Gene Activity List


Gene Activity List

Gene Compound Assay Inh Ic50 Ki View
sodium channel, voltage-gated, type IX, alpha CELECOXIB Sodium Channel, Site 2 62% 16.854uM 15.111uM View
sodium channel, voltage-gated, type VII, alpha CELECOXIB Sodium Channel, Site 2 62% 16.854uM 15.111uM View
amiloride-sensitive cation channel 5, intestinal CELECOXIB Sodium Channel, Site 2 62% 16.854uM 15.111uM View
sodium channel, voltage-gated, type I, beta PENTAMIDINE Sodium Channel, Site 2 62% NoneNone NoneNone View
sodium channel, voltage-gated, type 10, alpha polypeptide PENTAMIDINE Sodium Channel, Site 2 62% NoneNone NoneNone View
sodium channel, voltage-gated, type IV, alpha polypeptide PENTAMIDINE Sodium Channel, Site 2 62% NoneNone NoneNone View
sodium channel, voltage-gated, type V, alpha polypeptide PENTAMIDINE Sodium Channel, Site 2 62% NoneNone NoneNone View
sodium channel, voltage-gated, type II, beta PENTAMIDINE Sodium Channel, Site 2 62% NoneNone NoneNone View
sodium channel, nonvoltage-gated 1 alpha PENTAMIDINE Sodium Channel, Site 2 62% NoneNone NoneNone View
sodium channel, nonvoltage-gated 1 gamma PENTAMIDINE Sodium Channel, Site 2 62% NoneNone NoneNone View
sodium channel, nonvoltage-gated 1 beta PENTAMIDINE Sodium Channel, Site 2 62% NoneNone NoneNone View
sodium channel, voltage-gated, type 2, alpha 1 polypeptide PENTAMIDINE Sodium Channel, Site 2 62% NoneNone NoneNone View
sodium channel, voltage-gated, type XI, alpha PENTAMIDINE Sodium Channel, Site 2 62% NoneNone NoneNone View
sodium channel, nonvoltage-gated 1, gamma PENTAMIDINE Sodium Channel, Site 2 62% NoneNone NoneNone View
sodium channel, nonvoltage-gated 1, delta PENTAMIDINE Sodium Channel, Site 2 62% NoneNone NoneNone View
sodium channel, nonvoltage-gated 1, beta (Liddle syndrome) PENTAMIDINE Sodium Channel, Site 2 62% NoneNone NoneNone View
sodium channel, nonvoltage-gated 1 alpha PENTAMIDINE Sodium Channel, Site 2 62% NoneNone NoneNone View
sodium channel, voltage-gated, type X, alpha PENTAMIDINE Sodium Channel, Site 2 62% NoneNone NoneNone View
sodium channel, voltage-gated, type IX, alpha PENTAMIDINE Sodium Channel, Site 2 62% NoneNone NoneNone View
sodium channel, voltage gated, type VIII, alpha PENTAMIDINE Sodium Channel, Site 2 62% NoneNone NoneNone View
5-hydroxytryptamine (serotonin) receptor 3a CYPROHEPTADINE Serotonin 5-HT3 62% NoneNone NoneNone View
5-hydroxytryptamine (serotonin) receptor 3b CYPROHEPTADINE Serotonin 5-HT3 62% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 8 GUANETHIDINE Calcium Channel Type L, Phenylalkylamine 62% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 7 GUANETHIDINE Calcium Channel Type L, Phenylalkylamine 62% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 6 GUANETHIDINE Calcium Channel Type L, Phenylalkylamine 62% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 5 GUANETHIDINE Calcium Channel Type L, Phenylalkylamine 62% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 4 GUANETHIDINE Calcium Channel Type L, Phenylalkylamine 62% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 3 GUANETHIDINE Calcium Channel Type L, Phenylalkylamine 62% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 2 GUANETHIDINE Calcium Channel Type L, Phenylalkylamine 62% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 1 GUANETHIDINE Calcium Channel Type L, Phenylalkylamine 62% NoneNone NoneNone View
