Gene Activity List


Gene Activity List

Gene Compound Assay Inh Ic50 Ki View
potassium voltage-gated channel, subfamily H (eag-related), member 2 CHLORPROMAZINE Potassium Channel HERG 72% 5.8275uM 4.7743uM View
potassium voltage-gated channel, subfamily H (eag-related), member 5 CHLORPROMAZINE Potassium Channel HERG 72% 5.8275uM 4.7743uM View
potassium voltage-gated channel, subfamily H (eag-related), member 3 CHLORPROMAZINE Potassium Channel HERG 72% 5.8275uM 4.7743uM View
potassium voltage-gated channel, subfamily H (eag-related), member 4 CHLORPROMAZINE Potassium Channel HERG 72% 5.8275uM 4.7743uM View
potassium voltage-gated channel, subfamily H (eag-related), member 1 CHLORPROMAZINE Potassium Channel HERG 72% 5.8275uM 4.7743uM View
calcium channel, voltage-dependent, L type, alpha 1E subunit BW-723C86 Calcium Channel Type L, Benzothiazepine 73% 3.4696uM 3.0841uM View
calcium channel, voltage-dependent, N type, alpha 1B subunit BW-723C86 Calcium Channel Type L, Benzothiazepine 73% 3.4696uM 3.0841uM View
calcium channel, voltage-dependent, alpha2/delta subunit 1 BW-723C86 Calcium Channel Type L, Benzothiazepine 73% 3.4696uM 3.0841uM View
cholinergic receptor, muscarinic 5 SULOCTIDIL Muscarinic M5 73% 4.4868uM 3.2235uM View
solute carrier family 6 (neurotransmitter transporter, serotonin), member 4 DOMPERIDONE Serotonin Transporter 73% 3.055uM 1.623uM View
mitogen activated protein kinase 3 ZAFIRLUKAST Protein Serine/Threonine Kinase, ERK1 73% 4.376uM NoneNone View
mitogen-activated protein kinase 3 ZAFIRLUKAST Protein Serine/Threonine Kinase, ERK1 73% 4.376uM NoneNone View
cholinergic receptor, muscarinic 1 MONTELUKAST Muscarinic M1 73% 8.045uM 1.938uM View
cholinergic receptor, muscarinic 1 METHAPYRILENE Muscarinic M1 73% 4.773uM 1.15uM View
dopamine receptor D3 MONTELUKAST Dopamine D3 73% 7.747uM 2.631uM View
calcium channel, voltage-dependent, gamma subunit 8 DESLORATADINE Calcium Channel Type L, Benzothiazepine 73% 5.791uM 5.148uM View
calcium channel, voltage-dependent, gamma subunit 7 DESLORATADINE Calcium Channel Type L, Benzothiazepine 73% 5.791uM 5.148uM View
calcium channel, voltage-dependent, gamma subunit 6 DESLORATADINE Calcium Channel Type L, Benzothiazepine 73% 5.791uM 5.148uM View
calcium channel, voltage-dependent, gamma subunit 5 DESLORATADINE Calcium Channel Type L, Benzothiazepine 73% 5.791uM 5.148uM View
calcium channel, voltage-dependent, gamma subunit 4 DESLORATADINE Calcium Channel Type L, Benzothiazepine 73% 5.791uM 5.148uM View
calcium channel, voltage-dependent, gamma subunit 3 DESLORATADINE Calcium Channel Type L, Benzothiazepine 73% 5.791uM 5.148uM View
calcium channel, voltage-dependent, gamma subunit 2 DESLORATADINE Calcium Channel Type L, Benzothiazepine 73% 5.791uM 5.148uM View
calcium channel, voltage-dependent, gamma subunit 1 DESLORATADINE Calcium Channel Type L, Benzothiazepine 73% 5.791uM 5.148uM View
calcium channel, voltage-dependent, beta 4 subunit DESLORATADINE Calcium Channel Type L, Benzothiazepine 73% 5.791uM 5.148uM View
calcium channel, voltage-dependent, beta 3 subunit DESLORATADINE Calcium Channel Type L, Benzothiazepine 73% 5.791uM 5.148uM View
calcium channel, voltage-dependent, beta 2 subunit DESLORATADINE Calcium Channel Type L, Benzothiazepine 73% 5.791uM 5.148uM View
