| 5-hydroxytryptamine (serotonin) receptor 2A | GUANFACINE | Serotonin 5-HT2A | 75% | 3.014uM | .861uM | View | 
          
            
                | potassium voltage-gated channel, subfamily H (eag-related), member 1 | FLUPHENAZINE | Potassium Channel HERG | 75% | 5.7058uM | 4.6746uM | View | 
          
            
                | potassium voltage-gated channel, subfamily H (eag-related), member 1 | FLUPHENAZINE | Potassium Channel HERG | 75% | 5.7058uM | 4.6746uM | View | 
          
            
                | potassium voltage-gated channel, subfamily H, member 8 | FLUPHENAZINE | Potassium Channel HERG | 75% | 5.7058uM | 4.6746uM | View | 
          
            
                | potassium voltage-gated channel, subfamily H (eag-related), member 6 | FLUPHENAZINE | Potassium Channel HERG | 75% | 5.7058uM | 4.6746uM | View | 
          
            
                | potassium voltage-gated channel, subfamily H (eag-related), member 7 | FLUPHENAZINE | Potassium Channel HERG | 75% | 5.7058uM | 4.6746uM | View | 
          
            
                | potassium voltage-gated channel, subfamily H (eag-related), member 2 | FLUPHENAZINE | Potassium Channel HERG | 75% | 5.7058uM | 4.6746uM | View | 
          
            
                | potassium voltage-gated channel, subfamily H (eag-related), member 5 | FLUPHENAZINE | Potassium Channel HERG | 75% | 5.7058uM | 4.6746uM | View | 
          
            
                | potassium voltage-gated channel, subfamily H (eag-related), member 3 | FLUPHENAZINE | Potassium Channel HERG | 75% | 5.7058uM | 4.6746uM | View | 
          
            
                | potassium voltage-gated channel, subfamily H (eag-related), member 4 | FLUPHENAZINE | Potassium Channel HERG | 75% | 5.7058uM | 4.6746uM | View | 
          
            
                | cholinergic receptor, muscarinic 5 | TRANS-PLATINUM(II)DIAMMINE DICHLORIDE | Muscarinic M5 | 75% | 5.9254uM | 4.2571uM | View | 
          
            
                | Cytochrom P450-2D6 monooxygenase | METHAPYRILENE | CYP450-2D6 Inhibition | 75% | 2.7564uM | NoneNone | View | 
          
            
                | Cytochrom P450-1A2 monooxygenase | PROPAFENONE | CYP450-1A2 Inhibition | 75% | 3.292uM | NoneNone | View | 
          
            
                | adrenergic receptor, beta 3 | SULOCTIDIL | Adrenergic beta3 | 75% | 4.9963uM | 3.7472uM | View | 
          
            
                | solute carrier family 6 (neurotransmitter transporter, serotonin), member 4 | LEVOBUNOLOL | Serotonin Transporter | 75% | 4.898uM | 2.602uM | View | 
          
            
                | 5-hydroxytryptamine (serotonin) receptor 2B | DIMENHYDRINATE | Serotonin 5-HT2B | 75% | 1.724uM | 1.097uM | View | 
          
            
                | mitogen activated protein kinase 14 | MONTELUKAST | Protein Serine/Threonine Kinase, p38alpha | 75% | .856uM | NoneNone | View | 
          
            
                | mitogen-activated protein kinase 14 | MONTELUKAST | Protein Serine/Threonine Kinase, p38alpha | 75% | .856uM | NoneNone | View | 
          
            
                | platelet-activating factor receptor | CILOSTAMIDE | Platelet Activating Factor (PAF) | 75% | 3.687uM | 1.917uM | View | 
          
            
                | cholinergic receptor, muscarinic 4 | FLUNARIZINE | Muscarinic M4 | 75% | 5.656uM | .789uM | View | 
          
            
                | dopamine receptor D4 | THIORIDAZINE | Dopamine D4.2 | 75% | 1.468uM | .515uM | View | 
          
            
                | calcium channel, voltage-dependent, L type, alpha 1E subunit | SPIRADOLINE | Calcium Channel Type L, Phenylalkylamine | 78% | 5.24uM | 5.095uM | View | 
          
            
                | calcium channel, voltage-dependent, N type, alpha 1B subunit | SPIRADOLINE | Calcium Channel Type L, Phenylalkylamine | 78% | 5.24uM | 5.095uM | View | 
          
            
                | calcium channel, voltage-dependent, alpha2/delta subunit 1 | SPIRADOLINE | Calcium Channel Type L, Phenylalkylamine | 78% | 5.24uM | 5.095uM | View | 
          
            
                | acetylcholinesterase (YT blood group) | BUTENAFINE | Acetylcholinesterase | 78% | 6.9071uM | NoneNone | View | 
          
