| calcium channel, voltage-dependent, P/Q type, alpha 1A subunit |
L-744832 |
Calcium Channel Type L, Benzothiazepine |
81% |
3.568uM |
3.172uM |
View
|
| calcium channel, voltage-dependent, beta 1 subunit |
L-744832 |
Calcium Channel Type L, Benzothiazepine |
81% |
3.568uM |
3.172uM |
View
|
| calcium channel, voltage-dependent, L type, alpha 1E subunit |
L-744832 |
Calcium Channel Type L, Benzothiazepine |
81% |
3.568uM |
3.172uM |
View
|
| calcium channel, voltage-dependent, N type, alpha 1B subunit |
L-744832 |
Calcium Channel Type L, Benzothiazepine |
81% |
3.568uM |
3.172uM |
View
|
| calcium channel, voltage-dependent, alpha2/delta subunit 1 |
L-744832 |
Calcium Channel Type L, Benzothiazepine |
81% |
3.568uM |
3.172uM |
View
|
| 5-hydroxytryptamine (serotonin) receptor 2A |
QUINACRINE |
Serotonin 5-HT2A |
81% |
2.663uM |
.761uM |
View
|
| acetylcholinesterase (YT blood group) |
QUINACRINE |
Acetylcholinesterase |
81% |
2.667uM |
NoneNone |
View
|
| collagen-like tail subunit (single strand of homotrimer) of asymmetric acetylcholinesterase |
QUINACRINE |
Acetylcholinesterase |
81% |
2.667uM |
NoneNone |
View
|
| acetylcholinesterase |
QUINACRINE |
Acetylcholinesterase |
81% |
2.667uM |
NoneNone |
View
|
| adrenergic receptor, alpha 2b |
KETOTIFEN |
Adrenergic alpha2B |
81% |
.71uM |
.324uM |
View
|
| arginine vasopressin receptor 1A |
RITONAVIR |
Vasopressin V1A |
81% |
12.416uM |
4.981uM |
View
|
| mu-opioid receptor MOR |
CYPROTERONE ACETATE |
Opiate mu |
81% |
2.183uM |
.886uM |
View
|
| 5-hydroxytryptamine (serotonin) receptor 1B |
OLANZAPINE |
Serotonin 5-HT1B |
81% |
.707uM |
.433uM |
View
|
| calcium channel, voltage-dependent, gamma subunit 8 |
OXYBUTYNIN |
Calcium Channel Type L, Phenylalkylamine |
81% |
2.358uM |
2.2925uM |
View
|
| calcium channel, voltage-dependent, gamma subunit 7 |
OXYBUTYNIN |
Calcium Channel Type L, Phenylalkylamine |
81% |
2.358uM |
2.2925uM |
View
|
| calcium channel, voltage-dependent, gamma subunit 6 |
OXYBUTYNIN |
Calcium Channel Type L, Phenylalkylamine |
81% |
2.358uM |
2.2925uM |
View
|
| calcium channel, voltage-dependent, gamma subunit 5 |
OXYBUTYNIN |
Calcium Channel Type L, Phenylalkylamine |
81% |
2.358uM |
2.2925uM |
View
|
| calcium channel, voltage-dependent, gamma subunit 4 |
OXYBUTYNIN |
Calcium Channel Type L, Phenylalkylamine |
81% |
2.358uM |
2.2925uM |
View
|
| calcium channel, voltage-dependent, gamma subunit 3 |
OXYBUTYNIN |
Calcium Channel Type L, Phenylalkylamine |
81% |
2.358uM |
2.2925uM |
View
|
| calcium channel, voltage-dependent, gamma subunit 2 |
OXYBUTYNIN |
Calcium Channel Type L, Phenylalkylamine |
81% |
2.358uM |
2.2925uM |
View
|
| calcium channel, voltage-dependent, gamma subunit 1 |
OXYBUTYNIN |
Calcium Channel Type L, Phenylalkylamine |
81% |
2.358uM |
2.2925uM |
View
|
| calcium channel, voltage-dependent, beta 4 subunit |
OXYBUTYNIN |
Calcium Channel Type L, Phenylalkylamine |
81% |
2.358uM |
2.2925uM |
View
|
| calcium channel, voltage-dependent, beta 3 subunit |
OXYBUTYNIN |
Calcium Channel Type L, Phenylalkylamine |
81% |
2.358uM |
2.2925uM |
View
|
| calcium channel, voltage-dependent, beta 2 subunit |
OXYBUTYNIN |
Calcium Channel Type L, Phenylalkylamine |
81% |
2.358uM |
2.2925uM |
View
|
| sodium channel associated protein 2 |