calcium channel, voltage-dependent, L type, alpha 1S subunit DESLORATADINE Calcium Channel Type L, Benzothiazepine 73% 5.791uM 5.148uM View
calcium channel, voltage-dependent, alpha 1F subunit DESLORATADINE Calcium Channel Type L, Benzothiazepine 73% 5.791uM 5.148uM View
calcium channel, voltage-dependent, L type, alpha 1D subunit DESLORATADINE Calcium Channel Type L, Benzothiazepine 73% 5.791uM 5.148uM View
calcium channel, voltage-dependent, L type, alpha 1C subunit DESLORATADINE Calcium Channel Type L, Benzothiazepine 73% 5.791uM 5.148uM View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit DESLORATADINE Calcium Channel Type L, Benzothiazepine 73% 5.791uM 5.148uM View
calcium channel, voltage-dependent, beta 1 subunit DESLORATADINE Calcium Channel Type L, Benzothiazepine 73% 5.791uM 5.148uM View
calcium channel, voltage-dependent, L type, alpha 1E subunit DESLORATADINE Calcium Channel Type L, Benzothiazepine 73% 5.791uM 5.148uM View
calcium channel, voltage-dependent, N type, alpha 1B subunit DESLORATADINE Calcium Channel Type L, Benzothiazepine 73% 5.791uM 5.148uM View
calcium channel, voltage-dependent, alpha2/delta subunit 1 DESLORATADINE Calcium Channel Type L, Benzothiazepine 73% 5.791uM 5.148uM View
Cytochrome P450, subfamily IIC (mephenytoin 4-hydroxylase) RESVERATROL CYP450-2C9 Inhibition 73% 7uM NoneNone View
cytochrome P450, family 2, subfamily C, polypeptide 9 RESVERATROL CYP450-2C9 Inhibition 73% 7uM NoneNone View
adrenergic receptor, beta 3 ALPHA-ERGOCRYPTINE Adrenergic beta3 73% 2.496uM 1.872uM View
5-hydroxytryptamine (serotonin) receptor 5B BERBERINE CHLORIDE Serotonin 5-HT4 73% 2.222uM .37uM View
5-hydroxytryptamine (serotonin) receptor 4 BERBERINE CHLORIDE Serotonin 5-HT4 73% 2.222uM .37uM View
calcium channel, voltage-dependent, gamma subunit 8 DIPHENIDOL Calcium Channel Type L, Phenylalkylamine 73% 4.501uM 4.376uM View
calcium channel, voltage-dependent, gamma subunit 7 DIPHENIDOL Calcium Channel Type L, Phenylalkylamine 73% 4.501uM 4.376uM View
calcium channel, voltage-dependent, gamma subunit 6 DIPHENIDOL Calcium Channel Type L, Phenylalkylamine 73% 4.501uM 4.376uM View
calcium channel, voltage-dependent, gamma subunit 5 DIPHENIDOL Calcium Channel Type L, Phenylalkylamine 73% 4.501uM 4.376uM View
calcium channel, voltage-dependent, gamma subunit 4 DIPHENIDOL Calcium Channel Type L, Phenylalkylamine 73% 4.501uM 4.376uM View
calcium channel, voltage-dependent, gamma subunit 3 DIPHENIDOL Calcium Channel Type L, Phenylalkylamine 73% 4.501uM 4.376uM View
calcium channel, voltage-dependent, gamma subunit 2 DIPHENIDOL Calcium Channel Type L, Phenylalkylamine 73% 4.501uM 4.376uM View
calcium channel, voltage-dependent, gamma subunit 1 DIPHENIDOL Calcium Channel Type L, Phenylalkylamine 73% 4.501uM 4.376uM View
calcium channel, voltage-dependent, beta 4 subunit DIPHENIDOL Calcium Channel Type L, Phenylalkylamine 73% 4.501uM 4.376uM View
calcium channel, voltage-dependent, beta 3 subunit DIPHENIDOL Calcium Channel Type L, Phenylalkylamine 73% 4.501uM 4.376uM View
calcium channel, voltage-dependent, beta 2 subunit DIPHENIDOL Calcium Channel Type L, Phenylalkylamine 73% 4.501uM 4.376uM View
