHLORPERAZINE Sodium Channel, Site 2 100% 1.265uM 1.154uM View
sodium channel, voltage gated, type VIII, alpha PROCHLORPERAZINE Sodium Channel, Site 2 100% 1.265uM 1.154uM View
sodium channel, voltage-gated, type VII, alpha PROCHLORPERAZINE Sodium Channel, Site 2 100% 1.265uM 1.154uM View
sodium channel, voltage-gated, type V, alpha (long QT syndrome 3) PROCHLORPERAZINE Sodium Channel, Site 2 100% 1.265uM 1.154uM View
protein kinase C, theta PACLITAXEL Phorbol Ester 19% NoneNone NoneNone View
sodium channel, voltage-gated, type IV, beta PROCHLORPERAZINE Sodium Channel, Site 2 100% 1.265uM 1.154uM View
sodium channel, voltage-gated, type IV, alpha PROCHLORPERAZINE Sodium Channel, Site 2 100% 1.265uM 1.154uM View
sodium channel, voltage-gated, type III, alpha PROCHLORPERAZINE Sodium Channel, Site 2 100% 1.265uM 1.154uM View
sodium channel, voltage-gated, type II, beta PROCHLORPERAZINE Sodium Channel, Site 2 100% 1.265uM 1.154uM View
sodium channel, voltage-gated, type II, alpha 2 PROCHLORPERAZINE Sodium Channel, Site 2 100% 1.265uM 1.154uM View
sodium channel, voltage-gated, type I, beta PROCHLORPERAZINE Sodium Channel, Site 2 100% 1.265uM 1.154uM View
sodium channel, voltage-gated, type I, alpha PROCHLORPERAZINE Sodium Channel, Site 2 100% 1.265uM 1.154uM View
adrenergic receptor, alpha 1b PROCHLORPERAZINE Adrenergic alpha1B 100% .089uM .049uM View
adrenergic receptor, alpha 2b PROCHLORPERAZINE Adrenergic alpha2B 100% .01uM .004741uM View
5-hydroxytryptamine (serotonin) receptor 2A PROCHLORPERAZINE Serotonin 5-HT2A 100% .007062uM .002018uM View
5-hydroxytryptamine (serotonin) receptor 1A PINDOLOL Serotonin 5-HT1A 100% .048uM .027uM View
adrenergic receptor, alpha 1d (Non-specific probe) PRAZOSIN Adrenergic alpha1D 100% .000656uM .000323uM View
adrenergic receptor, alpha 2a PROCHLORPERAZINE Adrenergic alpha2A 100% .169uM .063uM View
adrenergic receptor, alpha 1a PRAZOSIN Adrenergic alpha1A 100% .000218uM .000088uM View
adrenergic receptor, beta 2 PINDOLOL Adrenergic beta2 100% .000549uM .000377uM View
adrenergic receptor, alpha 2b PROCHLORPERAZINE Adrenergic alpha2C 100% .082uM .012uM View
adrenergic receptor, alpha 2c (Non-specific probe) PROCHLORPERAZINE Adrenergic alpha2C 100% .082uM .012uM View
dopamine receptor D3 PROCHLORPERAZINE Dopamine D3 100% .013uM .004454uM View
matrix metalloproteinase 1 (interstitial collagenase) PRAZOSIN Protease, Matrix Metalloprotease-1 (MMP-1) 100% 4.036uM NoneNone View
dopamine receptor D1A METERGOLINE Dopamine D1 100% .074uM .037uM View
5-hydroxytryptamine (serotonin) receptor 2B METERGOLINE Serotonin 5-HT2B 100% .000442uM .000281uM View
sodium channel, voltage-gated, type IV, beta METERGOLINE Sodium Channel, Site 2 100% .792uM .723uM View
sodium channel associated protein 1 METERGOLINE Sodium Channel, Site 2 100% .792uM .723uM View
sodium channel associated protein 2 METERGOLINE Sodium Channel, Site 2 100% .792uM .723uM View
sodium channel, voltage-gated, type III, beta METERGOLINE Sodium Channel, Site 2 100% .792uM .723uM View
