| cytochrome P450, family 2, subfamily C, polypeptide 9 | 
                CLOSANTEL | 
                CYP450-2C9 Inhibition | 
                89% | 
                2uM | 
                NoneNone | 
              
              
                View
               | 
              
            
          
            
                | Cytochrom P450-2C19 monooxygenase | 
                MOSAPRIDE | 
                CYP450-2C19 Inhibition | 
                89% | 
                1uM | 
                NoneNone | 
              
              
                View
               | 
              
            
          
            
                | cholinergic receptor, muscarinic 5 | 
                DIPHENIDOL | 
                Muscarinic M5 | 
                89% | 
                1.191uM | 
                .855uM | 
              
              
                View
               | 
              
            
          
            
                | thromboxane A synthase 1 | 
                BITHIONOL | 
                Thromboxane Synthetase | 
                89% | 
                1.84uM | 
                NoneNone | 
              
              
                View
               | 
              
            
          
            
                | thromboxane A synthase 1 (platelet, cytochrome P450, family 5, subfamily A) | 
                BITHIONOL | 
                Thromboxane Synthetase | 
                89% | 
                1.84uM | 
                NoneNone | 
              
              
                View
               | 
              
            
          
            
                | adrenergic receptor, alpha 2a | 
                AMITRAZ | 
                Adrenergic alpha2A | 
                89% | 
                .9269uM | 
                .3476uM | 
              
              
                View
               | 
              
            
          
            
                | FMS-like tyrosine kinase 1 | 
                DIGITONIN | 
                Vascular Endothelinal Growth Factor (VEGF) | 
                89% | 
                3.859uM | 
                1.001uM | 
              
              
                View
               | 
              
            
          
            
                | fms-related tyrosine kinase 1 (vascular endothelial growth factor/vascular permeability factor receptor) | 
                DIGITONIN | 
                Vascular Endothelinal Growth Factor (VEGF) | 
                89% | 
                3.859uM | 
                1.001uM | 
              
              
                View
               | 
              
            
          
            
                | adrenergic receptor, alpha 2a | 
                DIHYDROERGOCRISTINE MESYLATE | 
                Imidazoline I2, Central | 
                89% | 
                .005428uM | 
                .003619uM | 
              
              
                View
               | 
              
            
          
            
                | adrenergic receptor, alpha 2c (Non-specific probe) | 
                DIHYDROERGOCRISTINE MESYLATE | 
                Imidazoline I2, Central | 
                89% | 
                .005428uM | 
                .003619uM | 
              
              
                View
               | 
              
            
          
            
                | adrenergic receptor, alpha 1b | 
                EPINEPHRINE | 
                Adrenergic alpha1B | 
                89% | 
                1.766uM | 
                .977uM | 
              
              
                View
               | 
              
            
          
            
                | mu-opioid receptor MOR | 
                NELFINAVIR | 
                Opiate mu | 
                89% | 
                14.432uM | 
                5.859uM | 
              
              
                View
               | 
              
            
          
            
                | adrenergic receptor, alpha 1b | 
                CINNARIZINE | 
                Adrenergic alpha1B | 
                89% | 
                .906uM | 
                .502uM | 
              
              
                View
               | 
              
            
          
            
                | 5-hydroxytryptamine receptor 6 | 
                SULFADIMETHOXINE | 
                Serotonin 5-HT6 | 
                87% | 
                1.339uM | 
                .622uM | 
              
              
                View
               | 
              
            
          
            
                | Cytochrom P450-1A2 monooxygenase | 
                PROCHLORPERAZINE | 
                CYP450-1A2 Inhibition | 
                87% | 
                2uM | 
                NoneNone | 
              
              
                View
               | 
              
            
          
            
                | 5-hydroxytryptamine (serotonin) receptor 1A | 
                SAQUINAVIR | 
                Serotonin 5-HT1A | 
                87% | 
                4.273uM | 
                2.442uM | 
              
              
                View
               | 
              
            
          
            
                | adrenergic receptor, alpha 2a | 
                SELEGILINE | 
                Imidazoline I2, Central | 
                87% | 
                1.614uM | 
                1.076uM | 
              
              
                View
               | 
              
            
          
            
                | adrenergic receptor, alpha 2c (Non-specific probe) | 
                SELEGILINE | 
                Imidazoline I2, Central | 
                87% | 
                1.614uM | 
                1.076uM | 
              
              
                View
               | 
              
            
          
            
                | adrenergic receptor, beta 3 | 
                OXICONAZOLE | 
                Adrenergic beta3 | 
                87% | 
                4.7449uM | 
                3.5587uM | 
              
              
                View
               | 
              
            
          
            
                | dopamine receptor D1A | 
                EBASTINE | 
                Dopamine D1 | 
                87% | 
                1.1929uM | 
                .5965uM | 
              
              
                View
               | 
              
            
          
            
                | solute carrier family 6 (neurotransmitter transporter, noradrenalin), member 2 | 
                MONTELUKAST | 
                Adrenergic, Norepinephrine Transporter | 
                87% | 
                2.689uM | 
                2.667uM | 
              
              
                View
               | 
              
            
          
