Gene Activity List


Gene Activity List

Gene Compound Assay Inh Ic50 Ki View
calcium channel, voltage-dependent, beta 4 subunit SILDENAFIL Calcium Channel Type L, Phenylalkylamine 54% NoneNone NoneNone View
calcium channel, voltage-dependent, beta 3 subunit SILDENAFIL Calcium Channel Type L, Phenylalkylamine 54% NoneNone NoneNone View
calcium channel, voltage-dependent, beta 2 subunit SILDENAFIL Calcium Channel Type L, Phenylalkylamine 54% NoneNone NoneNone View
calcium channel, voltage-dependent, L type, alpha 1S subunit SILDENAFIL Calcium Channel Type L, Phenylalkylamine 54% NoneNone NoneNone View
calcium channel, voltage-dependent, alpha 1F subunit SILDENAFIL Calcium Channel Type L, Phenylalkylamine 54% NoneNone NoneNone View
calcium channel, voltage-dependent, L type, alpha 1D subunit SILDENAFIL Calcium Channel Type L, Phenylalkylamine 54% NoneNone NoneNone View
calcium channel, voltage-dependent, L type, alpha 1C subunit SILDENAFIL Calcium Channel Type L, Phenylalkylamine 54% NoneNone NoneNone View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit SILDENAFIL Calcium Channel Type L, Phenylalkylamine 54% NoneNone NoneNone View
calcium channel, voltage-dependent, beta 1 subunit SILDENAFIL Calcium Channel Type L, Phenylalkylamine 54% NoneNone NoneNone View
calcium channel, voltage-dependent, L type, alpha 1E subunit SILDENAFIL Calcium Channel Type L, Phenylalkylamine 54% NoneNone NoneNone View
calcium channel, voltage-dependent, N type, alpha 1B subunit SILDENAFIL Calcium Channel Type L, Phenylalkylamine 54% NoneNone NoneNone View
calcium channel, voltage-dependent, alpha2/delta subunit 1 SILDENAFIL Calcium Channel Type L, Phenylalkylamine 54% NoneNone NoneNone View
adrenergic receptor, beta 3 METERGOLINE Adrenergic beta3 54% NoneNone NoneNone View
dopamine receptor D4 PERGOLIDE Dopamine D4.2 54% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 8 GUANETHIDINE Calcium Channel Type L, Benzothiazepine 54% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 7 GUANETHIDINE Calcium Channel Type L, Benzothiazepine 54% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 6 GUANETHIDINE Calcium Channel Type L, Benzothiazepine 54% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 5 GUANETHIDINE Calcium Channel Type L, Benzothiazepine 54% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 4 GUANETHIDINE Calcium Channel Type L, Benzothiazepine 54% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 3 GUANETHIDINE Calcium Channel Type L, Benzothiazepine 54% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 2 GUANETHIDINE Calcium Channel Type L, Benzothiazepine 54% NoneNone NoneNone View
sodium channel, voltage-gated, type 2, alpha 1 polypeptide PREGNENOLONE-16ALPHA-CARBONITRILE Sodium Channel, Site 2 53% 24.848uM 22.278uM View
sodium channel, voltage-gated, type XI, alpha PREGNENOLONE-16ALPHA-CARBONITRILE Sodium Channel, Site 2 53% 24.848uM 22.278uM View
sodium channel, nonvoltage-gated 1, gamma PREGNENOLONE-16ALPHA-CARBONITRILE Sodium Channel, Site 2 53% 24.848uM 22.278uM View
sodium channel, nonvoltage-gated 1, delta PREGNENOLONE-16ALPHA-CARBONITRILE Sodium Channel, Site 2 53% 24.848uM 22.278uM View
sodium channel, nonvoltage-gated 1, beta (Liddle syndrome) PREGNENOLONE-16ALPHA-CARBONITRILE Sodium Channel, Site 2 53% 24.848uM 22.278uM View
