Gene Activity List


Gene Activity List

Gene Compound Assay Inh Ic50 Ki View
thromboxane A synthase 1 ROSIGLITAZONE Thromboxane Synthetase 88% 3.56uM NoneNone View
thromboxane A synthase 1 (platelet, cytochrome P450, family 5, subfamily A) ROSIGLITAZONE Thromboxane Synthetase 88% 3.56uM NoneNone View
adrenergic receptor, alpha 1d (Non-specific probe) DOMPERIDONE Adrenergic alpha1D 88% 1.065uM .524uM View
sodium channel, voltage gated, type VIII, alpha PERGOLIDE Sodium Channel, Site 2 88% 1.728uM 1.577uM View
sodium channel, voltage-gated, type VII, alpha PERGOLIDE Sodium Channel, Site 2 88% 1.728uM 1.577uM View
sodium channel, voltage-gated, type V, alpha (long QT syndrome 3) PERGOLIDE Sodium Channel, Site 2 88% 1.728uM 1.577uM View
sodium channel, voltage-gated, type IV, beta PERGOLIDE Sodium Channel, Site 2 88% 1.728uM 1.577uM View
sodium channel, voltage-gated, type IV, alpha PERGOLIDE Sodium Channel, Site 2 88% 1.728uM 1.577uM View
sodium channel, voltage-gated, type III, alpha PERGOLIDE Sodium Channel, Site 2 88% 1.728uM 1.577uM View
sodium channel, voltage-gated, type II, beta PERGOLIDE Sodium Channel, Site 2 88% 1.728uM 1.577uM View
sodium channel, voltage-gated, type II, alpha 2 PERGOLIDE Sodium Channel, Site 2 88% 1.728uM 1.577uM View
sodium channel, voltage-gated, type I, beta PERGOLIDE Sodium Channel, Site 2 88% 1.728uM 1.577uM View
sodium channel, voltage-gated, type I, alpha PERGOLIDE Sodium Channel, Site 2 88% 1.728uM 1.577uM View
sodium channel, voltage-gated, type IV, beta PERGOLIDE Sodium Channel, Site 2 88% 1.728uM 1.577uM View
sodium channel associated protein 1 PERGOLIDE Sodium Channel, Site 2 88% 1.728uM 1.577uM View
sodium channel associated protein 2 PERGOLIDE Sodium Channel, Site 2 88% 1.728uM 1.577uM View
sodium channel, voltage-gated, type III, beta PERGOLIDE Sodium Channel, Site 2 88% 1.728uM 1.577uM View
sodium channel, voltage-gated, type I, alpha PERGOLIDE Sodium Channel, Site 2 88% 1.728uM 1.577uM View
sodium channel, voltage-gated, type IX, alpha PERGOLIDE Sodium Channel, Site 2 88% 1.728uM 1.577uM View
sodium channel, voltage-gated, type VII, alpha PERGOLIDE Sodium Channel, Site 2 88% 1.728uM 1.577uM View
calcium channel, voltage-dependent, gamma subunit 7 CLOMIPHENE Calcium Channel Type L, Phenylalkylamine 86% .754uM .733uM View
calcium channel, voltage-dependent, gamma subunit 6 CLOMIPHENE Calcium Channel Type L, Phenylalkylamine 86% .754uM .733uM View
calcium channel, voltage-dependent, gamma subunit 5 CLOMIPHENE Calcium Channel Type L, Phenylalkylamine 86% .754uM .733uM View
calcium channel, voltage-dependent, gamma subunit 4 CLOMIPHENE Calcium Channel Type L, Phenylalkylamine 86% .754uM .733uM View
calcium channel, voltage-dependent, gamma subunit 3 CLOMIPHENE Calcium Channel Type L, Phenylalkylamine 86% .754uM .733uM View
calcium channel, voltage-dependent, gamma subunit 2 CLOMIPHENE Calcium Channel Type L, Phenylalkylamine 86% .754uM .733uM View
calcium channel, voltage-dependent, gamma subunit 1 CLOMIPHENE Calcium Channel Type L, Phenylalkylamine 86% .754uM .733uM View
calcium channel, voltage-dependent, beta 4 subunit CLOMIPHENE Calcium Channel Type L, Phenylalkylamine 86% .754uM .733uM View