PIPAMAZINE |
Sodium Channel, Site 2 |
80% |
2.686uM |
2.451uM |
View
|
| sodium channel, voltage-gated, type III, beta |
PIPAMAZINE |
Sodium Channel, Site 2 |
80% |
2.686uM |
2.451uM |
View
|
| sodium channel, voltage-gated, type I, alpha |
PIPAMAZINE |
Sodium Channel, Site 2 |
80% |
2.686uM |
2.451uM |
View
|
| sodium channel, voltage-gated, type IX, alpha |
PIPAMAZINE |
Sodium Channel, Site 2 |
80% |
2.686uM |
2.451uM |
View
|
| sodium channel, voltage-gated, type VII, alpha |
PIPAMAZINE |
Sodium Channel, Site 2 |
80% |
2.686uM |
2.451uM |
View
|
| amiloride-sensitive cation channel 5, intestinal |
PIPAMAZINE |
Sodium Channel, Site 2 |
80% |
2.686uM |
2.451uM |
View
|
| sodium channel, voltage-gated, type III, beta |
PIPAMAZINE |
Sodium Channel, Site 2 |
80% |
2.686uM |
2.451uM |
View
|
| sodium channel, voltage-gated, type VIII, alpha polypeptide |
PIPAMAZINE |
Sodium Channel, Site 2 |
80% |
2.686uM |
2.451uM |
View
|
| sodium channel, voltage-gated, type XI, alpha |
PIPAMAZINE |
Sodium Channel, Site 2 |
80% |
2.686uM |
2.451uM |
View
|
| sodium channel, voltage-gated, type I, beta |
PIPAMAZINE |
Sodium Channel, Site 2 |
80% |
2.686uM |
2.451uM |
View
|
| sodium channel, voltage-gated, type 10, alpha polypeptide |
PIPAMAZINE |
Sodium Channel, Site 2 |
80% |
2.686uM |
2.451uM |
View
|
| sodium channel, voltage-gated, type IV, alpha polypeptide |
PIPAMAZINE |
Sodium Channel, Site 2 |
80% |
2.686uM |
2.451uM |
View
|
| sodium channel, voltage-gated, type V, alpha polypeptide |
PIPAMAZINE |
Sodium Channel, Site 2 |
80% |
2.686uM |
2.451uM |
View
|
| sodium channel, voltage-gated, type II, beta |
PIPAMAZINE |
Sodium Channel, Site 2 |
80% |
2.686uM |
2.451uM |
View
|
| sodium channel, nonvoltage-gated 1 alpha |
PIPAMAZINE |
Sodium Channel, Site 2 |
80% |
2.686uM |
2.451uM |
View
|
| sodium channel, nonvoltage-gated 1 gamma |
PIPAMAZINE |
Sodium Channel, Site 2 |
80% |
2.686uM |
2.451uM |
View
|
| sodium channel, nonvoltage-gated 1 beta |
PIPAMAZINE |
Sodium Channel, Site 2 |
80% |
2.686uM |
2.451uM |
View
|
| sodium channel, voltage-gated, type 2, alpha 1 polypeptide |
PIPAMAZINE |
Sodium Channel, Site 2 |
80% |
2.686uM |
2.451uM |
View
|
| sodium channel, voltage-gated, type XI, alpha |
PIPAMAZINE |
Sodium Channel, Site 2 |
80% |
2.686uM |
2.451uM |
View
|
| sodium channel, nonvoltage-gated 1, gamma |
PIPAMAZINE |
Sodium Channel, Site 2 |
80% |
2.686uM |
2.451uM |
View
|
| sodium channel, nonvoltage-gated 1, delta |
PIPAMAZINE |
Sodium Channel, Site 2 |
80% |
2.686uM |
2.451uM |
View
|
| sodium channel, nonvoltage-gated 1, beta (Liddle syndrome) |
PIPAMAZINE |
Sodium Channel, Site 2 |
80% |
2.686uM |
2.451uM |
View
|
| sodium channel, nonvoltage-gated 1 alpha |
PIPAMAZINE |
Sodium Channel, Site 2 |
80% |
2.686uM |
2.451uM |
View
|
| sodium channel, voltage-gated, type X, alpha |
PIPAMAZINE |
Sodium Channel, Site 2 |
80% |
2.686uM |
2.451uM |
View
|
| sodium channel, voltage-gated, type IX, alpha |
PIPAMAZINE |
Sodium Channel, Site 2 |
80% |
2.686uM |
2.451uM |
View
|
| sodium channel, voltage gated, type VIII, alpha |
PIPAMAZINE |
Sodium Channel, Site 2 |
80% |
2.686uM |
2.451uM |
View
|
| sodium channel, voltage-gated, type VII, alpha |
PIPAMAZINE |
Sodium Channel, Site 2 |
80% |
2.686uM |
2.451uM |
View
|