ATPase, Na+/K+ transporting, alpha 3 polypeptide SODIUM ORTHOVANADATE ATPase, Na+/K+ 72% 1.853uM NoneNone View
ATPase, Na+/K+ transporting, alpha 2 polypeptide SODIUM ORTHOVANADATE ATPase, Na+/K+ 72% 1.853uM NoneNone View
ATPase, Na+/K+ transporting, alpha 1 polypeptide SODIUM ORTHOVANADATE ATPase, Na+/K+ 72% 1.853uM NoneNone View
ATPase, Na+/K+ transporting, beta 1 polypeptide SODIUM ORTHOVANADATE ATPase, Na+/K+ 72% 1.853uM NoneNone View
ATPase, Na+/K+ transporting, beta 3 polypeptide SODIUM ORTHOVANADATE ATPase, Na+/K+ 72% 1.853uM NoneNone View
ATPase, Na+/K+ transporting, beta 2 polypeptide SODIUM ORTHOVANADATE ATPase, Na+/K+ 72% 1.853uM NoneNone View
ATPase, (Na+)/K+ transporting, beta 4 polypeptide SODIUM ORTHOVANADATE ATPase, Na+/K+ 72% 1.853uM NoneNone View
matrix metallopeptidase 9 BUSULFAN Protease, Matrix Metalloprotease-9 (MMP-9) 72% 5.215uM NoneNone View
matrix metalloproteinase 9 (gelatinase B, 92kDa gelatinase, 92kDa type IV collagenase) BUSULFAN Protease, Matrix Metalloprotease-9 (MMP-9) 72% 5.215uM NoneNone View
solute carrier family 6 (neurotransmitter transporter, noradrenalin), member 2 PROMETHAZINE Adrenergic, Norepinephrine Transporter 72% 4.238uM 4.203uM View
5-hydroxytryptamine (serotonin) receptor 2B CETYLPYRIDINIUM BROMIDE Serotonin 5-HT2B 72% 5.69uM 3.621uM View
5-hydroxytryptamine (serotonin) receptor 2B PHENTOLAMINE Serotonin 5-HT2B 72% 3.807uM 2.422uM View
A3 adenosine receptor NISOLDIPINE Adenosine A3 72% 7.12uM 4.024uM View
adrenergic receptor, beta 3 ASTEMIZOLE Adrenergic beta3 72% 8.06uM 6.045uM View
lymphocyte protein tyrosine kinase (mapped) ASTEMIZOLE Protein Tyrosine Kinase, Lck 72% 19.92uM NoneNone View
5-hydroxytryptamine receptor 6 CLOMIPHENE Serotonin 5-HT6 72% 1.522uM .707uM View
adrenergic receptor, alpha 1b CLOMIPHENE Adrenergic alpha1B 72% 4.569uM 2.529uM View
cholinergic receptor, muscarinic 4 DROPERIDOL Muscarinic M4 72% 3.849uM .537uM View
5-hydroxytryptamine (serotonin) receptor 2B DROPERIDOL Serotonin 5-HT2B 72% 1.342uM .854uM View
sodium channel, voltage-gated, type I, beta DIHYDROERGOTAMINE Sodium Channel, Site 2 72% 5.058uM 4.614uM View
sodium channel, voltage-gated, type 10, alpha polypeptide DIHYDROERGOTAMINE Sodium Channel, Site 2 72% 5.058uM 4.614uM View
sodium channel, voltage-gated, type IV, alpha polypeptide DIHYDROERGOTAMINE Sodium Channel, Site 2 72% 5.058uM 4.614uM View
sodium channel, voltage-gated, type V, alpha polypeptide DIHYDROERGOTAMINE Sodium Channel, Site 2 72% 5.058uM 4.614uM View
sodium channel, voltage-gated, type II, beta DIHYDROERGOTAMINE Sodium Channel, Site 2 72% 5.058uM 4.614uM View
sodium channel, nonvoltage-gated 1 alpha DIHYDROERGOTAMINE Sodium Channel, Site 2 72% 5.058uM 4.614uM View
sodium channel, nonvoltage-gated 1 gamma DIHYDROERGOTAMINE Sodium Channel, Site 2 72% 5.058uM 4.614uM View
sodium channel, nonvoltage-gated 1 beta DIHYDROERGOTAMINE Sodium Channel, Site 2 72% 5.058uM 4.614uM View
sodium channel, voltage-gated, type 2, alpha 1 polypeptide DIHYDROERGOTAMINE Sodium Channel, Site 2 72% 5.058uM 4.614uM View
sodium channel, voltage-gated, type XI, alpha DIHYDROERGOTAMINE Sodium Channel, Site 2 72% 5.058uM 4.614uM View
sodium channel, nonvoltage-gated 1, gamma DIHYDROERGOTAMINE Sodium Channel, Site 2 72% 5.058uM 4.614uM View
