Gene Activity List


Gene Activity List

Gene Compound Assay Inh Ic50 Ki View
tachykinin receptor 2 TERFENADINE Tachykinin NK2 80% 2.677uM .892uM View
Sigma-2 Receptor THIORIDAZINE Sigma2 80% .845uM .52uM View
Protein-tyrosine kinase, Fyn MONTELUKAST Protein Tyrosine Kinase, Fyn 80% 4.702uM NoneNone View
Protein-tyrosine kinase, Fyn THIORIDAZINE Protein Tyrosine Kinase, Fyn 80% 5.05uM NoneNone View
cholinergic receptor, muscarinic 5 METHAPYRILENE Muscarinic M5 80% 3.265uM 2.346uM View
solute carrier family 6 (neurotransmitter transporter, dopamine), member 3 DIMENHYDRINATE Dopamine Transporter 80% 2.245uM 1.784uM View
solute carrier family 6 (neurotransmitter transporter, dopamine), member 3 METHAPYRILENE Dopamine Transporter 80% 2.757uM 2.19uM View
dopamine receptor D1A FLUNARIZINE Dopamine D1 80% 3.874uM 1.937uM View
cytochrome P450, family 3, subfamily a, polypeptide 13 CISAPRIDE CYP450-3A4 Inhibition 80% .3uM NoneNone View
Cytochrom P450-2D6 monooxygenase METOCLOPRAMIDE CYP450-2D6 Inhibition 80% .8uM NoneNone View
Cytochrom P450-2D6 monooxygenase NALTREXONE CYP450-2D6 Inhibition 80% 1uM NoneNone View
Cytochrom P450-2D6 monooxygenase CLEMASTINE CYP450-2D6 Inhibition 80% 3uM NoneNone View
Cytochrom P450-2C19 monooxygenase CHLORMADINONE ACETATE CYP450-2C19 Inhibition 80% 3uM NoneNone View
solute carrier family 6 (neurotransmitter transporter, serotonin), member 4 DOBUTAMINE Serotonin Transporter 80% 1.895uM 1.006uM View
lymphocyte protein tyrosine kinase (mapped) GRAMICIDIN Protein Tyrosine Kinase, Lck 80% 1.094uM NoneNone View
solute carrier family 6 (neurotransmitter transporter, noradrenalin), member 2 ETHYLESTRENOL Adrenergic, Norepinephrine Transporter 80% 2.098uM 2.08uM View
opioid receptor, sigma 1 QUETIAPINE Sigma1 80% 2.2935uM .9639uM View
calcium channel, voltage-dependent, gamma subunit 1 NITRENDIPINE Calcium Channel Type L, Benzothiazepine 80% .001565uM .001391uM View
calcium channel, voltage-dependent, beta 4 subunit NITRENDIPINE Calcium Channel Type L, Benzothiazepine 80% .001565uM .001391uM View
calcium channel, voltage-dependent, beta 3 subunit NITRENDIPINE Calcium Channel Type L, Benzothiazepine 80% .001565uM .001391uM View
calcium channel, voltage-dependent, beta 2 subunit NITRENDIPINE Calcium Channel Type L, Benzothiazepine 80% .001565uM .001391uM View
calcium channel, voltage-dependent, L type, alpha 1S subunit NITRENDIPINE Calcium Channel Type L, Benzothiazepine 80% .001565uM .001391uM View
calcium channel, voltage-dependent, alpha 1F subunit NITRENDIPINE Calcium Channel Type L, Benzothiazepine 80% .001565uM .001391uM View
calcium channel, voltage-dependent, L type, alpha 1D subunit NITRENDIPINE Calcium Channel Type L, Benzothiazepine 80% .001565uM .001391uM View
calcium channel, voltage-dependent, L type, alpha 1C subunit NITRENDIPINE Calcium Channel Type L, Benzothiazepine 80% .001565uM .001391uM View
prostaglandin-endoperoxide synthase 1 (prostaglandin G/H synthase and cyclooxygenase) TENOXICAM Cyclooxygenase COX-1 83% 1.14uM NoneNone View
adrenergic receptor, alpha 1d (Non-specific probe) CYCLIZINE Adrenergic alpha1D 83% 1.215uM .597uM View
Cytochrom P450-2D6 monooxygenase PAROXETINE CYP450-2D6 Inhibition 83% 1uM NoneNone View
adrenergic receptor, alpha 2a PENTAMIDINE Adrenergic alpha2A 83% 1.375uM .516uM View