sodium channel, nonvoltage-gated 1 alpha PREGNENOLONE-16ALPHA-CARBONITRILE Sodium Channel, Site 2 53% 24.848uM 22.278uM View
sodium channel, voltage-gated, type X, alpha PREGNENOLONE-16ALPHA-CARBONITRILE Sodium Channel, Site 2 53% 24.848uM 22.278uM View
sodium channel, voltage-gated, type IX, alpha PREGNENOLONE-16ALPHA-CARBONITRILE Sodium Channel, Site 2 53% 24.848uM 22.278uM View
sodium channel, voltage gated, type VIII, alpha PREGNENOLONE-16ALPHA-CARBONITRILE Sodium Channel, Site 2 53% 24.848uM 22.278uM View
sodium channel, voltage-gated, type VII, alpha PREGNENOLONE-16ALPHA-CARBONITRILE Sodium Channel, Site 2 53% 24.848uM 22.278uM View
mitogen activated protein kinase 14 BETA-NAPHTHOFLAVONE Protein Serine/Threonine Kinase, p38alpha 53% NoneNone NoneNone View
mitogen-activated protein kinase 14 BETA-NAPHTHOFLAVONE Protein Serine/Threonine Kinase, p38alpha 53% NoneNone NoneNone View
cholinergic receptor, muscarinic 2 SULOCTIDIL Muscarinic M2 53% NoneNone NoneNone View
dopamine receptor D4 PERHEXILINE Dopamine D4.2 53% NoneNone NoneNone View
tachykinin receptor 1 IODOQUINOL Tachykinin NK1 53% NoneNone NoneNone View
5-hydroxytryptamine (serotonin) receptor 2A DILTIAZEM Serotonin 5-HT2A 53% NoneNone NoneNone View
cholinergic receptor, muscarinic 5 TERFENADINE Muscarinic M5 53% NoneNone NoneNone View
cholinergic receptor, muscarinic 3 HYDROXYCHLOROQUINE Muscarinic M3 53% NoneNone NoneNone View
melanocortin 5 receptor TERFENADINE Melanocortin MC5 53% NoneNone NoneNone View
Cytochrom P450-2D6 monooxygenase DAUNORUBICIN CYP450-2D6 Inhibition 53% NoneNone NoneNone View
Cytochrome P450, subfamily IIC (mephenytoin 4-hydroxylase) WARFARIN CYP450-2C9 Inhibition 53% NoneNone NoneNone View
cytochrome P450, family 2, subfamily C, polypeptide 9 WARFARIN CYP450-2C9 Inhibition 53% NoneNone NoneNone View
Cytochrome P450, subfamily IIC (mephenytoin 4-hydroxylase) CYPROTERONE ACETATE CYP450-2C9 Inhibition 53% NoneNone NoneNone View
cytochrome P450, family 2, subfamily C, polypeptide 9 CYPROTERONE ACETATE CYP450-2C9 Inhibition 53% NoneNone NoneNone View
Cytochrom P450-2C19 monooxygenase PANTOPRAZOLE CYP450-2C19 Inhibition 53% NoneNone NoneNone View
mu-opioid receptor MOR CLOSANTEL Opiate mu 53% NoneNone NoneNone View
adrenergic receptor, beta 3 BITHIONOL Adrenergic beta3 53% NoneNone NoneNone View
adrenergic receptor, alpha 1d (Non-specific probe) DIPHENIDOL Adrenergic alpha1D 53% NoneNone NoneNone View
dopamine receptor D4 DOBUTAMINE Dopamine D4.2 53% NoneNone NoneNone View
mitogen activated protein kinase 1 COBALT(II) ACETYLACETONATE Protein Serine/Threonine Kinase, ERK2 53% NoneNone NoneNone View
mitogen-activated protein kinase 1 COBALT(II) ACETYLACETONATE Protein Serine/Threonine Kinase, ERK2 53% NoneNone NoneNone View
Cytochrom P450-2D6 monooxygenase DIHYDROERGOCRISTINE MESYLATE CYP450-2D6 Inhibition 53% NoneNone NoneNone View
thromboxane A synthase 1 DIHYDROERGOCRISTINE MESYLATE Thromboxane Synthetase 53% NoneNone NoneNone View
thromboxane A synthase 1 (platelet, cytochrome P450, family 5, subfamily A) DIHYDROERGOCRISTINE MESYLATE Thromboxane Synthetase 53% NoneNone NoneNone View
acetylcholinesterase (YT blood group) TERBINAFINE Acetylcholinesterase 53% NoneNone NoneNone View