| prostaglandin-endoperoxide synthase 2 |
KETOPROFEN |
Cyclooxygenase COX-2 |
80% |
.785uM |
NoneNone |
View
|
| prostaglandin-endoperoxide synthase 2 (prostaglandin G/H synthase and cyclooxygenase) |
KETOPROFEN |
Cyclooxygenase COX-2 |
80% |
.785uM |
NoneNone |
View
|
| v-erb-b2 erythroblastic leukemia viral oncogene homolog 2, neuro/glioblastoma derived oncogene homolog (avian) |
MICONAZOLE |
Protein Tyrosine Kinase, HER2 Receptor |
80% |
27.43uM |
NoneNone |
View
|
| v-erb-b2 erythroblastic leukemia viral oncogene homolog 2, neuro/glioblastoma derived oncogene homolog (avian) |
MICONAZOLE |
Protein Tyrosine Kinase, HER2 Receptor |
80% |
27.43uM |
NoneNone |
View
|
| epidermal growth factor receptor |
CIGLITAZONE |
Protein Tyrosine Kinase, EGF Receptor |
80% |
4.655uM |
NoneNone |
View
|
| matrix metallopeptidase 9 |
BUDESONIDE |
Protease, Matrix Metalloprotease-9 (MMP-9) |
80% |
1.989uM |
NoneNone |
View
|
| matrix metalloproteinase 9 (gelatinase B, 92kDa gelatinase, 92kDa type IV collagenase) |
BUDESONIDE |
Protease, Matrix Metalloprotease-9 (MMP-9) |
80% |
1.989uM |
NoneNone |
View
|
| Protein-tyrosine kinase, Fyn |
AURANOFIN |
Protein Tyrosine Kinase, Fyn |
80% |
1.197uM |
NoneNone |
View
|
| calcium channel, voltage-dependent, beta 1 subunit |
DANAZOL |
Calcium Channel Type L, Benzothiazepine |
80% |
14.649uM |
13.021uM |
View
|
| calcium channel, voltage-dependent, L type, alpha 1E subunit |
DANAZOL |
Calcium Channel Type L, Benzothiazepine |
80% |
14.649uM |
13.021uM |
View
|
| calcium channel, voltage-dependent, N type, alpha 1B subunit |
DANAZOL |
Calcium Channel Type L, Benzothiazepine |
80% |
14.649uM |
13.021uM |
View
|
| calcium channel, voltage-dependent, alpha2/delta subunit 1 |
DANAZOL |
Calcium Channel Type L, Benzothiazepine |
80% |
14.649uM |
13.021uM |
View
|
| calcium channel, voltage-dependent, gamma subunit 8 |
DANAZOL |
Calcium Channel Type L, Benzothiazepine |
80% |
14.649uM |
13.021uM |
View
|
| calcium channel, voltage-dependent, gamma subunit 7 |
DANAZOL |
Calcium Channel Type L, Benzothiazepine |
80% |
14.649uM |
13.021uM |
View
|
| calcium channel, voltage-dependent, gamma subunit 6 |
DANAZOL |
Calcium Channel Type L, Benzothiazepine |
80% |
14.649uM |
13.021uM |
View
|
| calcium channel, voltage-dependent, gamma subunit 5 |
DANAZOL |
Calcium Channel Type L, Benzothiazepine |
80% |
14.649uM |
13.021uM |
View
|
| calcium channel, voltage-dependent, gamma subunit 4 |
DANAZOL |
Calcium Channel Type L, Benzothiazepine |
80% |
14.649uM |
13.021uM |
View
|
| calcium channel, voltage-dependent, gamma subunit 3 |
DANAZOL |
Calcium Channel Type L, Benzothiazepine |
80% |
14.649uM |
13.021uM |
View
|
| calcium channel, voltage-dependent, gamma subunit 2 |
DANAZOL |
Calcium Channel Type L, Benzothiazepine |
80% |
14.649uM |
13.021uM |
View
|
| calcium channel, voltage-dependent, gamma subunit 1 |
DANAZOL |
Calcium Channel Type L, Benzothiazepine |
80% |
14.649uM |
13.021uM |
View
|
| calcium channel, voltage-dependent, beta 4 subunit |
DANAZOL |
Calcium Channel Type L, Benzothiazepine |
80% |
14.649uM |
13.021uM |
View
|
| calcium channel, voltage-dependent, beta 3 subunit |
DANAZOL |
Calcium Channel Type L, Benzothiazepine |
80% |
14.649uM |
13.021uM |
View
|
| calcium channel, voltage-dependent, L type, alpha 1E subunit |