calcium channel, voltage-dependent, beta 4 subunit GUANETHIDINE Calcium Channel Type L, Phenylalkylamine 62% NoneNone NoneNone View
calcium channel, voltage-dependent, beta 3 subunit GUANETHIDINE Calcium Channel Type L, Phenylalkylamine 62% NoneNone NoneNone View
calcium channel, voltage-dependent, beta 2 subunit GUANETHIDINE Calcium Channel Type L, Phenylalkylamine 62% NoneNone NoneNone View
potassium voltage-gated channel, subfamily H (eag-related), member 1 MYRTECAINE Potassium Channel HERG 65% 5.9024uM 4.8357uM View
potassium voltage-gated channel, subfamily H (eag-related), member 1 MYRTECAINE Potassium Channel HERG 65% 5.9024uM 4.8357uM View
potassium voltage-gated channel, subfamily H, member 8 MYRTECAINE Potassium Channel HERG 65% 5.9024uM 4.8357uM View
potassium voltage-gated channel, subfamily H (eag-related), member 6 MYRTECAINE Potassium Channel HERG 65% 5.9024uM 4.8357uM View
potassium voltage-gated channel, subfamily H (eag-related), member 7 MYRTECAINE Potassium Channel HERG 65% 5.9024uM 4.8357uM View
potassium voltage-gated channel, subfamily H (eag-related), member 2 MYRTECAINE Potassium Channel HERG 65% 5.9024uM 4.8357uM View
potassium voltage-gated channel, subfamily H (eag-related), member 5 MYRTECAINE Potassium Channel HERG 65% 5.9024uM 4.8357uM View
potassium voltage-gated channel, subfamily H (eag-related), member 3 MYRTECAINE Potassium Channel HERG 65% 5.9024uM 4.8357uM View
potassium voltage-gated channel, subfamily H, member 8 SERTRALINE Potassium Channel HERG 65% 8.3173uM 6.8141uM View
potassium voltage-gated channel, subfamily H (eag-related), member 6 SERTRALINE Potassium Channel HERG 65% 8.3173uM 6.8141uM View
potassium voltage-gated channel, subfamily H (eag-related), member 7 SERTRALINE Potassium Channel HERG 65% 8.3173uM 6.8141uM View
potassium voltage-gated channel, subfamily H (eag-related), member 2 SERTRALINE Potassium Channel HERG 65% 8.3173uM 6.8141uM View
potassium voltage-gated channel, subfamily H (eag-related), member 5 SERTRALINE Potassium Channel HERG 65% 8.3173uM 6.8141uM View
potassium voltage-gated channel, subfamily H (eag-related), member 3 SERTRALINE Potassium Channel HERG 65% 8.3173uM 6.8141uM View
potassium voltage-gated channel, subfamily H (eag-related), member 4 SERTRALINE Potassium Channel HERG 65% 8.3173uM 6.8141uM View
potassium voltage-gated channel, subfamily H (eag-related), member 1 SERTRALINE Potassium Channel HERG 65% 8.3173uM 6.8141uM View
potassium voltage-gated channel, subfamily H (eag-related), member 1 SERTRALINE Potassium Channel HERG 65% 8.3173uM 6.8141uM View
Cytochrom P450-2D6 monooxygenase FLUNARIZINE CYP450-2D6 Inhibition 65% NoneNone NoneNone View
Cytochrom P450-1A2 monooxygenase IODOQUINOL CYP450-1A2 Inhibition 65% NoneNone NoneNone View
opioid receptor, sigma 1 AMBROXOL Sigma1 65% NoneNone NoneNone View
solute carrier family 6 (neurotransmitter transporter, serotonin), member 4 DIMENHYDRINATE Serotonin Transporter 65% NoneNone NoneNone View
solute carrier family 6 (neurotransmitter transporter, serotonin), member 4 TRIMETAZIDINE Serotonin Transporter 65% NoneNone NoneNone View
opioid receptor, sigma 1 HYDROXYCHLOROQUINE Sigma1 65% NoneNone NoneNone View
