Gene Activity List


Gene Activity List

Gene Compound Assay Inh Ic50 Ki View
sodium channel, voltage-gated, type IV, beta DESLORATADINE Sodium Channel, Site 2 67% NoneNone NoneNone View
sodium channel, voltage-gated, type IV, alpha DESLORATADINE Sodium Channel, Site 2 67% NoneNone NoneNone View
sodium channel, voltage-gated, type III, alpha DESLORATADINE Sodium Channel, Site 2 67% NoneNone NoneNone View
sodium channel, voltage-gated, type II, beta DESLORATADINE Sodium Channel, Site 2 67% NoneNone NoneNone View
sodium channel, voltage-gated, type II, alpha 2 DESLORATADINE Sodium Channel, Site 2 67% NoneNone NoneNone View
sodium channel, voltage-gated, type I, beta DESLORATADINE Sodium Channel, Site 2 67% NoneNone NoneNone View
sodium channel, voltage-gated, type I, alpha DESLORATADINE Sodium Channel, Site 2 67% NoneNone NoneNone View
3-hydroxy-3-methylglutaryl-Coenzyme A reductase ZAFIRLUKAST HMG-CoA Reductase 67% NoneNone NoneNone View
3-hydroxy-3-methylglutaryl-Coenzyme A reductase ZAFIRLUKAST HMG-CoA Reductase 67% NoneNone NoneNone View
Cytochrom P450-2D6 monooxygenase KETOTIFEN CYP450-2D6 Inhibition 67% NoneNone NoneNone View
Cytochrome P450, subfamily IIC (mephenytoin 4-hydroxylase) ALOSETRON CYP450-2C9 Inhibition 67% NoneNone NoneNone View
cytochrome P450, family 2, subfamily C, polypeptide 9 ALOSETRON CYP450-2C9 Inhibition 67% NoneNone NoneNone View
Cytochrome P450, subfamily IIC (mephenytoin 4-hydroxylase) CHLORMADINONE ACETATE CYP450-2C9 Inhibition 67% NoneNone NoneNone View
cytochrome P450, family 2, subfamily C, polypeptide 9 CHLORMADINONE ACETATE CYP450-2C9 Inhibition 67% NoneNone NoneNone View
acetylcholinesterase (YT blood group) 4-NONYLPHENOL Acetylcholinesterase 67% NoneNone NoneNone View
collagen-like tail subunit (single strand of homotrimer) of asymmetric acetylcholinesterase 4-NONYLPHENOL Acetylcholinesterase 67% NoneNone NoneNone View
acetylcholinesterase 4-NONYLPHENOL Acetylcholinesterase 67% NoneNone NoneNone View
adenosine A2a receptor AMINOPHYLLINE Adenosine A2A 67% NoneNone NoneNone View
adrenergic receptor, alpha 1d (Non-specific probe) METHYLERGONOVINE Adrenergic alpha1D 67% NoneNone NoneNone View
adrenergic receptor, alpha 2b AMITRAZ Adrenergic alpha2B 67% NoneNone NoneNone View
solute carrier family 6 (neurotransmitter transporter, noradrenalin), member 2 GRAMICIDIN Adrenergic, Norepinephrine Transporter 67% NoneNone NoneNone View
bradykinin receptor, beta 2 GRAMICIDIN Bradykinin B2 67% NoneNone NoneNone View
bradykinin receptor B2 GRAMICIDIN Bradykinin B2 67% NoneNone NoneNone View
adrenergic receptor, alpha 2a MOXONIDINE Adrenergic alpha2A 67% NoneNone NoneNone View
A3 adenosine receptor DIGITONIN Adenosine A3 67% NoneNone NoneNone View
adrenergic receptor, alpha 2b O-ANISIDINE Adrenergic alpha2B 67% 2.508uM 1.145uM View
neuropeptide Y receptor Y2 DIHYDROERGOCRISTINE MESYLATE Neuropeptide Y2 67% NoneNone NoneNone View
calcium channel, voltage-dependent, beta 4 subunit DEXTROMETHORPHAN Calcium Channel Type L, Benzothiazepine 66% NoneNone NoneNone View
calcium channel, voltage-dependent, beta 3 subunit DEXTROMETHORPHAN Calcium Channel Type L, Benzothiazepine 66% NoneNone NoneNone View