FLUNARIZINE |
Calcium Channel Type L, Benzothiazepine |
83% |
1.12uM |
.995uM |
View
|
| calcium channel, voltage-dependent, N type, alpha 1B subunit |
FLUNARIZINE |
Calcium Channel Type L, Benzothiazepine |
83% |
1.12uM |
.995uM |
View
|
| calcium channel, voltage-dependent, alpha2/delta subunit 1 |
FLUNARIZINE |
Calcium Channel Type L, Benzothiazepine |
83% |
1.12uM |
.995uM |
View
|
| Cytochrome P450, subfamily IIC (mephenytoin 4-hydroxylase) |
NIFURSOL |
CYP450-2C9 Inhibition |
83% |
7uM |
NoneNone |
View
|
| cytochrome P450, family 2, subfamily C, polypeptide 9 |
NIFURSOL |
CYP450-2C9 Inhibition |
83% |
7uM |
NoneNone |
View
|
| Cytochrom P450-2C19 monooxygenase |
TICLOPIDINE |
CYP450-2C19 Inhibition |
83% |
.6678uM |
NoneNone |
View
|
| mitogen activated protein kinase 14 |
FENBENDAZOLE |
Protein Serine/Threonine Kinase, p38alpha |
83% |
3.188uM |
NoneNone |
View
|
| mitogen-activated protein kinase 14 |
FENBENDAZOLE |
Protein Serine/Threonine Kinase, p38alpha |
83% |
3.188uM |
NoneNone |
View
|
| cholinergic receptor, muscarinic 2 |
MAPROTILINE |
Muscarinic M2 |
83% |
1.927uM |
.685uM |
View
|
| sodium channel, voltage-gated, type IV, alpha |
SPIRADOLINE |
Sodium Channel, Site 2 |
83% |
3.086uM |
2.815uM |
View
|
| sodium channel, voltage-gated, type III, alpha |
SPIRADOLINE |
Sodium Channel, Site 2 |
83% |
3.086uM |
2.815uM |
View
|
| sodium channel, voltage-gated, type II, beta |
SPIRADOLINE |
Sodium Channel, Site 2 |
83% |
3.086uM |
2.815uM |
View
|
| sodium channel, voltage-gated, type II, alpha 2 |
SPIRADOLINE |
Sodium Channel, Site 2 |
83% |
3.086uM |
2.815uM |
View
|
| sodium channel, voltage-gated, type I, beta |
SPIRADOLINE |
Sodium Channel, Site 2 |
83% |
3.086uM |
2.815uM |
View
|
| sodium channel, voltage-gated, type I, alpha |
SPIRADOLINE |
Sodium Channel, Site 2 |
83% |
3.086uM |
2.815uM |
View
|
| sodium channel, voltage-gated, type IV, beta |
SPIRADOLINE |
Sodium Channel, Site 2 |
83% |
3.086uM |
2.815uM |
View
|
| sodium channel associated protein 1 |
SPIRADOLINE |
Sodium Channel, Site 2 |
83% |
3.086uM |
2.815uM |
View
|
| sodium channel associated protein 2 |
SPIRADOLINE |
Sodium Channel, Site 2 |
83% |
3.086uM |
2.815uM |
View
|
| sodium channel, voltage-gated, type III, beta |
SPIRADOLINE |
Sodium Channel, Site 2 |
83% |
3.086uM |
2.815uM |
View
|
| sodium channel, voltage-gated, type I, alpha |
SPIRADOLINE |
Sodium Channel, Site 2 |
83% |
3.086uM |
2.815uM |
View
|
| sodium channel, voltage-gated, type IX, alpha |
SPIRADOLINE |
Sodium Channel, Site 2 |
83% |
3.086uM |
2.815uM |
View
|
| sodium channel, voltage-gated, type VII, alpha |
SPIRADOLINE |
Sodium Channel, Site 2 |
83% |
3.086uM |
2.815uM |
View
|
| amiloride-sensitive cation channel 5, intestinal |
SPIRADOLINE |
Sodium Channel, Site 2 |
83% |
3.086uM |
2.815uM |
View
|
| sodium channel, voltage-gated, type III, beta |
SPIRADOLINE |
Sodium Channel, Site 2 |
83% |
3.086uM |
2.815uM |
View
|
| sodium channel, voltage-gated, type VIII, alpha polypeptide |
SPIRADOLINE |
Sodium Channel, Site 2 |
83% |
3.086uM |
2.815uM |
View
|
| sodium channel, voltage-gated, type XI, alpha |
SPIRADOLINE |
Sodium Channel, Site 2 |
83% |
3.086uM |
2.815uM |
View
|
| sodium channel, voltage-gated, type I, beta |
SPIRADOLINE |