calcium channel, voltage-dependent, beta 3 subunit CLOMIPHENE Calcium Channel Type L, Phenylalkylamine 86% .754uM .733uM View
calcium channel, voltage-dependent, beta 2 subunit CLOMIPHENE Calcium Channel Type L, Phenylalkylamine 86% .754uM .733uM View
calcium channel, voltage-dependent, L type, alpha 1S subunit CLOMIPHENE Calcium Channel Type L, Phenylalkylamine 86% .754uM .733uM View
calcium channel, voltage-dependent, alpha 1F subunit CLOMIPHENE Calcium Channel Type L, Phenylalkylamine 86% .754uM .733uM View
calcium channel, voltage-dependent, L type, alpha 1D subunit CLOMIPHENE Calcium Channel Type L, Phenylalkylamine 86% .754uM .733uM View
calcium channel, voltage-dependent, L type, alpha 1C subunit CLOMIPHENE Calcium Channel Type L, Phenylalkylamine 86% .754uM .733uM View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit CLOMIPHENE Calcium Channel Type L, Phenylalkylamine 86% .754uM .733uM View
calcium channel, voltage-dependent, beta 1 subunit CLOMIPHENE Calcium Channel Type L, Phenylalkylamine 86% .754uM .733uM View
calcium channel, voltage-dependent, L type, alpha 1E subunit CLOMIPHENE Calcium Channel Type L, Phenylalkylamine 86% .754uM .733uM View
calcium channel, voltage-dependent, N type, alpha 1B subunit CLOMIPHENE Calcium Channel Type L, Phenylalkylamine 86% .754uM .733uM View
calcium channel, voltage-dependent, alpha2/delta subunit 1 CLOMIPHENE Calcium Channel Type L, Phenylalkylamine 86% .754uM .733uM View
5-hydroxytryptamine receptor 6 S-(-)-PROPRANOLOL Serotonin 5-HT6 86% .998uM .463uM View
aldo-keto reductase family 1, member B4 (aldose reductase) TROGLITAZONE Aldose Reductase 86% 2.038uM NoneNone View
aldo-keto reductase family 1, member B1 (aldose reductase) TROGLITAZONE Aldose Reductase 86% 2.038uM NoneNone View
aldo-keto reductase family 7, member A2 (aflatoxin aldehyde reductase) TROGLITAZONE Aldose Reductase 86% 2.038uM NoneNone View
aldo-keto reductase family 7, member A3 (aflatoxin aldehyde reductase) TROGLITAZONE Aldose Reductase 86% 2.038uM NoneNone View
sodium channel, voltage-gated, type IV, beta PROMETHAZINE Sodium Channel, Site 2 86% 2.37uM 2.162uM View
sodium channel associated protein 1 PROMETHAZINE Sodium Channel, Site 2 86% 2.37uM 2.162uM View
sodium channel associated protein 2 PROMETHAZINE Sodium Channel, Site 2 86% 2.37uM 2.162uM View
sodium channel, voltage-gated, type III, beta PROMETHAZINE Sodium Channel, Site 2 86% 2.37uM 2.162uM View
sodium channel, voltage-gated, type I, alpha PROMETHAZINE Sodium Channel, Site 2 86% 2.37uM 2.162uM View
sodium channel, voltage-gated, type IX, alpha PROMETHAZINE Sodium Channel, Site 2 86% 2.37uM 2.162uM View
sodium channel, voltage-gated, type VII, alpha PROMETHAZINE Sodium Channel, Site 2 86% 2.37uM 2.162uM View
amiloride-sensitive cation channel 5, intestinal PROMETHAZINE Sodium Channel, Site 2 86% 2.37uM 2.162uM View
sodium channel, voltage-gated, type III, beta PROMETHAZINE Sodium Channel, Site 2 86% 2.37uM 2.162uM View
sodium channel, voltage-gated, type VIII, alpha polypeptide PROMETHAZINE Sodium Channel, Site 2 86% 2.37uM 2.162uM View
sodium channel, voltage-gated, type XI, alpha PROMETHAZINE Sodium Channel, Site 2 86% 2.37uM 2.162uM View
sodium channel, voltage-gated, type I, beta PROMETHAZINE Sodium Channel, Site 2 86% 2.37uM 2.162uM View
