Gene Activity List


Gene Activity List

Gene Compound Assay Inh Ic50 Ki View
adrenergic receptor, alpha 2a LEAD(IV) ACETATE Adrenergic alpha2A 68% NoneNone NoneNone View
sodium channel, nonvoltage-gated 1, beta (Liddle syndrome) MEDROXYPROGESTERONE ACETATE Sodium Channel, Site 2 68% 14.954uM 13.407uM View
sodium channel, nonvoltage-gated 1 alpha MEDROXYPROGESTERONE ACETATE Sodium Channel, Site 2 68% 14.954uM 13.407uM View
sodium channel, voltage-gated, type X, alpha MEDROXYPROGESTERONE ACETATE Sodium Channel, Site 2 68% 14.954uM 13.407uM View
sodium channel, voltage-gated, type IX, alpha MEDROXYPROGESTERONE ACETATE Sodium Channel, Site 2 68% 14.954uM 13.407uM View
sodium channel, voltage gated, type VIII, alpha MEDROXYPROGESTERONE ACETATE Sodium Channel, Site 2 68% 14.954uM 13.407uM View
sodium channel, voltage-gated, type VII, alpha MEDROXYPROGESTERONE ACETATE Sodium Channel, Site 2 68% 14.954uM 13.407uM View
sodium channel, voltage-gated, type V, alpha (long QT syndrome 3) MEDROXYPROGESTERONE ACETATE Sodium Channel, Site 2 68% 14.954uM 13.407uM View
sodium channel, voltage-gated, type IV, beta MEDROXYPROGESTERONE ACETATE Sodium Channel, Site 2 68% 14.954uM 13.407uM View
sodium channel, voltage-gated, type IV, alpha MEDROXYPROGESTERONE ACETATE Sodium Channel, Site 2 68% 14.954uM 13.407uM View
histamine receptor H 2 QUINACRINE Histamine H2 72% 3.535uM 3.476uM View
adrenergic receptor, alpha 1d (Non-specific probe) IMIQUIMOD Adrenergic alpha1D 72% 2.621uM 1.288uM View
calcium channel, voltage-dependent, beta 4 subunit BOPINDOLOL Calcium Channel Type L, Benzothiazepine 72% 2.805uM 2.493uM View
calcium channel, voltage-dependent, beta 3 subunit BOPINDOLOL Calcium Channel Type L, Benzothiazepine 72% 2.805uM 2.493uM View
calcium channel, voltage-dependent, beta 2 subunit BOPINDOLOL Calcium Channel Type L, Benzothiazepine 72% 2.805uM 2.493uM View
calcium channel, voltage-dependent, L type, alpha 1S subunit BOPINDOLOL Calcium Channel Type L, Benzothiazepine 72% 2.805uM 2.493uM View
calcium channel, voltage-dependent, alpha 1F subunit BOPINDOLOL Calcium Channel Type L, Benzothiazepine 72% 2.805uM 2.493uM View
calcium channel, voltage-dependent, L type, alpha 1D subunit BOPINDOLOL Calcium Channel Type L, Benzothiazepine 72% 2.805uM 2.493uM View
calcium channel, voltage-dependent, L type, alpha 1C subunit BOPINDOLOL Calcium Channel Type L, Benzothiazepine 72% 2.805uM 2.493uM View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit BOPINDOLOL Calcium Channel Type L, Benzothiazepine 72% 2.805uM 2.493uM View
calcium channel, voltage-dependent, beta 1 subunit BOPINDOLOL Calcium Channel Type L, Benzothiazepine 72% 2.805uM 2.493uM View
calcium channel, voltage-dependent, L type, alpha 1E subunit BOPINDOLOL Calcium Channel Type L, Benzothiazepine 72% 2.805uM 2.493uM View