sodium channel, nonvoltage-gated 1, delta DIHYDROERGOTAMINE Sodium Channel, Site 2 72% 5.058uM 4.614uM View
sodium channel, nonvoltage-gated 1, beta (Liddle syndrome) DIHYDROERGOTAMINE Sodium Channel, Site 2 72% 5.058uM 4.614uM View
sodium channel, nonvoltage-gated 1 alpha DIHYDROERGOTAMINE Sodium Channel, Site 2 72% 5.058uM 4.614uM View
sodium channel, voltage-gated, type X, alpha DIHYDROERGOTAMINE Sodium Channel, Site 2 72% 5.058uM 4.614uM View
sodium channel, voltage-gated, type IX, alpha DIHYDROERGOTAMINE Sodium Channel, Site 2 72% 5.058uM 4.614uM View
sodium channel, voltage gated, type VIII, alpha DIHYDROERGOTAMINE Sodium Channel, Site 2 72% 5.058uM 4.614uM View
sodium channel, voltage-gated, type VII, alpha DIHYDROERGOTAMINE Sodium Channel, Site 2 72% 5.058uM 4.614uM View
adrenergic receptor, alpha 2a YOHIMBINE Imidazoline I2, Central 72% .157uM .105uM View
adrenergic receptor, alpha 2c (Non-specific probe) YOHIMBINE Imidazoline I2, Central 72% .157uM .105uM View
adrenergic receptor, beta 1 TAMOXIFEN Adrenergic beta1 72% 17.289uM 9.984uM View
adrenergic, beta-1-, receptor TAMOXIFEN Adrenergic beta1 72% 17.289uM 9.984uM View
solute carrier family 6 (neurotransmitter transporter, dopamine), member 3 CLOMIPRAMINE Dopamine Transporter 72% 2.746uM 2.182uM View
adrenergic receptor, alpha 2b METHAPYRILENE Adrenergic alpha2B 72% 3.318uM 1.515uM View
5-hydroxytryptamine (serotonin) receptor 2A TETRACAINE Serotonin 5-HT2A 72% 3.415uM .976uM View
cholinergic receptor, muscarinic 3 FLUOXETINE Muscarinic M3 72% 3.595uM .762uM View
Sigma-2 Receptor FLUPHENAZINE Sigma2 72% .158uM .097uM View
Cytochrom P450-1A2 monooxygenase SULINDAC SULFIDE CYP450-1A2 Inhibition 72% 2uM NoneNone View
Cytochrom P450-1A2 monooxygenase NABUMETONE CYP450-1A2 Inhibition 72% 5uM NoneNone View
opioid receptor, sigma 1 R-(+)-PROPRANOLOL Sigma1 72% 3.974uM 1.67uM View
solute carrier family 6 (neurotransmitter transporter, serotonin), member 4 HALOPERIDOL Serotonin Transporter 72% 3.386uM 1.799uM View
5-hydroxytryptamine (serotonin) receptor 1A R-(+)-PROPRANOLOL Serotonin 5-HT1A 72% 4.88uM 2.789uM View
dopamine receptor D1A LYSERGOL Dopamine D1 72% 2.908uM 1.454uM View
adrenergic receptor, alpha 1d (Non-specific probe) LYSERGOL Adrenergic alpha1D 72% 1.128uM .554uM View
adrenergic receptor, alpha 2a METHYSERGIDE Imidazoline I2, Central 72% 2.519uM 1.68uM View
adrenergic receptor, alpha 2c (Non-specific probe) METHYSERGIDE Imidazoline I2, Central 72% 2.519uM 1.68uM View
potassium voltage-gated channel, subfamily H (eag-related), member 1 CHLORPROMAZINE Potassium Channel HERG 72% 5.8275uM 4.7743uM View
potassium voltage-gated channel, subfamily H, member 8 VERAPAMIL Potassium Channel HERG 72% NoneNone NoneNone View
potassium voltage-gated channel, subfamily H (eag-related), member 6 VERAPAMIL Potassium Channel HERG 72% NoneNone NoneNone View
potassium voltage-gated channel, subfamily H (eag-related), member 7 VERAPAMIL Potassium Channel HERG 72% NoneNone NoneNone View
potassium voltage-gated channel, subfamily H (eag-related), member 2 VERAPAMIL Potassium Channel HERG 72% NoneNone NoneNone View
potassium voltage-gated channel, subfamily H (eag-related), member 5 VERAPAMIL Potassium Channel HERG 72% NoneNone NoneNone View