            
                | collagen-like tail subunit (single strand of homotrimer) of asymmetric acetylcholinesterase | BUTENAFINE | Acetylcholinesterase | 78% | 6.9071uM | NoneNone | View | 
          
            
                | acetylcholinesterase | BUTENAFINE | Acetylcholinesterase | 78% | 6.9071uM | NoneNone | View | 
          
            
                | cholinergic receptor, muscarinic 1 | QUETIAPINE | Muscarinic M1 | 78% | 2.615uM | .6298uM | View | 
          
            
                | A3 adenosine receptor | VX-745 | Adenosine A3 | 78% | 8.547uM | 4.831uM | View | 
          
            
                | dopamine receptor D3 | TERCONAZOLE | Dopamine D3 | 78% | 4.712uM | 1.6uM | View | 
          
            
                | adrenergic receptor, alpha 2a | SEMUSTINE | Adrenergic alpha2A | 78% | 4.809uM | 1.803uM | View | 
          
            
                | histamine receptor H 1 | METERGOLINE | Histamine H1, Central | 78% | 4.133uM | .48uM | View | 
          
            
                | cholinergic receptor, muscarinic 5 | PENTAMIDINE | Muscarinic M5 | 78% | 2.885uM | 2.073uM | View | 
          
            
                | 5-hydroxytryptamine (serotonin) receptor 2C | PENTAMIDINE | Serotonin 5-HT2C | 78% | 3.278uM | 1.717uM | View | 
          
            
                | adrenergic receptor, alpha 2a | PRAZOSIN | Imidazoline I2, Central | 78% | .949uM | .633uM | View | 
          
            
                | adrenergic receptor, alpha 2c (Non-specific probe) | PRAZOSIN | Imidazoline I2, Central | 78% | .949uM | .633uM | View | 
          
            
                | Protein-tyrosine kinase, Fyn | PROCHLORPERAZINE | Protein Tyrosine Kinase, Fyn | 78% | 5.684uM | NoneNone | View | 
          
            
                | calcium channel, voltage-dependent, gamma subunit 8 | PERGOLIDE | Calcium Channel Type L, Benzothiazepine | 78% | 3.301uM | 2.934uM | View | 
          
            
                | calcium channel, voltage-dependent, gamma subunit 7 | PERGOLIDE | Calcium Channel Type L, Benzothiazepine | 78% | 3.301uM | 2.934uM | View | 
          
            
                | calcium channel, voltage-dependent, gamma subunit 6 | PERGOLIDE | Calcium Channel Type L, Benzothiazepine | 78% | 3.301uM | 2.934uM | View | 
          
            
                | calcium channel, voltage-dependent, gamma subunit 5 | PERGOLIDE | Calcium Channel Type L, Benzothiazepine | 78% | 3.301uM | 2.934uM | View | 
          
            
                | calcium channel, voltage-dependent, gamma subunit 4 | PERGOLIDE | Calcium Channel Type L, Benzothiazepine | 78% | 3.301uM | 2.934uM | View | 
          
            
                | calcium channel, voltage-dependent, gamma subunit 3 | PERGOLIDE | Calcium Channel Type L, Benzothiazepine | 78% | 3.301uM | 2.934uM | View | 
          
            
                | calcium channel, voltage-dependent, gamma subunit 2 | PERGOLIDE | Calcium Channel Type L, Benzothiazepine | 78% | 3.301uM | 2.934uM | View | 
          
            
                | calcium channel, voltage-dependent, gamma subunit 1 | PERGOLIDE | Calcium Channel Type L, Benzothiazepine | 78% | 3.301uM | 2.934uM | View | 
          
            
                | calcium channel, voltage-dependent, beta 4 subunit | PERGOLIDE | Calcium Channel Type L, Benzothiazepine | 78% | 3.301uM | 2.934uM | View | 
          
            
                | calcium channel, voltage-dependent, beta 3 subunit | PERGOLIDE | Calcium Channel Type L, Benzothiazepine | 78% | 3.301uM | 2.934uM | View | 
          
            
                | calcium channel, voltage-dependent, beta 2 subunit | PERGOLIDE | Calcium Channel Type L, Benzothiazepine | 78% | 3.301uM | 2.934uM | View | 
          
            
                | calcium channel, voltage-dependent, L type, alpha 1S subunit | PERGOLIDE | Calcium Channel Type L, Benzothiazepine | 78% | 3.301uM | 2.934uM | View | 
          
            
                | calcium channel, voltage-dependent, alpha 1F subunit | PERGOLIDE | Calcium Channel Type L, Benzothiazepine | 78% | 3.301uM | 2.934uM | View | 
          