solute carrier family 6 (neurotransmitter transporter, noradrenalin), member 2 PENTAMIDINE Adrenergic, Norepinephrine Transporter 83% 2.214uM 2.196uM View
cholinergic receptor, muscarinic 3 PROCHLORPERAZINE Muscarinic M3 83% 1.514uM .321uM View
potassium voltage-gated channel, subfamily H, member 8 DOXAZOSIN Potassium Channel HERG 83% 2.2155uM 1.8151uM View
potassium voltage-gated channel, subfamily H (eag-related), member 6 DOXAZOSIN Potassium Channel HERG 83% 2.2155uM 1.8151uM View
potassium voltage-gated channel, subfamily H (eag-related), member 7 DOXAZOSIN Potassium Channel HERG 83% 2.2155uM 1.8151uM View
potassium voltage-gated channel, subfamily H (eag-related), member 2 DOXAZOSIN Potassium Channel HERG 83% 2.2155uM 1.8151uM View
potassium voltage-gated channel, subfamily H (eag-related), member 5 DOXAZOSIN Potassium Channel HERG 83% 2.2155uM 1.8151uM View
potassium voltage-gated channel, subfamily H (eag-related), member 3 DOXAZOSIN Potassium Channel HERG 83% 2.2155uM 1.8151uM View
potassium voltage-gated channel, subfamily H (eag-related), member 4 DOXAZOSIN Potassium Channel HERG 83% 2.2155uM 1.8151uM View
potassium voltage-gated channel, subfamily H (eag-related), member 1 DOXAZOSIN Potassium Channel HERG 83% 2.2155uM 1.8151uM View
potassium voltage-gated channel, subfamily H (eag-related), member 1 DOXAZOSIN Potassium Channel HERG 83% 2.2155uM 1.8151uM View
potassium voltage-gated channel, subfamily H, member 8 PERPHENAZINE Potassium Channel HERG 83% 4.216uM 3.4541uM View
potassium voltage-gated channel, subfamily H (eag-related), member 6 PERPHENAZINE Potassium Channel HERG 83% 4.216uM 3.4541uM View
potassium voltage-gated channel, subfamily H (eag-related), member 7 PERPHENAZINE Potassium Channel HERG 83% 4.216uM 3.4541uM View
potassium voltage-gated channel, subfamily H (eag-related), member 2 PERPHENAZINE Potassium Channel HERG 83% 4.216uM 3.4541uM View
potassium voltage-gated channel, subfamily H (eag-related), member 5 PERPHENAZINE Potassium Channel HERG 83% 4.216uM 3.4541uM View
potassium voltage-gated channel, subfamily H (eag-related), member 3 PERPHENAZINE Potassium Channel HERG 83% 4.216uM 3.4541uM View
potassium voltage-gated channel, subfamily H (eag-related), member 4 PERPHENAZINE Potassium Channel HERG 83% 4.216uM 3.4541uM View
potassium voltage-gated channel, subfamily H (eag-related), member 1 PERPHENAZINE Potassium Channel HERG 83% 4.216uM 3.4541uM View
potassium voltage-gated channel, subfamily H (eag-related), member 1 PERPHENAZINE Potassium Channel HERG 83% 4.216uM 3.4541uM View
leukotriene B4 receptor 2 SULOCTIDIL Leukotriene B4 83% 1.4405uM .3655uM View
leukotriene B4 receptor SULOCTIDIL Leukotriene B4 83% 1.4405uM .3655uM View
leukotriene B4 receptor SULOCTIDIL Leukotriene B4 83% 1.4405uM .3655uM View
leukotriene B4 receptor 2 SULOCTIDIL Leukotriene B4 83% 1.4405uM .3655uM View
aldo-keto reductase family 1, member B4 (aldose reductase) PIRINIXIC ACID Aldose Reductase 83% 2.8169uM NoneNone View
aldo-keto reductase family 1, member B1 (aldose reductase) PIRINIXIC ACID Aldose Reductase 83% 2.8169uM NoneNone View
aldo-keto reductase family 7, member A2 (aflatoxin aldehyde reductase) PIRINIXIC ACID Aldose Reductase 83% 2.8169uM NoneNone View
aldo-keto reductase family 7, member A3 (aflatoxin aldehyde reductase) PIRINIXIC ACID Aldose Reductase 83% 2.8169uM NoneNone View