sodium channel, voltage-gated, type I, alpha METERGOLINE Sodium Channel, Site 2 100% .792uM .723uM View
sodium channel, voltage-gated, type IX, alpha METERGOLINE Sodium Channel, Site 2 100% .792uM .723uM View
sodium channel, voltage-gated, type VII, alpha METERGOLINE Sodium Channel, Site 2 100% .792uM .723uM View
amiloride-sensitive cation channel 5, intestinal METERGOLINE Sodium Channel, Site 2 100% .792uM .723uM View
sodium channel, voltage-gated, type III, beta METERGOLINE Sodium Channel, Site 2 100% .792uM .723uM View
sodium channel, voltage-gated, type VIII, alpha polypeptide METERGOLINE Sodium Channel, Site 2 100% .792uM .723uM View
sodium channel, voltage-gated, type XI, alpha METERGOLINE Sodium Channel, Site 2 100% .792uM .723uM View
sodium channel, voltage-gated, type I, beta METERGOLINE Sodium Channel, Site 2 100% .792uM .723uM View
sodium channel, voltage-gated, type 10, alpha polypeptide METERGOLINE Sodium Channel, Site 2 100% .792uM .723uM View
sodium channel, voltage-gated, type IV, alpha polypeptide METERGOLINE Sodium Channel, Site 2 100% .792uM .723uM View
sodium channel, voltage-gated, type V, alpha polypeptide METERGOLINE Sodium Channel, Site 2 100% .792uM .723uM View
sodium channel, voltage-gated, type II, beta METERGOLINE Sodium Channel, Site 2 100% .792uM .723uM View
sodium channel, nonvoltage-gated 1 alpha METERGOLINE Sodium Channel, Site 2 100% .792uM .723uM View
sodium channel, nonvoltage-gated 1 gamma METERGOLINE Sodium Channel, Site 2 100% .792uM .723uM View
sodium channel, nonvoltage-gated 1 beta METERGOLINE Sodium Channel, Site 2 100% .792uM .723uM View
sodium channel, voltage-gated, type 2, alpha 1 polypeptide METERGOLINE Sodium Channel, Site 2 100% .792uM .723uM View
sodium channel, voltage-gated, type XI, alpha METERGOLINE Sodium Channel, Site 2 100% .792uM .723uM View
sodium channel, nonvoltage-gated 1, gamma METERGOLINE Sodium Channel, Site 2 100% .792uM .723uM View
sodium channel, nonvoltage-gated 1, delta METERGOLINE Sodium Channel, Site 2 100% .792uM .723uM View
sodium channel, nonvoltage-gated 1, beta (Liddle syndrome) METERGOLINE Sodium Channel, Site 2 100% .792uM .723uM View
sodium channel, nonvoltage-gated 1 alpha METERGOLINE Sodium Channel, Site 2 100% .792uM .723uM View
sodium channel, voltage-gated, type X, alpha METERGOLINE Sodium Channel, Site 2 100% .792uM .723uM View
sodium channel, voltage-gated, type IX, alpha METERGOLINE Sodium Channel, Site 2 100% .792uM .723uM View
sodium channel, voltage gated, type VIII, alpha METERGOLINE Sodium Channel, Site 2 100% .792uM .723uM View
sodium channel, voltage-gated, type VII, alpha METERGOLINE Sodium Channel, Site 2 100% .792uM .723uM View
sodium channel, voltage-gated, type V, alpha (long QT syndrome 3) METERGOLINE Sodium Channel, Site 2 100% .792uM .723uM View
sodium channel, voltage-gated, type IV, beta METERGOLINE Sodium Channel, Site 2 100% .792uM .723uM View
sodium channel, voltage-gated, type IV, alpha METERGOLINE Sodium Channel, Site 2 100% .792uM .723uM View