calcium channel, voltage-dependent, N type, alpha 1B subunit BOPINDOLOL Calcium Channel Type L, Benzothiazepine 72% 2.805uM 2.493uM View
calcium channel, voltage-dependent, alpha2/delta subunit 1 BOPINDOLOL Calcium Channel Type L, Benzothiazepine 72% 2.805uM 2.493uM View
calcium channel, voltage-dependent, gamma subunit 8 BOPINDOLOL Calcium Channel Type L, Benzothiazepine 72% 2.805uM 2.493uM View
calcium channel, voltage-dependent, gamma subunit 7 BOPINDOLOL Calcium Channel Type L, Benzothiazepine 72% 2.805uM 2.493uM View
calcium channel, voltage-dependent, gamma subunit 6 BOPINDOLOL Calcium Channel Type L, Benzothiazepine 72% 2.805uM 2.493uM View
calcium channel, voltage-dependent, gamma subunit 5 BOPINDOLOL Calcium Channel Type L, Benzothiazepine 72% 2.805uM 2.493uM View
calcium channel, voltage-dependent, gamma subunit 4 BOPINDOLOL Calcium Channel Type L, Benzothiazepine 72% 2.805uM 2.493uM View
calcium channel, voltage-dependent, gamma subunit 3 BOPINDOLOL Calcium Channel Type L, Benzothiazepine 72% 2.805uM 2.493uM View
calcium channel, voltage-dependent, gamma subunit 2 BOPINDOLOL Calcium Channel Type L, Benzothiazepine 72% 2.805uM 2.493uM View
calcium channel, voltage-dependent, gamma subunit 1 BOPINDOLOL Calcium Channel Type L, Benzothiazepine 72% 2.805uM 2.493uM View
Cytochrom P450-2C19 monooxygenase NIMODIPINE CYP450-2C19 Inhibition 72% 4uM NoneNone View
dopamine receptor D1A OXICONAZOLE Dopamine D1 72% 4.1361uM 2.068uM View
opioid receptor, delta 1 OXICONAZOLE Opiate delta 72% 5.3081uM 1.8712uM View
5-hydroxytryptamine (serotonin) receptor 2B OXYMETAZOLINE Serotonin 5-HT2B 72% 3.056uM 1.945uM View
ATPase, Na+/K+ transporting, alpha 4 polypeptide SODIUM ORTHOVANADATE ATPase, Na+/K+ 72% 1.853uM NoneNone View
5-hydroxytryptamine (serotonin) receptor 1A PROMAZINE Serotonin 5-HT1A 72% 5.172uM 2.955uM View
solute carrier family 6 (neurotransmitter transporter, noradrenalin), member 2 VX-745 Adrenergic, Norepinephrine Transporter 72% 20.404uM 20.236uM View
opioid receptor, sigma 1 PAROXETINE Sigma1 72% 5.366uM 2.255uM View
tachykinin receptor 2 METERGOLINE Tachykinin NK2 72% 4.071uM 1.357uM View
adrenergic receptor, alpha 1b PERGOLIDE Adrenergic alpha1B 72% 2.622uM 1.452uM View
adrenergic receptor, alpha 2a PRAZOSIN Adrenergic alpha2A 72% 2.638uM .989uM View
adrenergic receptor, alpha 2a METOCLOPRAMIDE Adrenergic alpha2A 72% 2.721uM 1.02uM View
melanocortin 5 receptor ECONAZOLE Melanocortin MC5 72% 39.538uM 37.089uM View
Protein-tyrosine kinase, Fyn EPIRUBICIN Protein Tyrosine Kinase, Fyn 72% 5.181uM NoneNone View
5-hydroxytryptamine (serotonin) receptor 1B KETOCONAZOLE Serotonin 5-HT1B 72% 13.539uM 6.154uM View
adrenergic receptor, alpha 1b DEXCHLORPHENIRAMINE Adrenergic alpha1B 72% 15.56uM 8.613uM View
Sigma-2 Receptor LEVAMISOLE Sigma2 72% 4.392uM 2.703uM View
phosphodiesterase 5A, cGMP-specific LY-294002 Phosphodiesterase PDE5 72% 9.614uM NoneNone View