calcium channel, voltage-dependent, beta 2 subunit DEXTROMETHORPHAN Calcium Channel Type L, Benzothiazepine 66% NoneNone NoneNone View
calcium channel, voltage-dependent, L type, alpha 1S subunit DEXTROMETHORPHAN Calcium Channel Type L, Benzothiazepine 66% NoneNone NoneNone View
calcium channel, voltage-dependent, alpha 1F subunit DEXTROMETHORPHAN Calcium Channel Type L, Benzothiazepine 66% NoneNone NoneNone View
calcium channel, voltage-dependent, L type, alpha 1D subunit DEXTROMETHORPHAN Calcium Channel Type L, Benzothiazepine 66% NoneNone NoneNone View
adrenergic receptor, alpha 2b EPERISONE Adrenergic alpha2B 71% 3.034uM 1.385uM View
adrenergic receptor, beta 1 BROMOCRIPTINE Adrenergic beta1 71% 2.4uM 1.386uM View
adrenergic, beta-1-, receptor BROMOCRIPTINE Adrenergic beta1 71% 2.4uM 1.386uM View
histamine receptor H 1 CITALOPRAM Histamine H1, Central 71% 3.194uM .371uM View
adrenergic receptor, alpha 2a VERAPAMIL Imidazoline I2, Central 71% 5.524uM 3.683uM View
adrenergic receptor, alpha 2c (Non-specific probe) VERAPAMIL Imidazoline I2, Central 71% 5.524uM 3.683uM View
adrenergic receptor, alpha 1b LYSERGOL Adrenergic alpha1B 71% 4.726uM 2.616uM View
sodium channel, nonvoltage-gated 1, delta PYRILAMINE Sodium Channel, Site 2 71% 5.283uM 4.819uM View
sodium channel, nonvoltage-gated 1, beta (Liddle syndrome) PYRILAMINE Sodium Channel, Site 2 71% 5.283uM 4.819uM View
sodium channel, nonvoltage-gated 1 alpha PYRILAMINE Sodium Channel, Site 2 71% 5.283uM 4.819uM View
sodium channel, voltage-gated, type X, alpha PYRILAMINE Sodium Channel, Site 2 71% 5.283uM 4.819uM View
sodium channel, voltage-gated, type IX, alpha PYRILAMINE Sodium Channel, Site 2 71% 5.283uM 4.819uM View
sodium channel, voltage gated, type VIII, alpha PYRILAMINE Sodium Channel, Site 2 71% 5.283uM 4.819uM View
sodium channel, voltage-gated, type VII, alpha PYRILAMINE Sodium Channel, Site 2 71% 5.283uM 4.819uM View
sodium channel, voltage-gated, type V, alpha (long QT syndrome 3) PYRILAMINE Sodium Channel, Site 2 71% 5.283uM 4.819uM View
sodium channel, voltage-gated, type IV, beta PYRILAMINE Sodium Channel, Site 2 71% 5.283uM 4.819uM View
sodium channel, voltage-gated, type IV, alpha PYRILAMINE Sodium Channel, Site 2 71% 5.283uM 4.819uM View
sodium channel, voltage-gated, type III, alpha PYRILAMINE Sodium Channel, Site 2 71% 5.283uM 4.819uM View
sodium channel, voltage-gated, type II, beta PYRILAMINE Sodium Channel, Site 2 71% 5.283uM 4.819uM View
sodium channel, voltage-gated, type II, alpha 2 PYRILAMINE Sodium Channel, Site 2 71% 5.283uM 4.819uM View
sodium channel, voltage-gated, type I, beta PYRILAMINE Sodium Channel, Site 2 71% 5.283uM 4.819uM View
sodium channel, voltage-gated, type I, alpha PYRILAMINE Sodium Channel, Site 2 71% 5.283uM 4.819uM View
A3 adenosine receptor NELFINAVIR Adenosine A3 71% 14.796uM 8.363uM View
adrenergic receptor, alpha 1a TACRINE Adrenergic alpha1A 71% 2.749uM 1.113uM View
adrenergic receptor, beta 2 ZIDOVUDINE Adrenergic beta2 12% NoneNone NoneNone View
solute carrier family 6 (neurotransmitter transporter, dopamine), member 3 PROCHLORPERAZINE Dopamine Transporter 71% 1.735uM 1.379uM View
monoamine oxidase A PIOGLITAZONE Monoamine Oxidase MAOA 71% 35.069uM NoneNone View
monoamine oxidase A PIOGLITAZONE Monoamine Oxidase MAOA 71% 35.069uM NoneNone View
