Gene Activity List


Gene Activity List

Gene Compound Assay Inh Ic50 Ki View
gamma-aminobutyric acid (GABA-C) receptor, subunit rho 1 TROPISETRON GABAA, Agonist Site 71% 3.025uM 2.395uM View
gamma-aminobutyric acid A receptor, delta TROPISETRON GABAA, Agonist Site 71% 3.025uM 2.395uM View
gamma-aminobutyric acid (GABA-A) receptor, subunit alpha 3 TROPISETRON GABAA, Agonist Site 71% 3.025uM 2.395uM View
calcium channel, voltage-dependent, gamma subunit 8 KETOTIFEN Calcium Channel Type L, Benzothiazepine 71% 2.305uM 2.049uM View
calcium channel, voltage-dependent, gamma subunit 7 KETOTIFEN Calcium Channel Type L, Benzothiazepine 71% 2.305uM 2.049uM View
calcium channel, voltage-dependent, gamma subunit 6 KETOTIFEN Calcium Channel Type L, Benzothiazepine 71% 2.305uM 2.049uM View
calcium channel, voltage-dependent, gamma subunit 5 KETOTIFEN Calcium Channel Type L, Benzothiazepine 71% 2.305uM 2.049uM View
calcium channel, voltage-dependent, gamma subunit 4 KETOTIFEN Calcium Channel Type L, Benzothiazepine 71% 2.305uM 2.049uM View
calcium channel, voltage-dependent, gamma subunit 3 KETOTIFEN Calcium Channel Type L, Benzothiazepine 71% 2.305uM 2.049uM View
calcium channel, voltage-dependent, gamma subunit 2 KETOTIFEN Calcium Channel Type L, Benzothiazepine 71% 2.305uM 2.049uM View
calcium channel, voltage-dependent, gamma subunit 1 KETOTIFEN Calcium Channel Type L, Benzothiazepine 71% 2.305uM 2.049uM View
sodium channel associated protein 1 KETOCONAZOLE Sodium Channel, Site 2 70% 23.911uM 21.438uM View
sodium channel associated protein 2 KETOCONAZOLE Sodium Channel, Site 2 70% 23.911uM 21.438uM View
sodium channel, voltage-gated, type III, beta KETOCONAZOLE Sodium Channel, Site 2 70% 23.911uM 21.438uM View
sodium channel, voltage-gated, type I, alpha KETOCONAZOLE Sodium Channel, Site 2 70% 23.911uM 21.438uM View
sodium channel, voltage-gated, type IX, alpha KETOCONAZOLE Sodium Channel, Site 2 70% 23.911uM 21.438uM View
sodium channel, voltage-gated, type VII, alpha KETOCONAZOLE Sodium Channel, Site 2 70% 23.911uM 21.438uM View
thromboxane A synthase 1 KETOCONAZOLE Thromboxane Synthetase 70% 2.165uM NoneNone View
thromboxane A synthase 1 (platelet, cytochrome P450, family 5, subfamily A) KETOCONAZOLE Thromboxane Synthetase 70% 2.165uM NoneNone View
adrenergic receptor, beta 3 CIGLITAZONE Adrenergic beta3 70% 17.871uM 13.403uM View
aldo-keto reductase family 1, member B4 (aldose reductase) KETOROLAC Aldose Reductase 70% 6.109uM NoneNone View
aldo-keto reductase family 1, member B1 (aldose reductase) KETOROLAC Aldose Reductase 70% 6.109uM NoneNone View
aldo-keto reductase family 7, member A2 (aflatoxin aldehyde reductase) KETOROLAC Aldose Reductase 70% 6.109uM NoneNone View
aldo-keto reductase family 7, member A3 (aflatoxin aldehyde reductase) KETOROLAC Aldose Reductase 70% 6.109uM NoneNone View
monoamine oxidase A NOCODAZOLE Monoamine Oxidase MAOA 70% 24.099uM NoneNone View