phosphodiesterase 5A, cGMP-specific LY-294002 Phosphodiesterase PDE5 72% 9.614uM NoneNone View
opioid receptor, kappa 1 DANAZOL Opiate kappa 72% 15.518uM 6.207uM View
A3 adenosine receptor DANAZOL Adenosine A3 72% 11.16uM 6.309uM View
solute carrier family 6 (neurotransmitter transporter, serotonin), member 4 ESTRONE Serotonin Transporter 72% 5.301uM 2.816uM View
androgen receptor FLUTAMIDE Testosterone 72% 13.39uM 8.927uM View
5-hydroxytryptamine (serotonin) receptor 2B BETA-ESTRADIOL 3-BENZOATE Serotonin 5-HT2B 72% 11.565uM 7.359uM View
melanocortin 5 receptor CHLORPROMAZINE Melanocortin MC5 72% 7.617uM 7.145uM View
chemokine (C-C motif) receptor 2 AMIODARONE Chemokine CCR2B 72% 11.086uM 4.285uM View
calcium channel, voltage-dependent, gamma subunit 8 LOVASTATIN Calcium Channel Type L, Phenylalkylamine 72% 6.318uM 6.142uM View
calcium channel, voltage-dependent, gamma subunit 7 LOVASTATIN Calcium Channel Type L, Phenylalkylamine 72% 6.318uM 6.142uM View
calcium channel, voltage-dependent, gamma subunit 6 LOVASTATIN Calcium Channel Type L, Phenylalkylamine 72% 6.318uM 6.142uM View
calcium channel, voltage-dependent, gamma subunit 5 LOVASTATIN Calcium Channel Type L, Phenylalkylamine 72% 6.318uM 6.142uM View
calcium channel, voltage-dependent, gamma subunit 6 L-744832 Calcium Channel Type L, Dihydropyridine 70% 4.501uM 2.893uM View
calcium channel, voltage-dependent, gamma subunit 5 L-744832 Calcium Channel Type L, Dihydropyridine 70% 4.501uM 2.893uM View
calcium channel, voltage-dependent, gamma subunit 4 L-744832 Calcium Channel Type L, Dihydropyridine 70% 4.501uM 2.893uM View
calcium channel, voltage-dependent, gamma subunit 3 L-744832 Calcium Channel Type L, Dihydropyridine 70% 4.501uM 2.893uM View
adrenergic receptor, alpha 2b QUINACRINE Adrenergic alpha2C 70% 3.857uM .56uM View
adrenergic receptor, alpha 2c (Non-specific probe) QUINACRINE Adrenergic alpha2C 70% 3.857uM .56uM View
calcium channel, voltage-dependent, gamma subunit 8 QUINACRINE Calcium Channel Type L, Benzothiazepine 70% 1.076uM .956uM View
calcium channel, voltage-dependent, gamma subunit 7 QUINACRINE Calcium Channel Type L, Benzothiazepine 70% 1.076uM .956uM View
calcium channel, voltage-dependent, gamma subunit 6 QUINACRINE Calcium Channel Type L, Benzothiazepine 70% 1.076uM .956uM View
calcium channel, voltage-dependent, gamma subunit 5 QUINACRINE Calcium Channel Type L, Benzothiazepine 70% 1.076uM .956uM View
calcium channel, voltage-dependent, gamma subunit 4 QUINACRINE Calcium Channel Type L, Benzothiazepine 70% 1.076uM .956uM View
calcium channel, voltage-dependent, gamma subunit 3 QUINACRINE Calcium Channel Type L, Benzothiazepine 70% 1.076uM .956uM View
calcium channel, voltage-dependent, gamma subunit 2 QUINACRINE Calcium Channel Type L, Benzothiazepine 70% 1.076uM .956uM View
calcium channel, voltage-dependent, gamma subunit 1 QUINACRINE Calcium Channel Type L, Benzothiazepine 70% 1.076uM .956uM View