            
                | calcium channel, voltage-dependent, L type, alpha 1D subunit | PERGOLIDE | Calcium Channel Type L, Benzothiazepine | 78% | 3.301uM | 2.934uM | View | 
          
            
                | calcium channel, voltage-dependent, L type, alpha 1C subunit | PERGOLIDE | Calcium Channel Type L, Benzothiazepine | 78% | 3.301uM | 2.934uM | View | 
          
            
                | calcium channel, voltage-dependent, P/Q type, alpha 1A subunit | PERGOLIDE | Calcium Channel Type L, Benzothiazepine | 78% | 3.301uM | 2.934uM | View | 
          
            
                | calcium channel, voltage-dependent, beta 1 subunit | PERGOLIDE | Calcium Channel Type L, Benzothiazepine | 78% | 3.301uM | 2.934uM | View | 
          
            
                | Cytochrom P450-2C19 monooxygenase | ROTENONE | CYP450-2C19 Inhibition | 78% | 3.6486uM | NoneNone | View | 
          
            
                | solute carrier family 6 (neurotransmitter transporter, noradrenalin), member 2 | BW-723C86 | Adrenergic, Norepinephrine Transporter | 78% | 3.6257uM | 3.5957uM | View | 
          
            
                | Cytochrom P450-2D6 monooxygenase | CYCLIZINE | CYP450-2D6 Inhibition | 78% | 6.2175uM | NoneNone | View | 
          
            
                | epidermal growth factor receptor | THIORIDAZINE | Protein Tyrosine Kinase, EGF Receptor | 78% | 2.947uM | NoneNone | View | 
          
            
                | mitogen activated protein kinase 14 | ZAFIRLUKAST | Protein Serine/Threonine Kinase, p38alpha | 78% | .353uM | NoneNone | View | 
          
            
                | mitogen-activated protein kinase 14 | ZAFIRLUKAST | Protein Serine/Threonine Kinase, p38alpha | 78% | .353uM | NoneNone | View | 
          
            
                | cholinergic receptor, muscarinic 3 | MONTELUKAST | Muscarinic M3 | 78% | 6.626uM | 1.404uM | View | 
          
            
                | cannabinoid receptor 1 (brain) | FLUNARIZINE | Cannabinoid CB1 | 78% | 3.028uM | 2.391uM | View | 
          
            
                | calcium channel, voltage-dependent, gamma subunit 8 | DIMENHYDRINATE | Calcium Channel Type L, Phenylalkylamine | 78% | 3.344uM | 3.251uM | View | 
          
            
                | calcium channel, voltage-dependent, gamma subunit 7 | DIMENHYDRINATE | Calcium Channel Type L, Phenylalkylamine | 78% | 3.344uM | 3.251uM | View | 
          
            
                | calcium channel, voltage-dependent, gamma subunit 6 | DIMENHYDRINATE | Calcium Channel Type L, Phenylalkylamine | 78% | 3.344uM | 3.251uM | View | 
          
            
                | calcium channel, voltage-dependent, gamma subunit 5 | DIMENHYDRINATE | Calcium Channel Type L, Phenylalkylamine | 78% | 3.344uM | 3.251uM | View | 
          
            
                | calcium channel, voltage-dependent, gamma subunit 4 | DIMENHYDRINATE | Calcium Channel Type L, Phenylalkylamine | 78% | 3.344uM | 3.251uM | View | 
          
            
                | calcium channel, voltage-dependent, gamma subunit 3 | DIMENHYDRINATE | Calcium Channel Type L, Phenylalkylamine | 78% | 3.344uM | 3.251uM | View | 
          
            
                | calcium channel, voltage-dependent, gamma subunit 2 | DIMENHYDRINATE | Calcium Channel Type L, Phenylalkylamine | 78% | 3.344uM | 3.251uM | View | 
          
            
                | calcium channel, voltage-dependent, gamma subunit 1 | DIMENHYDRINATE | Calcium Channel Type L, Phenylalkylamine | 78% | 3.344uM | 3.251uM | View | 
          
            
                | sodium channel, voltage-gated, type III, beta | PROMAZINE | Sodium Channel, Site 2 | 77% | 2.573uM | 2.347uM | View | 
          
            
                | sodium channel, voltage-gated, type VIII, alpha polypeptide | PROMAZINE | Sodium Channel, Site 2 | 77% | 2.573uM | 2.347uM | View | 
          
            
                | 5-hydroxytryptamine (serotonin) receptor 2C | TERCONAZOLE | Serotonin 5-HT2C | 77% | 6.961uM | 3.646uM | View | 
          
            
                | adrenergic receptor, alpha 1d (Non-specific probe) | TERCONAZOLE | Adrenergic alpha1D | 77% | 14.385uM | 7.07uM | View | 
          