potassium voltage-gated channel, subfamily H (eag-related), member 3 VERAPAMIL Potassium Channel HERG 72% NoneNone NoneNone View
potassium voltage-gated channel, subfamily H (eag-related), member 4 VERAPAMIL Potassium Channel HERG 72% NoneNone NoneNone View
potassium voltage-gated channel, subfamily H (eag-related), member 1 VERAPAMIL Potassium Channel HERG 72% NoneNone NoneNone View
potassium voltage-gated channel, subfamily H (eag-related), member 1 VERAPAMIL Potassium Channel HERG 72% NoneNone NoneNone View
androgen receptor ZINC CHLORIDE Testosterone 72% 6.5086uM 4.3391uM View
5-hydroxytryptamine (serotonin) receptor 2B HEXACHLOROPHENE Serotonin 5-HT2B 72% 5.6947uM 3.6239uM View
mitogen activated protein kinase 14 NAFENOPIN Protein Serine/Threonine Kinase, p38alpha 72% 3.7405uM NoneNone View
mitogen-activated protein kinase 14 NAFENOPIN Protein Serine/Threonine Kinase, p38alpha 72% 3.7405uM NoneNone View
cholinergic receptor, muscarinic 1 SULOCTIDIL Muscarinic M1 72% 4.505uM 1.085uM View
Cytochrom P450-1A2 monooxygenase THIORIDAZINE CYP450-1A2 Inhibition 72% 9.3323uM NoneNone View
Sigma-2 Receptor TOLPERISONE Sigma2 72% 3.357uM 2.066uM View
5-hydroxytryptamine (serotonin) receptor 1A FLUNARIZINE Serotonin 5-HT1A 72% 4.281uM 2.446uM View
5-hydroxytryptamine (serotonin) receptor 1A LEVOBUNOLOL Serotonin 5-HT1A 72% 2.901uM 1.658uM View
calcium channel, voltage-dependent, gamma subunit 8 CYCLIZINE Calcium Channel Type L, Phenylalkylamine 72% 4.644uM 4.515uM View
calcium channel, voltage-dependent, gamma subunit 7 CYCLIZINE Calcium Channel Type L, Phenylalkylamine 72% 4.644uM 4.515uM View
calcium channel, voltage-dependent, gamma subunit 6 CYCLIZINE Calcium Channel Type L, Phenylalkylamine 72% 4.644uM 4.515uM View
calcium channel, voltage-dependent, gamma subunit 5 CYCLIZINE Calcium Channel Type L, Phenylalkylamine 72% 4.644uM 4.515uM View
calcium channel, voltage-dependent, gamma subunit 4 CYCLIZINE Calcium Channel Type L, Phenylalkylamine 72% 4.644uM 4.515uM View
calcium channel, voltage-dependent, gamma subunit 3 CYCLIZINE Calcium Channel Type L, Phenylalkylamine 72% 4.644uM 4.515uM View
calcium channel, voltage-dependent, gamma subunit 2 CYCLIZINE Calcium Channel Type L, Phenylalkylamine 72% 4.644uM 4.515uM View
calcium channel, voltage-dependent, gamma subunit 1 CYCLIZINE Calcium Channel Type L, Phenylalkylamine 72% 4.644uM 4.515uM View
calcium channel, voltage-dependent, beta 4 subunit CYCLIZINE Calcium Channel Type L, Phenylalkylamine 72% 4.644uM 4.515uM View
calcium channel, voltage-dependent, beta 3 subunit CYCLIZINE Calcium Channel Type L, Phenylalkylamine 72% 4.644uM 4.515uM View
calcium channel, voltage-dependent, beta 2 subunit CYCLIZINE Calcium Channel Type L, Phenylalkylamine 72% 4.644uM 4.515uM View
calcium channel, voltage-dependent, L type, alpha 1S subunit CYCLIZINE Calcium Channel Type L, Phenylalkylamine 72% 4.644uM 4.515uM View
calcium channel, voltage-dependent, alpha 1F subunit CYCLIZINE Calcium Channel Type L, Phenylalkylamine 72% 4.644uM 4.515uM View
calcium channel, voltage-dependent, L type, alpha 1D subunit CYCLIZINE Calcium Channel Type L, Phenylalkylamine 72% 4.644uM 4.515uM View