            
                | solute carrier family 6 (neurotransmitter transporter, noradrenalin), member 2 | 
                RESVERATROL | 
                Adrenergic, Norepinephrine Transporter | 
                87% | 
                2.312uM | 
                2.293uM | 
              
              
                View
               | 
              
            
          
            
                | solute carrier family 6 (neurotransmitter transporter, noradrenalin), member 2 | 
                CETYLPYRIDINIUM BROMIDE | 
                Adrenergic, Norepinephrine Transporter | 
                87% | 
                2.653uM | 
                2.631uM | 
              
              
                View
               | 
              
            
          
            
                | opioid receptor, sigma 1 | 
                RALOXIFENE | 
                Sigma1 | 
                87% | 
                .681uM | 
                .286uM | 
              
              
                View
               | 
              
            
          
            
                | 5-hydroxytryptamine (serotonin) receptor 1B | 
                RALOXIFENE | 
                Serotonin 5-HT1B | 
                87% | 
                1.861uM | 
                .846uM | 
              
              
                View
               | 
              
            
          
            
                | solute carrier family 6 (neurotransmitter transporter, dopamine), member 3 | 
                SIBUTRAMINE | 
                Dopamine Transporter | 
                87% | 
                .632uM | 
                .502uM | 
              
              
                View
               | 
              
            
          
            
                | Cytochrome P450, subfamily IIC (mephenytoin 4-hydroxylase) | 
                STANOZOLOL | 
                CYP450-2C9 Inhibition | 
                87% | 
                1.1276uM | 
                NoneNone | 
              
              
                View
               | 
              
            
          
            
                | cytochrome P450, family 2, subfamily C, polypeptide 9 | 
                STANOZOLOL | 
                CYP450-2C9 Inhibition | 
                87% | 
                1.1276uM | 
                NoneNone | 
              
              
                View
               | 
              
            
          
            
                | adrenergic receptor, alpha 2b | 
                BENZETHONIUM CHLORIDE | 
                Adrenergic alpha2B | 
                87% | 
                .643uM | 
                .294uM | 
              
              
                View
               | 
              
            
          
            
                | cholinergic receptor, muscarinic 5 | 
                BENZETHONIUM CHLORIDE | 
                Muscarinic M5 | 
                87% | 
                .134uM | 
                .096uM | 
              
              
                View
               | 
              
            
          
            
                | 5-hydroxytryptamine (serotonin) receptor 1A | 
                ASTEMIZOLE | 
                Serotonin 5-HT1A | 
                87% | 
                .767uM | 
                .438uM | 
              
              
                View
               | 
              
            
          
            
                | nuclear receptor subfamily 3, group C, member 1 | 
                SPIRONOLACTONE | 
                Glucocorticoid | 
                87% | 
                1.9025uM | 
                .8648uM | 
              
              
                View
               | 
              
            
          
            
                | dopamine receptor D3 | 
                BAY 11-7085 | 
                Dopamine D3 | 
                87% | 
                3.46uM | 
                1.175uM | 
              
              
                View
               | 
              
            
          
            
                | 5-hydroxytryptamine receptor 6 | 
                ASTEMIZOLE | 
                Serotonin 5-HT6 | 
                87% | 
                3.266uM | 
                1.516uM | 
              
              
                View
               | 
              
            
          
            
                | Sigma-2 Receptor | 
                CLOMIPHENE | 
                Sigma2 | 
                87% | 
                .049uM | 
                .03uM | 
              
              
                View
               | 
              
            
          
            
                | mitogen activated protein kinase 1 | 
                ANTIMYCIN A | 
                Protein Serine/Threonine Kinase, ERK2 | 
                87% | 
                2.116uM | 
                NoneNone | 
              
              
                View
               | 
              
            
          
            
                | mitogen-activated protein kinase 1 | 
                ANTIMYCIN A | 
                Protein Serine/Threonine Kinase, ERK2 | 
                87% | 
                2.116uM | 
                NoneNone | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, N type, alpha 1B subunit | 
                NELFINAVIR | 
                Calcium Channel Type L, Dihydropyridine | 
                87% | 
                9.84uM | 
                6.324uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, alpha2/delta subunit 1 | 
                NELFINAVIR | 
                Calcium Channel Type L, Dihydropyridine | 
                87% | 
                9.84uM | 
                6.324uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, gamma subunit 8 | 
                NELFINAVIR | 
                Calcium Channel Type L, Dihydropyridine | 
                87% | 
                9.84uM | 
                6.324uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, gamma subunit 7 | 
                NELFINAVIR | 
                Calcium Channel Type L, Dihydropyridine | 
                87% | 
                9.84uM | 
                6.324uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, gamma subunit 6 | 
                NELFINAVIR | 
                Calcium Channel Type L, Dihydropyridine | 
                87% | 
                9.84uM | 
                6.324uM | 
              
              
                View
               | 
              
            
          
            
                | Sigma-2 Receptor | 
                TERBINAFINE | 
                Sigma2 | 
                87% | 
                .0354uM | 
                .0218uM | 
              
              
                View
               | 
              
            
          
