Gene Activity List


Gene Activity List

Gene Compound Assay Inh Ic50 Ki View
calcium channel, voltage-dependent, beta 4 subunit SERTRALINE Calcium Channel Type L, Phenylalkylamine 83% 2.1436uM 2.0841uM View
calcium channel, voltage-dependent, beta 3 subunit SERTRALINE Calcium Channel Type L, Phenylalkylamine 83% 2.1436uM 2.0841uM View
calcium channel, voltage-dependent, beta 2 subunit SERTRALINE Calcium Channel Type L, Phenylalkylamine 83% 2.1436uM 2.0841uM View
calcium channel, voltage-dependent, L type, alpha 1S subunit SERTRALINE Calcium Channel Type L, Phenylalkylamine 83% 2.1436uM 2.0841uM View
calcium channel, voltage-dependent, alpha 1F subunit SERTRALINE Calcium Channel Type L, Phenylalkylamine 83% 2.1436uM 2.0841uM View
calcium channel, voltage-dependent, L type, alpha 1D subunit SERTRALINE Calcium Channel Type L, Phenylalkylamine 83% 2.1436uM 2.0841uM View
calcium channel, voltage-dependent, L type, alpha 1C subunit SERTRALINE Calcium Channel Type L, Phenylalkylamine 83% 2.1436uM 2.0841uM View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit SERTRALINE Calcium Channel Type L, Phenylalkylamine 83% 2.1436uM 2.0841uM View
calcium channel, voltage-dependent, beta 1 subunit SERTRALINE Calcium Channel Type L, Phenylalkylamine 83% 2.1436uM 2.0841uM View
calcium channel, voltage-dependent, L type, alpha 1E subunit SERTRALINE Calcium Channel Type L, Phenylalkylamine 83% 2.1436uM 2.0841uM View
calcium channel, voltage-dependent, N type, alpha 1B subunit SERTRALINE Calcium Channel Type L, Phenylalkylamine 83% 2.1436uM 2.0841uM View
calcium channel, voltage-dependent, alpha2/delta subunit 1 SERTRALINE Calcium Channel Type L, Phenylalkylamine 83% 2.1436uM 2.0841uM View
calcium channel, voltage-dependent, gamma subunit 8 NIMODIPINE Calcium Channel Type L, Benzothiazepine 83% .002093uM .00186uM View
calcium channel, voltage-dependent, gamma subunit 7 NIMODIPINE Calcium Channel Type L, Benzothiazepine 83% .002093uM .00186uM View
calcium channel, voltage-dependent, gamma subunit 6 NIMODIPINE Calcium Channel Type L, Benzothiazepine 83% .002093uM .00186uM View
calcium channel, voltage-dependent, gamma subunit 5 NIMODIPINE Calcium Channel Type L, Benzothiazepine 83% .002093uM .00186uM View
calcium channel, voltage-dependent, gamma subunit 4 NIMODIPINE Calcium Channel Type L, Benzothiazepine 83% .002093uM .00186uM View
calcium channel, voltage-dependent, gamma subunit 3 NIMODIPINE Calcium Channel Type L, Benzothiazepine 83% .002093uM .00186uM View
calcium channel, voltage-dependent, gamma subunit 2 NIMODIPINE Calcium Channel Type L, Benzothiazepine 83% .002093uM .00186uM View
calcium channel, voltage-dependent, gamma subunit 1 NIMODIPINE Calcium Channel Type L, Benzothiazepine 83% .002093uM .00186uM View
calcium channel, voltage-dependent, beta 4 subunit NIMODIPINE Calcium Channel Type L, Benzothiazepine 83% .002093uM .00186uM View
calcium channel, voltage-dependent, beta 3 subunit NIMODIPINE Calcium Channel Type L, Benzothiazepine 83% .002093uM .00186uM View