monoamine oxidase A NOCODAZOLE Monoamine Oxidase MAOA 70% 24.099uM NoneNone View
adenosine A2a receptor NOCODAZOLE Adenosine A2A 70% 7.509uM 4.219uM View
opioid receptor, sigma 1 PROGESTERONE Sigma1 70% 3.055uM 1.284uM View
adrenergic receptor, alpha 2a AMOXAPINE Imidazoline I2, Central 70% 3.466uM 2.31uM View
adrenergic receptor, alpha 2c (Non-specific probe) AMOXAPINE Imidazoline I2, Central 70% 3.466uM 2.31uM View
calcium channel, voltage-dependent, gamma subunit 8 CLOTRIMAZOLE Calcium Channel Type L, Benzothiazepine 70% 28.499uM 25.332uM View
calcium channel, voltage-dependent, gamma subunit 7 CLOTRIMAZOLE Calcium Channel Type L, Benzothiazepine 70% 28.499uM 25.332uM View
calcium channel, voltage-dependent, gamma subunit 6 CLOTRIMAZOLE Calcium Channel Type L, Benzothiazepine 70% 28.499uM 25.332uM View
calcium channel, voltage-dependent, gamma subunit 5 CLOTRIMAZOLE Calcium Channel Type L, Benzothiazepine 70% 28.499uM 25.332uM View
calcium channel, voltage-dependent, gamma subunit 4 CLOTRIMAZOLE Calcium Channel Type L, Benzothiazepine 70% 28.499uM 25.332uM View
calcium channel, voltage-dependent, gamma subunit 3 CLOTRIMAZOLE Calcium Channel Type L, Benzothiazepine 70% 28.499uM 25.332uM View
calcium channel, voltage-dependent, gamma subunit 2 CLOTRIMAZOLE Calcium Channel Type L, Benzothiazepine 70% 28.499uM 25.332uM View
calcium channel, voltage-dependent, gamma subunit 1 CLOTRIMAZOLE Calcium Channel Type L, Benzothiazepine 70% 28.499uM 25.332uM View
calcium channel, voltage-dependent, beta 4 subunit CLOTRIMAZOLE Calcium Channel Type L, Benzothiazepine 70% 28.499uM 25.332uM View
calcium channel, voltage-dependent, beta 3 subunit CLOTRIMAZOLE Calcium Channel Type L, Benzothiazepine 70% 28.499uM 25.332uM View
solute carrier family 6 (neurotransmitter transporter, serotonin), member 4 BW-723C86 Serotonin Transporter 70% 4.785uM 2.542uM View
cholinergic receptor, muscarinic 3 SULOCTIDIL Muscarinic M3 70% 4.6238uM .98uM View
opioid receptor, sigma 1 DIMENHYDRINATE Sigma1 70% 1.158uM .487uM View
mu-opioid receptor MOR CINNARIZINE Opiate mu 70% 2.272uM .922uM View
opioid receptor, kappa 1 DOMPERIDONE Opiate kappa 70% 6.994uM 2.798uM View
calcium channel, voltage-dependent, gamma subunit 8 VALETHAMATE BROMIDE Calcium Channel Type L, Benzothiazepine 70% 3.389uM 3.013uM View
calcium channel, voltage-dependent, gamma subunit 7 VALETHAMATE BROMIDE Calcium Channel Type L, Benzothiazepine 70% 3.389uM 3.013uM View
calcium channel, voltage-dependent, gamma subunit 6 VALETHAMATE BROMIDE Calcium Channel Type L, Benzothiazepine 70% 3.389uM 3.013uM View
calcium channel, voltage-dependent, gamma subunit 5 VALETHAMATE BROMIDE Calcium Channel Type L, Benzothiazepine 70% 3.389uM 3.013uM View
calcium channel, voltage-dependent, gamma subunit 4 VALETHAMATE BROMIDE Calcium Channel Type L, Benzothiazepine 70% 3.389uM 3.013uM View