            
                | adrenergic receptor, alpha 1d (Non-specific probe) | 
                CINNARIZINE | 
                Adrenergic alpha1D | 
                87% | 
                1.167uM | 
                .573uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, gamma subunit 3 | 
                PAROXETINE | 
                Calcium Channel Type L, Dihydropyridine | 
                87% | 
                1.476uM | 
                .949uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, gamma subunit 2 | 
                PAROXETINE | 
                Calcium Channel Type L, Dihydropyridine | 
                87% | 
                1.476uM | 
                .949uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, gamma subunit 1 | 
                PAROXETINE | 
                Calcium Channel Type L, Dihydropyridine | 
                87% | 
                1.476uM | 
                .949uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, beta 4 subunit | 
                PAROXETINE | 
                Calcium Channel Type L, Dihydropyridine | 
                87% | 
                1.476uM | 
                .949uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, beta 3 subunit | 
                PAROXETINE | 
                Calcium Channel Type L, Dihydropyridine | 
                87% | 
                1.476uM | 
                .949uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, beta 2 subunit | 
                PAROXETINE | 
                Calcium Channel Type L, Dihydropyridine | 
                87% | 
                1.476uM | 
                .949uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, L type, alpha 1S subunit | 
                PAROXETINE | 
                Calcium Channel Type L, Dihydropyridine | 
                87% | 
                1.476uM | 
                .949uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, alpha 1F subunit | 
                PAROXETINE | 
                Calcium Channel Type L, Dihydropyridine | 
                87% | 
                1.476uM | 
                .949uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, L type, alpha 1D subunit | 
                PAROXETINE | 
                Calcium Channel Type L, Dihydropyridine | 
                87% | 
                1.476uM | 
                .949uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, L type, alpha 1C subunit | 
                PAROXETINE | 
                Calcium Channel Type L, Dihydropyridine | 
                87% | 
                1.476uM | 
                .949uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, P/Q type, alpha 1A subunit | 
                PAROXETINE | 
                Calcium Channel Type L, Dihydropyridine | 
                87% | 
                1.476uM | 
                .949uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, beta 1 subunit | 
                PAROXETINE | 
                Calcium Channel Type L, Dihydropyridine | 
                87% | 
                1.476uM | 
                .949uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, L type, alpha 1E subunit | 
                PAROXETINE | 
                Calcium Channel Type L, Dihydropyridine | 
                87% | 
                1.476uM | 
                .949uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, N type, alpha 1B subunit | 
                PAROXETINE | 
                Calcium Channel Type L, Dihydropyridine | 
                87% | 
                1.476uM | 
                .949uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, alpha2/delta subunit 1 | 
                PAROXETINE | 
                Calcium Channel Type L, Dihydropyridine | 
                87% | 
                1.476uM | 
                .949uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, gamma subunit 8 | 
                PAROXETINE | 
                Calcium Channel Type L, Dihydropyridine | 
                87% | 
                1.476uM | 
                .949uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, gamma subunit 7 | 
                PAROXETINE | 
                Calcium Channel Type L, Dihydropyridine | 
                87% | 
                1.476uM | 
                .949uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, gamma subunit 6 | 
                PAROXETINE | 
                Calcium Channel Type L, Dihydropyridine | 
                87% | 
                1.476uM | 
                .949uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, gamma subunit 5 | 
                PAROXETINE | 
                Calcium Channel Type L, Dihydropyridine | 
                87% | 
                1.476uM | 
                .949uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, L type, alpha 1E subunit | 
                U-78517F | 
                Calcium Channel Type L, Dihydropyridine | 
                86% | 
                1.659uM | 
                1.066uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, N type, alpha 1B subunit | 
                U-78517F | 
                Calcium Channel Type L, Dihydropyridine | 
                86% | 
                1.659uM | 
                1.066uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, alpha2/delta subunit 1 | 
                U-78517F | 
                Calcium Channel Type L, Dihydropyridine | 
                86% | 
                1.659uM | 
                1.066uM | 
              
              
                View
               | 
              
            
          
            
                | mitogen activated protein kinase 14 | 
                U-78517F | 
                Protein Serine/Threonine Kinase, p38alpha | 
                86% | 
                5.596uM | 
                NoneNone | 
              
              
                View
               | 
              
            
          
            
                | mitogen-activated protein kinase 14 | 
                U-78517F | 
                Protein Serine/Threonine Kinase, p38alpha | 
                86% | 
                5.596uM | 
                NoneNone | 
              
              
                View
               | 
              
            
          
            
                | cholinergic receptor, muscarinic 3 | 
                AMOXAPINE | 
                Muscarinic M3 | 
                86% | 
                1.781uM | 
                .378uM | 
              
              
                View
               | 
              
            
          
            
                | melanocortin 4 receptor | 
                AMIODARONE | 
                Melanocortin MC4 | 
                86% | 
                13.755uM | 
                13.226uM | 
              
              
                View
               | 
              
            
          
            
                | cholinergic receptor, muscarinic 1 | 
                AMIODARONE | 
                Muscarinic M1 | 
                86% | 
                2.613uM | 
                .629uM | 
              
              
                View
               | 
              
            
          
            
                | epidermal growth factor receptor | 
                TAMOXIFEN | 
                Protein Tyrosine Kinase, EGF Receptor | 
                86% | 
                3.553uM | 
                NoneNone | 
              