calcium channel, voltage-dependent, beta 2 subunit NIMODIPINE Calcium Channel Type L, Benzothiazepine 83% .002093uM .00186uM View
calcium channel, voltage-dependent, L type, alpha 1S subunit NIMODIPINE Calcium Channel Type L, Benzothiazepine 83% .002093uM .00186uM View
calcium channel, voltage-dependent, alpha 1F subunit NIMODIPINE Calcium Channel Type L, Benzothiazepine 83% .002093uM .00186uM View
calcium channel, voltage-dependent, L type, alpha 1D subunit NIMODIPINE Calcium Channel Type L, Benzothiazepine 83% .002093uM .00186uM View
calcium channel, voltage-dependent, L type, alpha 1C subunit NIMODIPINE Calcium Channel Type L, Benzothiazepine 83% .002093uM .00186uM View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit NIMODIPINE Calcium Channel Type L, Benzothiazepine 83% .002093uM .00186uM View
calcium channel, voltage-dependent, beta 1 subunit NIMODIPINE Calcium Channel Type L, Benzothiazepine 83% .002093uM .00186uM View
calcium channel, voltage-dependent, L type, alpha 1E subunit NIMODIPINE Calcium Channel Type L, Benzothiazepine 83% .002093uM .00186uM View
calcium channel, voltage-dependent, N type, alpha 1B subunit NIMODIPINE Calcium Channel Type L, Benzothiazepine 83% .002093uM .00186uM View
calcium channel, voltage-dependent, alpha2/delta subunit 1 NIMODIPINE Calcium Channel Type L, Benzothiazepine 83% .002093uM .00186uM View
calcium channel, voltage-dependent, gamma subunit 8 RESERPINE Calcium Channel Type L, Phenylalkylamine 83% 2.05uM 1.993uM View
calcium channel, voltage-dependent, gamma subunit 7 RESERPINE Calcium Channel Type L, Phenylalkylamine 83% 2.05uM 1.993uM View
calcium channel, voltage-dependent, gamma subunit 6 RESERPINE Calcium Channel Type L, Phenylalkylamine 83% 2.05uM 1.993uM View
calcium channel, voltage-dependent, gamma subunit 5 RESERPINE Calcium Channel Type L, Phenylalkylamine 83% 2.05uM 1.993uM View
calcium channel, voltage-dependent, gamma subunit 4 RESERPINE Calcium Channel Type L, Phenylalkylamine 83% 2.05uM 1.993uM View
calcium channel, voltage-dependent, gamma subunit 3 RESERPINE Calcium Channel Type L, Phenylalkylamine 83% 2.05uM 1.993uM View
calcium channel, voltage-dependent, gamma subunit 2 RESERPINE Calcium Channel Type L, Phenylalkylamine 83% 2.05uM 1.993uM View
calcium channel, voltage-dependent, gamma subunit 1 RESERPINE Calcium Channel Type L, Phenylalkylamine 83% 2.05uM 1.993uM View
calcium channel, voltage-dependent, beta 4 subunit RESERPINE Calcium Channel Type L, Phenylalkylamine 83% 2.05uM 1.993uM View
calcium channel, voltage-dependent, beta 3 subunit RESERPINE Calcium Channel Type L, Phenylalkylamine 83% 2.05uM 1.993uM View
calcium channel, voltage-dependent, beta 2 subunit RESERPINE Calcium Channel Type L, Phenylalkylamine 83% 2.05uM 1.993uM View
calcium channel, voltage-dependent, L type, alpha 1S subunit RESERPINE Calcium Channel Type L, Phenylalkylamine 83% 2.05uM 1.993uM View
calcium channel, voltage-dependent, L type, alpha 1C subunit CLOMIPRAMINE Calcium Channel Type L, Benzothiazepine 83% 1.687uM 1.499uM View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit CLOMIPRAMINE Calcium Channel Type L, Benzothiazepine 83% 1.687uM 1.499uM View