calcium channel, voltage-dependent, gamma subunit 3 VALETHAMATE BROMIDE Calcium Channel Type L, Benzothiazepine 70% 3.389uM 3.013uM View
calcium channel, voltage-dependent, gamma subunit 2 VALETHAMATE BROMIDE Calcium Channel Type L, Benzothiazepine 70% 3.389uM 3.013uM View
calcium channel, voltage-dependent, gamma subunit 1 VALETHAMATE BROMIDE Calcium Channel Type L, Benzothiazepine 70% 3.389uM 3.013uM View
calcium channel, voltage-dependent, beta 4 subunit VALETHAMATE BROMIDE Calcium Channel Type L, Benzothiazepine 70% 3.389uM 3.013uM View
ATPase, Na+/K+ transporting, beta 2 polypeptide CLADRIBINE ATPase, Na+/K+ 13% NoneNone NoneNone View
calcium channel, voltage-dependent, beta 3 subunit VALETHAMATE BROMIDE Calcium Channel Type L, Benzothiazepine 70% 3.389uM 3.013uM View
calcium channel, voltage-dependent, beta 2 subunit VALETHAMATE BROMIDE Calcium Channel Type L, Benzothiazepine 70% 3.389uM 3.013uM View
calcium channel, voltage-dependent, L type, alpha 1S subunit VALETHAMATE BROMIDE Calcium Channel Type L, Benzothiazepine 70% 3.389uM 3.013uM View
calcium channel, voltage-dependent, alpha 1F subunit VALETHAMATE BROMIDE Calcium Channel Type L, Benzothiazepine 70% 3.389uM 3.013uM View
calcium channel, voltage-dependent, L type, alpha 1D subunit VALETHAMATE BROMIDE Calcium Channel Type L, Benzothiazepine 70% 3.389uM 3.013uM View
calcium channel, voltage-dependent, L type, alpha 1C subunit VALETHAMATE BROMIDE Calcium Channel Type L, Benzothiazepine 70% 3.389uM 3.013uM View
calcium channel, voltage-dependent, L type, alpha 1E subunit OXICONAZOLE Calcium Channel Type L, Benzothiazepine 67% NoneNone NoneNone View
calcium channel, voltage-dependent, N type, alpha 1B subunit OXICONAZOLE Calcium Channel Type L, Benzothiazepine 67% NoneNone NoneNone View
calcium channel, voltage-dependent, alpha2/delta subunit 1 OXICONAZOLE Calcium Channel Type L, Benzothiazepine 67% NoneNone NoneNone View
cholinergic receptor, muscarinic 5 OXICONAZOLE Muscarinic M5 67% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 5 OXYMETAZOLINE Calcium Channel Type L, Benzothiazepine 67% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 4 OXYMETAZOLINE Calcium Channel Type L, Benzothiazepine 67% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 3 OXYMETAZOLINE Calcium Channel Type L, Benzothiazepine 67% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 2 OXYMETAZOLINE Calcium Channel Type L, Benzothiazepine 67% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 1 OXYMETAZOLINE Calcium Channel Type L, Benzothiazepine 67% NoneNone NoneNone View
calcium channel, voltage-dependent, beta 4 subunit OXYMETAZOLINE Calcium Channel Type L, Benzothiazepine 67% NoneNone NoneNone View
calcium channel, voltage-dependent, beta 3 subunit OXYMETAZOLINE Calcium Channel Type L, Benzothiazepine 67% NoneNone NoneNone View
calcium channel, voltage-dependent, beta 2 subunit OXYMETAZOLINE Calcium Channel Type L, Benzothiazepine 67% NoneNone NoneNone View