            
                | cholinergic receptor, muscarinic 2 | PROCHLORPERAZINE | Muscarinic M2 | 77% | 3.112uM | 1.107uM | View | 
          
            
                | A3 adenosine receptor | TROGLITAZONE | Adenosine A3 | 77% | 5.208uM | 2.943uM | View | 
          
            
                | adrenergic receptor, alpha 1d (Non-specific probe) | ECONAZOLE | Adrenergic alpha1D | 77% | 8.897uM | 4.373uM | View | 
          
            
                | calcium channel, voltage-dependent, gamma subunit 8 | SULCONAZOLE | Calcium Channel Type L, Dihydropyridine | 77% | 2.427uM | 1.56uM | View | 
          
            
                | calcium channel, voltage-dependent, gamma subunit 7 | SULCONAZOLE | Calcium Channel Type L, Dihydropyridine | 77% | 2.427uM | 1.56uM | View | 
          
            
                | calcium channel, voltage-dependent, gamma subunit 6 | SULCONAZOLE | Calcium Channel Type L, Dihydropyridine | 77% | 2.427uM | 1.56uM | View | 
          
            
                | calcium channel, voltage-dependent, gamma subunit 5 | SULCONAZOLE | Calcium Channel Type L, Dihydropyridine | 77% | 2.427uM | 1.56uM | View | 
          
            
                | calcium channel, voltage-dependent, gamma subunit 4 | SULCONAZOLE | Calcium Channel Type L, Dihydropyridine | 77% | 2.427uM | 1.56uM | View | 
          
            
                | Protein-tyrosine kinase, Fyn | BETA-NAPHTHOFLAVONE | Protein Tyrosine Kinase, Fyn | 77% | 2.5149uM | NoneNone | View | 
          
            
                | epidermal growth factor receptor | PERHEXILINE | Protein Tyrosine Kinase, EGF Receptor | 77% | 1.4852uM | NoneNone | View | 
          
            
                | Cytochrom P450-2C19 monooxygenase | BUPROPION | CYP450-2C19 Inhibition | 77% | 1.9983uM | NoneNone | View | 
          
            
                | 5-hydroxytryptamine receptor 6 | PROPAFENONE | Serotonin 5-HT6 | 77% | 1.863uM | .865uM | View | 
          
            
                | solute carrier family 6 (neurotransmitter transporter, serotonin), member 4 | AMBROXOL | Serotonin Transporter | 77% | 3.391uM | 1.802uM | View | 
          
            
                | Protein-tyrosine kinase, Fyn | TERFENADINE | Protein Tyrosine Kinase, Fyn | 77% | 6.123uM | NoneNone | View | 
          
            
                | mu-opioid receptor MOR | DOMPERIDONE | Opiate mu | 77% | 4.218uM | 1.712uM | View | 
          
            
                | histamine receptor H 2 | IMATINIB | Histamine H2 | 77% | 1.963uM | 1.93uM | View | 
          
            
                | dopamine receptor D3 | CYCLIZINE | Dopamine D3 | 77% | 2.992uM | 1.016uM | View | 
          
            
                | Cytochrom P450-2D6 monooxygenase | LOPERAMIDE | CYP450-2D6 Inhibition | 77% | 2uM | NoneNone | View | 
          
            
                | Cytochrom P450-2C19 monooxygenase | ETHYLESTRENOL | CYP450-2C19 Inhibition | 77% | 1.2907uM | NoneNone | View | 
          
            
                | Cytochrom P450-2C19 monooxygenase | RAPAMYCIN | CYP450-2C19 Inhibition | 77% | 4uM | NoneNone | View | 
          
            
                | Cytochrom P450-2C19 monooxygenase | RESVERATROL | CYP450-2C19 Inhibition | 77% | 3uM | NoneNone | View | 
          
            
                | A3 adenosine receptor | HYDROXYPROGESTERONE | Adenosine A3 | 77% | 4.73uM | 2.674uM | View | 
          
            
                | 5-hydroxytryptamine (serotonin) receptor 2A | DIPHENIDOL | Serotonin 5-HT2A | 77% | 2.586uM | .739uM | View | 
          
            
                | estrogen receptor 1 | ETHYLESTRENOL | Estrogen ERalpha | 77% | 1.121uM | .32uM | View | 
          
            
                | estrogen receptor 1 | ETHYLESTRENOL | Estrogen ERalpha | 77% | 1.121uM | .32uM | View | 
          
            
                | adrenergic receptor, alpha 2a | MOXONIDINE | Imidazoline I2, Central | 77% | 1.4764uM | .9843uM | View | 
          