              
                View
               | 
              
            
          
            
                | dopamine receptor D3 | 
                DICYCLOMINE | 
                Dopamine D3 | 
                86% | 
                1.21uM | 
                .411uM | 
              
              
                View
               | 
              
            
          
            
                | adrenergic receptor, alpha 1d (Non-specific probe) | 
                CISAPRIDE | 
                Adrenergic alpha1D | 
                86% | 
                .189uM | 
                .093uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, gamma subunit 8 | 
                CLOMIPRAMINE | 
                Calcium Channel Type L, Phenylalkylamine | 
                86% | 
                .506uM | 
                .492uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, gamma subunit 7 | 
                CLOMIPRAMINE | 
                Calcium Channel Type L, Phenylalkylamine | 
                86% | 
                .506uM | 
                .492uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, gamma subunit 6 | 
                CLOMIPRAMINE | 
                Calcium Channel Type L, Phenylalkylamine | 
                86% | 
                .506uM | 
                .492uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, gamma subunit 5 | 
                CLOMIPRAMINE | 
                Calcium Channel Type L, Phenylalkylamine | 
                86% | 
                .506uM | 
                .492uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, gamma subunit 4 | 
                CLOMIPRAMINE | 
                Calcium Channel Type L, Phenylalkylamine | 
                86% | 
                .506uM | 
                .492uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, gamma subunit 3 | 
                CLOMIPRAMINE | 
                Calcium Channel Type L, Phenylalkylamine | 
                86% | 
                .506uM | 
                .492uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, gamma subunit 2 | 
                CLOMIPRAMINE | 
                Calcium Channel Type L, Phenylalkylamine | 
                86% | 
                .506uM | 
                .492uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, gamma subunit 1 | 
                CLOMIPRAMINE | 
                Calcium Channel Type L, Phenylalkylamine | 
                86% | 
                .506uM | 
                .492uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, beta 4 subunit | 
                CLOMIPRAMINE | 
                Calcium Channel Type L, Phenylalkylamine | 
                86% | 
                .506uM | 
                .492uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, beta 3 subunit | 
                CLOMIPRAMINE | 
                Calcium Channel Type L, Phenylalkylamine | 
                86% | 
                .506uM | 
                .492uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, beta 2 subunit | 
                CLOMIPRAMINE | 
                Calcium Channel Type L, Phenylalkylamine | 
                86% | 
                .506uM | 
                .492uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, L type, alpha 1S subunit | 
                CLOMIPRAMINE | 
                Calcium Channel Type L, Phenylalkylamine | 
                86% | 
                .506uM | 
                .492uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, alpha 1F subunit | 
                CLOMIPRAMINE | 
                Calcium Channel Type L, Phenylalkylamine | 
                86% | 
                .506uM | 
                .492uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, L type, alpha 1D subunit | 
                CLOMIPRAMINE | 
                Calcium Channel Type L, Phenylalkylamine | 
                86% | 
                .506uM | 
                .492uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, L type, alpha 1C subunit | 
                CLOMIPRAMINE | 
                Calcium Channel Type L, Phenylalkylamine | 
                86% | 
                .506uM | 
                .492uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, P/Q type, alpha 1A subunit | 
                CLOMIPRAMINE | 
                Calcium Channel Type L, Phenylalkylamine | 
                86% | 
                .506uM | 
                .492uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, beta 1 subunit | 
                CLOMIPRAMINE | 
                Calcium Channel Type L, Phenylalkylamine | 
                86% | 
                .506uM | 
                .492uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, L type, alpha 1E subunit | 
                CLOMIPRAMINE | 
                Calcium Channel Type L, Phenylalkylamine | 
                86% | 
                .506uM | 
                .492uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, N type, alpha 1B subunit | 
                CLOMIPRAMINE | 
                Calcium Channel Type L, Phenylalkylamine | 
                86% | 
                .506uM | 
                .492uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, alpha2/delta subunit 1 | 
                CLOMIPRAMINE | 
                Calcium Channel Type L, Phenylalkylamine | 
                86% | 
                .506uM | 
                .492uM | 
              
              
                View
               | 
              
            
          
            
                | 5-hydroxytryptamine (serotonin) receptor 5B | 
                CARVEDILOL | 
                Serotonin 5-HT4 | 
                86% | 
                1.088uM | 
                .181uM | 
              
              
                View
               | 
              
            
          