calcium channel, voltage-dependent, L type, alpha 1S subunit OXYMETAZOLINE Calcium Channel Type L, Benzothiazepine 67% NoneNone NoneNone View
calcium channel, voltage-dependent, alpha 1F subunit OXYMETAZOLINE Calcium Channel Type L, Benzothiazepine 67% NoneNone NoneNone View
calcium channel, voltage-dependent, L type, alpha 1D subunit OXYMETAZOLINE Calcium Channel Type L, Benzothiazepine 67% NoneNone NoneNone View
calcium channel, voltage-dependent, L type, alpha 1C subunit OXYMETAZOLINE Calcium Channel Type L, Benzothiazepine 67% NoneNone NoneNone View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit OXYMETAZOLINE Calcium Channel Type L, Benzothiazepine 67% NoneNone NoneNone View
calcium channel, voltage-dependent, beta 1 subunit OXYMETAZOLINE Calcium Channel Type L, Benzothiazepine 67% NoneNone NoneNone View
calcium channel, voltage-dependent, L type, alpha 1E subunit OXYMETAZOLINE Calcium Channel Type L, Benzothiazepine 67% NoneNone NoneNone View
calcium channel, voltage-dependent, N type, alpha 1B subunit OXYMETAZOLINE Calcium Channel Type L, Benzothiazepine 67% NoneNone NoneNone View
calcium channel, voltage-dependent, alpha2/delta subunit 1 OXYMETAZOLINE Calcium Channel Type L, Benzothiazepine 67% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 8 OXYMETAZOLINE Calcium Channel Type L, Benzothiazepine 67% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 7 OXYMETAZOLINE Calcium Channel Type L, Benzothiazepine 67% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 6 OXYMETAZOLINE Calcium Channel Type L, Benzothiazepine 67% NoneNone NoneNone View
Cytochrom P450-2C19 monooxygenase FELODIPINE CYP450-2C19 Inhibition 67% NoneNone NoneNone View
dopamine receptor D3 CANDESARTAN Dopamine D3 67% NoneNone NoneNone View
cholinergic receptor, muscarinic 2 RALOXIFENE Muscarinic M2 67% NoneNone NoneNone View
5-hydroxytryptamine (serotonin) receptor 5B SB-203580 Serotonin 5-HT4 67% 10.553uM 1.759uM View
5-hydroxytryptamine (serotonin) receptor 4 SB-203580 Serotonin 5-HT4 67% 10.553uM 1.759uM View
adrenergic receptor, beta 2 ATENOLOL Adrenergic beta2 67% 14.634uM 10.061uM View
lymphocyte protein tyrosine kinase (mapped) CLOMIPHENE Protein Tyrosine Kinase, Lck 67% NoneNone NoneNone View
mu-opioid receptor MOR DROPERIDOL Opiate mu 67% NoneNone NoneNone View
Cytochrome P450, subfamily IIC (mephenytoin 4-hydroxylase) ANTIMYCIN A CYP450-2C9 Inhibition 67% NoneNone NoneNone View
cytochrome P450, family 2, subfamily C, polypeptide 9 ANTIMYCIN A CYP450-2C9 Inhibition 67% NoneNone NoneNone View
neuropeptide Y receptor Y2 DIHYDROERGOCRISTINE MESYLATE Neuropeptide Y2 67% NoneNone NoneNone View
adrenergic receptor, beta 3 NELFINAVIR Adrenergic beta3 67% 34.08uM 25.566uM View
opioid receptor, sigma 1 STANOLONE Sigma1 67% NoneNone NoneNone View
leukotriene C4 synthase 6-METHOXY-2-NAPHTHYLACETIC ACID Leukotriene C4 Synthetase 67% 49.66uM NoneNone View