calcium channel, voltage-dependent, beta 1 subunit CLOMIPRAMINE Calcium Channel Type L, Benzothiazepine 83% 1.687uM 1.499uM View
calcium channel, voltage-dependent, L type, alpha 1E subunit CLOMIPRAMINE Calcium Channel Type L, Benzothiazepine 83% 1.687uM 1.499uM View
calcium channel, voltage-dependent, N type, alpha 1B subunit CLOMIPRAMINE Calcium Channel Type L, Benzothiazepine 83% 1.687uM 1.499uM View
calcium channel, voltage-dependent, alpha2/delta subunit 1 CLOMIPRAMINE Calcium Channel Type L, Benzothiazepine 83% 1.687uM 1.499uM View
adrenergic receptor, alpha 2a FLUPHENAZINE Imidazoline I2, Central 83% 4.369uM 2.912uM View
adrenergic receptor, alpha 2c (Non-specific probe) FLUPHENAZINE Imidazoline I2, Central 83% 4.369uM 2.912uM View
aldo-keto reductase family 1, member B4 (aldose reductase) TOLMETIN Aldose Reductase 83% 2.153uM NoneNone View
aldo-keto reductase family 1, member B1 (aldose reductase) TOLMETIN Aldose Reductase 83% 2.153uM NoneNone View
aldo-keto reductase family 7, member A2 (aflatoxin aldehyde reductase) TOLMETIN Aldose Reductase 83% 2.153uM NoneNone View
aldo-keto reductase family 7, member A3 (aflatoxin aldehyde reductase) TOLMETIN Aldose Reductase 83% 2.153uM NoneNone View
adrenergic receptor, alpha 2b DOMPERIDONE Adrenergic alpha2B 83% 2.125uM .97uM View
opioid receptor, sigma 1 LABETALOL Sigma1 83% 1.815uM .763uM View
histamine receptor H 2 GENTIAN VIOLET Histamine H2 83% 1.155uM 1.136uM View
mu-opioid receptor MOR GENTIAN VIOLET Opiate mu 83% 2.145uM .871uM View
calcium channel, voltage-dependent, gamma subunit 8 GENTIAN VIOLET Calcium Channel Type L, Dihydropyridine 83% 2.133uM 1.371uM View
calcium channel, voltage-dependent, gamma subunit 7 GENTIAN VIOLET Calcium Channel Type L, Dihydropyridine 83% 2.133uM 1.371uM View
calcium channel, voltage-dependent, gamma subunit 6 GENTIAN VIOLET Calcium Channel Type L, Dihydropyridine 83% 2.133uM 1.371uM View
calcium channel, voltage-dependent, gamma subunit 5 GENTIAN VIOLET Calcium Channel Type L, Dihydropyridine 83% 2.133uM 1.371uM View
calcium channel, voltage-dependent, gamma subunit 4 GENTIAN VIOLET Calcium Channel Type L, Dihydropyridine 83% 2.133uM 1.371uM View
calcium channel, voltage-dependent, gamma subunit 3 GENTIAN VIOLET Calcium Channel Type L, Dihydropyridine 83% 2.133uM 1.371uM View
calcium channel, voltage-dependent, gamma subunit 2 GENTIAN VIOLET Calcium Channel Type L, Dihydropyridine 83% 2.133uM 1.371uM View
calcium channel, voltage-dependent, gamma subunit 1 GENTIAN VIOLET Calcium Channel Type L, Dihydropyridine 83% 2.133uM 1.371uM View
calcium channel, voltage-dependent, beta 4 subunit GENTIAN VIOLET Calcium Channel Type L, Dihydropyridine 83% 2.133uM 1.371uM View
calcium channel, voltage-dependent, beta 3 subunit GENTIAN VIOLET Calcium Channel Type L, Dihydropyridine 83% 2.133uM 1.371uM View
calcium channel, voltage-dependent, beta 2 subunit GENTIAN VIOLET Calcium Channel Type L, Dihydropyridine 83% 2.133uM 1.371uM View