mu-opioid receptor MOR THIORIDAZINE Opiate mu 65% NoneNone NoneNone View
cholinergic receptor, muscarinic 2 CINNARIZINE Muscarinic M2 65% NoneNone NoneNone View
glutamate receptor, ionotropic, N-methyl D-aspartate 2D IODOQUINOL Glutamate, NMDA, Phencyclidine 65% NoneNone NoneNone View
glutamate receptor, ionotropic, NMDA2C IODOQUINOL Glutamate, NMDA, Phencyclidine 65% NoneNone NoneNone View
glutamate receptor, ionotropic, N-methyl D-aspartate 2B IODOQUINOL Glutamate, NMDA, Phencyclidine 65% NoneNone NoneNone View
glutamate receptor, ionotropic, N-methyl D-aspartate 2A IODOQUINOL Glutamate, NMDA, Phencyclidine 65% NoneNone NoneNone View
N-methyl-D-aspartate receptor 1 (Grin1) gene, exons 1 through 6 and partial cds; alternatively spliced (Rn.) IODOQUINOL Glutamate, NMDA, Phencyclidine 65% NoneNone NoneNone View
glutamate receptor, ionotropic, N-methyl-D-aspartate 3B IODOQUINOL Glutamate, NMDA, Phencyclidine 65% NoneNone NoneNone View
Cytochrom P450-2D6 monooxygenase DOXEPIN CYP450-2D6 Inhibition 65% NoneNone NoneNone View
Cytochrome P450, subfamily IIC (mephenytoin 4-hydroxylase) ANASTROZOLE CYP450-2C9 Inhibition 65% NoneNone NoneNone View
cytochrome P450, family 2, subfamily C, polypeptide 9 ANASTROZOLE CYP450-2C9 Inhibition 65% NoneNone NoneNone View
solute carrier family 6 (neurotransmitter transporter, noradrenalin), member 2 AMITRAZ Adrenergic, Norepinephrine Transporter 65% NoneNone NoneNone View
cholinergic receptor, muscarinic 4 ETHYLESTRENOL Muscarinic M4 65% NoneNone NoneNone View
adrenergic receptor, alpha 1a METHYLERGONOVINE Adrenergic alpha1A 65% NoneNone NoneNone View
histamine receptor H 1 BUSPIRONE Histamine H1, Central 65% NoneNone NoneNone View
histamine receptor H 1 ERGOTAMINE Histamine H1, Central 65% NoneNone NoneNone View
cytochrome P450, family 3, subfamily a, polypeptide 13 TERCONAZOLE CYP450-3A4 Inhibition 65% NoneNone NoneNone View
5-hydroxytryptamine (serotonin) receptor 2A TERBINAFINE Serotonin 5-HT2A 65% NoneNone NoneNone View
solute carrier family 28 (sodium-coupled nucleoside transporter), member 3 TERCONAZOLE Adenosine Transporter 65% 12.383uM 4.236uM View
concentrative Na+ nucleoside cotransporter (DBSS) TERCONAZOLE Adenosine Transporter 65% 12.383uM 4.236uM View
solute carrier family 28 (sodium-coupled nucleoside transporter), member 1 TERCONAZOLE Adenosine Transporter 65% 12.383uM 4.236uM View
adenine nucleotide translocase (DBSS) (Non-specific probe) TERCONAZOLE Adenosine Transporter 65% 12.383uM 4.236uM View
solute carrier family 25 (mitochondrial carrier; adenine nucleotide translocator), member 4 TERCONAZOLE Adenosine Transporter 65% 12.383uM 4.236uM View
melanocortin 5 receptor PROCHLORPERAZINE Melanocortin MC5 65% NoneNone NoneNone View
adrenergic receptor, alpha 1d (Non-specific probe) DESLORATADINE Adrenergic alpha1D 65% NoneNone NoneNone View
5-hydroxytryptamine receptor 6 GUANABENZ Serotonin 5-HT6 65% NoneNone NoneNone View
adenosine A1 receptor GW-1929 Adenosine A1 65% 14.966uM 8.73uM View
epidermal growth factor receptor ECONAZOLE Protein Tyrosine Kinase, EGF Receptor 65% 32.404uM NoneNone View
epidermal growth factor receptor MICONAZOLE Protein Tyrosine Kinase, EGF Receptor 65% 29.256uM NoneNone View
phosphodiesterase 4C, cAMP-specific LY-294002 Phosphodiesterase PDE4 64% 10.404uM NoneNone View