opioid receptor, sigma 1 THIORIDAZINE Sigma1 83% .363uM .153uM View
opioid receptor, sigma 1 1,3-DIPHENYLGUANIDINE Sigma1 83% 1.696uM .713uM View
mitogen activated protein kinase 3 IODOQUINOL Protein Serine/Threonine Kinase, ERK1 83% 5.264uM NoneNone View
mitogen-activated protein kinase 3 IODOQUINOL Protein Serine/Threonine Kinase, ERK1 83% 5.264uM NoneNone View
opioid receptor, kappa 1 THIORIDAZINE Opiate kappa 83% 2.49uM .996uM View
solute carrier family 6 (neurotransmitter transporter, dopamine), member 3 PROPAFENONE Dopamine Transporter 83% 1.868uM 1.484uM View
calcium channel, voltage-dependent, L type, alpha 1D subunit CINNARIZINE Calcium Channel Type L, Phenylalkylamine 83% .624uM .607uM View
calcium channel, voltage-dependent, L type, alpha 1C subunit CINNARIZINE Calcium Channel Type L, Phenylalkylamine 83% .624uM .607uM View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit CINNARIZINE Calcium Channel Type L, Phenylalkylamine 83% .624uM .607uM View
calcium channel, voltage-dependent, beta 1 subunit CINNARIZINE Calcium Channel Type L, Phenylalkylamine 83% .624uM .607uM View
calcium channel, voltage-dependent, L type, alpha 1E subunit CINNARIZINE Calcium Channel Type L, Phenylalkylamine 83% .624uM .607uM View
calcium channel, voltage-dependent, N type, alpha 1B subunit CINNARIZINE Calcium Channel Type L, Phenylalkylamine 83% .624uM .607uM View
calcium channel, voltage-dependent, alpha2/delta subunit 1 CINNARIZINE Calcium Channel Type L, Phenylalkylamine 83% .624uM .607uM View
calcium channel, voltage-dependent, gamma subunit 8 CINNARIZINE Calcium Channel Type L, Phenylalkylamine 83% .624uM .607uM View
calcium channel, voltage-dependent, gamma subunit 7 CINNARIZINE Calcium Channel Type L, Phenylalkylamine 83% .624uM .607uM View
calcium channel, voltage-dependent, gamma subunit 6 CINNARIZINE Calcium Channel Type L, Phenylalkylamine 83% .624uM .607uM View
calcium channel, voltage-dependent, gamma subunit 5 CINNARIZINE Calcium Channel Type L, Phenylalkylamine 83% .624uM .607uM View
sodium channel, nonvoltage-gated 1, beta (Liddle syndrome) TETRACAINE Sodium Channel, Site 2 81% 1.7uM 1.551uM View
sodium channel, nonvoltage-gated 1 alpha TETRACAINE Sodium Channel, Site 2 81% 1.7uM 1.551uM View
sodium channel, voltage-gated, type X, alpha TETRACAINE Sodium Channel, Site 2 81% 1.7uM 1.551uM View
sodium channel, voltage-gated, type IX, alpha TETRACAINE Sodium Channel, Site 2 81% 1.7uM 1.551uM View
sodium channel, voltage gated, type VIII, alpha TETRACAINE Sodium Channel, Site 2 81% 1.7uM 1.551uM View
sodium channel, voltage-gated, type VII, alpha TETRACAINE Sodium Channel, Site 2 81% 1.7uM 1.551uM View
sodium channel, voltage-gated, type V, alpha (long QT syndrome 3) TETRACAINE Sodium Channel, Site 2 81% 1.7uM 1.551uM View
sodium channel, voltage-gated, type IV, beta TETRACAINE Sodium Channel, Site 2 81% 1.7uM 1.551uM View
sodium channel, voltage-gated, type IV, alpha TETRACAINE Sodium Channel, Site 2 81% 1.7uM 1.551uM View
sodium channel, voltage-gated, type III, alpha TETRACAINE Sodium Channel, Site 2 81% 1.7uM 1.551uM View
sodium channel, voltage-gated, type II, beta TETRACAINE Sodium Channel, Site 2 81% 1.7uM 1.551uM View
sodium channel, voltage-gated, type II, alpha 2 TETRACAINE Sodium Channel, Site 2 81% 1.7uM 1.551uM View