calcium channel, voltage-dependent, L type, alpha 1S subunit GENTIAN VIOLET Calcium Channel Type L, Dihydropyridine 83% 2.133uM 1.371uM View
calcium channel, voltage-dependent, alpha 1F subunit GENTIAN VIOLET Calcium Channel Type L, Dihydropyridine 83% 2.133uM 1.371uM View
calcium channel, voltage-dependent, L type, alpha 1D subunit GENTIAN VIOLET Calcium Channel Type L, Dihydropyridine 83% 2.133uM 1.371uM View
calcium channel, voltage-dependent, L type, alpha 1C subunit GENTIAN VIOLET Calcium Channel Type L, Dihydropyridine 83% 2.133uM 1.371uM View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit GENTIAN VIOLET Calcium Channel Type L, Dihydropyridine 83% 2.133uM 1.371uM View
calcium channel, voltage-dependent, beta 1 subunit GENTIAN VIOLET Calcium Channel Type L, Dihydropyridine 83% 2.133uM 1.371uM View
calcium channel, voltage-dependent, L type, alpha 1E subunit GENTIAN VIOLET Calcium Channel Type L, Dihydropyridine 83% 2.133uM 1.371uM View
calcium channel, voltage-dependent, N type, alpha 1B subunit GENTIAN VIOLET Calcium Channel Type L, Dihydropyridine 83% 2.133uM 1.371uM View
calcium channel, voltage-dependent, alpha2/delta subunit 1 GENTIAN VIOLET Calcium Channel Type L, Dihydropyridine 83% 2.133uM 1.371uM View
calcium channel, voltage-dependent, L type, alpha 1S subunit CITALOPRAM Calcium Channel Type L, Benzothiazepine 83% 1.786uM 1.588uM View
calcium channel, voltage-dependent, alpha 1F subunit CITALOPRAM Calcium Channel Type L, Benzothiazepine 83% 1.786uM 1.588uM View
calcium channel, voltage-dependent, L type, alpha 1D subunit CITALOPRAM Calcium Channel Type L, Benzothiazepine 83% 1.786uM 1.588uM View
calcium channel, voltage-dependent, L type, alpha 1C subunit CITALOPRAM Calcium Channel Type L, Benzothiazepine 83% 1.786uM 1.588uM View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit CITALOPRAM Calcium Channel Type L, Benzothiazepine 83% 1.786uM 1.588uM View
calcium channel, voltage-dependent, beta 1 subunit CITALOPRAM Calcium Channel Type L, Benzothiazepine 83% 1.786uM 1.588uM View
calcium channel, voltage-dependent, L type, alpha 1E subunit CITALOPRAM Calcium Channel Type L, Benzothiazepine 83% 1.786uM 1.588uM View
calcium channel, voltage-dependent, N type, alpha 1B subunit CITALOPRAM Calcium Channel Type L, Benzothiazepine 83% 1.786uM 1.588uM View
calcium channel, voltage-dependent, alpha2/delta subunit 1 CITALOPRAM Calcium Channel Type L, Benzothiazepine 83% 1.786uM 1.588uM View
calcium channel, voltage-dependent, gamma subunit 8 CITALOPRAM Calcium Channel Type L, Benzothiazepine 83% 1.786uM 1.588uM View
calcium channel, voltage-dependent, gamma subunit 7 CITALOPRAM Calcium Channel Type L, Benzothiazepine 83% 1.786uM 1.588uM View
calcium channel, voltage-dependent, gamma subunit 6 CITALOPRAM Calcium Channel Type L, Benzothiazepine 83% 1.786uM 1.588uM View
calcium channel, voltage-dependent, gamma subunit 5 CITALOPRAM Calcium Channel Type L, Benzothiazepine 83% 1.786uM 1.588uM View