sodium channel, voltage-gated, type III, alpha METERGOLINE Sodium Channel, Site 2 100% .792uM .723uM View
sodium channel, voltage-gated, type II, beta METERGOLINE Sodium Channel, Site 2 100% .792uM .723uM View
sodium channel, voltage-gated, type II, alpha 2 METERGOLINE Sodium Channel, Site 2 100% .792uM .723uM View
sodium channel, voltage-gated, type I, beta METERGOLINE Sodium Channel, Site 2 100% .792uM .723uM View
sodium channel, voltage-gated, type I, alpha METERGOLINE Sodium Channel, Site 2 100% .792uM .723uM View
adrenergic receptor, alpha 1a METERGOLINE Adrenergic alpha1A 100% .095uM .038uM View
dopamine receptor D1A MICONAZOLE Dopamine D1 100% 6.247uM 3.124uM View
solute carrier family 6 (neurotransmitter transporter, noradrenalin), member 2 MICONAZOLE Adrenergic, Norepinephrine Transporter 100% 2.939uM 2.915uM View
solute carrier family 6 (neurotransmitter transporter, dopamine), member 3 MICONAZOLE Dopamine Transporter 100% 1.701uM 1.352uM View
tachykinin receptor 2 MICONAZOLE Tachykinin NK2 100% 4.839uM 1.613uM View
5-hydroxytryptamine receptor 6 MICONAZOLE Serotonin 5-HT6 100% 10.887uM 5.055uM View
solute carrier family 6 (neurotransmitter transporter, serotonin), member 4 MICONAZOLE Serotonin Transporter 100% .778uM .414uM View
5-hydroxytryptamine (serotonin) receptor 2C PIPAMAZINE Serotonin 5-HT2C 100% .022uM .011uM View
5-hydroxytryptamine (serotonin) receptor 2A PIPAMAZINE Serotonin 5-HT2A 100% .001938uM .000554uM View
adrenergic receptor, alpha 2b PIPAMAZINE Adrenergic alpha2B 100% .001722uM .000786uM View
dopamine receptor D3 CYPROHEPTADINE Dopamine D3 100% .048uM .016uM View
adrenergic receptor, alpha 1d (Non-specific probe) CYPROHEPTADINE Adrenergic alpha1D 100% .107uM .053uM View
dopamine receptor D1A PIPAMAZINE Dopamine D1 100% .032uM .016uM View
5-hydroxytryptamine receptor 6 PIPAMAZINE Serotonin 5-HT6 100% .112uM .052uM View
cholinergic receptor, muscarinic 1 CYPROHEPTADINE Muscarinic M1 100% .016uM .003943uM View
cholinergic receptor, muscarinic 4 CYPROHEPTADINE Muscarinic M4 100% .016uM .002186uM View
histamine receptor H 1 CYPROHEPTADINE Histamine H1, Central 100% .0037uM .00043uM View
5-hydroxytryptamine (serotonin) receptor 2A CYPROHEPTADINE Serotonin 5-HT2A 100% .000973uM .000278uM View
adrenergic receptor, alpha 2a GUANABENZ Imidazoline I2, Central 100% .018uM .012uM View
adrenergic receptor, alpha 2c (Non-specific probe) GUANABENZ Imidazoline I2, Central 100% .018uM .012uM View
5-hydroxytryptamine (serotonin) receptor 2B GUANABENZ Serotonin 5-HT2B 100% .097uM .062uM View
5-hydroxytryptamine (serotonin) receptor 1A S-(-)-PROPRANOLOL Serotonin 5-HT1A 100% .124uM .071uM View
adrenergic receptor, alpha 2b GUANABENZ Adrenergic alpha2B 100% .149uM .068uM View
3-hydroxy-3-methylglutaryl-Coenzyme A reductase FLUVASTATIN HMG-CoA Reductase 100% .000353uM NoneNone View
3-hydroxy-3-methylglutaryl-Coenzyme A reductase FLUVASTATIN HMG-CoA Reductase 100% .000353uM NoneNone View
nuclear receptor subfamily 3, group C, member 1 HALCINONIDE Glucocorticoid 100% .001611uM .000732uM View