leukotriene C4 synthase 6-METHOXY-2-NAPHTHYLACETIC ACID Leukotriene C4 Synthetase 67% 49.66uM NoneNone View
adrenergic receptor, alpha 2a PROCHLORPERAZINE Imidazoline I2, Central 67% NoneNone NoneNone View
adrenergic receptor, alpha 2c (Non-specific probe) PROCHLORPERAZINE Imidazoline I2, Central 67% NoneNone NoneNone View
adrenergic receptor, alpha 1d (Non-specific probe) PENTAMIDINE Adrenergic alpha1D 67% NoneNone NoneNone View
Sigma-2 Receptor CYPROHEPTADINE Sigma2 67% NoneNone NoneNone View
opioid receptor, sigma 1 METOCLOPRAMIDE Sigma1 67% NoneNone NoneNone View
5-hydroxytryptamine (serotonin) receptor 1B ECONAZOLE Serotonin 5-HT1B 67% 22.034uM 10.016uM View
Sigma-2 Receptor MICONAZOLE Sigma2 67% 3.305uM 2.034uM View
adrenergic receptor, alpha 2a KETOCONAZOLE Adrenergic alpha2A 67% 19.783uM 7.419uM View
progesterone receptor CIGLITAZONE Progesterone 67% 29.118uM 3.798uM View
progesterone receptor CIGLITAZONE Progesterone 67% 29.118uM 3.798uM View
thromboxane A synthase 1 AURANOFIN Thromboxane Synthetase 67% NoneNone NoneNone View
thromboxane A synthase 1 (platelet, cytochrome P450, family 5, subfamily A) AURANOFIN Thromboxane Synthetase 67% NoneNone NoneNone View
opioid receptor, kappa 1 SULCONAZOLE Opiate kappa 67% NoneNone NoneNone View
lymphocyte protein tyrosine kinase (mapped) 4-OCTYLPHENOL Protein Tyrosine Kinase, Lck 67% 22.054uM NoneNone View
acetylcholinesterase (YT blood group) 4-OCTYLPHENOL Acetylcholinesterase 67% 11.471uM NoneNone View
collagen-like tail subunit (single strand of homotrimer) of asymmetric acetylcholinesterase 4-OCTYLPHENOL Acetylcholinesterase 67% 11.471uM NoneNone View
calcium channel, voltage-dependent, beta 4 subunit KETOTIFEN Calcium Channel Type L, Benzothiazepine 71% 2.305uM 2.049uM View
calcium channel, voltage-dependent, beta 3 subunit KETOTIFEN Calcium Channel Type L, Benzothiazepine 71% 2.305uM 2.049uM View
calcium channel, voltage-dependent, beta 2 subunit KETOTIFEN Calcium Channel Type L, Benzothiazepine 71% 2.305uM 2.049uM View
calcium channel, voltage-dependent, L type, alpha 1S subunit KETOTIFEN Calcium Channel Type L, Benzothiazepine 71% 2.305uM 2.049uM View
calcium channel, voltage-dependent, alpha 1F subunit KETOTIFEN Calcium Channel Type L, Benzothiazepine 71% 2.305uM 2.049uM View
calcium channel, voltage-dependent, L type, alpha 1D subunit KETOTIFEN Calcium Channel Type L, Benzothiazepine 71% 2.305uM 2.049uM View
calcium channel, voltage-dependent, L type, alpha 1C subunit KETOTIFEN Calcium Channel Type L, Benzothiazepine 71% 2.305uM 2.049uM View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit KETOTIFEN Calcium Channel Type L, Benzothiazepine 71% 2.305uM 2.049uM View
calcium channel, voltage-dependent, beta 1 subunit KETOTIFEN Calcium Channel Type L, Benzothiazepine 71% 2.305uM 2.049uM View
calcium channel, voltage-dependent, L type, alpha 1E subunit KETOTIFEN Calcium Channel Type L, Benzothiazepine 71% 2.305uM 2.049uM View