calcium channel, voltage-dependent, gamma subunit 4 CITALOPRAM Calcium Channel Type L, Benzothiazepine 83% 1.786uM 1.588uM View
calcium channel, voltage-dependent, gamma subunit 3 CITALOPRAM Calcium Channel Type L, Benzothiazepine 83% 1.786uM 1.588uM View
calcium channel, voltage-dependent, gamma subunit 2 CITALOPRAM Calcium Channel Type L, Benzothiazepine 83% 1.786uM 1.588uM View
calcium channel, voltage-dependent, gamma subunit 1 CITALOPRAM Calcium Channel Type L, Benzothiazepine 83% 1.786uM 1.588uM View
calcium channel, voltage-dependent, beta 4 subunit CITALOPRAM Calcium Channel Type L, Benzothiazepine 83% 1.786uM 1.588uM View
calcium channel, voltage-dependent, beta 3 subunit CITALOPRAM Calcium Channel Type L, Benzothiazepine 83% 1.786uM 1.588uM View
calcium channel, voltage-dependent, beta 2 subunit CITALOPRAM Calcium Channel Type L, Benzothiazepine 83% 1.786uM 1.588uM View
ATPase, Na+/K+ transporting, alpha 4 polypeptide CISPLATIN ATPase, Na+/K+ 83% 9.427uM NoneNone View
ATPase, Na+/K+ transporting, alpha 3 polypeptide CISPLATIN ATPase, Na+/K+ 83% 9.427uM NoneNone View
ATPase, Na+/K+ transporting, alpha 2 polypeptide CISPLATIN ATPase, Na+/K+ 83% 9.427uM NoneNone View
ATPase, Na+/K+ transporting, alpha 1 polypeptide CISPLATIN ATPase, Na+/K+ 83% 9.427uM NoneNone View
ATPase, Na+/K+ transporting, beta 1 polypeptide CISPLATIN ATPase, Na+/K+ 83% 9.427uM NoneNone View
ATPase, Na+/K+ transporting, beta 3 polypeptide CISPLATIN ATPase, Na+/K+ 83% 9.427uM NoneNone View
ATPase, Na+/K+ transporting, beta 2 polypeptide CISPLATIN ATPase, Na+/K+ 83% 9.427uM NoneNone View
ATPase, (Na+)/K+ transporting, beta 4 polypeptide CISPLATIN ATPase, Na+/K+ 83% 9.427uM NoneNone View
5-hydroxytryptamine (serotonin) receptor 5B PROCHLORPERAZINE Serotonin 5-HT4 83% 1.164uM .194uM View
5-hydroxytryptamine (serotonin) receptor 4 PROCHLORPERAZINE Serotonin 5-HT4 83% 1.164uM .194uM View
progesterone receptor ETHYNODIOL DIACETATE Progesterone 83% .16uM .021uM View
progesterone receptor ETHYNODIOL DIACETATE Progesterone 83% .16uM .021uM View
mitogen-activated protein kinase 1 TROGLITAZONE Protein Serine/Threonine Kinase, ERK2 83% 1.238uM NoneNone View
mitogen activated protein kinase 1 TROGLITAZONE Protein Serine/Threonine Kinase, ERK2 83% 1.238uM NoneNone View
acetylcholinesterase (YT blood group) MICONAZOLE Acetylcholinesterase 83% 18.659uM NoneNone View
collagen-like tail subunit (single strand of homotrimer) of asymmetric acetylcholinesterase MICONAZOLE Acetylcholinesterase 83% 18.659uM NoneNone View
acetylcholinesterase MICONAZOLE Acetylcholinesterase 83% 18.659uM NoneNone View
thromboxane A synthase 1 MICONAZOLE Thromboxane Synthetase 83% .263uM NoneNone View
thromboxane A synthase 1 (platelet, cytochrome P450, family 5, subfamily A) MICONAZOLE Thromboxane Synthetase 83% .263uM NoneNone View
cytochrome P450, family 3, subfamily a, polypeptide 13 METYRAPONE CYP450-3A4 Inhibition 83% .8uM NoneNone View
adrenergic receptor, alpha 2a ERGOCORNINE Imidazoline I2, Central 83% .004487uM .002991uM View
adrenergic receptor, alpha 2c (Non-specific probe) ERGOCORNINE Imidazoline I2, Central 83% .004487uM .002991uM View