            
                | 5-hydroxytryptamine (serotonin) receptor 4 | 
                CARVEDILOL | 
                Serotonin 5-HT4 | 
                86% | 
                1.088uM | 
                .181uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, gamma subunit 8 | 
                CLOZAPINE | 
                Calcium Channel Type L, Benzothiazepine | 
                86% | 
                3.752uM | 
                3.335uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, gamma subunit 7 | 
                CLOZAPINE | 
                Calcium Channel Type L, Benzothiazepine | 
                86% | 
                3.752uM | 
                3.335uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, gamma subunit 6 | 
                CLOZAPINE | 
                Calcium Channel Type L, Benzothiazepine | 
                86% | 
                3.752uM | 
                3.335uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, gamma subunit 5 | 
                CLOZAPINE | 
                Calcium Channel Type L, Benzothiazepine | 
                86% | 
                3.752uM | 
                3.335uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, gamma subunit 4 | 
                CLOZAPINE | 
                Calcium Channel Type L, Benzothiazepine | 
                86% | 
                3.752uM | 
                3.335uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, gamma subunit 3 | 
                CLOZAPINE | 
                Calcium Channel Type L, Benzothiazepine | 
                86% | 
                3.752uM | 
                3.335uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, gamma subunit 2 | 
                CLOZAPINE | 
                Calcium Channel Type L, Benzothiazepine | 
                86% | 
                3.752uM | 
                3.335uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, gamma subunit 1 | 
                CLOZAPINE | 
                Calcium Channel Type L, Benzothiazepine | 
                86% | 
                3.752uM | 
                3.335uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, beta 4 subunit | 
                CLOZAPINE | 
                Calcium Channel Type L, Benzothiazepine | 
                86% | 
                3.752uM | 
                3.335uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, beta 3 subunit | 
                CLOZAPINE | 
                Calcium Channel Type L, Benzothiazepine | 
                86% | 
                3.752uM | 
                3.335uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, beta 2 subunit | 
                CLOZAPINE | 
                Calcium Channel Type L, Benzothiazepine | 
                86% | 
                3.752uM | 
                3.335uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, L type, alpha 1S subunit | 
                CLOZAPINE | 
                Calcium Channel Type L, Benzothiazepine | 
                86% | 
                3.752uM | 
                3.335uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, alpha 1F subunit | 
                CLOZAPINE | 
                Calcium Channel Type L, Benzothiazepine | 
                86% | 
                3.752uM | 
                3.335uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, L type, alpha 1D subunit | 
                CLOZAPINE | 
                Calcium Channel Type L, Benzothiazepine | 
                86% | 
                3.752uM | 
                3.335uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, L type, alpha 1C subunit | 
                FLUNARIZINE | 
                Calcium Channel Type L, Dihydropyridine | 
                90% | 
                1.012uM | 
                .65uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, P/Q type, alpha 1A subunit | 
                FLUNARIZINE | 
                Calcium Channel Type L, Dihydropyridine | 
                90% | 
                1.012uM | 
                .65uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, beta 1 subunit | 
                FLUNARIZINE | 
                Calcium Channel Type L, Dihydropyridine | 
                90% | 
                1.012uM | 
                .65uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, L type, alpha 1E subunit | 
                FLUNARIZINE | 
                Calcium Channel Type L, Dihydropyridine | 
                90% | 
                1.012uM | 
                .65uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, N type, alpha 1B subunit | 
                FLUNARIZINE | 
                Calcium Channel Type L, Dihydropyridine | 
                90% | 
                1.012uM | 
                .65uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, alpha2/delta subunit 1 | 
                FLUNARIZINE | 
                Calcium Channel Type L, Dihydropyridine | 
                90% | 
                1.012uM | 
                .65uM | 
              
              
                View
               | 
              
            
          
            
                | Cytochrom P450-2D6 monooxygenase | 
                TICLOPIDINE | 
                CYP450-2D6 Inhibition | 
                90% | 
                6.2928uM | 
                NoneNone | 
              
              
                View
               | 
              
            
          
            
                | Cytochrom P450-2D6 monooxygenase | 
                YOHIMBINE | 
                CYP450-2D6 Inhibition | 
                90% | 
                2.0317uM | 
                NoneNone | 
              
              
                View
               | 
              
            
          
            
                | Cytochrom P450-2D6 monooxygenase | 
                PHENTOLAMINE | 
                CYP450-2D6 Inhibition | 
                90% | 
                10uM | 
                NoneNone | 
              
              
                View
               | 
              
            
          
            
                | Cytochrom P450-2D6 monooxygenase | 
                PYRILAMINE | 
                CYP450-2D6 Inhibition | 
                90% | 
                .3uM | 
                NoneNone | 
              
              
                View
               | 
              
            
          
            
                | Cytochrom P450-2D6 monooxygenase | 
                CISAPRIDE | 
                CYP450-2D6 Inhibition | 
                90% | 
                .07uM | 
                NoneNone | 
              
              
                View
               | 
              
            
          
            
                | Cytochrome P450, subfamily IIC (mephenytoin 4-hydroxylase) | 
                FELODIPINE | 
                CYP450-2C9 Inhibition | 
                90% | 
                4.5795uM | 
                NoneNone | 
              
              
                View
               | 
              
            
          
            
                | cytochrome P450, family 2, subfamily C, polypeptide 9 | 
                FELODIPINE | 
                CYP450-2C9 Inhibition | 
                90% | 
                4.5795uM | 
                NoneNone | 
              
              
                View
               | 
              
            
          
            
                | mitogen activated protein kinase 1 | 
                3,3',4',5-TETRACHLOROSALICYLANILIDE | 
                Protein Serine/Threonine Kinase, ERK2 | 
                90% | 
                .886uM | 
                NoneNone | 
              
              
                View
               | 
              
            
          