calcium channel, voltage-dependent, beta 4 subunit QUINACRINE Calcium Channel Type L, Benzothiazepine 70% 1.076uM .956uM View
adrenergic receptor, alpha 2a DIMENHYDRINATE Adrenergic alpha2A 70% 4.313uM 1.617uM View
5-hydroxytryptamine (serotonin) receptor 1B PIPAMAZINE Serotonin 5-HT1B 70% 3.007uM 1.367uM View
5-hydroxytryptamine (serotonin) receptor 5B EPIRUBICIN Serotonin 5-HT4 70% 7.935uM 1.323uM View
5-hydroxytryptamine (serotonin) receptor 4 EPIRUBICIN Serotonin 5-HT4 70% 7.935uM 1.323uM View
amiloride-sensitive cation channel 5, intestinal KETOCONAZOLE Sodium Channel, Site 2 70% 23.911uM 21.438uM View
sodium channel, voltage-gated, type III, beta KETOCONAZOLE Sodium Channel, Site 2 70% 23.911uM 21.438uM View
sodium channel, voltage-gated, type VIII, alpha polypeptide KETOCONAZOLE Sodium Channel, Site 2 70% 23.911uM 21.438uM View
sodium channel, voltage-gated, type XI, alpha KETOCONAZOLE Sodium Channel, Site 2 70% 23.911uM 21.438uM View
sodium channel, voltage-gated, type I, beta KETOCONAZOLE Sodium Channel, Site 2 70% 23.911uM 21.438uM View
sodium channel, voltage-gated, type 10, alpha polypeptide KETOCONAZOLE Sodium Channel, Site 2 70% 23.911uM 21.438uM View
sodium channel, voltage-gated, type IV, alpha polypeptide KETOCONAZOLE Sodium Channel, Site 2 70% 23.911uM 21.438uM View
sodium channel, voltage-gated, type V, alpha polypeptide KETOCONAZOLE Sodium Channel, Site 2 70% 23.911uM 21.438uM View
sodium channel, voltage-gated, type II, beta KETOCONAZOLE Sodium Channel, Site 2 70% 23.911uM 21.438uM View
sodium channel, nonvoltage-gated 1 alpha KETOCONAZOLE Sodium Channel, Site 2 70% 23.911uM 21.438uM View
sodium channel, nonvoltage-gated 1 gamma KETOCONAZOLE Sodium Channel, Site 2 70% 23.911uM 21.438uM View
sodium channel, nonvoltage-gated 1 beta KETOCONAZOLE Sodium Channel, Site 2 70% 23.911uM 21.438uM View
sodium channel, voltage-gated, type 2, alpha 1 polypeptide KETOCONAZOLE Sodium Channel, Site 2 70% 23.911uM 21.438uM View
sodium channel, voltage-gated, type XI, alpha KETOCONAZOLE Sodium Channel, Site 2 70% 23.911uM 21.438uM View
sodium channel, nonvoltage-gated 1, gamma KETOCONAZOLE Sodium Channel, Site 2 70% 23.911uM 21.438uM View
sodium channel, nonvoltage-gated 1, delta KETOCONAZOLE Sodium Channel, Site 2 70% 23.911uM 21.438uM View
sodium channel, nonvoltage-gated 1, beta (Liddle syndrome) KETOCONAZOLE Sodium Channel, Site 2 70% 23.911uM 21.438uM View
sodium channel, nonvoltage-gated 1 alpha KETOCONAZOLE Sodium Channel, Site 2 70% 23.911uM 21.438uM View
sodium channel, voltage-gated, type X, alpha KETOCONAZOLE Sodium Channel, Site 2 70% 23.911uM 21.438uM View
sodium channel, voltage-gated, type IX, alpha KETOCONAZOLE Sodium Channel, Site 2 70% 23.911uM 21.438uM View
sodium channel, voltage gated, type VIII, alpha KETOCONAZOLE Sodium Channel, Site 2 70% 23.911uM 21.438uM View