nuclear receptor subfamily 3, group C, member 1 DANAZOL Glucocorticoid 83% 4.314uM 1.961uM View
gamma-aminobutyric acid (GABA-A) receptor, subunit alpha 4 DIETHYLSTILBESTROL GABAA, Chloride Channel, TBOB 83% 15.09uM 13.529uM View
gamma-aminobutyric acid A receptor, gamma 1 DIETHYLSTILBESTROL GABAA, Chloride Channel, TBOB 83% 15.09uM 13.529uM View
gamma-aminobutyric acid A receptor, pi DIETHYLSTILBESTROL GABAA, Chloride Channel, TBOB 83% 15.09uM 13.529uM View
AT hook, DNA binding motif, containing 1 (DBSS) DIETHYLSTILBESTROL GABAA, Chloride Channel, TBOB 83% 15.09uM 13.529uM View
gamma-aminobutyric acid A receptor, theta DIETHYLSTILBESTROL GABAA, Chloride Channel, TBOB 83% 15.09uM 13.529uM View
gamma-aminobutyric acid A receptor, gamma 2 DIETHYLSTILBESTROL GABAA, Chloride Channel, TBOB 83% 15.09uM 13.529uM View
gamma-aminobutyric acid (GABA-A) receptor, subunit alpha 6 DIETHYLSTILBESTROL GABAA, Chloride Channel, TBOB 83% 15.09uM 13.529uM View
gamma-aminobutyric acid (GABA-A) receptor, subunit alpha 5 DIETHYLSTILBESTROL GABAA, Chloride Channel, TBOB 83% 15.09uM 13.529uM View
gamma-aminobutyric acid A receptor, alpha 2 DIETHYLSTILBESTROL GABAA, Chloride Channel, TBOB 83% 15.09uM 13.529uM View
gamma-aminobutyric acid A receptor, alpha 1 DIETHYLSTILBESTROL GABAA, Chloride Channel, TBOB 83% 15.09uM 13.529uM View
gamma-aminobutyric acid (GABA-C) receptor, subunit rho 2 DIETHYLSTILBESTROL GABAA, Chloride Channel, TBOB 83% 15.09uM 13.529uM View
gamma-aminobutyric acid (GABA-C) receptor, subunit rho 1 DIETHYLSTILBESTROL GABAA, Chloride Channel, TBOB 83% 15.09uM 13.529uM View
gamma-aminobutyric acid A receptor, delta DIETHYLSTILBESTROL GABAA, Chloride Channel, TBOB 83% 15.09uM 13.529uM View
gamma-aminobutyric acid (GABA-A) receptor, subunit alpha 3 DIETHYLSTILBESTROL GABAA, Chloride Channel, TBOB 83% 15.09uM 13.529uM View
adrenergic receptor, beta 1 METOPROLOL Adrenergic beta1 83% .176uM .102uM View
adrenergic, beta-1-, receptor METOPROLOL Adrenergic beta1 83% .176uM .102uM View
adrenergic receptor, alpha 1d (Non-specific probe) DIMENHYDRINATE Adrenergic alpha1D 83% 2.894uM 1.423uM View
epidermal growth factor receptor BACITRACIN Protein Tyrosine Kinase, EGF Receptor 83% 5.377uM NoneNone View
progesterone receptor TESTOSTERONE Progesterone 83% 1.935uM .252uM View
progesterone receptor TESTOSTERONE Progesterone 83% 1.935uM .252uM View
solute carrier family 6 (neurotransmitter transporter, serotonin), member 4 BETA-ESTRADIOL 3-BENZOATE Serotonin Transporter 83% 3.672uM 1.951uM View
mitogen activated protein kinase 3 TANNIC ACID Protein Serine/Threonine Kinase, ERK1 83% 4.052uM NoneNone View
mitogen-activated protein kinase 3 TANNIC ACID Protein Serine/Threonine Kinase, ERK1 83% 4.052uM NoneNone View
adrenergic receptor, alpha 2b EPINEPHRINE Adrenergic alpha2C 83% 2.449uM .356uM View
adrenergic receptor, alpha 2c (Non-specific probe) EPINEPHRINE Adrenergic alpha2C 83% 2.449uM .356uM View
Protein-tyrosine kinase, Fyn TANNIC ACID Protein Tyrosine Kinase, Fyn 83% .022uM NoneNone View