sodium channel, voltage-gated, type I, beta TETRACAINE Sodium Channel, Site 2 81% 1.7uM 1.551uM View
sodium channel, voltage-gated, type I, alpha TETRACAINE Sodium Channel, Site 2 81% 1.7uM 1.551uM View
cholinergic receptor, muscarinic 2 GALLAMINE TRIETHIODIDE Muscarinic M2 81% 1.999uM .711uM View
solute carrier family 6 (neurotransmitter transporter, noradrenalin), member 2 THIMEROSAL Adrenergic, Norepinephrine Transporter 81% .931uM .923uM View
dopamine receptor D1A BENZOTHIAZYL DISULFIDE Dopamine D1 81% 1.189uM .595uM View
aldo-keto reductase family 1, member B4 (aldose reductase) CAFFEIC ACID PHENETHYL ESTER Aldose Reductase 81% 1.414uM NoneNone View
aldo-keto reductase family 1, member B1 (aldose reductase) CAFFEIC ACID PHENETHYL ESTER Aldose Reductase 81% 1.414uM NoneNone View
aldo-keto reductase family 7, member A2 (aflatoxin aldehyde reductase) CAFFEIC ACID PHENETHYL ESTER Aldose Reductase 81% 1.414uM NoneNone View
aldo-keto reductase family 7, member A3 (aflatoxin aldehyde reductase) CAFFEIC ACID PHENETHYL ESTER Aldose Reductase 81% 1.414uM NoneNone View
prostaglandin-endoperoxide synthase 1 CAPSAICIN Cyclooxygenase COX-1 81% 1.551uM NoneNone View
prostaglandin-endoperoxide synthase 1 (prostaglandin G/H synthase and cyclooxygenase) CAPSAICIN Cyclooxygenase COX-1 81% 1.551uM NoneNone View
solute carrier family 6 (neurotransmitter transporter, noradrenalin), member 2 LABETALOL Adrenergic, Norepinephrine Transporter 81% 3.354uM 3.326uM View
adrenergic receptor, alpha 2c (Non-specific probe) TRAZODONE Adrenergic alpha2C 81% 1.942uM .282uM View
adrenergic receptor, alpha 2b TRAZODONE Adrenergic alpha2C 81% 1.942uM .282uM View
Sigma-2 Receptor TRAZODONE Sigma2 81% 1.342uM .826uM View
aldo-keto reductase family 1, member B4 (aldose reductase) TICRYNAFEN Aldose Reductase 81% 3.206uM NoneNone View
aldo-keto reductase family 1, member B1 (aldose reductase) TICRYNAFEN Aldose Reductase 81% 3.206uM NoneNone View
aldo-keto reductase family 7, member A2 (aflatoxin aldehyde reductase) TICRYNAFEN Aldose Reductase 81% 3.206uM NoneNone View
aldo-keto reductase family 7, member A3 (aflatoxin aldehyde reductase) TICRYNAFEN Aldose Reductase 81% 3.206uM NoneNone View
adrenergic receptor, alpha 2a MOSAPRIDE Adrenergic alpha2A 81% 3.6794uM 1.3798uM View
adrenergic receptor, alpha 1a CITALOPRAM Adrenergic alpha1A 81% 1.756uM .711uM View
adrenergic receptor, alpha 2b LYSERGOL Adrenergic alpha2C 81% 1.61uM .234uM View
adrenergic receptor, alpha 2c (Non-specific probe) LYSERGOL Adrenergic alpha2C 81% 1.61uM .234uM View
Cytochrome P450, subfamily IIC (mephenytoin 4-hydroxylase) 1-(2-CHLOROBENZOYL)-4-(PHENYLMETHYL)-PIPERIDINE CYP450-2C9 Inhibition 81% 2uM NoneNone View
sodium channel, voltage-gated, type II, beta CYCLIZINE Sodium Channel, Site 2 81% 3.091uM 2.82uM View
sodium channel, voltage-gated, type II, alpha 2 CYCLIZINE Sodium Channel, Site 2 81% 3.091uM 2.82uM View
sodium channel, voltage-gated, type I, beta CYCLIZINE Sodium Channel, Site 2 81% 3.091uM 2.82uM View
sodium channel, voltage-gated, type I, alpha CYCLIZINE Sodium Channel, Site 2 81% 3.091uM 2.82uM View
cholinergic receptor, muscarinic 2 HYDROXYCHLOROQUINE Muscarinic M2 81% 2.951uM 1.049uM View
Cytochrome P450, subfamily IIC (mephenytoin 4-hydroxylase) PHENELZINE CYP450-2C9 Inhibition 81% 4uM NoneNone View