Sodium Channel, Site 2 |
83% |
3.086uM |
2.815uM |
View
|
| sodium channel, voltage-gated, type 10, alpha polypeptide |
SPIRADOLINE |
Sodium Channel, Site 2 |
83% |
3.086uM |
2.815uM |
View
|
| sodium channel, voltage-gated, type IV, alpha polypeptide |
SPIRADOLINE |
Sodium Channel, Site 2 |
83% |
3.086uM |
2.815uM |
View
|
| sodium channel, voltage-gated, type V, alpha polypeptide |
SPIRADOLINE |
Sodium Channel, Site 2 |
83% |
3.086uM |
2.815uM |
View
|
| sodium channel, voltage-gated, type II, beta |
SPIRADOLINE |
Sodium Channel, Site 2 |
83% |
3.086uM |
2.815uM |
View
|
| sodium channel, nonvoltage-gated 1 alpha |
SPIRADOLINE |
Sodium Channel, Site 2 |
83% |
3.086uM |
2.815uM |
View
|
| sodium channel, nonvoltage-gated 1 gamma |
SPIRADOLINE |
Sodium Channel, Site 2 |
83% |
3.086uM |
2.815uM |
View
|
| sodium channel, nonvoltage-gated 1 beta |
SPIRADOLINE |
Sodium Channel, Site 2 |
83% |
3.086uM |
2.815uM |
View
|
| sodium channel, voltage-gated, type 2, alpha 1 polypeptide |
SPIRADOLINE |
Sodium Channel, Site 2 |
83% |
3.086uM |
2.815uM |
View
|
| sodium channel, voltage-gated, type XI, alpha |
SPIRADOLINE |
Sodium Channel, Site 2 |
83% |
3.086uM |
2.815uM |
View
|
| sodium channel, nonvoltage-gated 1, gamma |
SPIRADOLINE |
Sodium Channel, Site 2 |
83% |
3.086uM |
2.815uM |
View
|
| sodium channel, nonvoltage-gated 1, delta |
SPIRADOLINE |
Sodium Channel, Site 2 |
83% |
3.086uM |
2.815uM |
View
|
| sodium channel, nonvoltage-gated 1, beta (Liddle syndrome) |
SPIRADOLINE |
Sodium Channel, Site 2 |
83% |
3.086uM |
2.815uM |
View
|
| sodium channel, nonvoltage-gated 1 alpha |
SPIRADOLINE |
Sodium Channel, Site 2 |
83% |
3.086uM |
2.815uM |
View
|
| sodium channel, voltage-gated, type X, alpha |
SPIRADOLINE |
Sodium Channel, Site 2 |
83% |
3.086uM |
2.815uM |
View
|
| sodium channel, voltage-gated, type IX, alpha |
SPIRADOLINE |
Sodium Channel, Site 2 |
83% |
3.086uM |
2.815uM |
View
|
| sodium channel, voltage gated, type VIII, alpha |
SPIRADOLINE |
Sodium Channel, Site 2 |
83% |
3.086uM |
2.815uM |
View
|
| sodium channel, voltage-gated, type VII, alpha |
SPIRADOLINE |
Sodium Channel, Site 2 |
83% |
3.086uM |
2.815uM |
View
|
| sodium channel, voltage-gated, type V, alpha (long QT syndrome 3) |
SPIRADOLINE |
Sodium Channel, Site 2 |
83% |
3.086uM |
2.815uM |
View
|
| sodium channel, voltage-gated, type IV, beta |
SPIRADOLINE |
Sodium Channel, Site 2 |
83% |
3.086uM |
2.815uM |
View
|
| adrenergic receptor, alpha 2a |
IVERMECTIN |
Adrenergic alpha2A |
83% |
5.8398uM |
2.1899uM |
View
|
| adrenergic receptor, alpha 2a |
QUETIAPINE |
Adrenergic alpha2A |
83% |
2.4914uM |
.9343uM |
View
|
| cholinergic receptor, muscarinic 4 |
QUETIAPINE |
Muscarinic M4 |
83% |
1.5787uM |
.2202uM |
View
|
| adrenergic receptor, alpha 2a |
PROMAZINE |
Imidazoline I2, Central |
83% |
1.098uM |
.732uM |
View
|
| adrenergic receptor, alpha 2c (Non-specific probe) |
PROMAZINE |
Imidazoline I2, Central |
83% |
1.098uM |
.732uM |
View
|
| 5-hydroxytryptamine (serotonin) receptor 2A |
TERCONAZOLE |
Serotonin 5-HT2A |
83% |
8.175uM |
2.336uM |
View
|
| prostaglandin-endoperoxide synthase 1 |
TENOXICAM |
Cyclooxygenase COX-1 |
83% |
1.14uM |
NoneNone |
View
|
| calcium channel, voltage-dependent, L type, alpha 1S subunit |
OXYBUTYNIN |