calcium channel, voltage-dependent, L type, alpha 1C subunit CYCLIZINE Calcium Channel Type L, Phenylalkylamine 72% 4.644uM 4.515uM View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit CYCLIZINE Calcium Channel Type L, Phenylalkylamine 72% 4.644uM 4.515uM View
calcium channel, voltage-dependent, beta 1 subunit CYCLIZINE Calcium Channel Type L, Phenylalkylamine 72% 4.644uM 4.515uM View
calcium channel, voltage-dependent, L type, alpha 1E subunit CYCLIZINE Calcium Channel Type L, Phenylalkylamine 72% 4.644uM 4.515uM View
calcium channel, voltage-dependent, N type, alpha 1B subunit CYCLIZINE Calcium Channel Type L, Phenylalkylamine 72% 4.644uM 4.515uM View
calcium channel, voltage-dependent, alpha2/delta subunit 1 CYCLIZINE Calcium Channel Type L, Phenylalkylamine 72% 4.644uM 4.515uM View
cytochrome P450, family 3, subfamily a, polypeptide 13 RWJ-68354 CYP450-3A4 Inhibition 72% 1uM NoneNone View
Cytochrom P450-2D6 monooxygenase TRIHEXYPHENIDYL CYP450-2D6 Inhibition 72% 2.4498uM NoneNone View
Cytochrom P450-2D6 monooxygenase NALOXONE CYP450-2D6 Inhibition 72% 2uM NoneNone View
Cytochrom P450-2C19 monooxygenase SPIRONOLACTONE CYP450-2C19 Inhibition 72% 3uM NoneNone View
5-hydroxytryptamine (serotonin) receptor 2C BITHIONOL Serotonin 5-HT2C 72% 8.78uM 4.599uM View
dopamine receptor D3 DIPHENIDOL Dopamine D3 72% 2.311uM .785uM View
dopamine receptor D3 DOBUTAMINE Dopamine D3 72% 4.985uM 1.693uM View
adrenergic receptor, alpha 2b CLOSANTEL Adrenergic alpha2C 72% 7.1uM 1uM View
adrenergic receptor, alpha 2c (Non-specific probe) CLOSANTEL Adrenergic alpha2C 72% 7.1uM 1uM View
solute carrier family 6 (neurotransmitter transporter, dopamine), member 3 CLOSANTEL Dopamine Transporter 72% 4.8uM 3.8uM View
opioid receptor, sigma 1 DOBUTAMINE Sigma1 72% 2.518uM 1.058uM View
lymphocyte protein tyrosine kinase (mapped) DOBUTAMINE Protein Tyrosine Kinase, Lck 72% 5.519uM NoneNone View
phosphodiesterase 4A, cAMP specific CELECOXIB Phosphodiesterase PDE4 68% 9.26uM NoneNone View
Sigma-2 Receptor AMITRIPTYLINE Sigma2 68% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 8 AMOXAPINE Calcium Channel Type L, Benzothiazepine 68% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 7 AMOXAPINE Calcium Channel Type L, Benzothiazepine 68% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 6 AMOXAPINE Calcium Channel Type L, Benzothiazepine 68% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 5 AMOXAPINE Calcium Channel Type L, Benzothiazepine 68% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 4 AMOXAPINE Calcium Channel Type L, Benzothiazepine 68% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 3 AMOXAPINE Calcium Channel Type L, Benzothiazepine 68% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 2 AMOXAPINE Calcium Channel Type L, Benzothiazepine 68% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 1 AMOXAPINE Calcium Channel Type L, Benzothiazepine 68% NoneNone NoneNone View
calcium channel, voltage-dependent, beta 4 subunit AMOXAPINE Calcium Channel Type L, Benzothiazepine 68% NoneNone NoneNone View
calcium channel, voltage-dependent, beta 3 subunit AMOXAPINE Calcium Channel Type L, Benzothiazepine 68% NoneNone NoneNone View
calcium channel, voltage-dependent, beta 2 subunit AMOXAPINE Calcium Channel Type L, Benzothiazepine 68% NoneNone NoneNone View