            
                | adrenergic receptor, alpha 2c (Non-specific probe) | MOXONIDINE | Imidazoline I2, Central | 77% | 1.4764uM | .9843uM | View | 
          
            
                | Protein-tyrosine kinase, Fyn | METHYLDOPA | Protein Tyrosine Kinase, Fyn | 77% | 5.176uM | NoneNone | View | 
          
            
                | calcium channel, voltage-dependent, gamma subunit 8 | LISURIDE | Calcium Channel Type L, Benzothiazepine | 77% | 3.522uM | 3.131uM | View | 
          
            
                | calcium channel, voltage-dependent, gamma subunit 7 | LISURIDE | Calcium Channel Type L, Benzothiazepine | 77% | 3.522uM | 3.131uM | View | 
          
            
                | calcium channel, voltage-dependent, gamma subunit 6 | LISURIDE | Calcium Channel Type L, Benzothiazepine | 77% | 3.522uM | 3.131uM | View | 
          
            
                | calcium channel, voltage-dependent, gamma subunit 5 | LISURIDE | Calcium Channel Type L, Benzothiazepine | 77% | 3.522uM | 3.131uM | View | 
          
            
                | calcium channel, voltage-dependent, gamma subunit 4 | LISURIDE | Calcium Channel Type L, Benzothiazepine | 77% | 3.522uM | 3.131uM | View | 
          
            
                | calcium channel, voltage-dependent, gamma subunit 3 | LISURIDE | Calcium Channel Type L, Benzothiazepine | 77% | 3.522uM | 3.131uM | View | 
          
            
                | calcium channel, voltage-dependent, gamma subunit 2 | LISURIDE | Calcium Channel Type L, Benzothiazepine | 77% | 3.522uM | 3.131uM | View | 
          
            
                | calcium channel, voltage-dependent, gamma subunit 1 | LISURIDE | Calcium Channel Type L, Benzothiazepine | 77% | 3.522uM | 3.131uM | View | 
          
            
                | calcium channel, voltage-dependent, beta 4 subunit | LISURIDE | Calcium Channel Type L, Benzothiazepine | 77% | 3.522uM | 3.131uM | View | 
          
            
                | calcium channel, voltage-dependent, beta 3 subunit | LISURIDE | Calcium Channel Type L, Benzothiazepine | 77% | 3.522uM | 3.131uM | View | 
          
            
                | calcium channel, voltage-dependent, beta 2 subunit | LISURIDE | Calcium Channel Type L, Benzothiazepine | 77% | 3.522uM | 3.131uM | View | 
          
            
                | calcium channel, voltage-dependent, L type, alpha 1S subunit | LISURIDE | Calcium Channel Type L, Benzothiazepine | 77% | 3.522uM | 3.131uM | View | 
          
            
                | calcium channel, voltage-dependent, alpha 1F subunit | LISURIDE | Calcium Channel Type L, Benzothiazepine | 77% | 3.522uM | 3.131uM | View | 
          
            
                | calcium channel, voltage-dependent, L type, alpha 1D subunit | LISURIDE | Calcium Channel Type L, Benzothiazepine | 77% | 3.522uM | 3.131uM | View | 
          
            
                | calcium channel, voltage-dependent, L type, alpha 1C subunit | LISURIDE | Calcium Channel Type L, Benzothiazepine | 77% | 3.522uM | 3.131uM | View | 
          
            
                | calcium channel, voltage-dependent, P/Q type, alpha 1A subunit | LISURIDE | Calcium Channel Type L, Benzothiazepine | 77% | 3.522uM | 3.131uM | View | 
          
            
                | calcium channel, voltage-dependent, beta 1 subunit | LISURIDE | Calcium Channel Type L, Benzothiazepine | 77% | 3.522uM | 3.131uM | View | 
          
            
                | calcium channel, voltage-dependent, L type, alpha 1E subunit | LISURIDE | Calcium Channel Type L, Benzothiazepine | 77% | 3.522uM | 3.131uM | View | 
          
            
                | calcium channel, voltage-dependent, N type, alpha 1B subunit | LISURIDE | Calcium Channel Type L, Benzothiazepine | 77% | 3.522uM | 3.131uM | View | 
          
            
                | calcium channel, voltage-dependent, alpha2/delta subunit 1 | LISURIDE | Calcium Channel Type L, Benzothiazepine | 77% | 3.522uM | 3.131uM | View | 
          
            
                | epidermal growth factor receptor | TERFENADINE | Protein Tyrosine Kinase, EGF Receptor | 76% | 3.566uM | NoneNone | View | 
          
            
                | epidermal growth factor receptor | ZAFIRLUKAST | Protein Tyrosine Kinase, EGF Receptor | 76% | 5.751uM | NoneNone | View | 
          