Calcium Channel Type L, Phenylalkylamine |
81% |
2.358uM |
2.2925uM |
View
|
| calcium channel, voltage-dependent, alpha 1F subunit |
OXYBUTYNIN |
Calcium Channel Type L, Phenylalkylamine |
81% |
2.358uM |
2.2925uM |
View
|
| calcium channel, voltage-dependent, L type, alpha 1D subunit |
OXYBUTYNIN |
Calcium Channel Type L, Phenylalkylamine |
81% |
2.358uM |
2.2925uM |
View
|
| calcium channel, voltage-dependent, L type, alpha 1C subunit |
OXYBUTYNIN |
Calcium Channel Type L, Phenylalkylamine |
81% |
2.358uM |
2.2925uM |
View
|
| calcium channel, voltage-dependent, P/Q type, alpha 1A subunit |
OXYBUTYNIN |
Calcium Channel Type L, Phenylalkylamine |
81% |
2.358uM |
2.2925uM |
View
|
| calcium channel, voltage-dependent, beta 1 subunit |
OXYBUTYNIN |
Calcium Channel Type L, Phenylalkylamine |
81% |
2.358uM |
2.2925uM |
View
|
| calcium channel, voltage-dependent, L type, alpha 1E subunit |
OXYBUTYNIN |
Calcium Channel Type L, Phenylalkylamine |
81% |
2.358uM |
2.2925uM |
View
|
| calcium channel, voltage-dependent, N type, alpha 1B subunit |
OXYBUTYNIN |
Calcium Channel Type L, Phenylalkylamine |
81% |
2.358uM |
2.2925uM |
View
|
| calcium channel, voltage-dependent, alpha2/delta subunit 1 |
OXYBUTYNIN |
Calcium Channel Type L, Phenylalkylamine |
81% |
2.358uM |
2.2925uM |
View
|
| histamine receptor H 2 |
ORPHENADRINE |
Histamine H2 |
81% |
6.961uM |
6.845uM |
View
|
| 5-hydroxytryptamine receptor 6 |
EBASTINE |
Serotonin 5-HT6 |
81% |
2.1974uM |
1.0202uM |
View
|
| cytochrome P450, family 3, subfamily a, polypeptide 13 |
AMPRENAVIR |
CYP450-3A4 Inhibition |
81% |
1uM |
NoneNone |
View
|
| epidermal growth factor receptor |
CETYLPYRIDINIUM BROMIDE |
Protein Tyrosine Kinase, EGF Receptor |
81% |
3.472uM |
NoneNone |
View
|
| thromboxane A synthase 1 |
CETYLPYRIDINIUM BROMIDE |
Thromboxane Synthetase |
81% |
6.452uM |
NoneNone |
View
|
| thromboxane A synthase 1 (platelet, cytochrome P450, family 5, subfamily A) |
CETYLPYRIDINIUM BROMIDE |
Thromboxane Synthetase |
81% |
6.452uM |
NoneNone |
View
|
| tachykinin receptor 2 |
RALOXIFENE |
Tachykinin NK2 |
81% |
3.989uM |
1.33uM |
View
|
| Protein-tyrosine kinase, Fyn |
RALOXIFENE |
Protein Tyrosine Kinase, Fyn |
81% |
3.666uM |
NoneNone |
View
|
| arachidonate 15-lipoxygenase, second type |
PROPOFOL |
Lipoxygenase 15-LO |
81% |
7.596uM |
NoneNone |
View
|
| arachidonate 15-lipoxygenase |
PROPOFOL |
Lipoxygenase 15-LO |
81% |
7.596uM |
NoneNone |
View
|
| arachidonate 15-lipoxygenase |
PROPOFOL |
Lipoxygenase 15-LO |
81% |
7.596uM |
NoneNone |
View
|
| cholinergic receptor, muscarinic 1 |
SB-203580 |
Muscarinic M1 |
81% |
10.666uM |
2.569uM |
View
|
| dopamine receptor D1A |
BAY 11-7085 |
Dopamine D1 |
81% |
4.412uM |
2.206uM |
View
|
| v-erb-b2 erythroblastic leukemia viral oncogene homolog 2, neuro/glioblastoma derived oncogene homolog (avian) |
ASTEMIZOLE |
Protein Tyrosine Kinase, HER2 Receptor |
81% |
13.084uM |
NoneNone |
View
|
| calcium channel, voltage-dependent, beta 1 subunit |
NIFEDIPINE |
Calcium Channel Type L, Benzothiazepine |
81% |
.00867uM |
.007707uM |
View
|
| calcium channel, voltage-dependent, L type, alpha 1E subunit |
NIFEDIPINE |
Calcium Channel Type L, Benzothiazepine |
81% |
.00867uM |
.007707uM |
View
|
| calcium channel, voltage-dependent, N type, alpha 1B subunit |