sodium channel, voltage-gated, type VII, alpha KETOCONAZOLE Sodium Channel, Site 2 70% 23.911uM 21.438uM View
sodium channel, voltage-gated, type V, alpha (long QT syndrome 3) KETOCONAZOLE Sodium Channel, Site 2 70% 23.911uM 21.438uM View
sodium channel, voltage-gated, type IV, beta KETOCONAZOLE Sodium Channel, Site 2 70% 23.911uM 21.438uM View
sodium channel, voltage-gated, type IV, alpha KETOCONAZOLE Sodium Channel, Site 2 70% 23.911uM 21.438uM View
sodium channel, voltage-gated, type III, alpha KETOCONAZOLE Sodium Channel, Site 2 70% 23.911uM 21.438uM View
sodium channel, voltage-gated, type II, beta KETOCONAZOLE Sodium Channel, Site 2 70% 23.911uM 21.438uM View
sodium channel, voltage-gated, type II, alpha 2 KETOCONAZOLE Sodium Channel, Site 2 70% 23.911uM 21.438uM View
sodium channel, voltage-gated, type I, beta KETOCONAZOLE Sodium Channel, Site 2 70% 23.911uM 21.438uM View
sodium channel, voltage-gated, type I, alpha KETOCONAZOLE Sodium Channel, Site 2 70% 23.911uM 21.438uM View
sodium channel, voltage-gated, type IV, beta KETOCONAZOLE Sodium Channel, Site 2 70% 23.911uM 21.438uM View
sodium channel, voltage-gated, type III, alpha MEDROXYPROGESTERONE ACETATE Sodium Channel, Site 2 68% 14.954uM 13.407uM View
sodium channel, voltage-gated, type II, beta MEDROXYPROGESTERONE ACETATE Sodium Channel, Site 2 68% 14.954uM 13.407uM View
sodium channel, voltage-gated, type II, alpha 2 MEDROXYPROGESTERONE ACETATE Sodium Channel, Site 2 68% 14.954uM 13.407uM View
sodium channel, voltage-gated, type I, beta MEDROXYPROGESTERONE ACETATE Sodium Channel, Site 2 68% 14.954uM 13.407uM View
sodium channel, voltage-gated, type I, alpha MEDROXYPROGESTERONE ACETATE Sodium Channel, Site 2 68% 14.954uM 13.407uM View
sodium channel, voltage-gated, type IV, beta MEDROXYPROGESTERONE ACETATE Sodium Channel, Site 2 68% 14.954uM 13.407uM View
sodium channel associated protein 1 MEDROXYPROGESTERONE ACETATE Sodium Channel, Site 2 68% 14.954uM 13.407uM View
sodium channel associated protein 2 MEDROXYPROGESTERONE ACETATE Sodium Channel, Site 2 68% 14.954uM 13.407uM View
sodium channel, voltage-gated, type III, beta MEDROXYPROGESTERONE ACETATE Sodium Channel, Site 2 68% 14.954uM 13.407uM View
sodium channel, voltage-gated, type I, alpha MEDROXYPROGESTERONE ACETATE Sodium Channel, Site 2 68% 14.954uM 13.407uM View
sodium channel, voltage-gated, type IX, alpha MEDROXYPROGESTERONE ACETATE Sodium Channel, Site 2 68% 14.954uM 13.407uM View
sodium channel, voltage-gated, type VII, alpha MEDROXYPROGESTERONE ACETATE Sodium Channel, Site 2 68% 14.954uM 13.407uM View
amiloride-sensitive cation channel 5, intestinal MEDROXYPROGESTERONE ACETATE Sodium Channel, Site 2 68% 14.954uM 13.407uM View
sodium channel, voltage-gated, type III, beta MEDROXYPROGESTERONE ACETATE Sodium Channel, Site 2 68% 14.954uM 13.407uM View