5-hydroxytryptamine (serotonin) receptor 1A PIPAMAZINE Serotonin 5-HT1A 71% 1.782uM 1.018uM View
Cytochrome P450, subfamily IIC (mephenytoin 4-hydroxylase) GW-1929 CYP450-2C9 Inhibition 71% 4uM NoneNone View
cytochrome P450, family 2, subfamily C, polypeptide 9 GW-1929 CYP450-2C9 Inhibition 71% 4uM NoneNone View
epidermal growth factor receptor GW-1929 Protein Tyrosine Kinase, EGF Receptor 71% 10.896uM NoneNone View
calcium channel, voltage-dependent, gamma subunit 8 MICONAZOLE Calcium Channel Type L, Benzothiazepine 71% 18.034uM 16.03uM View
calcium channel, voltage-dependent, gamma subunit 7 MICONAZOLE Calcium Channel Type L, Benzothiazepine 71% 18.034uM 16.03uM View
calcium channel, voltage-dependent, gamma subunit 6 MICONAZOLE Calcium Channel Type L, Benzothiazepine 71% 18.034uM 16.03uM View
calcium channel, voltage-dependent, gamma subunit 5 MICONAZOLE Calcium Channel Type L, Benzothiazepine 71% 18.034uM 16.03uM View
calcium channel, voltage-dependent, gamma subunit 4 MICONAZOLE Calcium Channel Type L, Benzothiazepine 71% 18.034uM 16.03uM View
calcium channel, voltage-dependent, gamma subunit 3 MICONAZOLE Calcium Channel Type L, Benzothiazepine 71% 18.034uM 16.03uM View
calcium channel, voltage-dependent, gamma subunit 2 MICONAZOLE Calcium Channel Type L, Benzothiazepine 71% 18.034uM 16.03uM View
calcium channel, voltage-dependent, gamma subunit 1 MICONAZOLE Calcium Channel Type L, Benzothiazepine 71% 18.034uM 16.03uM View
calcium channel, voltage-dependent, beta 4 subunit MICONAZOLE Calcium Channel Type L, Benzothiazepine 71% 18.034uM 16.03uM View
calcium channel, voltage-dependent, beta 3 subunit MICONAZOLE Calcium Channel Type L, Benzothiazepine 71% 18.034uM 16.03uM View
calcium channel, voltage-dependent, beta 2 subunit MICONAZOLE Calcium Channel Type L, Benzothiazepine 71% 18.034uM 16.03uM View
calcium channel, voltage-dependent, L type, alpha 1S subunit MICONAZOLE Calcium Channel Type L, Benzothiazepine 71% 18.034uM 16.03uM View
calcium channel, voltage-dependent, alpha 1F subunit MICONAZOLE Calcium Channel Type L, Benzothiazepine 71% 18.034uM 16.03uM View
calcium channel, voltage-dependent, L type, alpha 1D subunit MICONAZOLE Calcium Channel Type L, Benzothiazepine 71% 18.034uM 16.03uM View
calcium channel, voltage-dependent, L type, alpha 1C subunit MICONAZOLE Calcium Channel Type L, Benzothiazepine 71% 18.034uM 16.03uM View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit MICONAZOLE Calcium Channel Type L, Benzothiazepine 71% 18.034uM 16.03uM View
calcium channel, voltage-dependent, beta 1 subunit MICONAZOLE Calcium Channel Type L, Benzothiazepine 71% 18.034uM 16.03uM View
calcium channel, voltage-dependent, L type, alpha 1E subunit MICONAZOLE Calcium Channel Type L, Benzothiazepine 71% 18.034uM 16.03uM View
calcium channel, voltage-dependent, N type, alpha 1B subunit MICONAZOLE Calcium Channel Type L, Benzothiazepine 71% 18.034uM 16.03uM View
calcium channel, voltage-dependent, alpha2/delta subunit 1 MICONAZOLE Calcium Channel Type L, Benzothiazepine 71% 18.034uM 16.03uM View
sodium channel, nonvoltage-gated 1 alpha AMOXAPINE Sodium Channel, Site 2 69% NoneNone NoneNone View