calcium channel, voltage-dependent, N type, alpha 1B subunit KETOTIFEN Calcium Channel Type L, Benzothiazepine 71% 2.305uM 2.049uM View
calcium channel, voltage-dependent, alpha2/delta subunit 1 KETOTIFEN Calcium Channel Type L, Benzothiazepine 71% 2.305uM 2.049uM View
AT hook, DNA binding motif, containing 1 (DBSS) NORETHINDRONE GABAA, Benzodiazepine, Central 71% 13.343uM 10.872uM View
gamma-aminobutyric acid A receptor, theta NORETHINDRONE GABAA, Benzodiazepine, Central 71% 13.343uM 10.872uM View
gamma-aminobutyric acid A receptor, gamma 2 NORETHINDRONE GABAA, Benzodiazepine, Central 71% 13.343uM 10.872uM View
gamma-aminobutyric acid (GABA-A) receptor, subunit alpha 6 NORETHINDRONE GABAA, Benzodiazepine, Central 71% 13.343uM 10.872uM View
gamma-aminobutyric acid (GABA-A) receptor, subunit alpha 5 NORETHINDRONE GABAA, Benzodiazepine, Central 71% 13.343uM 10.872uM View
gamma-aminobutyric acid A receptor, alpha 2 NORETHINDRONE GABAA, Benzodiazepine, Central 71% 13.343uM 10.872uM View
gamma-aminobutyric acid A receptor, alpha 1 NORETHINDRONE GABAA, Benzodiazepine, Central 71% 13.343uM 10.872uM View
gamma-aminobutyric acid (GABA-C) receptor, subunit rho 2 NORETHINDRONE GABAA, Benzodiazepine, Central 71% 13.343uM 10.872uM View
gamma-aminobutyric acid (GABA-C) receptor, subunit rho 1 NORETHINDRONE GABAA, Benzodiazepine, Central 71% 13.343uM 10.872uM View
gamma-aminobutyric acid A receptor, delta NORETHINDRONE GABAA, Benzodiazepine, Central 71% 13.343uM 10.872uM View
gamma-aminobutyric acid (GABA-A) receptor, subunit alpha 3 NORETHINDRONE GABAA, Benzodiazepine, Central 71% 13.343uM 10.872uM View
gamma-aminobutyric acid (GABA-A) receptor, subunit alpha 4 NORETHINDRONE GABAA, Benzodiazepine, Central 71% 13.343uM 10.872uM View
gamma-aminobutyric acid A receptor, gamma 1 NORETHINDRONE GABAA, Benzodiazepine, Central 71% 13.343uM 10.872uM View
gamma-aminobutyric acid A receptor, pi NORETHINDRONE GABAA, Benzodiazepine, Central 71% 13.343uM 10.872uM View
solute carrier family 6 (neurotransmitter transporter, noradrenalin), member 2 PROPAFENONE Adrenergic, Norepinephrine Transporter 71% 3.016uM 2.991uM View
progesterone receptor STANOZOLOL Progesterone 71% 3.705uM .483uM View
progesterone receptor STANOZOLOL Progesterone 71% 3.705uM .483uM View
solute carrier family 6 (neurotransmitter transporter, serotonin), member 4 SIBUTRAMINE Serotonin Transporter 71% 2.085uM 1.108uM View
calcium channel, voltage-dependent, gamma subunit 5 RALOXIFENE Calcium Channel Type L, Dihydropyridine 71% .388uM .249uM View
calcium channel, voltage-dependent, gamma subunit 4 RALOXIFENE Calcium Channel Type L, Dihydropyridine 71% .388uM .249uM View
calcium channel, voltage-dependent, gamma subunit 3 RALOXIFENE Calcium Channel Type L, Dihydropyridine 71% .388uM .249uM View
calcium channel, voltage-dependent, gamma subunit 2 RALOXIFENE Calcium Channel Type L, Dihydropyridine 71% .388uM .249uM View