            
                | mitogen-activated protein kinase 1 | 
                3,3',4',5-TETRACHLOROSALICYLANILIDE | 
                Protein Serine/Threonine Kinase, ERK2 | 
                90% | 
                .886uM | 
                NoneNone | 
              
              
                View
               | 
              
            
          
            
                | adenosine A2a receptor | 
                BITHIONOL | 
                Adenosine A2A | 
                90% | 
                1.167uM | 
                .655uM | 
              
              
                View
               | 
              
            
          
            
                | A3 adenosine receptor | 
                CLOSANTEL | 
                Adenosine A3 | 
                90% | 
                .096uM | 
                .054uM | 
              
              
                View
               | 
              
            
          
            
                | acetylcholinesterase (YT blood group) | 
                CLOSANTEL | 
                Acetylcholinesterase | 
                90% | 
                2.951uM | 
                NoneNone | 
              
              
                View
               | 
              
            
          
            
                | collagen-like tail subunit (single strand of homotrimer) of asymmetric acetylcholinesterase | 
                CLOSANTEL | 
                Acetylcholinesterase | 
                90% | 
                2.951uM | 
                NoneNone | 
              
              
                View
               | 
              
            
          
            
                | acetylcholinesterase | 
                CLOSANTEL | 
                Acetylcholinesterase | 
                90% | 
                2.951uM | 
                NoneNone | 
              
              
                View
               | 
              
            
          
            
                | Protein-tyrosine kinase, Fyn | 
                GRAMICIDIN | 
                Protein Tyrosine Kinase, Fyn | 
                90% | 
                3.331uM | 
                NoneNone | 
              
              
                View
               | 
              
            
          
            
                | adrenergic receptor, alpha 2a | 
                CINNARIZINE | 
                Adrenergic alpha2A | 
                90% | 
                .444uM | 
                .167uM | 
              
              
                View
               | 
              
            
          
            
                | 5-hydroxytryptamine (serotonin) receptor 2B | 
                BUSPIRONE | 
                Serotonin 5-HT2B | 
                90% | 
                .75uM | 
                .477uM | 
              
              
                View
               | 
              
            
          
            
                | 5-hydroxytryptamine (serotonin) receptor 1A | 
                QUETIAPINE | 
                Serotonin 5-HT1A | 
                90% | 
                1.4264uM | 
                .8151uM | 
              
              
                View
               | 
              
            
          
            
                | mu-opioid receptor MOR | 
                DIHYDROERGOCRISTINE MESYLATE | 
                Opiate mu | 
                90% | 
                .85uM | 
                .345uM | 
              
              
                View
               | 
              
            
          
            
                | 5-hydroxytryptamine (serotonin) receptor 2A | 
                PYRILAMINE | 
                Serotonin 5-HT2A | 
                90% | 
                .997uM | 
                .285uM | 
              
              
                View
               | 
              
            
          
            
                | dopamine receptor 2 | 
                PROMAZINE | 
                Dopamine D2L | 
                90% | 
                .505uM | 
                .168uM | 
              
              
                View
               | 
              
            
          
            
                | adrenergic receptor, alpha 2a | 
                TERCONAZOLE | 
                Imidazoline I2, Central | 
                90% | 
                2.226uM | 
                1.484uM | 
              
              
                View
               | 
              
            
          
            
                | gamma-aminobutyric acid (GABA-A) receptor, subunit alpha 3 | 
                CHLORDIAZEPOXIDE | 
                GABAA, Benzodiazepine, Central | 
                89% | 
                1.429uM | 
                1.164uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, beta 2 subunit | 
                PROMETHAZINE | 
                Calcium Channel Type L, Phenylalkylamine | 
                89% | 
                .866uM | 
                .842uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, L type, alpha 1S subunit | 
                PROMETHAZINE | 
                Calcium Channel Type L, Phenylalkylamine | 
                89% | 
                .866uM | 
                .842uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, alpha 1F subunit | 
                PROMETHAZINE | 
                Calcium Channel Type L, Phenylalkylamine | 
                89% | 
                .866uM | 
                .842uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, L type, alpha 1D subunit | 
                PROMETHAZINE | 
                Calcium Channel Type L, Phenylalkylamine | 
                89% | 
                .866uM | 
                .842uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, L type, alpha 1C subunit | 
                PROMETHAZINE | 
                Calcium Channel Type L, Phenylalkylamine | 
                89% | 
                .866uM | 
                .842uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, P/Q type, alpha 1A subunit | 
                PROMETHAZINE | 
                Calcium Channel Type L, Phenylalkylamine | 
                89% | 
                .866uM | 
                .842uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, beta 1 subunit | 
                PROMETHAZINE | 
                Calcium Channel Type L, Phenylalkylamine | 
                89% | 
                .866uM | 
                .842uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, L type, alpha 1E subunit | 
                PROMETHAZINE | 
                Calcium Channel Type L, Phenylalkylamine | 
                89% | 
                .866uM | 
                .842uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, N type, alpha 1B subunit | 
                PROMETHAZINE | 
                Calcium Channel Type L, Phenylalkylamine | 
                89% | 
                .866uM | 
                .842uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, alpha2/delta subunit 1 | 
                PROMETHAZINE | 
                Calcium Channel Type L, Phenylalkylamine | 
                89% | 
                .866uM | 
                .842uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, gamma subunit 8 | 
                PROMETHAZINE | 
                Calcium Channel Type L, Phenylalkylamine | 
                89% | 
                .866uM | 
                .842uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, gamma subunit 7 | 
                PROMETHAZINE | 
                Calcium Channel Type L, Phenylalkylamine | 
                89% | 
                .866uM | 
                .842uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, gamma subunit 6 | 
                PROMETHAZINE | 
                Calcium Channel Type L, Phenylalkylamine | 
                89% | 
                .866uM | 
                .842uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, gamma subunit 5 | 
                PROMETHAZINE | 
                Calcium Channel Type L, Phenylalkylamine | 
                89% | 
                .866uM | 
                .842uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, gamma subunit 4 | 
                PROMETHAZINE | 
                Calcium Channel Type L, Phenylalkylamine | 
                89% | 
                .866uM | 
                .842uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, gamma subunit 3 | 
                PROMETHAZINE | 
                Calcium Channel Type L, Phenylalkylamine | 
                89% | 
                .866uM | 
                .842uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, gamma subunit 2 | 
                PROMETHAZINE | 
                Calcium Channel Type L, Phenylalkylamine | 
                89% | 
                .866uM | 
                .842uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, gamma subunit 1 | 
                PROMETHAZINE | 
                Calcium Channel Type L, Phenylalkylamine | 
                89% | 
                .866uM | 
                .842uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, beta 4 subunit | 
                PROMETHAZINE | 
                Calcium Channel Type L, Phenylalkylamine | 
                89% | 
                .866uM | 
                .842uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, beta 3 subunit | 
                PROMETHAZINE | 
                Calcium Channel Type L, Phenylalkylamine | 
                89% | 
                .866uM | 
                .842uM | 
              