phosphodiesterase 4D LY-294002 Phosphodiesterase PDE4 64% 10.404uM NoneNone View
phosphodiesterase 4B, cAMP specific LY-294002 Phosphodiesterase PDE4 64% 10.404uM NoneNone View
calcium channel, voltage-dependent, gamma subunit 8 ETHINYLESTRADIOL Calcium Channel Type L, Benzothiazepine 64% 15.42uM 13.706uM View
calcium channel, voltage-dependent, gamma subunit 7 ETHINYLESTRADIOL Calcium Channel Type L, Benzothiazepine 64% 15.42uM 13.706uM View
calcium channel, voltage-dependent, gamma subunit 6 ETHINYLESTRADIOL Calcium Channel Type L, Benzothiazepine 64% 15.42uM 13.706uM View
calcium channel, voltage-dependent, gamma subunit 5 ETHINYLESTRADIOL Calcium Channel Type L, Benzothiazepine 64% 15.42uM 13.706uM View
calcium channel, voltage-dependent, gamma subunit 4 ETHINYLESTRADIOL Calcium Channel Type L, Benzothiazepine 64% 15.42uM 13.706uM View
calcium channel, voltage-dependent, gamma subunit 3 ETHINYLESTRADIOL Calcium Channel Type L, Benzothiazepine 64% 15.42uM 13.706uM View
calcium channel, voltage-dependent, gamma subunit 2 ETHINYLESTRADIOL Calcium Channel Type L, Benzothiazepine 64% 15.42uM 13.706uM View
calcium channel, voltage-dependent, gamma subunit 1 ETHINYLESTRADIOL Calcium Channel Type L, Benzothiazepine 64% 15.42uM 13.706uM View
calcium channel, voltage-dependent, beta 4 subunit ETHINYLESTRADIOL Calcium Channel Type L, Benzothiazepine 64% 15.42uM 13.706uM View
calcium channel, voltage-dependent, beta 3 subunit ETHINYLESTRADIOL Calcium Channel Type L, Benzothiazepine 64% 15.42uM 13.706uM View
calcium channel, voltage-dependent, beta 2 subunit ETHINYLESTRADIOL Calcium Channel Type L, Benzothiazepine 64% 15.42uM 13.706uM View
calcium channel, voltage-dependent, L type, alpha 1S subunit ETHINYLESTRADIOL Calcium Channel Type L, Benzothiazepine 64% 15.42uM 13.706uM View
calcium channel, voltage-dependent, alpha 1F subunit ETHINYLESTRADIOL Calcium Channel Type L, Benzothiazepine 64% 15.42uM 13.706uM View
calcium channel, voltage-dependent, L type, alpha 1D subunit ETHINYLESTRADIOL Calcium Channel Type L, Benzothiazepine 64% 15.42uM 13.706uM View
calcium channel, voltage-dependent, L type, alpha 1C subunit ETHINYLESTRADIOL Calcium Channel Type L, Benzothiazepine 64% 15.42uM 13.706uM View
melanocortin 5 receptor SULOCTIDIL Melanocortin MC5 64% NoneNone NoneNone View
thromboxane A synthase 1 GLYBURIDE Thromboxane Synthetase 64% NoneNone NoneNone View
thromboxane A synthase 1 (platelet, cytochrome P450, family 5, subfamily A) GLYBURIDE Thromboxane Synthetase 64% NoneNone NoneNone View
opioid receptor, sigma 1 CYCLIZINE Sigma1 64% NoneNone NoneNone View
5-hydroxytryptamine receptor 6 CYCLIZINE Serotonin 5-HT6 64% NoneNone NoneNone View
lymphocyte protein tyrosine kinase (mapped) IMATINIB Protein Tyrosine Kinase, Lck 64% NoneNone NoneNone View
opioid receptor, delta 1 CINNARIZINE Opiate delta 64% NoneNone NoneNone View
Cytochrom P450-2C19 monooxygenase MOCLOBEMIDE CYP450-2C19 Inhibition 64% NoneNone NoneNone View
Cytochrom P450-2C19 monooxygenase 4-NONYLPHENOL CYP450-2C19 Inhibition 64% NoneNone NoneNone View
opioid receptor, kappa 1 BITHIONOL Opiate kappa 64% NoneNone NoneNone View
adrenergic receptor, alpha 2b DOBUTAMINE Adrenergic alpha2C 64% NoneNone NoneNone View
adrenergic receptor, alpha 2c (Non-specific probe) DOBUTAMINE Adrenergic alpha2C 64% NoneNone NoneNone View