calcium channel, voltage-dependent, gamma subunit 1 RALOXIFENE Calcium Channel Type L, Dihydropyridine 71% .388uM .249uM View
calcium channel, voltage-dependent, beta 4 subunit RALOXIFENE Calcium Channel Type L, Dihydropyridine 71% .388uM .249uM View
calcium channel, voltage-dependent, beta 3 subunit RALOXIFENE Calcium Channel Type L, Dihydropyridine 71% .388uM .249uM View
ATPase, Na+/K+ transporting, beta 1 polypeptide CHLORMADINONE ACETATE ATPase, Na+/K+ 71% 4.5696uM NoneNone View
ATPase, Na+/K+ transporting, beta 3 polypeptide CHLORMADINONE ACETATE ATPase, Na+/K+ 71% 4.5696uM NoneNone View
ATPase, Na+/K+ transporting, beta 2 polypeptide CHLORMADINONE ACETATE ATPase, Na+/K+ 71% 4.5696uM NoneNone View
ATPase, (Na+)/K+ transporting, beta 4 polypeptide CHLORMADINONE ACETATE ATPase, Na+/K+ 71% 4.5696uM NoneNone View
nuclear receptor subfamily 3, group C, member 1 CORTISONE ACETATE Glucocorticoid 71% 3.911uM 1.778uM View
5-hydroxytryptamine (serotonin) receptor 2B BENZBROMARONE Serotonin 5-HT2B 71% 1.804uM 1.148uM View
tachykinin receptor 2 FLUPHENAZINE Tachykinin NK2 71% 22.484uM 7.495uM View
Sigma-2 Receptor DOXEPIN Sigma2 71% 2.143uM 1.319uM View
mitogen activated protein kinase 1 DICUMAROL Protein Serine/Threonine Kinase, ERK2 71% 4.426uM NoneNone View
mitogen-activated protein kinase 1 DICUMAROL Protein Serine/Threonine Kinase, ERK2 71% 4.426uM NoneNone View
cholinergic receptor, muscarinic 5 HALOPERIDOL Muscarinic M5 71% 3.89uM 2.795uM View
opioid receptor, sigma 1 TRAZODONE Sigma1 71% 2.203uM .926uM View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit VALETHAMATE BROMIDE Calcium Channel Type L, Benzothiazepine 70% 3.389uM 3.013uM View
calcium channel, voltage-dependent, beta 1 subunit VALETHAMATE BROMIDE Calcium Channel Type L, Benzothiazepine 70% 3.389uM 3.013uM View
calcium channel, voltage-dependent, L type, alpha 1E subunit VALETHAMATE BROMIDE Calcium Channel Type L, Benzothiazepine 70% 3.389uM 3.013uM View
calcium channel, voltage-dependent, N type, alpha 1B subunit VALETHAMATE BROMIDE Calcium Channel Type L, Benzothiazepine 70% 3.389uM 3.013uM View
calcium channel, voltage-dependent, alpha2/delta subunit 1 VALETHAMATE BROMIDE Calcium Channel Type L, Benzothiazepine 70% 3.389uM 3.013uM View
cytochrome P450, family 3, subfamily a, polypeptide 13 CLOSANTEL CYP450-3A4 Inhibition 70% 5uM NoneNone View
cytochrome P450, family 3, subfamily a, polypeptide 13 IDEBENONE CYP450-3A4 Inhibition 70% 7uM NoneNone View
Cytochrom P450-2D6 monooxygenase BAMBUTEROL CYP450-2D6 Inhibition 70% 2uM NoneNone View
Cytochrome P450, subfamily IIC (mephenytoin 4-hydroxylase) LOSARTAN CYP450-2C9 Inhibition 70% 2.882uM NoneNone View
cytochrome P450, family 2, subfamily C, polypeptide 9 LOSARTAN CYP450-2C9 Inhibition 70% 2.882uM NoneNone View
adrenergic receptor, alpha 1a PROPAFENONE Adrenergic alpha1A 70% 6.147uM 2.488uM View
adrenergic receptor, alpha 2a DOMPERIDONE Adrenergic alpha2A 70% 2.74uM 1.027uM View