sodium channel, voltage-gated, type VIII, alpha polypeptide MEDROXYPROGESTERONE ACETATE Sodium Channel, Site 2 68% 14.954uM 13.407uM View
sodium channel, voltage-gated, type XI, alpha MEDROXYPROGESTERONE ACETATE Sodium Channel, Site 2 68% 14.954uM 13.407uM View
sodium channel, voltage-gated, type I, beta MEDROXYPROGESTERONE ACETATE Sodium Channel, Site 2 68% 14.954uM 13.407uM View
sodium channel, voltage-gated, type 10, alpha polypeptide MEDROXYPROGESTERONE ACETATE Sodium Channel, Site 2 68% 14.954uM 13.407uM View
sodium channel, voltage-gated, type IV, alpha polypeptide MEDROXYPROGESTERONE ACETATE Sodium Channel, Site 2 68% 14.954uM 13.407uM View
sodium channel, voltage-gated, type V, alpha polypeptide MEDROXYPROGESTERONE ACETATE Sodium Channel, Site 2 68% 14.954uM 13.407uM View
sodium channel, voltage-gated, type II, beta MEDROXYPROGESTERONE ACETATE Sodium Channel, Site 2 68% 14.954uM 13.407uM View
sodium channel, nonvoltage-gated 1 alpha MEDROXYPROGESTERONE ACETATE Sodium Channel, Site 2 68% 14.954uM 13.407uM View
sodium channel, nonvoltage-gated 1 gamma MEDROXYPROGESTERONE ACETATE Sodium Channel, Site 2 68% 14.954uM 13.407uM View
sodium channel, nonvoltage-gated 1 beta MEDROXYPROGESTERONE ACETATE Sodium Channel, Site 2 68% 14.954uM 13.407uM View
sodium channel, voltage-gated, type 2, alpha 1 polypeptide MEDROXYPROGESTERONE ACETATE Sodium Channel, Site 2 68% 14.954uM 13.407uM View
sodium channel, voltage-gated, type XI, alpha MEDROXYPROGESTERONE ACETATE Sodium Channel, Site 2 68% 14.954uM 13.407uM View
sodium channel, nonvoltage-gated 1, gamma MEDROXYPROGESTERONE ACETATE Sodium Channel, Site 2 68% 14.954uM 13.407uM View
sodium channel, nonvoltage-gated 1, delta MEDROXYPROGESTERONE ACETATE Sodium Channel, Site 2 68% 14.954uM 13.407uM View
5-hydroxytryptamine (serotonin) receptor 2C BUSPIRONE Serotonin 5-HT2C 68% NoneNone NoneNone View
solute carrier family 6 (neurotransmitter transporter, dopamine), member 3 (S)-(-)-PINDOLOL Dopamine Transporter 68% NoneNone NoneNone View
cannabinoid receptor 1 (brain) NITRENDIPINE Cannabinoid CB1 68% NoneNone NoneNone View
cholinergic receptor, muscarinic 3 TERCONAZOLE Muscarinic M3 68% 14.537uM 3.081uM View
5-hydroxytryptamine (serotonin) receptor 1B DAUNORUBICIN Serotonin 5-HT1B 68% NoneNone NoneNone View
aldo-keto reductase family 1, member B4 (aldose reductase) FLUVASTATIN Aldose Reductase 68% NoneNone NoneNone View
aldo-keto reductase family 1, member B1 (aldose reductase) FLUVASTATIN Aldose Reductase 68% NoneNone NoneNone View
aldo-keto reductase family 7, member A2 (aflatoxin aldehyde reductase) FLUVASTATIN Aldose Reductase 68% NoneNone NoneNone View
aldo-keto reductase family 7, member A3 (aflatoxin aldehyde reductase) FLUVASTATIN Aldose Reductase 68% NoneNone NoneNone View
nuclear receptor subfamily 3, group C, member 1 ETHYNODIOL DIACETATE Glucocorticoid 68% NoneNone NoneNone View