sodium channel, voltage-gated, type X, alpha AMOXAPINE Sodium Channel, Site 2 69% NoneNone NoneNone View
sodium channel, voltage-gated, type IX, alpha AMOXAPINE Sodium Channel, Site 2 69% NoneNone NoneNone View
sodium channel, voltage gated, type VIII, alpha AMOXAPINE Sodium Channel, Site 2 69% NoneNone NoneNone View
sodium channel, voltage-gated, type VII, alpha AMOXAPINE Sodium Channel, Site 2 69% NoneNone NoneNone View
sodium channel, voltage-gated, type V, alpha (long QT syndrome 3) AMOXAPINE Sodium Channel, Site 2 69% NoneNone NoneNone View
sodium channel, voltage-gated, type IV, beta AMOXAPINE Sodium Channel, Site 2 69% NoneNone NoneNone View
sodium channel, voltage-gated, type IV, alpha AMOXAPINE Sodium Channel, Site 2 69% NoneNone NoneNone View
sodium channel, voltage-gated, type III, alpha AMOXAPINE Sodium Channel, Site 2 69% NoneNone NoneNone View
sodium channel, voltage-gated, type II, beta AMOXAPINE Sodium Channel, Site 2 69% NoneNone NoneNone View
sodium channel, voltage-gated, type II, alpha 2 AMOXAPINE Sodium Channel, Site 2 69% NoneNone NoneNone View
sodium channel, voltage-gated, type I, beta AMOXAPINE Sodium Channel, Site 2 69% NoneNone NoneNone View
sodium channel, voltage-gated, type I, alpha AMOXAPINE Sodium Channel, Site 2 69% NoneNone NoneNone View
sodium channel, voltage-gated, type IV, beta AMOXAPINE Sodium Channel, Site 2 69% NoneNone NoneNone View
sodium channel associated protein 1 AMOXAPINE Sodium Channel, Site 2 69% NoneNone NoneNone View
5-hydroxytryptamine (serotonin) receptor 2C CHLOROXYLENOL Serotonin 5-HT2C 69% NoneNone NoneNone View
nuclear receptor subfamily 3, group C, member 1 PREGNENOLONE-16ALPHA-CARBONITRILE Glucocorticoid 69% 13.957uM 6.344uM View
adrenergic receptor, alpha 1b ERGONOVINE Adrenergic alpha1B 69% NoneNone NoneNone View
androgen receptor FLUOCINONIDE Testosterone 69% NoneNone NoneNone View
calcium channel, voltage-dependent, L type, alpha 1D subunit FLUOXETINE Calcium Channel Type L, Dihydropyridine 69% NoneNone NoneNone View
calcium channel, voltage-dependent, L type, alpha 1C subunit FLUOXETINE Calcium Channel Type L, Dihydropyridine 69% NoneNone NoneNone View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit FLUOXETINE Calcium Channel Type L, Dihydropyridine 69% NoneNone NoneNone View
calcium channel, voltage-dependent, beta 1 subunit FLUOXETINE Calcium Channel Type L, Dihydropyridine 69% NoneNone NoneNone View
calcium channel, voltage-dependent, L type, alpha 1E subunit FLUOXETINE Calcium Channel Type L, Dihydropyridine 69% NoneNone NoneNone View
calcium channel, voltage-dependent, N type, alpha 1B subunit FLUOXETINE Calcium Channel Type L, Dihydropyridine 69% NoneNone NoneNone View
calcium channel, voltage-dependent, alpha2/delta subunit 1 FLUOXETINE Calcium Channel Type L, Dihydropyridine 69% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 8 FLUOXETINE Calcium Channel Type L, Dihydropyridine 69% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 7 FLUOXETINE Calcium Channel Type L, Dihydropyridine 69% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 6 FLUOXETINE Calcium Channel Type L, Dihydropyridine 69% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 5 FLUOXETINE Calcium Channel Type L, Dihydropyridine 69% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 4 FLUOXETINE Calcium Channel Type L, Dihydropyridine 69% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 3 FLUOXETINE Calcium Channel Type L, Dihydropyridine 69% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 2 FLUOXETINE Calcium Channel Type L, Dihydropyridine 69% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 1 FLUOXETINE Calcium Channel Type L, Dihydropyridine 69% NoneNone NoneNone View