collagen-like tail subunit (single strand of homotrimer) of asymmetric acetylcholinesterase TERBINAFINE Acetylcholinesterase 53% NoneNone NoneNone View
acetylcholinesterase TERBINAFINE Acetylcholinesterase 53% NoneNone NoneNone View
mu-opioid receptor MOR PAROXETINE Opiate mu 53% NoneNone NoneNone View
cannabinoid receptor 1 (brain) PAROXETINE Cannabinoid CB1 53% NoneNone NoneNone View
adrenergic receptor, alpha 2a DESLORATADINE Adrenergic alpha2A 53% NoneNone NoneNone View
adrenergic receptor, alpha 2a PROPAFENONE Adrenergic alpha2A 53% NoneNone NoneNone View
adrenergic receptor, alpha 2a TACRINE Imidazoline I2, Central 53% NoneNone NoneNone View
adrenergic receptor, alpha 2c (Non-specific probe) TACRINE Imidazoline I2, Central 53% NoneNone NoneNone View
aldo-keto reductase family 1, member B4 (aldose reductase) ROSIGLITAZONE Aldose Reductase 53% NoneNone NoneNone View
aldo-keto reductase family 1, member B1 (aldose reductase) ROSIGLITAZONE Aldose Reductase 53% NoneNone NoneNone View
aldo-keto reductase family 7, member A2 (aflatoxin aldehyde reductase) ROSIGLITAZONE Aldose Reductase 53% NoneNone NoneNone View
aldo-keto reductase family 7, member A3 (aflatoxin aldehyde reductase) ROSIGLITAZONE Aldose Reductase 53% NoneNone NoneNone View
opioid receptor, sigma 1 METERGOLINE Sigma1 53% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 8 PROCHLORPERAZINE Calcium Channel Type L, Benzothiazepine 53% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 7 PROCHLORPERAZINE Calcium Channel Type L, Benzothiazepine 53% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 6 PROCHLORPERAZINE Calcium Channel Type L, Benzothiazepine 53% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 5 PROCHLORPERAZINE Calcium Channel Type L, Benzothiazepine 53% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 4 PROCHLORPERAZINE Calcium Channel Type L, Benzothiazepine 53% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 3 PROCHLORPERAZINE Calcium Channel Type L, Benzothiazepine 53% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 2 PROCHLORPERAZINE Calcium Channel Type L, Benzothiazepine 53% NoneNone NoneNone View
sodium channel, voltage-gated, type I, beta DIMENHYDRINATE Sodium Channel, Site 2 52% NoneNone NoneNone View
sodium channel, voltage-gated, type 10, alpha polypeptide DIMENHYDRINATE Sodium Channel, Site 2 52% NoneNone NoneNone View
sodium channel, voltage-gated, type IV, alpha polypeptide DIMENHYDRINATE Sodium Channel, Site 2 52% NoneNone NoneNone View
sodium channel, voltage-gated, type V, alpha polypeptide DIMENHYDRINATE Sodium Channel, Site 2 52% NoneNone NoneNone View
sodium channel, voltage-gated, type II, beta DIMENHYDRINATE Sodium Channel, Site 2 52% NoneNone NoneNone View
sodium channel, nonvoltage-gated 1 alpha DIMENHYDRINATE Sodium Channel, Site 2 52% NoneNone NoneNone View
sodium channel, nonvoltage-gated 1 gamma DIMENHYDRINATE Sodium Channel, Site 2 52% NoneNone NoneNone View
sodium channel, nonvoltage-gated 1 beta DIMENHYDRINATE Sodium Channel, Site 2 52% NoneNone NoneNone View
sodium channel, voltage-gated, type 2, alpha 1 polypeptide DIMENHYDRINATE Sodium Channel, Site 2 52% NoneNone NoneNone View