sodium channel, voltage-gated, type 10, alpha polypeptide PROMETHAZINE Sodium Channel, Site 2 86% 2.37uM 2.162uM View
sodium channel, voltage-gated, type IV, alpha polypeptide PROMETHAZINE Sodium Channel, Site 2 86% 2.37uM 2.162uM View
sodium channel, voltage-gated, type V, alpha polypeptide PROMETHAZINE Sodium Channel, Site 2 86% 2.37uM 2.162uM View
sodium channel, voltage-gated, type II, beta PROMETHAZINE Sodium Channel, Site 2 86% 2.37uM 2.162uM View
sodium channel, nonvoltage-gated 1 alpha PROMETHAZINE Sodium Channel, Site 2 86% 2.37uM 2.162uM View
sodium channel, nonvoltage-gated 1 gamma PROMETHAZINE Sodium Channel, Site 2 86% 2.37uM 2.162uM View
sodium channel, nonvoltage-gated 1 beta PROMETHAZINE Sodium Channel, Site 2 86% 2.37uM 2.162uM View
sodium channel, voltage-gated, type 2, alpha 1 polypeptide PROMETHAZINE Sodium Channel, Site 2 86% 2.37uM 2.162uM View
sodium channel, voltage-gated, type XI, alpha PROMETHAZINE Sodium Channel, Site 2 86% 2.37uM 2.162uM View
sodium channel, nonvoltage-gated 1, gamma PROMETHAZINE Sodium Channel, Site 2 86% 2.37uM 2.162uM View
sodium channel, nonvoltage-gated 1, delta PROMETHAZINE Sodium Channel, Site 2 86% 2.37uM 2.162uM View
sodium channel, nonvoltage-gated 1, beta (Liddle syndrome) PROMETHAZINE Sodium Channel, Site 2 86% 2.37uM 2.162uM View
sodium channel, nonvoltage-gated 1 alpha PROMETHAZINE Sodium Channel, Site 2 86% 2.37uM 2.162uM View
sodium channel, voltage-gated, type XI, alpha THIORIDAZINE Sodium Channel, Site 2 86% 2.056uM 1.876uM View
sodium channel, nonvoltage-gated 1, gamma THIORIDAZINE Sodium Channel, Site 2 86% 2.056uM 1.876uM View
sodium channel, nonvoltage-gated 1, delta THIORIDAZINE Sodium Channel, Site 2 86% 2.056uM 1.876uM View
amiloride-sensitive cation channel 5, intestinal PUROMYCIN Sodium Channel, Site 2 12% NoneNone NoneNone View
sodium channel, nonvoltage-gated 1, beta (Liddle syndrome) THIORIDAZINE Sodium Channel, Site 2 86% 2.056uM 1.876uM View
sodium channel, nonvoltage-gated 1 alpha THIORIDAZINE Sodium Channel, Site 2 86% 2.056uM 1.876uM View
sodium channel, voltage-gated, type X, alpha THIORIDAZINE Sodium Channel, Site 2 86% 2.056uM 1.876uM View
sodium channel, voltage-gated, type IX, alpha THIORIDAZINE Sodium Channel, Site 2 86% 2.056uM 1.876uM View
sodium channel, voltage gated, type VIII, alpha THIORIDAZINE Sodium Channel, Site 2 86% 2.056uM 1.876uM View
sodium channel, voltage-gated, type VII, alpha THIORIDAZINE Sodium Channel, Site 2 86% 2.056uM 1.876uM View
sodium channel, voltage-gated, type V, alpha (long QT syndrome 3) THIORIDAZINE Sodium Channel, Site 2 86% 2.056uM 1.876uM View
sodium channel, voltage-gated, type IV, beta THIORIDAZINE Sodium Channel, Site 2 86% 2.056uM 1.876uM View
sodium channel, voltage-gated, type IV, alpha THIORIDAZINE Sodium Channel, Site 2 86% 2.056uM 1.876uM View
sodium channel, voltage-gated, type III, alpha THIORIDAZINE Sodium Channel, Site 2 86% 2.056uM 1.876uM View
sodium channel, voltage-gated, type II, beta THIORIDAZINE Sodium Channel, Site 2 86% 2.056uM 1.876uM View
sodium channel, voltage-gated, type II, alpha 2 THIORIDAZINE Sodium Channel, Site 2 86% 2.056uM 1.876uM View
sodium channel, voltage-gated, type I, beta THIORIDAZINE Sodium Channel, Site 2 86% 2.056uM 1.876uM View