calcium channel, voltage-dependent, beta 4 subunit FLUOXETINE Calcium Channel Type L, Dihydropyridine 69% NoneNone NoneNone View
calcium channel, voltage-dependent, beta 3 subunit FLUOXETINE Calcium Channel Type L, Dihydropyridine 69% NoneNone NoneNone View
calcium channel, voltage-dependent, beta 2 subunit FLUOXETINE Calcium Channel Type L, Dihydropyridine 69% NoneNone NoneNone View
calcium channel, voltage-dependent, L type, alpha 1S subunit FLUOXETINE Calcium Channel Type L, Dihydropyridine 69% NoneNone NoneNone View
calcium channel, voltage-dependent, alpha 1F subunit FLUOXETINE Calcium Channel Type L, Dihydropyridine 69% NoneNone NoneNone View
epidermal growth factor receptor FLUPHENAZINE Protein Tyrosine Kinase, EGF Receptor 69% 40.107uM NoneNone View
calcium channel, voltage-dependent, gamma subunit 8 DOXEPIN Calcium Channel Type L, Benzothiazepine 69% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 7 DOXEPIN Calcium Channel Type L, Benzothiazepine 69% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 6 DOXEPIN Calcium Channel Type L, Benzothiazepine 69% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 5 DOXEPIN Calcium Channel Type L, Benzothiazepine 69% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 4 DOXEPIN Calcium Channel Type L, Benzothiazepine 69% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 3 DOXEPIN Calcium Channel Type L, Benzothiazepine 69% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 2 DOXEPIN Calcium Channel Type L, Benzothiazepine 69% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 1 DOXEPIN Calcium Channel Type L, Benzothiazepine 69% NoneNone NoneNone View
calcium channel, voltage-dependent, beta 4 subunit DOXEPIN Calcium Channel Type L, Benzothiazepine 69% NoneNone NoneNone View
calcium channel, voltage-dependent, beta 3 subunit DOXEPIN Calcium Channel Type L, Benzothiazepine 69% NoneNone NoneNone View
calcium channel, voltage-dependent, beta 2 subunit DOXEPIN Calcium Channel Type L, Benzothiazepine 69% NoneNone NoneNone View
calcium channel, voltage-dependent, L type, alpha 1S subunit DOXEPIN Calcium Channel Type L, Benzothiazepine 69% NoneNone NoneNone View
calcium channel, voltage-dependent, L type, alpha 1C subunit DEXTROMETHORPHAN Calcium Channel Type L, Benzothiazepine 66% NoneNone NoneNone View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit DEXTROMETHORPHAN Calcium Channel Type L, Benzothiazepine 66% NoneNone NoneNone View
calcium channel, voltage-dependent, beta 1 subunit DEXTROMETHORPHAN Calcium Channel Type L, Benzothiazepine 66% NoneNone NoneNone View
calcium channel, voltage-dependent, L type, alpha 1E subunit DEXTROMETHORPHAN Calcium Channel Type L, Benzothiazepine 66% NoneNone NoneNone View