NIFEDIPINE |
Calcium Channel Type L, Benzothiazepine |
81% |
.00867uM |
.007707uM |
View
|
| calcium channel, voltage-dependent, alpha2/delta subunit 1 |
NIFEDIPINE |
Calcium Channel Type L, Benzothiazepine |
81% |
.00867uM |
.007707uM |
View
|
| 5-hydroxytryptamine (serotonin) receptor 2B |
DICYCLOMINE |
Serotonin 5-HT2B |
81% |
1.301uM |
.828uM |
View
|
| sodium channel, voltage-gated, type IV, beta |
TETRACAINE |
Sodium Channel, Site 2 |
81% |
1.7uM |
1.551uM |
View
|
| sodium channel associated protein 1 |
TETRACAINE |
Sodium Channel, Site 2 |
81% |
1.7uM |
1.551uM |
View
|
| sodium channel associated protein 2 |
TETRACAINE |
Sodium Channel, Site 2 |
81% |
1.7uM |
1.551uM |
View
|
| sodium channel, voltage-gated, type III, beta |
TETRACAINE |
Sodium Channel, Site 2 |
81% |
1.7uM |
1.551uM |
View
|
| sodium channel, voltage-gated, type I, alpha |
TETRACAINE |
Sodium Channel, Site 2 |
81% |
1.7uM |
1.551uM |
View
|
| sodium channel, voltage-gated, type IX, alpha |
TETRACAINE |
Sodium Channel, Site 2 |
81% |
1.7uM |
1.551uM |
View
|
| sodium channel, voltage-gated, type VII, alpha |
TETRACAINE |
Sodium Channel, Site 2 |
81% |
1.7uM |
1.551uM |
View
|
| amiloride-sensitive cation channel 5, intestinal |
TETRACAINE |
Sodium Channel, Site 2 |
81% |
1.7uM |
1.551uM |
View
|
| sodium channel, voltage-gated, type III, beta |
TETRACAINE |
Sodium Channel, Site 2 |
81% |
1.7uM |
1.551uM |
View
|
| sodium channel, voltage-gated, type VIII, alpha polypeptide |
TETRACAINE |
Sodium Channel, Site 2 |
81% |
1.7uM |
1.551uM |
View
|
| sodium channel, voltage-gated, type XI, alpha |
TETRACAINE |
Sodium Channel, Site 2 |
81% |
1.7uM |
1.551uM |
View
|
| sodium channel, voltage-gated, type I, beta |
TETRACAINE |
Sodium Channel, Site 2 |
81% |
1.7uM |
1.551uM |
View
|
| sodium channel, voltage-gated, type 10, alpha polypeptide |
TETRACAINE |
Sodium Channel, Site 2 |
81% |
1.7uM |
1.551uM |
View
|
| sodium channel, voltage-gated, type IV, alpha polypeptide |
TETRACAINE |
Sodium Channel, Site 2 |
81% |
1.7uM |
1.551uM |
View
|
| sodium channel, voltage-gated, type V, alpha polypeptide |
TETRACAINE |
Sodium Channel, Site 2 |
81% |
1.7uM |
1.551uM |
View
|
| sodium channel, voltage-gated, type II, beta |
TETRACAINE |
Sodium Channel, Site 2 |
81% |
1.7uM |
1.551uM |
View
|
| sodium channel, nonvoltage-gated 1 alpha |
TETRACAINE |
Sodium Channel, Site 2 |
81% |
1.7uM |
1.551uM |
View
|
| sodium channel, nonvoltage-gated 1 gamma |
TETRACAINE |
Sodium Channel, Site 2 |
81% |
1.7uM |
1.551uM |
View
|
| sodium channel, nonvoltage-gated 1 beta |
TETRACAINE |
Sodium Channel, Site 2 |
81% |
1.7uM |
1.551uM |
View
|
| sodium channel, voltage-gated, type 2, alpha 1 polypeptide |
TETRACAINE |
Sodium Channel, Site 2 |
81% |
1.7uM |
1.551uM |
View
|
| sodium channel, voltage-gated, type XI, alpha |
TETRACAINE |
Sodium Channel, Site 2 |
81% |
1.7uM |
1.551uM |
View
|
| sodium channel, nonvoltage-gated 1, gamma |
TETRACAINE |
Sodium Channel, Site 2 |
81% |
1.7uM |
1.551uM |
View
|
| sodium channel, nonvoltage-gated 1, delta |
TETRACAINE |
Sodium Channel, Site 2 |
81% |
1.7uM |
1.551uM |
View
|
| calcium channel, voltage-dependent, beta 2 subunit |
DANAZOL |
Calcium Channel Type L, Benzothiazepine |
80% |
14.649uM |
13.021uM |
View
|