sodium channel, voltage-gated, type I, alpha THIORIDAZINE Sodium Channel, Site 2 86% 2.056uM 1.876uM View
opioid receptor, sigma 1 LEVOBUNOLOL Sigma1 86% .773uM .325uM View
opioid receptor, sigma 1 VALETHAMATE BROMIDE Sigma1 86% .475uM .2uM View
solute carrier family 6 (neurotransmitter transporter, serotonin), member 4 IMATINIB Serotonin Transporter 86% 1.402uM .745uM View
5-hydroxytryptamine receptor 6 THIORIDAZINE Serotonin 5-HT6 86% .071uM .033uM View
5-hydroxytryptamine (serotonin) receptor 2C DOMPERIDONE Serotonin 5-HT2C 86% 1.332uM .698uM View
cholinergic receptor, muscarinic 2 METHAPYRILENE Muscarinic M2 86% 1.665uM .592uM View
estrogen receptor 1 4-NONYLPHENOL Estrogen ERalpha 86% .377uM .108uM View
estrogen receptor 1 4-NONYLPHENOL Estrogen ERalpha 86% .377uM .108uM View
Cytochrom P450-2D6 monooxygenase ORPHENADRINE CYP450-2D6 Inhibition 86% .4uM NoneNone View
Cytochrome P450, subfamily IIC (mephenytoin 4-hydroxylase) RAPAMYCIN CYP450-2C9 Inhibition 86% 2uM NoneNone View
cytochrome P450, family 2, subfamily C, polypeptide 9 RAPAMYCIN CYP450-2C9 Inhibition 86% 2uM NoneNone View
Cytochrome P450, subfamily IIC (mephenytoin 4-hydroxylase) MOSAPRIDE CYP450-2C9 Inhibition 86% 1uM NoneNone View
cytochrome P450, family 2, subfamily C, polypeptide 9 MOSAPRIDE CYP450-2C9 Inhibition 86% 1uM NoneNone View
Cytochrome P450, subfamily IIC (mephenytoin 4-hydroxylase) TENIDAP CYP450-2C9 Inhibition 86% .7uM NoneNone View
cytochrome P450, family 2, subfamily C, polypeptide 9 TENIDAP CYP450-2C9 Inhibition 86% .7uM NoneNone View
Sigma-2 Receptor BERBERINE CHLORIDE Sigma2 86% .095uM .059uM View
tachykinin receptor 2 DOCETAXEL Tachykinin NK2 86% 1.563uM .521uM View
cholinergic receptor, muscarinic 2 PROMAZINE Muscarinic M2 86% 1.089uM .387uM View
Sigma-2 Receptor TERCONAZOLE Sigma2 86% .317uM .195uM View
solute carrier family 6 (neurotransmitter transporter, dopamine), member 3 VX-745 Dopamine Transporter 86% 8.098uM 6.434uM View
histamine receptor H 2 METERGOLINE Histamine H2 86% .975uM .959uM View
5-hydroxytryptamine (serotonin) receptor 1B PROCHLORPERAZINE Serotonin 5-HT1B 86% 2.651uM 1.205uM View
dopamine receptor D1A PERGOLIDE Dopamine D1 86% .679uM .339uM View
adrenergic receptor, alpha 1d (Non-specific probe) PERGOLIDE Adrenergic alpha1D 86% 1.513uM .744uM View
amiloride-sensitive cation channel 5, intestinal MEPAZINE Sodium Channel, Site 2 85% 2.521uM 2.3uM View
sodium channel, voltage-gated, type III, beta MEPAZINE Sodium Channel, Site 2 85% 2.521uM 2.3uM View
sodium channel, voltage-gated, type VIII, alpha polypeptide MEPAZINE Sodium Channel, Site 2 85% 2.521uM 2.3uM View
sodium channel, voltage-gated, type XI, alpha MEPAZINE Sodium Channel, Site 2 85% 2.521uM 2.3uM View
sodium channel, voltage-gated, type I, beta MEPAZINE Sodium Channel, Site 2 85% 2.521uM 2.3uM View
sodium channel, voltage-gated, type 10, alpha polypeptide MEPAZINE Sodium Channel, Site 2 85% 2.521uM 2.3uM View
sodium channel, voltage-gated, type IV, alpha polypeptide MEPAZINE Sodium Channel, Site 2 85% 2.521uM 2.3uM View
sodium channel, voltage-gated, type V, alpha polypeptide MEPAZINE Sodium Channel, Site 2 85% 2.521uM 2.3uM View