calcium channel, voltage-dependent, N type, alpha 1B subunit DEXTROMETHORPHAN Calcium Channel Type L, Benzothiazepine 66% NoneNone NoneNone View
calcium channel, voltage-dependent, alpha2/delta subunit 1 DEXTROMETHORPHAN Calcium Channel Type L, Benzothiazepine 66% NoneNone NoneNone View
solute carrier family 6 (neurotransmitter transporter, serotonin), member 4 LABETALOL Serotonin Transporter 66% NoneNone NoneNone View
adrenergic receptor, beta 2 BROMOCRIPTINE Adrenergic beta2 66% NoneNone NoneNone View
prostaglandin-endoperoxide synthase 1 ISOEUGENOL Cyclooxygenase COX-1 66% NoneNone NoneNone View
prostaglandin-endoperoxide synthase 1 (prostaglandin G/H synthase and cyclooxygenase) ISOEUGENOL Cyclooxygenase COX-1 66% NoneNone NoneNone View
chemokine (C-C motif) receptor 2 CISPLATIN Chemokine CCR2B 66% 18.142uM 7.012uM View
5-hydroxytryptamine (serotonin) receptor 2A LOPERAMIDE Serotonin 5-HT2A 66% NoneNone NoneNone View
A3 adenosine receptor N,N'-DIPHENYL-P-PHENYLENEDIAMINE Adenosine A3 66% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 8 ITRACONAZOLE Calcium Channel Type L, Dihydropyridine 66% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 7 ITRACONAZOLE Calcium Channel Type L, Dihydropyridine 66% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 6 ITRACONAZOLE Calcium Channel Type L, Dihydropyridine 66% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 5 ITRACONAZOLE Calcium Channel Type L, Dihydropyridine 66% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 4 ITRACONAZOLE Calcium Channel Type L, Dihydropyridine 66% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 3 ITRACONAZOLE Calcium Channel Type L, Dihydropyridine 66% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 2 ITRACONAZOLE Calcium Channel Type L, Dihydropyridine 66% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 1 ITRACONAZOLE Calcium Channel Type L, Dihydropyridine 66% NoneNone NoneNone View
calcium channel, voltage-dependent, beta 4 subunit ITRACONAZOLE Calcium Channel Type L, Dihydropyridine 66% NoneNone NoneNone View
calcium channel, voltage-dependent, beta 3 subunit ITRACONAZOLE Calcium Channel Type L, Dihydropyridine 66% NoneNone NoneNone View
calcium channel, voltage-dependent, beta 2 subunit ITRACONAZOLE Calcium Channel Type L, Dihydropyridine 66% NoneNone NoneNone View
calcium channel, voltage-dependent, L type, alpha 1S subunit ITRACONAZOLE Calcium Channel Type L, Dihydropyridine 66% NoneNone NoneNone View
calcium channel, voltage-dependent, alpha 1F subunit ITRACONAZOLE Calcium Channel Type L, Dihydropyridine 66% NoneNone NoneNone View
calcium channel, voltage-dependent, L type, alpha 1D subunit ITRACONAZOLE Calcium Channel Type L, Dihydropyridine 66% NoneNone NoneNone View
calcium channel, voltage-dependent, L type, alpha 1C subunit ITRACONAZOLE Calcium Channel Type L, Dihydropyridine 66% NoneNone NoneNone View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit ITRACONAZOLE Calcium Channel Type L, Dihydropyridine 66% NoneNone NoneNone View
calcium channel, voltage-dependent, beta 1 subunit ITRACONAZOLE Calcium Channel Type L, Dihydropyridine 66% NoneNone NoneNone View
calcium channel, voltage-dependent, L type, alpha 1E subunit ITRACONAZOLE Calcium Channel Type L, Dihydropyridine 66% NoneNone NoneNone View