            
                | angiotensin 1 converting enzyme 1 | IODOQUINOL | Protease, Angiotensin Converting Enzyme | 76% | .906uM | NoneNone | View | 
          
            
                | angiotensin I converting enzyme (peptidyl-dipeptidase A) 1 | IODOQUINOL | Protease, Angiotensin Converting Enzyme | 76% | .906uM | NoneNone | View | 
          
            
                | nitric oxide synthase 3 (endothelial cell) | CHLORZOXAZONE | Nitric Oxide Synthase, Constitutive (cNOS) | 76% | 2.794uM | NoneNone | View | 
          
            
                | nitric oxide synthase 3, endothelial cell | CHLORZOXAZONE | Nitric Oxide Synthase, Constitutive (cNOS) | 76% | 2.794uM | NoneNone | View | 
          
            
                | cholinergic receptor, muscarinic 4 | CINNARIZINE | Muscarinic M4 | 76% | 3.66uM | .51uM | View | 
          
            
                | Cytochrome P450, subfamily IIC (mephenytoin 4-hydroxylase) | ALPHA-ERGOCRYPTINE | CYP450-2C9 Inhibition | 76% | 6uM | NoneNone | View | 
          
            
                | cytochrome P450, family 2, subfamily C, polypeptide 9 | ALPHA-ERGOCRYPTINE | CYP450-2C9 Inhibition | 76% | 6uM | NoneNone | View | 
          
            
                | Cytochrome P450, subfamily IIC (mephenytoin 4-hydroxylase) | RWJ-68354 | CYP450-2C9 Inhibition | 76% | 1uM | NoneNone | View | 
          
            
                | cytochrome P450, family 2, subfamily C, polypeptide 9 | RWJ-68354 | CYP450-2C9 Inhibition | 76% | 1uM | NoneNone | View | 
          
            
                | Cytochrome P450, subfamily IIC (mephenytoin 4-hydroxylase) | PHENYLHYDRAZINE | CYP450-2C9 Inhibition | 76% | 6uM | NoneNone | View | 
          
            
                | cytochrome P450, family 2, subfamily C, polypeptide 9 | PHENYLHYDRAZINE | CYP450-2C9 Inhibition | 76% | 6uM | NoneNone | View | 
          
            
                | Cytochrom P450-2C19 monooxygenase | NOSCAPINE | CYP450-2C19 Inhibition | 76% | .4003uM | NoneNone | View | 
          
            
                | adrenergic receptor, alpha 2b | BERBERINE CHLORIDE | Adrenergic alpha2C | 76% | 2.837uM | .412uM | View | 
          
            
                | adrenergic receptor, alpha 2c (Non-specific probe) | BERBERINE CHLORIDE | Adrenergic alpha2C | 76% | 2.837uM | .412uM | View | 
          
            
                | phosphodiesterase 3B | MILRINONE | Phosphodiesterase PDE3 | 76% | .9585uM | NoneNone | View | 
          
            
                | phosphodiesterase 3A | MILRINONE | Phosphodiesterase PDE3 | 76% | .9585uM | NoneNone | View | 
          
            
                | melanocortin 5 receptor | DIGITONIN | Melanocortin MC5 | 76% | 3.88uM | 3.639uM | View | 
          
            
                | sodium channel, voltage-gated, type IV, beta | MAPROTILINE | Sodium Channel, Site 2 | 76% | 2.572uM | 2.346uM | View | 
          
            
                | sodium channel associated protein 1 | MAPROTILINE | Sodium Channel, Site 2 | 76% | 2.572uM | 2.346uM | View | 
          
            
                | sodium channel associated protein 2 | MAPROTILINE | Sodium Channel, Site 2 | 76% | 2.572uM | 2.346uM | View | 
          
            
                | sodium channel, voltage-gated, type III, beta | MAPROTILINE | Sodium Channel, Site 2 | 76% | 2.572uM | 2.346uM | View | 
          
            
                | sodium channel, voltage-gated, type I, alpha | MAPROTILINE | Sodium Channel, Site 2 | 76% | 2.572uM | 2.346uM | View | 
          
            
                | sodium channel, voltage-gated, type IX, alpha | MAPROTILINE | Sodium Channel, Site 2 | 76% | 2.572uM | 2.346uM | View | 
          
            
                | sodium channel, voltage-gated, type VII, alpha | MAPROTILINE | Sodium Channel, Site 2 | 76% | 2.572uM | 2.346uM | View | 
          
            
                | amiloride-sensitive cation channel 5, intestinal | MAPROTILINE | Sodium Channel, Site 2 | 76% | 2.572uM | 2.346uM | View | 
          
            
                | sodium channel, voltage-gated, type III, beta | MAPROTILINE | Sodium Channel, Site 2 | 76% | 2.572uM | 2.346uM | View | 
          