adrenergic receptor, alpha 1a AMITRAZ Adrenergic alpha1A 64% NoneNone NoneNone View
phosphodiesterase 5A, cGMP-specific CLOSANTEL Phosphodiesterase PDE5 64% NoneNone NoneNone View
phosphodiesterase 5A, cGMP-specific CLOSANTEL Phosphodiesterase PDE5 64% NoneNone NoneNone View
adrenergic receptor, beta 3 ERGOTAMINE Adrenergic beta3 64% NoneNone NoneNone View
cholinergic receptor, muscarinic 2 TERCONAZOLE Muscarinic M2 64% 12.909uM 4.59uM View
calcium channel, voltage-dependent, gamma subunit 8 NELFINAVIR Calcium Channel Type L, Benzothiazepine 64% 14.59uM 12.969uM View
calcium channel, voltage-dependent, gamma subunit 7 NELFINAVIR Calcium Channel Type L, Benzothiazepine 64% 14.59uM 12.969uM View
calcium channel, voltage-dependent, gamma subunit 6 NELFINAVIR Calcium Channel Type L, Benzothiazepine 64% 14.59uM 12.969uM View
calcium channel, voltage-dependent, gamma subunit 5 NELFINAVIR Calcium Channel Type L, Benzothiazepine 64% 14.59uM 12.969uM View
calcium channel, voltage-dependent, gamma subunit 4 NELFINAVIR Calcium Channel Type L, Benzothiazepine 64% 14.59uM 12.969uM View
calcium channel, voltage-dependent, gamma subunit 3 NELFINAVIR Calcium Channel Type L, Benzothiazepine 64% 14.59uM 12.969uM View
calcium channel, voltage-dependent, gamma subunit 2 NELFINAVIR Calcium Channel Type L, Benzothiazepine 64% 14.59uM 12.969uM View
calcium channel, voltage-dependent, gamma subunit 1 NELFINAVIR Calcium Channel Type L, Benzothiazepine 64% 14.59uM 12.969uM View
calcium channel, voltage-dependent, beta 4 subunit NELFINAVIR Calcium Channel Type L, Benzothiazepine 64% 14.59uM 12.969uM View
calcium channel, voltage-dependent, beta 3 subunit NELFINAVIR Calcium Channel Type L, Benzothiazepine 64% 14.59uM 12.969uM View
calcium channel, voltage-dependent, beta 2 subunit NELFINAVIR Calcium Channel Type L, Benzothiazepine 64% 14.59uM 12.969uM View
calcium channel, voltage-dependent, L type, alpha 1S subunit NELFINAVIR Calcium Channel Type L, Benzothiazepine 64% 14.59uM 12.969uM View
interleukin 1 receptor, type I AURANOFIN Interleukin IL-1 alpha 9% NoneNone NoneNone View
calcium channel, voltage-dependent, alpha 1F subunit NELFINAVIR Calcium Channel Type L, Benzothiazepine 64% 14.59uM 12.969uM View
calcium channel, voltage-dependent, L type, alpha 1D subunit NELFINAVIR Calcium Channel Type L, Benzothiazepine 64% 14.59uM 12.969uM View
calcium channel, voltage-dependent, L type, alpha 1C subunit NELFINAVIR Calcium Channel Type L, Benzothiazepine 64% 14.59uM 12.969uM View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit NELFINAVIR Calcium Channel Type L, Benzothiazepine 64% 14.59uM 12.969uM View
estrogen receptor 1 STANOLONE Estrogen ERalpha 63% NoneNone NoneNone View
estrogen receptor 1 STANOLONE Estrogen ERalpha 63% NoneNone NoneNone View
cholinergic receptor, muscarinic 2 TACRINE Muscarinic M2 63% NoneNone NoneNone View
5-hydroxytryptamine (serotonin) receptor 2B TACRINE Serotonin 5-HT2B 63% NoneNone NoneNone View
opioid receptor, kappa 1 METERGOLINE Opiate kappa 63% NoneNone NoneNone View
Sigma-2 Receptor METERGOLINE Sigma2 63% NoneNone NoneNone View
opioid receptor, sigma 1 CYPROHEPTADINE Sigma1 63% NoneNone NoneNone View
androgen receptor ECONAZOLE Testosterone 63% 10.125uM 6.75uM View
acetylcholinesterase (YT blood group) BENZO[A]PYRENE Acetylcholinesterase 63% 28uM NoneNone View