              
                View
               | 
              
            
          
            
                | A3 adenosine receptor | 
                LACIDIPINE | 
                Adenosine A3 | 
                89% | 
                4.036uM | 
                2.281uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, beta 3 subunit | 
                HALOPERIDOL | 
                Calcium Channel Type L, Phenylalkylamine | 
                88% | 
                .552uM | 
                .536uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, beta 2 subunit | 
                HALOPERIDOL | 
                Calcium Channel Type L, Phenylalkylamine | 
                88% | 
                .552uM | 
                .536uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, L type, alpha 1S subunit | 
                HALOPERIDOL | 
                Calcium Channel Type L, Phenylalkylamine | 
                88% | 
                .552uM | 
                .536uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, alpha 1F subunit | 
                HALOPERIDOL | 
                Calcium Channel Type L, Phenylalkylamine | 
                88% | 
                .552uM | 
                .536uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, L type, alpha 1D subunit | 
                HALOPERIDOL | 
                Calcium Channel Type L, Phenylalkylamine | 
                88% | 
                .552uM | 
                .536uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, L type, alpha 1C subunit | 
                HALOPERIDOL | 
                Calcium Channel Type L, Phenylalkylamine | 
                88% | 
                .552uM | 
                .536uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, P/Q type, alpha 1A subunit | 
                HALOPERIDOL | 
                Calcium Channel Type L, Phenylalkylamine | 
                88% | 
                .552uM | 
                .536uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, beta 1 subunit | 
                HALOPERIDOL | 
                Calcium Channel Type L, Phenylalkylamine | 
                88% | 
                .552uM | 
                .536uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, L type, alpha 1E subunit | 
                HALOPERIDOL | 
                Calcium Channel Type L, Phenylalkylamine | 
                88% | 
                .552uM | 
                .536uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, N type, alpha 1B subunit | 
                HALOPERIDOL | 
                Calcium Channel Type L, Phenylalkylamine | 
                88% | 
                .552uM | 
                .536uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, alpha2/delta subunit 1 | 
                HALOPERIDOL | 
                Calcium Channel Type L, Phenylalkylamine | 
                88% | 
                .552uM | 
                .536uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, gamma subunit 8 | 
                HALOPERIDOL | 
                Calcium Channel Type L, Phenylalkylamine | 
                88% | 
                .552uM | 
                .536uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, gamma subunit 7 | 
                HALOPERIDOL | 
                Calcium Channel Type L, Phenylalkylamine | 
                88% | 
                .552uM | 
                .536uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, gamma subunit 6 | 
                HALOPERIDOL | 
                Calcium Channel Type L, Phenylalkylamine | 
                88% | 
                .552uM | 
                .536uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, gamma subunit 5 | 
                HALOPERIDOL | 
                Calcium Channel Type L, Phenylalkylamine | 
                88% | 
                .552uM | 
                .536uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, gamma subunit 4 | 
                HALOPERIDOL | 
                Calcium Channel Type L, Phenylalkylamine | 
                88% | 
                .552uM | 
                .536uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, gamma subunit 3 | 
                HALOPERIDOL | 
                Calcium Channel Type L, Phenylalkylamine | 
                88% | 
                .552uM | 
                .536uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, gamma subunit 2 | 
                HALOPERIDOL | 
                Calcium Channel Type L, Phenylalkylamine | 
                88% | 
                .552uM | 
                .536uM | 
              