opioid receptor, kappa 1 AMIODARONE Opiate kappa 83% 16.68uM 6.672uM View
melanocortin 3 receptor AMIODARONE Melanocortin MC3 83% 12.372uM 10.797uM View
melanocortin 3 receptor AMIODARONE Melanocortin MC3 83% 12.372uM 10.797uM View
opioid receptor, kappa 1 CHLORPROMAZINE Opiate kappa 83% 11.082uM 4.433uM View
Cytochrom P450-2C19 monooxygenase TROPICAMIDE CYP450-2C19 Inhibition 83% 1uM NoneNone View
opioid receptor, delta 1 TAMOXIFEN Opiate delta 83% 13.339uM 4.702uM View
phosphodiesterase 3B CILOSTAMIDE Phosphodiesterase PDE3 83% .055uM NoneNone View
phosphodiesterase 3A CILOSTAMIDE Phosphodiesterase PDE3 83% .055uM NoneNone View
opioid receptor, sigma 1 TETRACAINE Sigma1 83% 1.673uM .703uM View
calcium channel, voltage-dependent, gamma subunit 8 CLOMIPRAMINE Calcium Channel Type L, Benzothiazepine 83% 1.687uM 1.499uM View
calcium channel, voltage-dependent, gamma subunit 7 CLOMIPRAMINE Calcium Channel Type L, Benzothiazepine 83% 1.687uM 1.499uM View
calcium channel, voltage-dependent, gamma subunit 6 CLOMIPRAMINE Calcium Channel Type L, Benzothiazepine 83% 1.687uM 1.499uM View
calcium channel, voltage-dependent, gamma subunit 5 CLOMIPRAMINE Calcium Channel Type L, Benzothiazepine 83% 1.687uM 1.499uM View
calcium channel, voltage-dependent, gamma subunit 4 CLOMIPRAMINE Calcium Channel Type L, Benzothiazepine 83% 1.687uM 1.499uM View
calcium channel, voltage-dependent, gamma subunit 3 CLOMIPRAMINE Calcium Channel Type L, Benzothiazepine 83% 1.687uM 1.499uM View
calcium channel, voltage-dependent, gamma subunit 2 CLOMIPRAMINE Calcium Channel Type L, Benzothiazepine 83% 1.687uM 1.499uM View
calcium channel, voltage-dependent, gamma subunit 1 CLOMIPRAMINE Calcium Channel Type L, Benzothiazepine 83% 1.687uM 1.499uM View
calcium channel, voltage-dependent, beta 4 subunit CLOMIPRAMINE Calcium Channel Type L, Benzothiazepine 83% 1.687uM 1.499uM View
calcium channel, voltage-dependent, beta 3 subunit CLOMIPRAMINE Calcium Channel Type L, Benzothiazepine 83% 1.687uM 1.499uM View
calcium channel, voltage-dependent, beta 2 subunit CLOMIPRAMINE Calcium Channel Type L, Benzothiazepine 83% 1.687uM 1.499uM View
calcium channel, voltage-dependent, L type, alpha 1S subunit CLOMIPRAMINE Calcium Channel Type L, Benzothiazepine 83% 1.687uM 1.499uM View
calcium channel, voltage-dependent, alpha 1F subunit CLOMIPRAMINE Calcium Channel Type L, Benzothiazepine 83% 1.687uM 1.499uM View
calcium channel, voltage-dependent, L type, alpha 1D subunit CLOMIPRAMINE Calcium Channel Type L, Benzothiazepine 83% 1.687uM 1.499uM View
calcium channel, voltage-dependent, alpha 1F subunit FLUNARIZINE Calcium Channel Type L, Benzothiazepine 83% 1.12uM .995uM View
calcium channel, voltage-dependent, L type, alpha 1D subunit FLUNARIZINE Calcium Channel Type L, Benzothiazepine 83% 1.12uM .995uM View
calcium channel, voltage-dependent, L type, alpha 1C subunit FLUNARIZINE Calcium Channel Type L, Benzothiazepine 83% 1.12uM .995uM View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit FLUNARIZINE Calcium Channel Type L, Benzothiazepine 83% 1.12uM .995uM View