sodium channel, voltage-gated, type II, beta MEPAZINE Sodium Channel, Site 2 85% 2.521uM 2.3uM View
sodium channel, nonvoltage-gated 1 alpha MEPAZINE Sodium Channel, Site 2 85% 2.521uM 2.3uM View
sodium channel, nonvoltage-gated 1 gamma MEPAZINE Sodium Channel, Site 2 85% 2.521uM 2.3uM View
sodium channel, nonvoltage-gated 1 beta MEPAZINE Sodium Channel, Site 2 85% 2.521uM 2.3uM View
sodium channel, voltage-gated, type 2, alpha 1 polypeptide MEPAZINE Sodium Channel, Site 2 85% 2.521uM 2.3uM View
sodium channel, voltage-gated, type XI, alpha MEPAZINE Sodium Channel, Site 2 85% 2.521uM 2.3uM View
calcium channel, voltage-dependent, gamma subunit 3 TIRILAZAD Calcium Channel Type L, Benzothiazepine 89% 2.694uM 2.395uM View
calcium channel, voltage-dependent, gamma subunit 2 TIRILAZAD Calcium Channel Type L, Benzothiazepine 89% 2.694uM 2.395uM View
calcium channel, voltage-dependent, gamma subunit 1 TIRILAZAD Calcium Channel Type L, Benzothiazepine 89% 2.694uM 2.395uM View
calcium channel, voltage-dependent, beta 4 subunit TIRILAZAD Calcium Channel Type L, Benzothiazepine 89% 2.694uM 2.395uM View
calcium channel, voltage-dependent, beta 3 subunit TIRILAZAD Calcium Channel Type L, Benzothiazepine 89% 2.694uM 2.395uM View
calcium channel, voltage-dependent, beta 2 subunit TIRILAZAD Calcium Channel Type L, Benzothiazepine 89% 2.694uM 2.395uM View
calcium channel, voltage-dependent, L type, alpha 1S subunit TIRILAZAD Calcium Channel Type L, Benzothiazepine 89% 2.694uM 2.395uM View
calcium channel, voltage-dependent, alpha 1F subunit TIRILAZAD Calcium Channel Type L, Benzothiazepine 89% 2.694uM 2.395uM View
calcium channel, voltage-dependent, L type, alpha 1D subunit TIRILAZAD Calcium Channel Type L, Benzothiazepine 89% 2.694uM 2.395uM View
calcium channel, voltage-dependent, L type, alpha 1C subunit TIRILAZAD Calcium Channel Type L, Benzothiazepine 89% 2.694uM 2.395uM View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit TIRILAZAD Calcium Channel Type L, Benzothiazepine 89% 2.694uM 2.395uM View
calcium channel, voltage-dependent, beta 1 subunit TIRILAZAD Calcium Channel Type L, Benzothiazepine 89% 2.694uM 2.395uM View
calcium channel, voltage-dependent, L type, alpha 1E subunit TIRILAZAD Calcium Channel Type L, Benzothiazepine 89% 2.694uM 2.395uM View
calcium channel, voltage-dependent, N type, alpha 1B subunit TIRILAZAD Calcium Channel Type L, Benzothiazepine 89% 2.694uM 2.395uM View
calcium channel, voltage-dependent, alpha2/delta subunit 1 TIRILAZAD Calcium Channel Type L, Benzothiazepine 89% 2.694uM 2.395uM View
calcium channel, voltage-dependent, gamma subunit 8 TIRILAZAD Calcium Channel Type L, Benzothiazepine 89% 2.694uM 2.395uM View
calcium channel, voltage-dependent, gamma subunit 7 TIRILAZAD Calcium Channel Type L, Benzothiazepine 89% 2.694uM 2.395uM View
calcium channel, voltage-dependent, gamma subunit 6 TIRILAZAD Calcium Channel Type L, Benzothiazepine 89% 2.694uM 2.395uM View
calcium channel, voltage-dependent, gamma subunit 5 TIRILAZAD Calcium Channel Type L, Benzothiazepine 89% 2.694uM 2.395uM View
calcium channel, voltage-dependent, gamma subunit 8 AMIODARONE Calcium Channel Type L, Benzothiazepine 89% .054uM .048uM View
calcium channel, voltage-dependent, gamma subunit 7 AMIODARONE Calcium Channel Type L, Benzothiazepine 89% .054uM .048uM View