cytochrome P450, family 2, subfamily C, polypeptide 9 PHENELZINE CYP450-2C9 Inhibition 81% 4uM NoneNone View
Cytochrom P450-2C19 monooxygenase NORETHINDRONE ACETATE CYP450-2C19 Inhibition 81% .8uM NoneNone View
adrenergic receptor, alpha 2a BERBERINE CHLORIDE Imidazoline I2, Central 81% 1.278uM .852uM View
adrenergic receptor, alpha 2c (Non-specific probe) BERBERINE CHLORIDE Imidazoline I2, Central 81% 1.278uM .852uM View
mu-opioid receptor MOR BITHIONOL Opiate mu 81% 5.507uM 2.236uM View
5-hydroxytryptamine (serotonin) receptor 1A BITHIONOL Serotonin 5-HT1A 81% 5.515uM 3.152uM View
thromboxane A synthase 1 VINBLASTINE Thromboxane Synthetase 81% 1.87uM NoneNone View
thromboxane A synthase 1 (platelet, cytochrome P450, family 5, subfamily A) VINBLASTINE Thromboxane Synthetase 81% 1.87uM NoneNone View
Sigma-2 Receptor DOBUTAMINE Sigma2 81% 2.6uM 1.6uM View
solute carrier family 6 (neurotransmitter transporter, noradrenalin), member 2 BENZTROPINE Adrenergic, Norepinephrine Transporter 81% 1.391uM 1.379uM View
5-hydroxytryptamine (serotonin) receptor 2A BUSPIRONE Serotonin 5-HT2A 81% 2.286uM .653uM View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit NITRENDIPINE Calcium Channel Type L, Benzothiazepine 80% .001565uM .001391uM View
calcium channel, voltage-dependent, beta 1 subunit NITRENDIPINE Calcium Channel Type L, Benzothiazepine 80% .001565uM .001391uM View
calcium channel, voltage-dependent, L type, alpha 1E subunit NITRENDIPINE Calcium Channel Type L, Benzothiazepine 80% .001565uM .001391uM View
calcium channel, voltage-dependent, N type, alpha 1B subunit NITRENDIPINE Calcium Channel Type L, Benzothiazepine 80% .001565uM .001391uM View
calcium channel, voltage-dependent, alpha2/delta subunit 1 NITRENDIPINE Calcium Channel Type L, Benzothiazepine 80% .001565uM .001391uM View
calcium channel, voltage-dependent, gamma subunit 8 NITRENDIPINE Calcium Channel Type L, Benzothiazepine 80% .001565uM .001391uM View
calcium channel, voltage-dependent, gamma subunit 7 NITRENDIPINE Calcium Channel Type L, Benzothiazepine 80% .001565uM .001391uM View
calcium channel, voltage-dependent, gamma subunit 6 NITRENDIPINE Calcium Channel Type L, Benzothiazepine 80% .001565uM .001391uM View
calcium channel, voltage-dependent, gamma subunit 5 NITRENDIPINE Calcium Channel Type L, Benzothiazepine 80% .001565uM .001391uM View
calcium channel, voltage-dependent, gamma subunit 4 NITRENDIPINE Calcium Channel Type L, Benzothiazepine 80% .001565uM .001391uM View
calcium channel, voltage-dependent, gamma subunit 3 NITRENDIPINE Calcium Channel Type L, Benzothiazepine 80% .001565uM .001391uM View
calcium channel, voltage-dependent, gamma subunit 2 NITRENDIPINE Calcium Channel Type L, Benzothiazepine 80% .001565uM .001391uM View
solute carrier family 6 (neurotransmitter transporter, noradrenalin), member 2 NELFINAVIR Adrenergic, Norepinephrine Transporter 80% 8.852uM 8.779uM View
nuclear receptor subfamily 3, group C, member 1 17-METHYLTESTOSTERONE Glucocorticoid 80% 1.843uM .838uM View
adrenergic receptor, alpha 1b TERFENADINE Adrenergic alpha1B 80% 3.335uM 1.846uM View
progesterone receptor FLUOROMETHOLONE Progesterone 80% .815uM .106uM View
progesterone receptor FLUOROMETHOLONE Progesterone 80% .815uM .106uM View