            
                | sodium channel, voltage-gated, type VIII, alpha polypeptide | MAPROTILINE | Sodium Channel, Site 2 | 76% | 2.572uM | 2.346uM | View | 
          
            
                | sodium channel, voltage-gated, type XI, alpha | MAPROTILINE | Sodium Channel, Site 2 | 76% | 2.572uM | 2.346uM | View | 
          
            
                | sodium channel, voltage-gated, type I, beta | MAPROTILINE | Sodium Channel, Site 2 | 76% | 2.572uM | 2.346uM | View | 
          
            
                | sodium channel, voltage-gated, type 10, alpha polypeptide | MAPROTILINE | Sodium Channel, Site 2 | 76% | 2.572uM | 2.346uM | View | 
          
            
                | sodium channel, voltage-gated, type IV, alpha polypeptide | MAPROTILINE | Sodium Channel, Site 2 | 76% | 2.572uM | 2.346uM | View | 
          
            
                | sodium channel, voltage-gated, type V, alpha polypeptide | MAPROTILINE | Sodium Channel, Site 2 | 76% | 2.572uM | 2.346uM | View | 
          
            
                | sodium channel, voltage-gated, type II, beta | MAPROTILINE | Sodium Channel, Site 2 | 76% | 2.572uM | 2.346uM | View | 
          
            
                | sodium channel, nonvoltage-gated 1 alpha | MAPROTILINE | Sodium Channel, Site 2 | 76% | 2.572uM | 2.346uM | View | 
          
            
                | sodium channel, nonvoltage-gated 1 gamma | MAPROTILINE | Sodium Channel, Site 2 | 76% | 2.572uM | 2.346uM | View | 
          
            
                | sodium channel, nonvoltage-gated 1 beta | MAPROTILINE | Sodium Channel, Site 2 | 76% | 2.572uM | 2.346uM | View | 
          
            
                | sodium channel, voltage-gated, type 2, alpha 1 polypeptide | MAPROTILINE | Sodium Channel, Site 2 | 76% | 2.572uM | 2.346uM | View | 
          
            
                | sodium channel, voltage-gated, type XI, alpha | MAPROTILINE | Sodium Channel, Site 2 | 76% | 2.572uM | 2.346uM | View | 
          
            
                | sodium channel, nonvoltage-gated 1, gamma | MAPROTILINE | Sodium Channel, Site 2 | 76% | 2.572uM | 2.346uM | View | 
          
            
                | sodium channel, nonvoltage-gated 1, delta | MAPROTILINE | Sodium Channel, Site 2 | 76% | 2.572uM | 2.346uM | View | 
          
            
                | sodium channel, nonvoltage-gated 1, beta (Liddle syndrome) | MAPROTILINE | Sodium Channel, Site 2 | 76% | 2.572uM | 2.346uM | View | 
          
            
                | sodium channel, nonvoltage-gated 1 alpha | MAPROTILINE | Sodium Channel, Site 2 | 76% | 2.572uM | 2.346uM | View | 
          
            
                | sodium channel, voltage-gated, type X, alpha | MAPROTILINE | Sodium Channel, Site 2 | 76% | 2.572uM | 2.346uM | View | 
          
            
                | sodium channel, voltage-gated, type IX, alpha | MAPROTILINE | Sodium Channel, Site 2 | 76% | 2.572uM | 2.346uM | View | 
          
            
                | sodium channel, voltage gated, type VIII, alpha | MAPROTILINE | Sodium Channel, Site 2 | 76% | 2.572uM | 2.346uM | View | 
          
            
                | sodium channel, voltage-gated, type VII, alpha | MAPROTILINE | Sodium Channel, Site 2 | 76% | 2.572uM | 2.346uM | View | 
          
            
                | sodium channel, voltage-gated, type V, alpha (long QT syndrome 3) | MAPROTILINE | Sodium Channel, Site 2 | 76% | 2.572uM | 2.346uM | View | 
          
            
                | sodium channel, voltage-gated, type IV, beta | MAPROTILINE | Sodium Channel, Site 2 | 76% | 2.572uM | 2.346uM | View | 
          
            
                | sodium channel, voltage-gated, type IV, alpha | MAPROTILINE | Sodium Channel, Site 2 | 76% | 2.572uM | 2.346uM | View | 
          
            
                | sodium channel, voltage-gated, type III, alpha | MAPROTILINE | Sodium Channel, Site 2 | 76% | 2.572uM | 2.346uM | View | 
          
            
                | sodium channel, voltage-gated, type II, beta | MAPROTILINE | Sodium Channel, Site 2 | 76% | 2.572uM | 2.346uM | View | 
          