calcium channel, voltage-dependent, beta 1 subunit FLUNARIZINE Calcium Channel Type L, Benzothiazepine 83% 1.12uM .995uM View
calcium channel, voltage-dependent, L type, alpha 1E subunit DROPERIDOL Calcium Channel Type L, Phenylalkylamine 81% 4.165uM 4.049uM View
calcium channel, voltage-dependent, N type, alpha 1B subunit DROPERIDOL Calcium Channel Type L, Phenylalkylamine 81% 4.165uM 4.049uM View
calcium channel, voltage-dependent, alpha2/delta subunit 1 DROPERIDOL Calcium Channel Type L, Phenylalkylamine 81% 4.165uM 4.049uM View
adrenergic receptor, beta 1 ESMOLOL Adrenergic beta1 81% .197uM .1137uM View
adrenergic, beta-1-, receptor ESMOLOL Adrenergic beta1 81% .197uM .1137uM View
5-hydroxytryptamine (serotonin) receptor 2B 1-(2-METHYLBENZOYL)-4-(PHENYLMETHYL)-PIPERIDINE Serotonin 5-HT2B 81% 1.86uM 1.183uM View
cytochrome P450, family 2, subfamily C, polypeptide 9 1-(2-CHLOROBENZOYL)-4-(PHENYLMETHYL)-PIPERIDINE CYP450-2C9 Inhibition 81% 2uM NoneNone View
adrenergic receptor, alpha 2a MITOTANE Adrenergic alpha2A 81% 7.347uM 2.755uM View
calcium channel, voltage-dependent, gamma subunit 8 L-744832 Calcium Channel Type L, Benzothiazepine 81% 3.568uM 3.172uM View
calcium channel, voltage-dependent, gamma subunit 7 L-744832 Calcium Channel Type L, Benzothiazepine 81% 3.568uM 3.172uM View
calcium channel, voltage-dependent, gamma subunit 6 L-744832 Calcium Channel Type L, Benzothiazepine 81% 3.568uM 3.172uM View
calcium channel, voltage-dependent, gamma subunit 5 L-744832 Calcium Channel Type L, Benzothiazepine 81% 3.568uM 3.172uM View
calcium channel, voltage-dependent, gamma subunit 4 L-744832 Calcium Channel Type L, Benzothiazepine 81% 3.568uM 3.172uM View
calcium channel, voltage-dependent, gamma subunit 3 L-744832 Calcium Channel Type L, Benzothiazepine 81% 3.568uM 3.172uM View
calcium channel, voltage-dependent, gamma subunit 2 L-744832 Calcium Channel Type L, Benzothiazepine 81% 3.568uM 3.172uM View
calcium channel, voltage-dependent, gamma subunit 1 L-744832 Calcium Channel Type L, Benzothiazepine 81% 3.568uM 3.172uM View
calcium channel, voltage-dependent, beta 4 subunit L-744832 Calcium Channel Type L, Benzothiazepine 81% 3.568uM 3.172uM View
calcium channel, voltage-dependent, beta 3 subunit L-744832 Calcium Channel Type L, Benzothiazepine 81% 3.568uM 3.172uM View
calcium channel, voltage-dependent, beta 2 subunit L-744832 Calcium Channel Type L, Benzothiazepine 81% 3.568uM 3.172uM View
calcium channel, voltage-dependent, L type, alpha 1S subunit L-744832 Calcium Channel Type L, Benzothiazepine 81% 3.568uM 3.172uM View
calcium channel, voltage-dependent, alpha 1F subunit L-744832 Calcium Channel Type L, Benzothiazepine 81% 3.568uM 3.172uM View
calcium channel, voltage-dependent, L type, alpha 1D subunit L-744832 Calcium Channel Type L, Benzothiazepine 81% 3.568uM 3.172uM View
calcium channel, voltage-dependent, L type, alpha 1C subunit L-744832 Calcium Channel Type L, Benzothiazepine 81% 3.568uM 3.172uM View