collagen-like tail subunit (single strand of homotrimer) of asymmetric acetylcholinesterase BENZO[A]PYRENE Acetylcholinesterase 63% 28uM NoneNone View
acetylcholinesterase BENZO[A]PYRENE Acetylcholinesterase 63% 28uM NoneNone View
sodium channel, voltage-gated, type IX, alpha DEXCHLORPHENIRAMINE Sodium Channel, Site 2 63% 15.017uM 13.464uM View
sodium channel, voltage-gated, type VII, alpha DEXCHLORPHENIRAMINE Sodium Channel, Site 2 63% 15.017uM 13.464uM View
amiloride-sensitive cation channel 5, intestinal DEXCHLORPHENIRAMINE Sodium Channel, Site 2 63% 15.017uM 13.464uM View
sodium channel, voltage-gated, type III, beta DEXCHLORPHENIRAMINE Sodium Channel, Site 2 63% 15.017uM 13.464uM View
sodium channel, voltage-gated, type VIII, alpha polypeptide DEXCHLORPHENIRAMINE Sodium Channel, Site 2 63% 15.017uM 13.464uM View
sodium channel, voltage-gated, type XI, alpha DEXCHLORPHENIRAMINE Sodium Channel, Site 2 63% 15.017uM 13.464uM View
sodium channel, voltage-gated, type I, beta DEXCHLORPHENIRAMINE Sodium Channel, Site 2 63% 15.017uM 13.464uM View
sodium channel, voltage-gated, type 10, alpha polypeptide DEXCHLORPHENIRAMINE Sodium Channel, Site 2 63% 15.017uM 13.464uM View
sodium channel, voltage-gated, type IV, alpha polypeptide DEXCHLORPHENIRAMINE Sodium Channel, Site 2 63% 15.017uM 13.464uM View
sodium channel, voltage-gated, type V, alpha polypeptide DEXCHLORPHENIRAMINE Sodium Channel, Site 2 63% 15.017uM 13.464uM View
sodium channel, voltage-gated, type II, beta DEXCHLORPHENIRAMINE Sodium Channel, Site 2 63% 15.017uM 13.464uM View
sodium channel, nonvoltage-gated 1 alpha DEXCHLORPHENIRAMINE Sodium Channel, Site 2 63% 15.017uM 13.464uM View
sodium channel, nonvoltage-gated 1 gamma DEXCHLORPHENIRAMINE Sodium Channel, Site 2 63% 15.017uM 13.464uM View
sodium channel, nonvoltage-gated 1 beta DEXCHLORPHENIRAMINE Sodium Channel, Site 2 63% 15.017uM 13.464uM View
sodium channel, voltage-gated, type 2, alpha 1 polypeptide DEXCHLORPHENIRAMINE Sodium Channel, Site 2 63% 15.017uM 13.464uM View
sodium channel, voltage-gated, type XI, alpha DEXCHLORPHENIRAMINE Sodium Channel, Site 2 63% 15.017uM 13.464uM View
sodium channel, nonvoltage-gated 1, gamma DEXCHLORPHENIRAMINE Sodium Channel, Site 2 63% 15.017uM 13.464uM View
sodium channel, nonvoltage-gated 1, delta DEXCHLORPHENIRAMINE Sodium Channel, Site 2 63% 15.017uM 13.464uM View
sodium channel, nonvoltage-gated 1, beta (Liddle syndrome) DEXCHLORPHENIRAMINE Sodium Channel, Site 2 63% 15.017uM 13.464uM View
sodium channel, nonvoltage-gated 1 alpha DEXCHLORPHENIRAMINE Sodium Channel, Site 2 63% 15.017uM 13.464uM View
sodium channel, voltage-gated, type X, alpha DEXCHLORPHENIRAMINE Sodium Channel, Site 2 63% 15.017uM 13.464uM View
sodium channel, voltage-gated, type IX, alpha DEXCHLORPHENIRAMINE Sodium Channel, Site 2 63% 15.017uM 13.464uM View
sodium channel, voltage gated, type VIII, alpha DEXCHLORPHENIRAMINE Sodium Channel, Site 2 63% 15.017uM 13.464uM View
sodium channel, voltage-gated, type VII, alpha DEXCHLORPHENIRAMINE Sodium Channel, Site 2 63% 15.017uM 13.464uM View
sodium channel, voltage-gated, type V, alpha (long QT syndrome 3) DEXCHLORPHENIRAMINE Sodium Channel, Site 2 63% 15.017uM 13.464uM View