calcium channel, voltage-dependent, gamma subunit 6 AMIODARONE Calcium Channel Type L, Benzothiazepine 89% .054uM .048uM View
calcium channel, voltage-dependent, gamma subunit 5 AMIODARONE Calcium Channel Type L, Benzothiazepine 89% .054uM .048uM View
calcium channel, voltage-dependent, gamma subunit 4 AMIODARONE Calcium Channel Type L, Benzothiazepine 89% .054uM .048uM View
calcium channel, voltage-dependent, gamma subunit 3 AMIODARONE Calcium Channel Type L, Benzothiazepine 89% .054uM .048uM View
calcium channel, voltage-dependent, gamma subunit 2 AMIODARONE Calcium Channel Type L, Benzothiazepine 89% .054uM .048uM View
calcium channel, voltage-dependent, gamma subunit 1 AMIODARONE Calcium Channel Type L, Benzothiazepine 89% .054uM .048uM View
calcium channel, voltage-dependent, beta 4 subunit AMIODARONE Calcium Channel Type L, Benzothiazepine 89% .054uM .048uM View
calcium channel, voltage-dependent, beta 3 subunit AMIODARONE Calcium Channel Type L, Benzothiazepine 89% .054uM .048uM View
calcium channel, voltage-dependent, beta 2 subunit AMIODARONE Calcium Channel Type L, Benzothiazepine 89% .054uM .048uM View
calcium channel, voltage-dependent, L type, alpha 1S subunit AMIODARONE Calcium Channel Type L, Benzothiazepine 89% .054uM .048uM View
calcium channel, voltage-dependent, alpha 1F subunit AMIODARONE Calcium Channel Type L, Benzothiazepine 89% .054uM .048uM View
calcium channel, voltage-dependent, L type, alpha 1D subunit AMIODARONE Calcium Channel Type L, Benzothiazepine 89% .054uM .048uM View
calcium channel, voltage-dependent, L type, alpha 1C subunit AMIODARONE Calcium Channel Type L, Benzothiazepine 89% .054uM .048uM View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit AMIODARONE Calcium Channel Type L, Benzothiazepine 89% .054uM .048uM View
calcium channel, voltage-dependent, beta 1 subunit AMIODARONE Calcium Channel Type L, Benzothiazepine 89% .054uM .048uM View
calcium channel, voltage-dependent, L type, alpha 1E subunit AMIODARONE Calcium Channel Type L, Benzothiazepine 89% .054uM .048uM View
calcium channel, voltage-dependent, N type, alpha 1B subunit AMIODARONE Calcium Channel Type L, Benzothiazepine 89% .054uM .048uM View
calcium channel, voltage-dependent, alpha2/delta subunit 1 AMIODARONE Calcium Channel Type L, Benzothiazepine 89% .054uM .048uM View
adrenergic receptor, alpha 1a YOHIMBINE Adrenergic alpha1A 89% 1.235uM .5uM View
adrenergic receptor, alpha 1b YOHIMBINE Adrenergic alpha1B 89% 1.188uM .658uM View
adrenergic receptor, alpha 2a DIHYDROERGOTAMINE Imidazoline I2, Central 89% .002503uM .001669uM View
adrenergic receptor, alpha 2c (Non-specific probe) DIHYDROERGOTAMINE Imidazoline I2, Central 89% .002503uM .001669uM View
adenosine A2a receptor TAMOXIFEN Adenosine A2A 89% 7.099uM 3.985uM View
5-hydroxytryptamine (serotonin) receptor 2C TAMOXIFEN Serotonin 5-HT2C 89% .46uM .241uM View
5-hydroxytryptamine (serotonin) receptor 2C CISAPRIDE Serotonin 5-HT2C 89% .767uM .402uM View
adrenergic receptor, alpha 2b CISAPRIDE Adrenergic alpha2B 89% 1.148uM .524uM View