sodium channel, voltage-gated, type XI, alpha DIMENHYDRINATE Sodium Channel, Site 2 52% NoneNone NoneNone View
sodium channel, nonvoltage-gated 1, gamma DIMENHYDRINATE Sodium Channel, Site 2 52% NoneNone NoneNone View
sodium channel, nonvoltage-gated 1, delta DIMENHYDRINATE Sodium Channel, Site 2 52% NoneNone NoneNone View
sodium channel, nonvoltage-gated 1, beta (Liddle syndrome) DIMENHYDRINATE Sodium Channel, Site 2 52% NoneNone NoneNone View
sodium channel, nonvoltage-gated 1 alpha DIMENHYDRINATE Sodium Channel, Site 2 52% NoneNone NoneNone View
sodium channel, voltage-gated, type X, alpha DIMENHYDRINATE Sodium Channel, Site 2 52% NoneNone NoneNone View
sodium channel, voltage-gated, type IX, alpha DIMENHYDRINATE Sodium Channel, Site 2 52% NoneNone NoneNone View
sodium channel, voltage gated, type VIII, alpha DIMENHYDRINATE Sodium Channel, Site 2 52% NoneNone NoneNone View
sodium channel, voltage-gated, type VII, alpha DIMENHYDRINATE Sodium Channel, Site 2 52% NoneNone NoneNone View
sodium channel, voltage-gated, type V, alpha (long QT syndrome 3) DIMENHYDRINATE Sodium Channel, Site 2 52% NoneNone NoneNone View
sodium channel, voltage-gated, type IV, beta DIMENHYDRINATE Sodium Channel, Site 2 52% NoneNone NoneNone View
sodium channel, voltage-gated, type IV, alpha DIMENHYDRINATE Sodium Channel, Site 2 52% NoneNone NoneNone View
sodium channel, voltage-gated, type III, alpha DIMENHYDRINATE Sodium Channel, Site 2 52% NoneNone NoneNone View
sodium channel, voltage-gated, type II, beta DIMENHYDRINATE Sodium Channel, Site 2 52% NoneNone NoneNone View
sodium channel, voltage-gated, type II, alpha 2 DIMENHYDRINATE Sodium Channel, Site 2 52% NoneNone NoneNone View
sodium channel, voltage-gated, type I, beta DIMENHYDRINATE Sodium Channel, Site 2 52% NoneNone NoneNone View
sodium channel, voltage-gated, type I, alpha DIMENHYDRINATE Sodium Channel, Site 2 52% NoneNone NoneNone View
Sigma-2 Receptor LEVOBUNOLOL Sigma2 52% NoneNone NoneNone View
5-hydroxytryptamine receptor 6 FLUNARIZINE Serotonin 5-HT6 52% NoneNone NoneNone View
cholinergic receptor, muscarinic 1 4-NONYLPHENOL Muscarinic M1 52% NoneNone NoneNone View
glutamate receptor, ionotropic, N-methyl-D-aspartate 3B 1,3-DIPHENYLGUANIDINE Glutamate, NMDA, Phencyclidine 52% NoneNone NoneNone View
glutamate receptor, ionotropic, N-methyl D-aspartate 2D 1,3-DIPHENYLGUANIDINE Glutamate, NMDA, Phencyclidine 52% NoneNone NoneNone View
glutamate receptor, ionotropic, NMDA2C 1,3-DIPHENYLGUANIDINE Glutamate, NMDA, Phencyclidine 52% NoneNone NoneNone View
glutamate receptor, ionotropic, N-methyl D-aspartate 2B 1,3-DIPHENYLGUANIDINE Glutamate, NMDA, Phencyclidine 52% NoneNone NoneNone View
glutamate receptor, ionotropic, N-methyl D-aspartate 2A 1,3-DIPHENYLGUANIDINE Glutamate, NMDA, Phencyclidine 52% NoneNone NoneNone View
N-methyl-D-aspartate receptor 1 (Grin1) gene, exons 1 through 6 and partial cds; alternatively spliced (Rn.) 1,3-DIPHENYLGUANIDINE Glutamate, NMDA, Phencyclidine 52% NoneNone NoneNone View
cytochrome P450, family 3, subfamily a, polypeptide 13 HARRINGTONINE CYP450-3A4 Inhibition 52% NoneNone NoneNone View
cytochrome P450, family 3, subfamily a, polypeptide 13 PUROMYCIN CYP450-3A4 Inhibition 52% NoneNone NoneNone View