solute carrier family 6 (neurotransmitter transporter, dopamine), member 3 IVERMECTIN Dopamine Transporter 70% 4.4552uM 3.5397uM View
calcium channel, voltage-dependent, gamma subunit 8 SPIRADOLINE Calcium Channel Type L, Benzothiazepine 70% 8.513uM 7.567uM View
calcium channel, voltage-dependent, gamma subunit 7 SPIRADOLINE Calcium Channel Type L, Benzothiazepine 70% 8.513uM 7.567uM View
calcium channel, voltage-dependent, gamma subunit 6 SPIRADOLINE Calcium Channel Type L, Benzothiazepine 70% 8.513uM 7.567uM View
calcium channel, voltage-dependent, gamma subunit 5 SPIRADOLINE Calcium Channel Type L, Benzothiazepine 70% 8.513uM 7.567uM View
calcium channel, voltage-dependent, gamma subunit 4 SPIRADOLINE Calcium Channel Type L, Benzothiazepine 70% 8.513uM 7.567uM View
calcium channel, voltage-dependent, gamma subunit 3 SPIRADOLINE Calcium Channel Type L, Benzothiazepine 70% 8.513uM 7.567uM View
ATPase, (Na+)/K+ transporting, beta 4 polypeptide CLADRIBINE ATPase, Na+/K+ 13% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 2 SPIRADOLINE Calcium Channel Type L, Benzothiazepine 70% 8.513uM 7.567uM View
calcium channel, voltage-dependent, gamma subunit 1 SPIRADOLINE Calcium Channel Type L, Benzothiazepine 70% 8.513uM 7.567uM View
calcium channel, voltage-dependent, beta 4 subunit SPIRADOLINE Calcium Channel Type L, Benzothiazepine 70% 8.513uM 7.567uM View
calcium channel, voltage-dependent, beta 3 subunit SPIRADOLINE Calcium Channel Type L, Benzothiazepine 70% 8.513uM 7.567uM View
calcium channel, voltage-dependent, beta 2 subunit SPIRADOLINE Calcium Channel Type L, Benzothiazepine 70% 8.513uM 7.567uM View
calcium channel, voltage-dependent, L type, alpha 1S subunit SPIRADOLINE Calcium Channel Type L, Benzothiazepine 70% 8.513uM 7.567uM View
calcium channel, voltage-dependent, alpha 1F subunit SPIRADOLINE Calcium Channel Type L, Benzothiazepine 70% 8.513uM 7.567uM View
calcium channel, voltage-dependent, L type, alpha 1D subunit SPIRADOLINE Calcium Channel Type L, Benzothiazepine 70% 8.513uM 7.567uM View
calcium channel, voltage-dependent, L type, alpha 1C subunit SPIRADOLINE Calcium Channel Type L, Benzothiazepine 70% 8.513uM 7.567uM View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit SPIRADOLINE Calcium Channel Type L, Benzothiazepine 70% 8.513uM 7.567uM View
calcium channel, voltage-dependent, beta 1 subunit SPIRADOLINE Calcium Channel Type L, Benzothiazepine 70% 8.513uM 7.567uM View
calcium channel, voltage-dependent, L type, alpha 1E subunit SPIRADOLINE Calcium Channel Type L, Benzothiazepine 70% 8.513uM 7.567uM View
calcium channel, voltage-dependent, N type, alpha 1B subunit SPIRADOLINE Calcium Channel Type L, Benzothiazepine 70% 8.513uM 7.567uM View
calcium channel, voltage-dependent, alpha2/delta subunit 1 SPIRADOLINE Calcium Channel Type L, Benzothiazepine 70% 8.513uM 7.567uM View
adrenergic receptor, alpha 2a BUTENAFINE Adrenergic alpha2A 70% 3.6443uM 1.3666uM View