calcium channel, voltage-dependent, L type, alpha 1S subunit AMOXAPINE Calcium Channel Type L, Benzothiazepine 68% NoneNone NoneNone View
calcium channel, voltage-dependent, alpha 1F subunit AMOXAPINE Calcium Channel Type L, Benzothiazepine 68% NoneNone NoneNone View
calcium channel, voltage-dependent, L type, alpha 1D subunit AMOXAPINE Calcium Channel Type L, Benzothiazepine 68% NoneNone NoneNone View
calcium channel, voltage-dependent, L type, alpha 1C subunit AMOXAPINE Calcium Channel Type L, Benzothiazepine 68% NoneNone NoneNone View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit AMOXAPINE Calcium Channel Type L, Benzothiazepine 68% NoneNone NoneNone View
calcium channel, voltage-dependent, beta 1 subunit AMOXAPINE Calcium Channel Type L, Benzothiazepine 68% NoneNone NoneNone View
calcium channel, voltage-dependent, L type, alpha 1E subunit AMOXAPINE Calcium Channel Type L, Benzothiazepine 68% NoneNone NoneNone View
calcium channel, voltage-dependent, N type, alpha 1B subunit AMOXAPINE Calcium Channel Type L, Benzothiazepine 68% NoneNone NoneNone View
calcium channel, voltage-dependent, alpha2/delta subunit 1 AMOXAPINE Calcium Channel Type L, Benzothiazepine 68% NoneNone NoneNone View
adrenergic receptor, alpha 2a AMIODARONE Imidazoline I2, Central 68% 7.826uM 5.217uM View
adrenergic receptor, alpha 2c (Non-specific probe) AMIODARONE Imidazoline I2, Central 68% 7.826uM 5.217uM View
Cytochrom P450-1A2 monooxygenase CHLORPROMAZINE CYP450-1A2 Inhibition 68% NoneNone NoneNone View
Cytochrome P450, subfamily IIC (mephenytoin 4-hydroxylase) 1-BENZYLIMIDAZOLE CYP450-2C9 Inhibition 68% NoneNone NoneNone View
cytochrome P450, family 2, subfamily C, polypeptide 9 1-BENZYLIMIDAZOLE CYP450-2C9 Inhibition 68% NoneNone NoneNone View
A3 adenosine receptor NIFEDIPINE Adenosine A3 68% 7.214uM 4.078uM View
mu-opioid receptor MOR CISAPRIDE Opiate mu 68% NoneNone NoneNone View
cytochrome P450, family 3, subfamily a, polypeptide 13 PAPAVERINE CYP450-3A4 Inhibition 68% NoneNone NoneNone View
Sigma-2 Receptor PERHEXILINE Sigma2 68% NoneNone NoneNone View
cholinergic receptor, muscarinic 3 HEXACHLOROPHENE Muscarinic M3 68% NoneNone NoneNone View
cytochrome P450, family 3, subfamily a, polypeptide 13 HEXACHLOROPHENE CYP450-3A4 Inhibition 68% NoneNone NoneNone View
Cytochrom P450-2C19 monooxygenase PROPAFENONE CYP450-2C19 Inhibition 68% NoneNone NoneNone View
matrix metallopeptidase 9 MESNA Protease, Matrix Metalloprotease-9 (MMP-9) 68% NoneNone NoneNone View
matrix metalloproteinase 9 (gelatinase B, 92kDa gelatinase, 92kDa type IV collagenase) MESNA Protease, Matrix Metalloprotease-9 (MMP-9) 68% NoneNone NoneNone View
dopamine receptor D4 1,3-DIPHENYLGUANIDINE Dopamine D4.2 68% NoneNone NoneNone View
dopamine receptor 2 DESLORATADINE Dopamine D2L 68% NoneNone NoneNone View
Cytochrom P450-2D6 monooxygenase MONOBENZONE CYP450-2D6 Inhibition 68% NoneNone NoneNone View
Cytochrom P450-2D6 monooxygenase NALOXONAZINE CYP450-2D6 Inhibition 68% NoneNone NoneNone View
arachidonate 15-lipoxygenase, second type RIFAPENTINE Lipoxygenase 15-LO 68% NoneNone NoneNone View
arachidonate 15-lipoxygenase RIFAPENTINE Lipoxygenase 15-LO 68% NoneNone NoneNone View
arachidonate 15-lipoxygenase RIFAPENTINE Lipoxygenase 15-LO 68% NoneNone NoneNone View