solute carrier family 6 (neurotransmitter transporter, dopamine), member 3 PIPAMAZINE Dopamine Transporter 68% NoneNone NoneNone View
Cytochrom P450-1A2 monooxygenase MICONAZOLE CYP450-1A2 Inhibition 68% NoneNone NoneNone View
calcium channel, voltage-dependent, beta 4 subunit OXICONAZOLE Calcium Channel Type L, Benzothiazepine 67% NoneNone NoneNone View
calcium channel, voltage-dependent, beta 3 subunit OXICONAZOLE Calcium Channel Type L, Benzothiazepine 67% NoneNone NoneNone View
calcium channel, voltage-dependent, beta 2 subunit OXICONAZOLE Calcium Channel Type L, Benzothiazepine 67% NoneNone NoneNone View
calcium channel, voltage-dependent, L type, alpha 1S subunit OXICONAZOLE Calcium Channel Type L, Benzothiazepine 67% NoneNone NoneNone View
calcium channel, voltage-dependent, alpha 1F subunit OXICONAZOLE Calcium Channel Type L, Benzothiazepine 67% NoneNone NoneNone View
calcium channel, voltage-dependent, L type, alpha 1D subunit OXICONAZOLE Calcium Channel Type L, Benzothiazepine 67% NoneNone NoneNone View
calcium channel, voltage-dependent, L type, alpha 1C subunit OXICONAZOLE Calcium Channel Type L, Benzothiazepine 67% NoneNone NoneNone View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit OXICONAZOLE Calcium Channel Type L, Benzothiazepine 67% NoneNone NoneNone View
calcium channel, voltage-dependent, beta 1 subunit OXICONAZOLE Calcium Channel Type L, Benzothiazepine 67% NoneNone NoneNone View
nuclear receptor subfamily 3, group C, member 1 CORTISONE Glucocorticoid 72% 2.378uM 1.081uM View
adrenergic receptor, alpha 1a BUSPIRONE Adrenergic alpha1A 72% 3.482uM 1.41uM View
cytochrome P450, family 3, subfamily a, polypeptide 13 DOCETAXEL CYP450-3A4 Inhibition 72% 2uM NoneNone View
adrenergic receptor, beta 3 DIHYDROERGOCRISTINE MESYLATE Adrenergic beta3 72% 3.308uM 2.481uM View
cholinergic receptor, muscarinic 2 QUETIAPINE Muscarinic M2 72% 3.3447uM 1.1892uM View
calcium channel, voltage-dependent, beta 2 subunit RALOXIFENE Calcium Channel Type L, Dihydropyridine 71% .388uM .249uM View
calcium channel, voltage-dependent, L type, alpha 1S subunit RALOXIFENE Calcium Channel Type L, Dihydropyridine 71% .388uM .249uM View
calcium channel, voltage-dependent, alpha 1F subunit RALOXIFENE Calcium Channel Type L, Dihydropyridine 71% .388uM .249uM View
calcium channel, voltage-dependent, L type, alpha 1D subunit RALOXIFENE Calcium Channel Type L, Dihydropyridine 71% .388uM .249uM View
calcium channel, voltage-dependent, L type, alpha 1C subunit RALOXIFENE Calcium Channel Type L, Dihydropyridine 71% .388uM .249uM View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit RALOXIFENE Calcium Channel Type L, Dihydropyridine 71% .388uM .249uM View
calcium channel, voltage-dependent, beta 1 subunit RALOXIFENE Calcium Channel Type L, Dihydropyridine 71% .388uM .249uM View
calcium channel, voltage-dependent, L type, alpha 1E subunit RALOXIFENE Calcium Channel Type L, Dihydropyridine 71% .388uM .249uM View