adrenergic receptor, alpha 2a CYPROHEPTADINE Adrenergic alpha2A 100% .283uM .106uM View
adrenergic receptor, alpha 2b CYPROHEPTADINE Adrenergic alpha2B 100% .038uM .017uM View
adrenergic receptor, alpha 2a PERGOLIDE Adrenergic alpha2A 100% .264uM .099uM View
prostaglandin-endoperoxide synthase 1 PIROXICAM Cyclooxygenase COX-1 100% 1.313uM NoneNone View
prostaglandin-endoperoxide synthase 1 (prostaglandin G/H synthase and cyclooxygenase) PIROXICAM Cyclooxygenase COX-1 100% 1.313uM NoneNone View
5-hydroxytryptamine (serotonin) receptor 1B PERGOLIDE Serotonin 5-HT1B 100% .087uM .04uM View
adrenergic receptor, alpha 2b PERGOLIDE Adrenergic alpha2B 100% .064uM .029uM View
dopamine receptor D3 PERGOLIDE Dopamine D3 100% .005393uM .001832uM View
5-hydroxytryptamine (serotonin) receptor 1A PERGOLIDE Serotonin 5-HT1A 100% .015uM .008468uM View
5-hydroxytryptamine receptor 6 PERGOLIDE Serotonin 5-HT6 100% .039uM .018uM View
dopamine receptor 2 PROCHLORPERAZINE Dopamine D2L 100% .011uM .003608uM View
5-hydroxytryptamine (serotonin) receptor 2B PERGOLIDE Serotonin 5-HT2B 100% .076uM .049uM View
monoamine oxidase A PHENELZINE Monoamine Oxidase MAOA 100% .146uM NoneNone View
monoamine oxidase A PHENELZINE Monoamine Oxidase MAOA 100% .146uM NoneNone View
sodium channel, voltage-gated, type IV, beta PROCHLORPERAZINE Sodium Channel, Site 2 100% 1.265uM 1.154uM View
calcium channel, voltage-dependent, beta 4 subunit METERGOLINE Calcium Channel Type L, Phenylalkylamine 100% .278uM .27uM View
calcium channel, voltage-dependent, beta 3 subunit METERGOLINE Calcium Channel Type L, Phenylalkylamine 100% .278uM .27uM View
calcium channel, voltage-dependent, beta 2 subunit METERGOLINE Calcium Channel Type L, Phenylalkylamine 100% .278uM .27uM View
calcium channel, voltage-dependent, L type, alpha 1S subunit METERGOLINE Calcium Channel Type L, Phenylalkylamine 100% .278uM .27uM View
calcium channel, voltage-dependent, alpha 1F subunit METERGOLINE Calcium Channel Type L, Phenylalkylamine 100% .278uM .27uM View
calcium channel, voltage-dependent, L type, alpha 1D subunit METERGOLINE Calcium Channel Type L, Phenylalkylamine 100% .278uM .27uM View
calcium channel, voltage-dependent, L type, alpha 1C subunit METERGOLINE Calcium Channel Type L, Phenylalkylamine 100% .278uM .27uM View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit METERGOLINE Calcium Channel Type L, Phenylalkylamine 100% .278uM .27uM View
calcium channel, voltage-dependent, beta 1 subunit METERGOLINE Calcium Channel Type L, Phenylalkylamine 100% .278uM .27uM View
calcium channel, voltage-dependent, L type, alpha 1E subunit METERGOLINE Calcium Channel Type L, Phenylalkylamine 100% .278uM .27uM View
calcium channel, voltage-dependent, N type, alpha 1B subunit METERGOLINE Calcium Channel Type L, Phenylalkylamine 100% .278uM .27uM View
calcium channel, voltage-dependent, alpha2/delta subunit 1 METERGOLINE Calcium Channel Type L, Phenylalkylamine 100% .278uM .27uM View