sodium channel, voltage-gated, type IV, beta DEXCHLORPHENIRAMINE Sodium Channel, Site 2 63% 15.017uM 13.464uM View
sodium channel, voltage-gated, type IV, alpha DEXCHLORPHENIRAMINE Sodium Channel, Site 2 63% 15.017uM 13.464uM View
sodium channel, voltage-gated, type III, alpha DEXCHLORPHENIRAMINE Sodium Channel, Site 2 63% 15.017uM 13.464uM View
adrenergic receptor, alpha 2a DIPHENHYDRAMINE Adrenergic alpha2A 62% NoneNone NoneNone View
5-hydroxytryptamine (serotonin) receptor 1B S-(-)-PROPRANOLOL Serotonin 5-HT1B 62% NoneNone NoneNone View
calcium channel, voltage-dependent, L type, alpha 1C subunit MEPAZINE Calcium Channel Type L, Benzothiazepine 62% NoneNone NoneNone View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit MEPAZINE Calcium Channel Type L, Benzothiazepine 62% NoneNone NoneNone View
calcium channel, voltage-dependent, beta 1 subunit MEPAZINE Calcium Channel Type L, Benzothiazepine 62% NoneNone NoneNone View
calcium channel, voltage-dependent, L type, alpha 1E subunit MEPAZINE Calcium Channel Type L, Benzothiazepine 62% NoneNone NoneNone View
calcium channel, voltage-dependent, N type, alpha 1B subunit MEPAZINE Calcium Channel Type L, Benzothiazepine 62% NoneNone NoneNone View
calcium channel, voltage-dependent, alpha2/delta subunit 1 MEPAZINE Calcium Channel Type L, Benzothiazepine 62% NoneNone NoneNone View
Cytochrom P450-2D6 monooxygenase LORATADINE CYP450-2D6 Inhibition 62% NoneNone NoneNone View
adrenergic receptor, alpha 2a 2-ACETYLAMINOFLUORENE Adrenergic alpha2A 62% 21.061uM 7.898uM View
5-hydroxytryptamine (serotonin) receptor 2B 1-(2-FLUOROBENZOYL)-4-(PHENYLMETHYL)-PIPERIDINE Serotonin 5-HT2B 62% NoneNone NoneNone View
5-hydroxytryptamine (serotonin) receptor 2B 1-NAPHTHYL ISOTHIOCYANATE Serotonin 5-HT2B 62% 25.158uM 16.009uM View
thromboxane A synthase 1 ITRACONAZOLE Thromboxane Synthetase 62% NoneNone NoneNone View
thromboxane A synthase 1 (platelet, cytochrome P450, family 5, subfamily A) ITRACONAZOLE Thromboxane Synthetase 62% NoneNone NoneNone View
calcium channel, voltage-dependent, L type, alpha 1S subunit GUANETHIDINE Calcium Channel Type L, Phenylalkylamine 62% NoneNone NoneNone View
calcium channel, voltage-dependent, alpha 1F subunit GUANETHIDINE Calcium Channel Type L, Phenylalkylamine 62% NoneNone NoneNone View
calcium channel, voltage-dependent, L type, alpha 1D subunit GUANETHIDINE Calcium Channel Type L, Phenylalkylamine 62% NoneNone NoneNone View
calcium channel, voltage-dependent, L type, alpha 1C subunit GUANETHIDINE Calcium Channel Type L, Phenylalkylamine 62% NoneNone NoneNone View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit GUANETHIDINE Calcium Channel Type L, Phenylalkylamine 62% NoneNone NoneNone View
calcium channel, voltage-dependent, beta 1 subunit GUANETHIDINE Calcium Channel Type L, Phenylalkylamine 62% NoneNone NoneNone View
calcium channel, voltage-dependent, L type, alpha 1E subunit GUANETHIDINE Calcium Channel Type L, Phenylalkylamine 62% NoneNone NoneNone View
calcium channel, voltage-dependent, N type, alpha 1B subunit GUANETHIDINE Calcium Channel Type L, Phenylalkylamine 62% NoneNone NoneNone View
calcium channel, voltage-dependent, alpha2/delta subunit 1 GUANETHIDINE Calcium Channel Type L, Phenylalkylamine 62% NoneNone NoneNone View
histamine receptor H 2 TROGLITAZONE Histamine H2 62% NoneNone NoneNone View