calcium channel, voltage-dependent, N type, alpha 1B subunit RALOXIFENE Calcium Channel Type L, Dihydropyridine 71% .388uM .249uM View
calcium channel, voltage-dependent, alpha2/delta subunit 1 RALOXIFENE Calcium Channel Type L, Dihydropyridine 71% .388uM .249uM View
calcium channel, voltage-dependent, gamma subunit 8 RALOXIFENE Calcium Channel Type L, Dihydropyridine 71% .388uM .249uM View
calcium channel, voltage-dependent, gamma subunit 7 RALOXIFENE Calcium Channel Type L, Dihydropyridine 71% .388uM .249uM View
calcium channel, voltage-dependent, gamma subunit 6 RALOXIFENE Calcium Channel Type L, Dihydropyridine 71% .388uM .249uM View
Cytochrom P450-2D6 monooxygenase SB-203580 CYP450-2D6 Inhibition 71% 2uM NoneNone View
5-hydroxytryptamine (serotonin) receptor 2C PROPOFOL Serotonin 5-HT2C 71% 11.553uM 6.051uM View
solute carrier family 6 (neurotransmitter transporter, serotonin), member 4 DOXAZOSIN Serotonin Transporter 71% 2.688uM 1.428uM View
5-hydroxytryptamine (serotonin) receptor 2C TRIOXSALEN Serotonin 5-HT2C 71% 2.356uM 1.234uM View
opioid receptor, sigma 1 S-(-)-PROPRANOLOL Sigma1 71% 6.665uM 2.801uM View
histamine receptor H 2 LOPERAMIDE Histamine H2 71% 3.081uM 3.03uM View
5-hydroxytryptamine (serotonin) receptor 2B LOPERAMIDE Serotonin 5-HT2B 71% 4.105uM 2.613uM View
prostaglandin-endoperoxide synthase 1 ETODOLAC Cyclooxygenase COX-1 71% 2.649uM NoneNone View
prostaglandin-endoperoxide synthase 1 (prostaglandin G/H synthase and cyclooxygenase) ETODOLAC Cyclooxygenase COX-1 71% 2.649uM NoneNone View
solute carrier family 6 (neurotransmitter transporter, noradrenalin), member 2 MITOXANTRONE Adrenergic, Norepinephrine Transporter 71% 4.9898uM 4.9485uM View
gamma-aminobutyric acid (GABA-A) receptor, subunit alpha 4 TROPISETRON GABAA, Agonist Site 71% 3.025uM 2.395uM View
gamma-aminobutyric acid A receptor, gamma 1 TROPISETRON GABAA, Agonist Site 71% 3.025uM 2.395uM View
gamma-aminobutyric acid A receptor, pi TROPISETRON GABAA, Agonist Site 71% 3.025uM 2.395uM View
AT hook, DNA binding motif, containing 1 (DBSS) TROPISETRON GABAA, Agonist Site 71% 3.025uM 2.395uM View
gamma-aminobutyric acid A receptor, theta TROPISETRON GABAA, Agonist Site 71% 3.025uM 2.395uM View
gamma-aminobutyric acid A receptor, gamma 2 TROPISETRON GABAA, Agonist Site 71% 3.025uM 2.395uM View
gamma-aminobutyric acid (GABA-A) receptor, subunit alpha 6 TROPISETRON GABAA, Agonist Site 71% 3.025uM 2.395uM View
gamma-aminobutyric acid (GABA-A) receptor, subunit alpha 5 TROPISETRON GABAA, Agonist Site 71% 3.025uM 2.395uM View
gamma-aminobutyric acid A receptor, alpha 2 TROPISETRON GABAA, Agonist Site 71% 3.025uM 2.395uM View
gamma-aminobutyric acid A receptor, alpha 1 TROPISETRON GABAA, Agonist Site 71% 3.025uM 2.395uM View
gamma-aminobutyric acid (GABA-C) receptor, subunit rho 2 TROPISETRON GABAA, Agonist Site 71% 3.025uM 2.395uM View