5-hydroxytryptamine (serotonin) receptor 1B METERGOLINE Serotonin 5-HT1B 100% .019uM .011uM View
adrenergic receptor, alpha 1b DOMPERIDONE Adrenergic alpha1B 100% .158uM .087uM View
5-hydroxytryptamine (serotonin) receptor 5B METERGOLINE Serotonin 5-HT4 100% 1.641uM .274uM View
5-hydroxytryptamine (serotonin) receptor 4 METERGOLINE Serotonin 5-HT4 100% 1.641uM .274uM View
androgen receptor STANOLONE Testosterone 100% .002305uM .001537uM View
adrenergic receptor, alpha 2a METERGOLINE Adrenergic alpha2A 100% .058uM .022uM View
dopamine receptor D3 METERGOLINE Dopamine D3 100% .007689uM .002611uM View
5-hydroxytryptamine receptor 6 METERGOLINE Serotonin 5-HT6 100% .028uM .013uM View
calcium channel, voltage-dependent, gamma subunit 8 METERGOLINE Calcium Channel Type L, Benzothiazepine 100% .268uM .238uM View
calcium channel, voltage-dependent, gamma subunit 7 METERGOLINE Calcium Channel Type L, Benzothiazepine 100% .268uM .238uM View
calcium channel, voltage-dependent, gamma subunit 6 METERGOLINE Calcium Channel Type L, Benzothiazepine 100% .268uM .238uM View
calcium channel, voltage-dependent, gamma subunit 5 METERGOLINE Calcium Channel Type L, Benzothiazepine 100% .268uM .238uM View
calcium channel, voltage-dependent, gamma subunit 4 METERGOLINE Calcium Channel Type L, Benzothiazepine 100% .268uM .238uM View
calcium channel, voltage-dependent, gamma subunit 3 METERGOLINE Calcium Channel Type L, Benzothiazepine 100% .268uM .238uM View
calcium channel, voltage-dependent, gamma subunit 2 METERGOLINE Calcium Channel Type L, Benzothiazepine 100% .268uM .238uM View
calcium channel, voltage-dependent, gamma subunit 1 METERGOLINE Calcium Channel Type L, Benzothiazepine 100% .268uM .238uM View
calcium channel, voltage-dependent, beta 4 subunit METERGOLINE Calcium Channel Type L, Benzothiazepine 100% .268uM .238uM View
calcium channel, voltage-dependent, beta 3 subunit METERGOLINE Calcium Channel Type L, Benzothiazepine 100% .268uM .238uM View
calcium channel, voltage-dependent, beta 2 subunit METERGOLINE Calcium Channel Type L, Benzothiazepine 100% .268uM .238uM View
calcium channel, voltage-dependent, L type, alpha 1S subunit METERGOLINE Calcium Channel Type L, Benzothiazepine 100% .268uM .238uM View
calcium channel, voltage-dependent, alpha 1F subunit METERGOLINE Calcium Channel Type L, Benzothiazepine 100% .268uM .238uM View
calcium channel, voltage-dependent, L type, alpha 1D subunit METERGOLINE Calcium Channel Type L, Benzothiazepine 100% .268uM .238uM View
phosphodiesterase 4B, cAMP specific GENISTEIN Phosphodiesterase PDE4 74% 10.924uM NoneNone View
calcium channel, voltage-dependent, L type, alpha 1C subunit METERGOLINE Calcium Channel Type L, Benzothiazepine 100% .268uM .238uM View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit METERGOLINE Calcium Channel Type L, Benzothiazepine 100% .268uM .238uM View
calcium channel, voltage-dependent, beta 1 subunit METERGOLINE Calcium Channel Type L, Benzothiazepine 100% .268uM .238uM View
calcium channel, voltage-dependent, L type, alpha 1E subunit METERGOLINE Calcium Channel Type L, Benzothiazepine 100% .268uM .238uM View