calcium channel, voltage-dependent, N type, alpha 1B subunit ITRACONAZOLE Calcium Channel Type L, Dihydropyridine 66% NoneNone NoneNone View
calcium channel, voltage-dependent, alpha2/delta subunit 1 ITRACONAZOLE Calcium Channel Type L, Dihydropyridine 66% NoneNone NoneNone View
Sigma-2 Receptor IRINOTECAN Sigma2 66% NoneNone NoneNone View
adrenergic receptor, alpha 2a IMIQUIMOD Adrenergic alpha2A 66% NoneNone NoneNone View
opioid receptor, kappa 1 RITONAVIR Opiate kappa 66% 13.655uM 5.462uM View
Sigma-2 Receptor NORETHINDRONE ACETATE Sigma2 66% NoneNone NoneNone View
v-erb-b2 erythroblastic leukemia viral oncogene homolog 2, neuro/glioblastoma derived oncogene homolog (avian) OXICONAZOLE Protein Tyrosine Kinase, HER2 Receptor 66% NoneNone NoneNone View
v-erb-b2 erythroblastic leukemia viral oncogene homolog 2, neuro/glioblastoma derived oncogene homolog (avian) OXICONAZOLE Protein Tyrosine Kinase, HER2 Receptor 66% NoneNone NoneNone View
mitogen activated protein kinase 14 EPALRESTAT Protein Serine/Threonine Kinase, p38alpha 66% NoneNone NoneNone View
mitogen-activated protein kinase 14 EPALRESTAT Protein Serine/Threonine Kinase, p38alpha 66% NoneNone NoneNone View
opioid receptor, sigma 1 ORPHENADRINE Sigma1 66% NoneNone NoneNone View
arachidonate 15-lipoxygenase, second type RESVERATROL Lipoxygenase 15-LO 66% NoneNone NoneNone View
arachidonate 15-lipoxygenase RESVERATROL Lipoxygenase 15-LO 66% NoneNone NoneNone View
arachidonate 15-lipoxygenase RESVERATROL Lipoxygenase 15-LO 66% NoneNone NoneNone View
Sigma-2 Receptor CETYLPYRIDINIUM BROMIDE Sigma2 66% NoneNone NoneNone View
cholinergic receptor, muscarinic 5 RALOXIFENE Muscarinic M5 66% NoneNone NoneNone View
solute carrier family 6 (neurotransmitter transporter, dopamine), member 3 DIPHENHYDRAMINE Dopamine Transporter 66% NoneNone NoneNone View
mu-opioid receptor MOR HALOPROGIN Opiate mu 66% NoneNone NoneNone View
chemokine (C-C motif) receptor 5 DISULFIRAM Chemokine CCR5 66% 23.661uM 18.284uM View
ATPase, Na+/K+ transporting, beta 1 polypeptide MICONAZOLE ATPase, Na+/K+ 66% 19.279uM NoneNone View
ATPase, Na+/K+ transporting, beta 3 polypeptide MICONAZOLE ATPase, Na+/K+ 66% 19.279uM NoneNone View
ATPase, Na+/K+ transporting, beta 2 polypeptide MICONAZOLE ATPase, Na+/K+ 66% 19.279uM NoneNone View
histamine receptor H 2 DEXCHLORPHENIRAMINE Histamine H2 71% 8.368uM 8.228uM View
thromboxane A synthase 1 ERGOCORNINE Thromboxane Synthetase 71% 1.993uM NoneNone View
thromboxane A synthase 1 (platelet, cytochrome P450, family 5, subfamily A) ERGOCORNINE Thromboxane Synthetase 71% 1.993uM NoneNone View
5-hydroxytryptamine (serotonin) receptor 2A SULCONAZOLE Serotonin 5-HT2A 71% 3.929uM 1.122uM View
5-hydroxytryptamine (serotonin) receptor 2C SULCONAZOLE Serotonin 5-HT2C 71% 2.785uM 1.459uM View
Cytochrom P450-2C19 monooxygenase MC 258714 CYP450-2C19 Inhibition 71% 3uM NoneNone View
Cytochrom P450-2D6 monooxygenase CELECOXIB CYP450-2D6 Inhibition 71% 1uM NoneNone View
5-hydroxytryptamine (serotonin) receptor 2C U-78517F Serotonin 5-HT2C 71% 7.563uM 3.962uM View
cholinergic receptor, muscarinic 2 AMOXAPINE Muscarinic M2 71% 2.623uM .933uM View
endothelin receptor type A AMIODARONE Endothelin ETA 71% 26.288uM 16.177uM View