            
                | solute carrier family 6 (neurotransmitter transporter, dopamine), member 3 | CLEMASTINE | Dopamine Transporter | 89% | .678uM | .538uM | View | 
          
            
                | adrenergic receptor, alpha 1d (Non-specific probe) | CLEMASTINE | Adrenergic alpha1D | 89% | .032uM | .015uM | View | 
          
            
                | 5-hydroxytryptamine (serotonin) receptor 1B | CLEMASTINE | Serotonin 5-HT1B | 89% | .359uM | .22uM | View | 
          
            
                | calcium channel, voltage-dependent, gamma subunit 4 | CLEMASTINE | Calcium Channel Type L, Phenylalkylamine | 89% | .508uM | .493uM | View | 
          
            
                | calcium channel, voltage-dependent, gamma subunit 3 | CLEMASTINE | Calcium Channel Type L, Phenylalkylamine | 89% | .508uM | .493uM | View | 
          
            
                | calcium channel, voltage-dependent, gamma subunit 2 | CLEMASTINE | Calcium Channel Type L, Phenylalkylamine | 89% | .508uM | .493uM | View | 
          
            
                | calcium channel, voltage-dependent, gamma subunit 1 | CLEMASTINE | Calcium Channel Type L, Phenylalkylamine | 89% | .508uM | .493uM | View | 
          
            
                | calcium channel, voltage-dependent, beta 4 subunit | CLEMASTINE | Calcium Channel Type L, Phenylalkylamine | 89% | .508uM | .493uM | View | 
          
            
                | calcium channel, voltage-dependent, beta 3 subunit | CLEMASTINE | Calcium Channel Type L, Phenylalkylamine | 89% | .508uM | .493uM | View | 
          
            
                | calcium channel, voltage-dependent, beta 2 subunit | CLEMASTINE | Calcium Channel Type L, Phenylalkylamine | 89% | .508uM | .493uM | View | 
          
            
                | calcium channel, voltage-dependent, L type, alpha 1S subunit | CLEMASTINE | Calcium Channel Type L, Phenylalkylamine | 89% | .508uM | .493uM | View | 
          
            
                | calcium channel, voltage-dependent, alpha 1F subunit | CLEMASTINE | Calcium Channel Type L, Phenylalkylamine | 89% | .508uM | .493uM | View | 
          
            
                | calcium channel, voltage-dependent, L type, alpha 1D subunit | CLEMASTINE | Calcium Channel Type L, Phenylalkylamine | 89% | .508uM | .493uM | View | 
          
            
                | calcium channel, voltage-dependent, L type, alpha 1C subunit | CLEMASTINE | Calcium Channel Type L, Phenylalkylamine | 89% | .508uM | .493uM | View | 
          
            
                | calcium channel, voltage-dependent, P/Q type, alpha 1A subunit | CLEMASTINE | Calcium Channel Type L, Phenylalkylamine | 89% | .508uM | .493uM | View | 
          
            
                | calcium channel, voltage-dependent, beta 1 subunit | CLEMASTINE | Calcium Channel Type L, Phenylalkylamine | 89% | .508uM | .493uM | View | 
          
            
                | calcium channel, voltage-dependent, L type, alpha 1E subunit | CLEMASTINE | Calcium Channel Type L, Phenylalkylamine | 89% | .508uM | .493uM | View | 
          
            
                | adrenergic receptor, alpha 2b | DOMPERIDONE | Adrenergic alpha2C | 89% | 1.011uM | .147uM | View | 
          
            
                | adrenergic receptor, alpha 2c (Non-specific probe) | DOMPERIDONE | Adrenergic alpha2C | 89% | 1.011uM | .147uM | View | 
          
            
                | cholinergic receptor, muscarinic 2 | PENTAMIDINE | Muscarinic M2 | 89% | 1.425uM | .507uM | View | 
          
            
                | adrenergic receptor, alpha 2b | EPINEPHRINE | Adrenergic alpha2B | 89% | .869uM | .397uM | View | 
          
            
                | adrenergic receptor, alpha 2a | METOCLOPRAMIDE | Imidazoline I2, Central | 89% | .708uM | .472uM | View | 
          
            
                | adrenergic receptor, alpha 2c (Non-specific probe) | METOCLOPRAMIDE | Imidazoline I2, Central | 89% | .708uM | .472uM | View | 
          
            
                | calcium channel, voltage-dependent, gamma subunit 8 | MICONAZOLE | Calcium Channel Type L, Phenylalkylamine | 89% | 3.788uM | 3.683uM | View | 
          
            
                | calcium channel, voltage-dependent, gamma subunit 7 | MICONAZOLE | Calcium Channel Type L, Phenylalkylamine | 89% | 3.788uM | 3.683uM | View |