calcium channel, voltage-dependent, N type, alpha 1B subunit METERGOLINE Calcium Channel Type L, Benzothiazepine 100% .268uM .238uM View
calcium channel, voltage-dependent, alpha2/delta subunit 1 METERGOLINE Calcium Channel Type L, Benzothiazepine 100% .268uM .238uM View
phosphodiesterase 5A, cGMP-specific SILDENAFIL Phosphodiesterase PDE5 100% .004577uM NoneNone View
phosphodiesterase 5A, cGMP-specific SILDENAFIL Phosphodiesterase PDE5 100% .004577uM NoneNone View
acetylcholinesterase (YT blood group) TACRINE Acetylcholinesterase 100% .33uM NoneNone View
collagen-like tail subunit (single strand of homotrimer) of asymmetric acetylcholinesterase TACRINE Acetylcholinesterase 100% .33uM NoneNone View
acetylcholinesterase TACRINE Acetylcholinesterase 100% .33uM NoneNone View
aldo-keto reductase family 1, member B4 (aldose reductase) SULINDAC SULFONE Aldose Reductase 100% .269uM NoneNone View
aldo-keto reductase family 1, member B1 (aldose reductase) SULINDAC SULFONE Aldose Reductase 100% .269uM NoneNone View
aldo-keto reductase family 7, member A2 (aflatoxin aldehyde reductase) SULINDAC SULFONE Aldose Reductase 100% .269uM NoneNone View
prostaglandin-endoperoxide synthase 2 (prostaglandin G/H synthase and cyclooxygenase) 3,3',4',5-TETRACHLOROSALICYLANILIDE Cyclooxygenase COX-2 100% .542uM NoneNone View
A3 adenosine receptor MONTELUKAST Adenosine A3 100% .434uM .245uM View
Cytochrom P450-2C19 monooxygenase OXICONAZOLE CYP450-2C19 Inhibition 100% .04uM NoneNone View
Cytochrom P450-2D6 monooxygenase TRIAMTERENE CYP450-2D6 Inhibition 100% 10uM NoneNone View
Cytochrom P450-2D6 monooxygenase BROMHEXINE CYP450-2D6 Inhibition 100% .1958uM NoneNone View
calcium channel, voltage-dependent, gamma subunit 8 TERFENADINE Calcium Channel Type L, Phenylalkylamine 100% .624uM .607uM View
calcium channel, voltage-dependent, gamma subunit 7 TERFENADINE Calcium Channel Type L, Phenylalkylamine 100% .624uM .607uM View
calcium channel, voltage-dependent, gamma subunit 6 TERFENADINE Calcium Channel Type L, Phenylalkylamine 100% .624uM .607uM View
calcium channel, voltage-dependent, gamma subunit 5 TERFENADINE Calcium Channel Type L, Phenylalkylamine 100% .624uM .607uM View
calcium channel, voltage-dependent, gamma subunit 4 TERFENADINE Calcium Channel Type L, Phenylalkylamine 100% .624uM .607uM View
calcium channel, voltage-dependent, gamma subunit 3 TERFENADINE Calcium Channel Type L, Phenylalkylamine 100% .624uM .607uM View
calcium channel, voltage-dependent, gamma subunit 2 TERFENADINE Calcium Channel Type L, Phenylalkylamine 100% .624uM .607uM View
calcium channel, voltage-dependent, gamma subunit 1 TERFENADINE Calcium Channel Type L, Phenylalkylamine 100% .624uM .607uM View
calcium channel, voltage-dependent, beta 4 subunit TERFENADINE Calcium Channel Type L, Phenylalkylamine 100% .624uM .607uM View
calcium channel, voltage-dependent, beta 3 subunit TERFENADINE Calcium Channel Type L, Phenylalkylamine 100% .624uM .607uM View