cytochrome P450, family 3, subfamily a, polypeptide 13 QUETIAPINE CYP450-3A4 Inhibition 52% NoneNone NoneNone View
Cytochrom P450-2D6 monooxygenase BUFLOMEDIL CYP450-2D6 Inhibition 52% NoneNone NoneNone View
Cytochrom P450-2D6 monooxygenase PRIMAQUINE CYP450-2D6 Inhibition 52% NoneNone NoneNone View
Cytochrom P450-2D6 monooxygenase RIMANTADINE CYP450-2D6 Inhibition 52% NoneNone NoneNone View
Cytochrom P450-2C19 monooxygenase BROMHEXINE CYP450-2C19 Inhibition 52% NoneNone NoneNone View
Cytochrom P450-2C19 monooxygenase PERGOLIDE CYP450-2C19 Inhibition 52% NoneNone NoneNone View
Cytochrom P450-2C19 monooxygenase RABEPRAZOLE CYP450-2C19 Inhibition 52% NoneNone NoneNone View
adrenergic receptor, alpha 1d (Non-specific probe) BERBERINE CHLORIDE Adrenergic alpha1D 52% NoneNone NoneNone View
adenosine A1 receptor AMINOPHYLLINE Adenosine A1 52% NoneNone NoneNone View
matrix metallopeptidase 9 PRIMAQUINE Protease, Matrix Metalloprotease-9 (MMP-9) 51% NoneNone NoneNone View
matrix metalloproteinase 9 (gelatinase B, 92kDa gelatinase, 92kDa type IV collagenase) PRIMAQUINE Protease, Matrix Metalloprotease-9 (MMP-9) 51% NoneNone NoneNone View
acetylcholinesterase (YT blood group) CARMOFUR Acetylcholinesterase 51% NoneNone NoneNone View
collagen-like tail subunit (single strand of homotrimer) of asymmetric acetylcholinesterase CARMOFUR Acetylcholinesterase 51% NoneNone NoneNone View
acetylcholinesterase CARMOFUR Acetylcholinesterase 51% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 4 LACIDIPINE Calcium Channel Type L, Phenylalkylamine 51% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 3 LACIDIPINE Calcium Channel Type L, Phenylalkylamine 51% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 2 LACIDIPINE Calcium Channel Type L, Phenylalkylamine 51% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 1 LACIDIPINE Calcium Channel Type L, Phenylalkylamine 51% NoneNone NoneNone View
N-methyl-D-aspartate receptor 1 (Grin1) gene, exons 1 through 6 and partial cds; alternatively spliced (Rn.) AMANTADINE Glutamate, NMDA, Phencyclidine 51% 31.983uM 21.666uM View
glutamate receptor, ionotropic, N-methyl-D-aspartate 3B AMANTADINE Glutamate, NMDA, Phencyclidine 51% 31.983uM 21.666uM View
adrenergic receptor, beta 2 TIRILAZAD Adrenergic beta2 51% 22.659uM 15.578uM View
cholinergic receptor, muscarinic 3 ALPHA-NAPHTHOFLAVONE Muscarinic M3 51% NoneNone NoneNone View
phosphodiesterase 5A, cGMP-specific COBALT (II) CHLORIDE Phosphodiesterase PDE5 51% NoneNone NoneNone View
phosphodiesterase 5A, cGMP-specific COBALT (II) CHLORIDE Phosphodiesterase PDE5 51% NoneNone NoneNone View
mitogen activated protein kinase 14 BENZO[E]PYRENE Protein Serine/Threonine Kinase, p38alpha 51% NoneNone NoneNone View
mitogen-activated protein kinase 14 BENZO[E]PYRENE Protein Serine/Threonine Kinase, p38alpha 51% NoneNone NoneNone View
solute carrier family 6 (neurotransmitter transporter, serotonin), member 4 2-HYDROXYPROPYL-BETA-CYCLODEXTRIN Serotonin Transporter 51% NoneNone NoneNone View
Sigma-2 Receptor AMOXAPINE Sigma2 51% NoneNone NoneNone View
cytochrome P450, family 3, subfamily a, polypeptide 13 4-METHYLPYRAZOLE CYP450-3A4 Inhibition 51% NoneNone NoneNone View
Cytochrom P450-2D6 monooxygenase TOLPERISONE CYP450-2D6 Inhibition 51% NoneNone NoneNone View