calcium channel, voltage-dependent, gamma subunit 6 ERGOTAMINE Calcium Channel Type L, Phenylalkylamine 54% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 5 ERGOTAMINE Calcium Channel Type L, Phenylalkylamine 54% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 4 ERGOTAMINE Calcium Channel Type L, Phenylalkylamine 54% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 3 ERGOTAMINE Calcium Channel Type L, Phenylalkylamine 54% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 2 ERGOTAMINE Calcium Channel Type L, Phenylalkylamine 54% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 1 ERGOTAMINE Calcium Channel Type L, Phenylalkylamine 54% NoneNone NoneNone View
calcium channel, voltage-dependent, beta 4 subunit ERGOTAMINE Calcium Channel Type L, Phenylalkylamine 54% NoneNone NoneNone View
calcium channel, voltage-dependent, beta 3 subunit ERGOTAMINE Calcium Channel Type L, Phenylalkylamine 54% NoneNone NoneNone View
calcium channel, voltage-dependent, beta 2 subunit ERGOTAMINE Calcium Channel Type L, Phenylalkylamine 54% NoneNone NoneNone View
calcium channel, voltage-dependent, L type, alpha 1S subunit ERGOTAMINE Calcium Channel Type L, Phenylalkylamine 54% NoneNone NoneNone View
calcium channel, voltage-dependent, alpha 1F subunit ERGOTAMINE Calcium Channel Type L, Phenylalkylamine 54% NoneNone NoneNone View
calcium channel, voltage-dependent, L type, alpha 1D subunit ERGOTAMINE Calcium Channel Type L, Phenylalkylamine 54% NoneNone NoneNone View
calcium channel, voltage-dependent, L type, alpha 1C subunit ERGOTAMINE Calcium Channel Type L, Phenylalkylamine 54% NoneNone NoneNone View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit ERGOTAMINE Calcium Channel Type L, Phenylalkylamine 54% NoneNone NoneNone View
calcium channel, voltage-dependent, beta 1 subunit ERGOTAMINE Calcium Channel Type L, Phenylalkylamine 54% NoneNone NoneNone View
calcium channel, voltage-dependent, L type, alpha 1E subunit ERGOTAMINE Calcium Channel Type L, Phenylalkylamine 54% NoneNone NoneNone View
calcium channel, voltage-dependent, N type, alpha 1B subunit ERGOTAMINE Calcium Channel Type L, Phenylalkylamine 54% NoneNone NoneNone View
calcium channel, voltage-dependent, alpha2/delta subunit 1 ERGOTAMINE Calcium Channel Type L, Phenylalkylamine 54% NoneNone NoneNone View
opioid receptor, delta 1 NELFINAVIR Opiate delta 54% 66.149uM 23.319uM View
5-hydroxytryptamine receptor 6 SUMATRIPTAN Serotonin 5-HT6 54% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 8 SILDENAFIL Calcium Channel Type L, Phenylalkylamine 54% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 7 SILDENAFIL Calcium Channel Type L, Phenylalkylamine 54% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 6 SILDENAFIL Calcium Channel Type L, Phenylalkylamine 54% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 5 SILDENAFIL Calcium Channel Type L, Phenylalkylamine 54% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 4 SILDENAFIL Calcium Channel Type L, Phenylalkylamine 54% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 3 SILDENAFIL Calcium Channel Type L, Phenylalkylamine 54% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 2 SILDENAFIL Calcium Channel Type L, Phenylalkylamine 54% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 1 SILDENAFIL Calcium Channel Type L, Phenylalkylamine 54% NoneNone NoneNone View