adrenergic receptor, alpha 2a PERGOLIDE Imidazoline I2, Central 80% 3.075uM 2.05uM View
adrenergic receptor, alpha 2c (Non-specific probe) PERGOLIDE Imidazoline I2, Central 80% 3.075uM 2.05uM View
thromboxane A synthase 1 GW-1929 Thromboxane Synthetase 80% 2.953uM NoneNone View
thromboxane A synthase 1 (platelet, cytochrome P450, family 5, subfamily A) GW-1929 Thromboxane Synthetase 80% 2.953uM NoneNone View
sodium channel, voltage-gated, type V, alpha (long QT syndrome 3) PIPAMAZINE Sodium Channel, Site 2 80% 2.686uM 2.451uM View
sodium channel, voltage-gated, type IV, beta PIPAMAZINE Sodium Channel, Site 2 80% 2.686uM 2.451uM View
sodium channel, voltage-gated, type IV, alpha PIPAMAZINE Sodium Channel, Site 2 80% 2.686uM 2.451uM View
potassium voltage-gated channel, subfamily H (eag-related), member 7 RISPERIDONE Potassium Channel HERG 80% 4.1901uM 3.4328uM View
potassium voltage-gated channel, subfamily H (eag-related), member 2 RISPERIDONE Potassium Channel HERG 80% 4.1901uM 3.4328uM View
potassium voltage-gated channel, subfamily H (eag-related), member 5 RISPERIDONE Potassium Channel HERG 80% 4.1901uM 3.4328uM View
potassium voltage-gated channel, subfamily H (eag-related), member 3 RISPERIDONE Potassium Channel HERG 80% 4.1901uM 3.4328uM View
potassium voltage-gated channel, subfamily H (eag-related), member 4 RISPERIDONE Potassium Channel HERG 80% 4.1901uM 3.4328uM View
potassium voltage-gated channel, subfamily H (eag-related), member 1 RISPERIDONE Potassium Channel HERG 80% 4.1901uM 3.4328uM View
potassium voltage-gated channel, subfamily H (eag-related), member 1 RISPERIDONE Potassium Channel HERG 80% 4.1901uM 3.4328uM View
potassium voltage-gated channel, subfamily H, member 8 RISPERIDONE Potassium Channel HERG 80% 4.1901uM 3.4328uM View
potassium voltage-gated channel, subfamily H (eag-related), member 6 RISPERIDONE Potassium Channel HERG 80% 4.1901uM 3.4328uM View
sodium channel, voltage-gated, type IV, beta BW-723C86 Sodium Channel, Site 2 80% 2.1739uM 1.9833uM View
sodium channel, voltage-gated, type IV, alpha BW-723C86 Sodium Channel, Site 2 80% 2.1739uM 1.9833uM View
sodium channel, voltage-gated, type III, alpha BW-723C86 Sodium Channel, Site 2 80% 2.1739uM 1.9833uM View
sodium channel, voltage-gated, type II, beta BW-723C86 Sodium Channel, Site 2 80% 2.1739uM 1.9833uM View
sodium channel, voltage-gated, type II, alpha 2 BW-723C86 Sodium Channel, Site 2 80% 2.1739uM 1.9833uM View
sodium channel, voltage-gated, type I, beta BW-723C86 Sodium Channel, Site 2 80% 2.1739uM 1.9833uM View
sodium channel, voltage-gated, type I, alpha BW-723C86 Sodium Channel, Site 2 80% 2.1739uM 1.9833uM View
sodium channel, voltage-gated, type IV, beta BW-723C86 Sodium Channel, Site 2 80% 2.1739uM 1.9833uM View
sodium channel associated protein 1 BW-723C86 Sodium Channel, Site 2 80% 2.1739uM 1.9833uM View
sodium channel associated protein 2 BW-723C86 Sodium Channel, Site 2 80% 2.1739uM 1.9833uM View
sodium channel, voltage-gated, type III, beta BW-723C86 Sodium Channel, Site 2 80% 2.1739uM 1.9833uM View
sodium channel, voltage-gated, type I, alpha BW-723C86 Sodium Channel, Site 2 80% 2.1739uM 1.9833uM View
sodium channel, voltage-gated, type IX, alpha BW-723C86 Sodium Channel, Site 2 80% 2.1739uM 1.9833uM View