Cytochrom P450-2C19 monooxygenase PERHEXILINE CYP450-2C19 Inhibition 51% NoneNone NoneNone View
Sigma-2 Receptor CYCLIZINE Sigma2 51% NoneNone NoneNone View
Sigma-2 Receptor HYDROXYPROGESTERONE Sigma2 51% NoneNone NoneNone View
5-hydroxytryptamine receptor 6 SULFAMETHAZINE Serotonin 5-HT6 51% NoneNone NoneNone View
platelet-activating factor receptor DILTIAZEM Platelet Activating Factor (PAF) 51% NoneNone NoneNone View
dopamine receptor D1A MONTELUKAST Dopamine D1 51% NoneNone NoneNone View
cytochrome P450, family 3, subfamily a, polypeptide 13 SERTRALINE CYP450-3A4 Inhibition 51% NoneNone NoneNone View
cytochrome P450, family 3, subfamily a, polypeptide 13 DOXAZOSIN CYP450-3A4 Inhibition 51% NoneNone NoneNone View
Cytochrom P450-2D6 monooxygenase MELATONIN CYP450-2D6 Inhibition 51% NoneNone NoneNone View
Cytochrom P450-2D6 monooxygenase DOBUTAMINE CYP450-2D6 Inhibition 51% NoneNone NoneNone View
Cytochrom P450-2C19 monooxygenase TANNIC ACID CYP450-2C19 Inhibition 51% NoneNone NoneNone View
A3 adenosine receptor IMATINIB Adenosine A3 51% NoneNone NoneNone View
acetylcholinesterase (YT blood group) FLUNARIZINE Acetylcholinesterase 51% NoneNone NoneNone View
collagen-like tail subunit (single strand of homotrimer) of asymmetric acetylcholinesterase FLUNARIZINE Acetylcholinesterase 51% NoneNone NoneNone View
acetylcholinesterase FLUNARIZINE Acetylcholinesterase 51% NoneNone NoneNone View
v-erb-b2 erythroblastic leukemia viral oncogene homolog 2, neuro/glioblastoma derived oncogene homolog (avian) 3,3',4',5-TETRACHLOROSALICYLANILIDE Protein Tyrosine Kinase, HER2 Receptor 51% NoneNone NoneNone View
v-erb-b2 erythroblastic leukemia viral oncogene homolog 2, neuro/glioblastoma derived oncogene homolog (avian) 3,3',4',5-TETRACHLOROSALICYLANILIDE Protein Tyrosine Kinase, HER2 Receptor 51% NoneNone NoneNone View
solute carrier family 6 (neurotransmitter transporter, dopamine), member 3 ETHYLESTRENOL Dopamine Transporter 51% NoneNone NoneNone View
A3 adenosine receptor AMITRAZ Adenosine A3 51% NoneNone NoneNone View
solute carrier family 6 (neurotransmitter transporter, serotonin), member 4 GRAMICIDIN Serotonin Transporter 51% NoneNone NoneNone View
tachykinin receptor 1 GRAMICIDIN Tachykinin NK1 51% NoneNone NoneNone View
solute carrier family 28 (sodium-coupled nucleoside transporter), member 3 KITASAMYCIN Adenosine Transporter 51% NoneNone NoneNone View
concentrative Na+ nucleoside cotransporter (DBSS) KITASAMYCIN Adenosine Transporter 51% NoneNone NoneNone View
solute carrier family 28 (sodium-coupled nucleoside transporter), member 1 KITASAMYCIN Adenosine Transporter 51% NoneNone NoneNone View
adenine nucleotide translocase (DBSS) (Non-specific probe) KITASAMYCIN Adenosine Transporter 51% NoneNone NoneNone View
solute carrier family 25 (mitochondrial carrier; adenine nucleotide translocator), member 4 KITASAMYCIN Adenosine Transporter 51% NoneNone NoneNone View
tachykinin receptor 2 IVERMECTIN Tachykinin NK2 51% NoneNone NoneNone View
Cytochrom P450-2D6 monooxygenase SPIRADOLINE CYP450-2D6 Inhibition 51% NoneNone NoneNone View
sodium channel, voltage-gated, type IV, beta ERGOTAMINE Sodium Channel, Site 2 51% NoneNone NoneNone View
sodium channel associated protein 1 ERGOTAMINE Sodium Channel, Site 2 51% NoneNone NoneNone View