| calcium channel, voltage-dependent, L type, alpha 1S subunit |
DANAZOL |
Calcium Channel Type L, Benzothiazepine |
80% |
14.649uM |
13.021uM |
View
|
| calcium channel, voltage-dependent, alpha 1F subunit |
DANAZOL |
Calcium Channel Type L, Benzothiazepine |
80% |
14.649uM |
13.021uM |
View
|
| calcium channel, voltage-dependent, L type, alpha 1D subunit |
DANAZOL |
Calcium Channel Type L, Benzothiazepine |
80% |
14.649uM |
13.021uM |
View
|
| calcium channel, voltage-dependent, L type, alpha 1C subunit |
DANAZOL |
Calcium Channel Type L, Benzothiazepine |
80% |
14.649uM |
13.021uM |
View
|
| calcium channel, voltage-dependent, P/Q type, alpha 1A subunit |
DANAZOL |
Calcium Channel Type L, Benzothiazepine |
80% |
14.649uM |
13.021uM |
View
|
| solute carrier family 6 (neurotransmitter transporter, serotonin), member 4 |
BETA-ESTRADIOL |
Serotonin Transporter |
80% |
10.755uM |
5.714uM |
View
|
| cholinergic receptor, muscarinic 1 |
4-OCTYLPHENOL |
Muscarinic M1 |
80% |
18.013uM |
4.338uM |
View
|
| calcium channel, voltage-dependent, gamma subunit 2 |
PERHEXILINE |
Calcium Channel Type L, Phenylalkylamine |
80% |
1.3499uM |
1.3124uM |
View
|
| calcium channel, voltage-dependent, gamma subunit 1 |
PERHEXILINE |
Calcium Channel Type L, Phenylalkylamine |
80% |
1.3499uM |
1.3124uM |
View
|
| calcium channel, voltage-dependent, beta 4 subunit |
PERHEXILINE |
Calcium Channel Type L, Phenylalkylamine |
80% |
1.3499uM |
1.3124uM |
View
|
| calcium channel, voltage-dependent, beta 3 subunit |
PERHEXILINE |
Calcium Channel Type L, Phenylalkylamine |
80% |
1.3499uM |
1.3124uM |
View
|
| calcium channel, voltage-dependent, beta 2 subunit |
PERHEXILINE |
Calcium Channel Type L, Phenylalkylamine |
80% |
1.3499uM |
1.3124uM |
View
|
| calcium channel, voltage-dependent, L type, alpha 1S subunit |
PERHEXILINE |
Calcium Channel Type L, Phenylalkylamine |
80% |
1.3499uM |
1.3124uM |
View
|
| calcium channel, voltage-dependent, alpha 1F subunit |
PERHEXILINE |
Calcium Channel Type L, Phenylalkylamine |
80% |
1.3499uM |
1.3124uM |
View
|
| calcium channel, voltage-dependent, L type, alpha 1D subunit |
PERHEXILINE |
Calcium Channel Type L, Phenylalkylamine |
80% |
1.3499uM |
1.3124uM |
View
|
| calcium channel, voltage-dependent, L type, alpha 1C subunit |
PERHEXILINE |
Calcium Channel Type L, Phenylalkylamine |
80% |
1.3499uM |
1.3124uM |
View
|
| calcium channel, voltage-dependent, P/Q type, alpha 1A subunit |
PERHEXILINE |
Calcium Channel Type L, Phenylalkylamine |
80% |
1.3499uM |
1.3124uM |
View
|
| calcium channel, voltage-dependent, beta 1 subunit |
PERHEXILINE |
Calcium Channel Type L, Phenylalkylamine |
80% |
1.3499uM |
1.3124uM |
View
|
| calcium channel, voltage-dependent, L type, alpha 1E subunit |
PERHEXILINE |
Calcium Channel Type L, Phenylalkylamine |
80% |
1.3499uM |
1.3124uM |
View
|
| calcium channel, voltage-dependent, N type, alpha 1B subunit |
PERHEXILINE |
Calcium Channel Type L, Phenylalkylamine |
80% |
1.3499uM |
1.3124uM |
View
|
| cytochrome P450, family 3, subfamily a, polypeptide 13 |
DILTIAZEM |
CYP450-3A4 Inhibition |
80% |
1.8366uM |
NoneNone |
View
|
| solute carrier family 6 (neurotransmitter transporter, noradrenalin), member 2 |
PERHEXILINE |
Adrenergic, Norepinephrine Transporter |
80% |
3.2942uM |
3.267uM |
View
|