              
                View
               | 
              
            
          
            
                | calcium channel, voltage-dependent, gamma subunit 1 | 
                HALOPERIDOL | 
                Calcium Channel Type L, Phenylalkylamine | 
                88% | 
                .552uM | 
                .536uM | 
              
              
                View
               | 
              
            
          
            
                | Protein-tyrosine kinase, Fyn | 
                GENTIAN VIOLET | 
                Protein Tyrosine Kinase, Fyn | 
                88% | 
                2.148uM | 
                NoneNone | 
              
              
                View
               | 
              
            
          
            
                | opioid receptor, sigma 1 | 
                MEPAZINE | 
                Sigma1 | 
                88% | 
                .18uM | 
                .076uM | 
              
              
                View
               | 
              
            
          
            
                | dopamine receptor D3 | 
                LOPERAMIDE | 
                Dopamine D3 | 
                88% | 
                1.337uM | 
                .454uM | 
              
              
                View
               | 
              
            
          
            
                | opioid receptor, delta 1 | 
                LOPERAMIDE | 
                Opiate delta | 
                88% | 
                .896uM | 
                .316uM | 
              
              
                View
               | 
              
            
          
            
                | dopamine receptor D1A | 
                METHYSERGIDE | 
                Dopamine D1 | 
                88% | 
                .943uM | 
                .472uM | 
              
              
                View
               | 
              
            
          
            
                | arachidonate 15-lipoxygenase, second type | 
                MITOXANTRONE | 
                Lipoxygenase 15-LO | 
                88% | 
                1.7853uM | 
                NoneNone | 
              
              
                View
               | 
              
            
          
            
                | arachidonate 15-lipoxygenase | 
                MITOXANTRONE | 
                Lipoxygenase 15-LO | 
                88% | 
                1.7853uM | 
                NoneNone | 
              
              
                View
               | 
              
            
          
            
                | arachidonate 15-lipoxygenase | 
                MITOXANTRONE | 
                Lipoxygenase 15-LO | 
                88% | 
                1.7853uM | 
                NoneNone | 
              
              
                View
               | 
              
            
          
            
                | epidermal growth factor receptor | 
                L-744832 | 
                Protein Tyrosine Kinase, EGF Receptor | 
                88% | 
                3.216uM | 
                NoneNone | 
              
              
                View
               | 
              
            
          
            
                | matrix metalloproteinase 1 (interstitial collagenase) | 
                IRINOTECAN | 
                Protease, Matrix Metalloprotease-1 (MMP-1) | 
                88% | 
                6.06uM | 
                NoneNone | 
              
              
                View
               | 
              
            
          
            
                | 5-hydroxytryptamine receptor 6 | 
                KETOTIFEN | 
                Serotonin 5-HT6 | 
                88% | 
                1.141uM | 
                .53uM | 
              
              
                View
               | 
              
            
          
            
                | adrenergic receptor, alpha 2a | 
                KETOTIFEN | 
                Adrenergic alpha2A | 
                88% | 
                2.187uM | 
                .82uM | 
              
              
                View
               | 
              
            
          
            
                | thromboxane A synthase 1 | 
                RITONAVIR | 
                Thromboxane Synthetase | 
                88% | 
                .076uM | 
                NoneNone | 
              
              
                View
               | 
              
            
          
            
                | thromboxane A synthase 1 (platelet, cytochrome P450, family 5, subfamily A) | 
                RITONAVIR | 
                Thromboxane Synthetase | 
                88% | 
                .076uM | 
                NoneNone | 
              
              
                View
               | 
              
            
          
            
                | adrenergic receptor, beta 3 | 
                MONTELUKAST | 
                Adrenergic beta3 | 
                88% | 
                4.3uM | 
                3.2uM | 
              
              
                View
               | 
              
            
          
            
                | phosphodiesterase 4A, cAMP specific | 
                PAPAVERINE | 
                Phosphodiesterase PDE4 | 
                88% | 
                .817uM | 
                NoneNone | 
              
              
                View
               | 
              
            
          
            
                | phosphodiesterase 4C, cAMP-specific | 
                PAPAVERINE | 
                Phosphodiesterase PDE4 | 
                88% | 
                .817uM | 
                NoneNone | 
              
              
                View
               | 
              
            
          
            
                | phosphodiesterase 4D | 
                PAPAVERINE | 
                Phosphodiesterase PDE4 | 
                88% | 
                .817uM | 
                NoneNone | 
              
              
                View
               | 
              
            
          
            
                | phosphodiesterase 4B, cAMP specific | 
                PAPAVERINE | 
                Phosphodiesterase PDE4 | 
                88% | 
                .817uM | 
                NoneNone | 
              
              
                View
               | 
              
            
          
            
                | phosphodiesterase 3B | 
                PAPAVERINE | 
                Phosphodiesterase PDE3 | 
                88% | 
                .665uM | 
                NoneNone | 
              
              
                View
               | 
              
            
          
            
                | phosphodiesterase 3A | 
                PAPAVERINE | 
                Phosphodiesterase PDE3 | 
                88% | 
                .665uM | 
                NoneNone | 
              
              
                View
               |