sodium channel associated protein 2 ERGOTAMINE Sodium Channel, Site 2 51% NoneNone NoneNone View
sodium channel, voltage-gated, type III, beta ERGOTAMINE Sodium Channel, Site 2 51% NoneNone NoneNone View
sodium channel, voltage-gated, type I, alpha ERGOTAMINE Sodium Channel, Site 2 51% NoneNone NoneNone View
sodium channel, voltage-gated, type IX, alpha ERGOTAMINE Sodium Channel, Site 2 51% NoneNone NoneNone View
sodium channel, voltage-gated, type VII, alpha ERGOTAMINE Sodium Channel, Site 2 51% NoneNone NoneNone View
amiloride-sensitive cation channel 5, intestinal ERGOTAMINE Sodium Channel, Site 2 51% NoneNone NoneNone View
sodium channel, voltage-gated, type III, beta ERGOTAMINE Sodium Channel, Site 2 51% NoneNone NoneNone View
sodium channel, voltage-gated, type VIII, alpha polypeptide ERGOTAMINE Sodium Channel, Site 2 51% NoneNone NoneNone View
sodium channel, voltage-gated, type XI, alpha ERGOTAMINE Sodium Channel, Site 2 51% NoneNone NoneNone View
sodium channel, voltage-gated, type I, beta ERGOTAMINE Sodium Channel, Site 2 51% NoneNone NoneNone View
sodium channel, voltage-gated, type 10, alpha polypeptide ERGOTAMINE Sodium Channel, Site 2 51% NoneNone NoneNone View
sodium channel, voltage-gated, type IV, alpha polypeptide ERGOTAMINE Sodium Channel, Site 2 51% NoneNone NoneNone View
sodium channel, voltage-gated, type V, alpha polypeptide ERGOTAMINE Sodium Channel, Site 2 51% NoneNone NoneNone View
sodium channel, voltage-gated, type II, beta ERGOTAMINE Sodium Channel, Site 2 51% NoneNone NoneNone View
sodium channel, nonvoltage-gated 1 alpha ERGOTAMINE Sodium Channel, Site 2 51% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 1 GUANETHIDINE Calcium Channel Type L, Benzothiazepine 54% NoneNone NoneNone View
calcium channel, voltage-dependent, beta 4 subunit GUANETHIDINE Calcium Channel Type L, Benzothiazepine 54% NoneNone NoneNone View
calcium channel, voltage-dependent, beta 3 subunit GUANETHIDINE Calcium Channel Type L, Benzothiazepine 54% NoneNone NoneNone View
calcium channel, voltage-dependent, beta 2 subunit GUANETHIDINE Calcium Channel Type L, Benzothiazepine 54% NoneNone NoneNone View
calcium channel, voltage-dependent, L type, alpha 1S subunit GUANETHIDINE Calcium Channel Type L, Benzothiazepine 54% NoneNone NoneNone View
calcium channel, voltage-dependent, alpha 1F subunit GUANETHIDINE Calcium Channel Type L, Benzothiazepine 54% NoneNone NoneNone View
calcium channel, voltage-dependent, L type, alpha 1D subunit GUANETHIDINE Calcium Channel Type L, Benzothiazepine 54% NoneNone NoneNone View
calcium channel, voltage-dependent, L type, alpha 1C subunit GUANETHIDINE Calcium Channel Type L, Benzothiazepine 54% NoneNone NoneNone View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit GUANETHIDINE Calcium Channel Type L, Benzothiazepine 54% NoneNone NoneNone View
calcium channel, voltage-dependent, beta 1 subunit GUANETHIDINE Calcium Channel Type L, Benzothiazepine 54% NoneNone NoneNone View
calcium channel, voltage-dependent, L type, alpha 1E subunit GUANETHIDINE Calcium Channel Type L, Benzothiazepine 54% NoneNone NoneNone View
potassium voltage-gated channel, subfamily H, member 8 PENTAMIDINE Potassium Channel HERG 54% 15.7215uM 12.8802uM View