sodium channel, voltage-gated, type VII, alpha BW-723C86 Sodium Channel, Site 2 80% 2.1739uM 1.9833uM View
amiloride-sensitive cation channel 5, intestinal BW-723C86 Sodium Channel, Site 2 80% 2.1739uM 1.9833uM View
sodium channel, voltage-gated, type III, beta BW-723C86 Sodium Channel, Site 2 80% 2.1739uM 1.9833uM View
sodium channel, voltage-gated, type VIII, alpha polypeptide BW-723C86 Sodium Channel, Site 2 80% 2.1739uM 1.9833uM View
calcium channel, voltage-dependent, gamma subunit 4 CINNARIZINE Calcium Channel Type L, Phenylalkylamine 83% .624uM .607uM View
calcium channel, voltage-dependent, gamma subunit 3 CINNARIZINE Calcium Channel Type L, Phenylalkylamine 83% .624uM .607uM View
calcium channel, voltage-dependent, gamma subunit 2 CINNARIZINE Calcium Channel Type L, Phenylalkylamine 83% .624uM .607uM View
calcium channel, voltage-dependent, gamma subunit 1 CINNARIZINE Calcium Channel Type L, Phenylalkylamine 83% .624uM .607uM View
sodium channel, voltage-gated, type IX, alpha PUROMYCIN Sodium Channel, Site 2 12% NoneNone NoneNone View
calcium channel, voltage-dependent, beta 4 subunit CINNARIZINE Calcium Channel Type L, Phenylalkylamine 83% .624uM .607uM View
calcium channel, voltage-dependent, beta 3 subunit CINNARIZINE Calcium Channel Type L, Phenylalkylamine 83% .624uM .607uM View
calcium channel, voltage-dependent, beta 2 subunit CINNARIZINE Calcium Channel Type L, Phenylalkylamine 83% .624uM .607uM View
calcium channel, voltage-dependent, L type, alpha 1S subunit CINNARIZINE Calcium Channel Type L, Phenylalkylamine 83% .624uM .607uM View
calcium channel, voltage-dependent, alpha 1F subunit CINNARIZINE Calcium Channel Type L, Phenylalkylamine 83% .624uM .607uM View
calcium channel, voltage-dependent, gamma subunit 8 FLUNARIZINE Calcium Channel Type L, Benzothiazepine 83% 1.12uM .995uM View
calcium channel, voltage-dependent, gamma subunit 7 FLUNARIZINE Calcium Channel Type L, Benzothiazepine 83% 1.12uM .995uM View
calcium channel, voltage-dependent, gamma subunit 6 FLUNARIZINE Calcium Channel Type L, Benzothiazepine 83% 1.12uM .995uM View
calcium channel, voltage-dependent, gamma subunit 5 FLUNARIZINE Calcium Channel Type L, Benzothiazepine 83% 1.12uM .995uM View
calcium channel, voltage-dependent, gamma subunit 4 FLUNARIZINE Calcium Channel Type L, Benzothiazepine 83% 1.12uM .995uM View
calcium channel, voltage-dependent, gamma subunit 3 FLUNARIZINE Calcium Channel Type L, Benzothiazepine 83% 1.12uM .995uM View
calcium channel, voltage-dependent, gamma subunit 2 FLUNARIZINE Calcium Channel Type L, Benzothiazepine 83% 1.12uM .995uM View
calcium channel, voltage-dependent, gamma subunit 1 FLUNARIZINE Calcium Channel Type L, Benzothiazepine 83% 1.12uM .995uM View
calcium channel, voltage-dependent, beta 4 subunit FLUNARIZINE Calcium Channel Type L, Benzothiazepine 83% 1.12uM .995uM View
calcium channel, voltage-dependent, beta 3 subunit FLUNARIZINE Calcium Channel Type L, Benzothiazepine 83% 1.12uM .995uM View
calcium channel, voltage-dependent, beta 2 subunit FLUNARIZINE Calcium Channel Type L, Benzothiazepine 83% 1.12uM .995uM View
calcium channel, voltage-dependent, L type, alpha 1S subunit FLUNARIZINE Calcium Channel Type L, Benzothiazepine 83% 1.12uM .995uM View
cytochrome P450, family 3, subfamily a, polypeptide 13 VINORELBINE CYP450-3A4 Inhibition 82.5% 1uM NoneNone View